PDB
Resolution
2.8 Å
Released
Aug. 27, 2025
Receptor
Class
A
Species
Homo sapiens
Ligand
DSO-5a
Function
Agonist
Reference
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Ligand Amino Acid Generic Number Segment Interaction Type
DSO-5a L128 3.33x33 TM3 hydrophobic
DSO-5a V131 3.36x36 TM3 hydrophobic
DSO-5a S205 45.52x52 ECL2 polar (hydrogen bond)
DSO-5a S205 45.52x52 ECL2 polar (hydrogen bond)
DSO-5a S205 45.52x52 ECL2 polar (hydrogen bond with backbone)
DSO-5a C221 5.42x43 TM5 Van der Waals
DSO-5a F225 5.46x461 TM5 hydrophobic
DSO-5a F225 5.46x461 TM5 Van der Waals
DSO-5a W284 6.48x48 TM6 hydrophobic
DSO-5a N287 6.51x51 TM6 polar (hydrogen bond)
DSO-5a N287 6.51x51 TM6 polar (hydrogen bond)
DSO-5a H288 6.52x52 TM6 Van der Waals
DSO-5a Y291 6.55x55 TM6 hydrophobic
DSO-5a Y291 6.55x55 TM6 Van der Waals
DSO-5a R316 7.39x38 TM7 polar (charge-assisted hydrogen bond)

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Snake plot — Download: PNG | SVG
ICL1 K S M Q ICL1ECL1 E G W L F ECL1ICL2 P L E R Q P S N ICL2ECL2 N V Y T F R D P N K N M T F E S C T S Y P V S ECL2ICL3 P T E E Q S ICL3ECL3 Q T Y V D P ECL3N-term M A Q R Q P H S P N Q T L I S I T N D T E S S S S V V S N D N T N K G W S G D N S P G N-termC-term C C K A E R P E P P V A D T S L T T L A V M G T V P G T G S I Q M S E I S V T S F T G C S V K Q A E D R F C-term I E A L C A I Y I T Y A V I I S V G I L G N A I L I K V F F K T T V P N I F I T S L A F G D L L L L L T C V P V D A T H Y L A G R I G C K V L S F I R L T S V G V S V F T L T I L S A D R Y K A V V K A I L K T C V K A G C V W I V S M I F A L P E A I F S K K L L Q E I H S L L C F L V F Y I I P L S I I S V Y Y S L I A R T L Y K S T L N I H A R K Q I E S R K R I A R T V L V L V A L F A L C W L P N H L L Y L Y H S F T S S A M H F I F T I F S R V L A F S N S C V N P F A L Y W L S K S F K A F Q K H Q L F
Helix box plot — Download: PNG | SVG A N G L I G V S I I V A Y T I Y I A C L 1 T S L A F G D L L L L T L C V P V D A T H 2 I T L T F V S V G V S T L R I F S L V K 3 T C V K A G C V W I V S M I F A L P E 4 Y Y V S I I S L P I I Y F V L F C L L S H 5 L V L V A L F A L C W L P N H L L Y L Y 6 F P N V C S N S F A L V R S F I T F I 7

GPCRdb(A)
GPCRdb(A)
BB3 receptor
TM3
3x33 3.33x33 L128
3x36 3.36x36 V131
ECL2
45x52 45.52x52 S205
TM5
5x43 5.42x43 C221
5x461 5.46x461 F225
TM6
6x48 6.48x48 W284
6x51 6.51x51 N287
6x52 6.52x52 H288
6x55 6.55x55 Y291
TM7
7x38 7.39x38 R316