PDB
Resolution
2.7 Å
Released
July 3, 2024
Receptor
Class
A
Species
Homo sapiens
Ligand
Function
L-797591
Agonist
Reference
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Ligand Amino Acid Generic Number Segment Interaction Type
L-797591 S110 2.56x56 TM2 Van der Waals
L-797591 L114 2.60x60 TM2 hydrophobic
L-797591 V133 3.28x28 TM3 hydrophobic
L-797591 L134 3.29x29 TM3 hydrophobic
L-797591 D137 3.32x32 TM3 Van der Waals
L-797591 A138 3.33x33 TM3 hydrophobic
L-797591 M141 3.36x36 TM3 hydrophobic
L-797591 I192 4.60x61 TM4 Van der Waals
L-797591 N209 45.51x51 ECL2 Van der Waals
L-797591 M210 45.52x52 ECL2 hydrophobic
L-797591 L220 5.35x36 TM5 hydrophobic
L-797591 F223 5.38x39 TM5 aromatic (edge-to-face)
L-797591 F223 5.38x39 TM5 hydrophobic
L-797591 T227 5.42x43 TM5 hydrophobic
L-797591 W284 6.48x48 TM6 hydrophobic
L-797591 F287 6.51x51 TM6 hydrophobic
L-797591 F287 6.51x51 TM6 aromatic (edge-to-face)
L-797591 Q291 6.55x55 TM6 Van der Waals
L-797591 V309 7.39x38 TM7 hydrophobic
L-797591 G312 7.42x41 TM7 Van der Waals
L-797591 Y313 7.43x42 TM7 hydrophobic
L-797591 Y313 7.43x42 TM7 aromatic (face-to-face)

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Snake plot — Download: PNG | SVG
ICL1 A K M K ICL1ECL1 R H W P F ECL1ICL2 P I K A A R Y R ICL2ECL2 R T A A N S D G T V A C N M L M P E ECL2ICL3 W Q Q R K R S ICL3ECL3 E Q D ECL3N-term M F P N G T A S S P S S S P S P S P G S C G E G G G S R G P G A G A A D G M E E P G R N A S Q N G T L S N-termC-term L S W M D N A A E E P V D Y Y A T A L K S R A Y S V E D F Q P E N L E S G G V F R N G T C T S R I T T L C-term E G Q G S A I L I S F I Y S V V C L V G L C G N S M V I Y V I L R Y T A T N I Y I L N L A I A D E L L M L S V P F L V T S T L L G A L L C R L V L S V D A V N M F T S I Y C L T V L S V D R Y V A V V H R P T V A K V V N L G V W V L S L L V I L P I V V F S P A Q R W L V G F V L Y T F L M G F L L P V G A I C L C Y V L I I A K M R M V A L K A G E R K I T L M V M M V V M V F V I C W M P F Y V V Q L V N V F A D A T V S Q L S V I L G Y A N S C A N P I L Y G F L S D N F Q R F K R S I L C
Helix box plot — Download: PNG | SVG S N G C L G V L C V V S Y I F S I L I A 1 L N L A I A D E L L M L S V P F L V T S 2 V T L C Y I S T F M N V A D V S L V L R 3 A K V V N L G V W V L S L L V I L P I 4 Y C L C I A G V P L L F G M L F T Y L V F 5 M M V V M V F V I C W M P F Y V V Q L V 6 I P N A C S N A Y G L I V S L Q S V T 7

GPCRdb(A)
GPCRdb(A)
SST1 receptor
TM2
2x56 2.56x56 S110
2x60 2.60x60 L114
TM3
3x28 3.28x28 V133
3x29 3.29x29 L134
3x32 3.32x32 D137
3x33 3.33x33 A138
3x36 3.36x36 M141
TM4
4x61 4.60x61 I192
ECL2
45x51 45.51x51 N209
45x52 45.52x52 M210
TM5
5x36 5.35x36 L220
5x39 5.38x39 F223
5x43 5.42x43 T227
TM6
6x48 6.48x48 W284
6x51 6.51x51 F287
6x55 6.55x55 Q291
TM7
7x38 7.39x38 V309
7x41 7.42x41 G312
7x42 7.43x42 Y313