Ligands
Function
Agonist
Agonist
Reference
| Ligand | Amino Acid | Generic Number | Segment | Interaction Type |
|---|---|---|---|---|
| D-tryptophan | S147 | N-term | polar (hydrogen bond) | |
| D-tryptophan | S147 | N-term | Van der Waals | |
| D-tryptophan | A168 | N-term | polar (hydrogen bond with backbone) | |
| D-tryptophan | A168 | N-term | Van der Waals | |
| D-tryptophan | S170 | N-term | polar (hydrogen bond) | |
| D-tryptophan | S170 | N-term | Van der Waals | |
| D-tryptophan | Y218 | N-term | hydrophobic | |
| D-tryptophan | Y218 | N-term | Van der Waals | |
| Calcium | D234 | N-term | polar (charge-charge) | |
| D-tryptophan | E297 | N-term | polar (charge-assisted hydrogen bond) | |
| D-tryptophan | A298 | N-term | Van der Waals | |
| D-tryptophan | A298 | N-term | hydrophobic |
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GPCRdb(A)
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GPCRdb(C)
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CaS receptor
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