PDB
Resolution
2.9 Å
Released
March 4, 2026
Receptor
Class
A
Species
Homo sapiens
Ligand
oridonin
Function
Agonist
Reference
—

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Ligand Amino Acid Generic Number Segment Interaction Type
oridonin C221 5.42x43 TM5 hydrophobic
oridonin N287 6.51x51 TM6 polar (hydrogen bond)
oridonin N287 6.51x51 TM6 Van der Waals
oridonin H288 6.52x52 TM6 Van der Waals
oridonin Y291 6.55x55 TM6 hydrophobic
oridonin Y291 6.55x55 TM6 Van der Waals
oridonin R316 7.39x38 TM7 Van der Waals

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Snake plot — Download: PNG | SVG
ICL1 K S M Q ICL1ECL1 E G W L F ECL1ICL2 P L E R Q P S N ICL2ECL2 N V Y T F R D P N K N M T F E S C T S Y P V S ECL2ICL3 P T E E Q S ICL3ECL3 Q T Y V D P ECL3N-term M A Q R Q P H S P N Q T L I S I T N D T E S S S S V V S N D N T N K G W S G D N S P G N-termC-term C C K A E R P E P P V A D T S L T T L A V M G T V P G T G S I Q M S E I S V T S F T G C S V K Q A E D R F C-term I E A L C A I Y I T Y A V I I S V G I L G N A I L I K V F F K T T V P N I F I T S L A F G D L L L L L T C V P V D A T H Y L A G R I G C K V L S F I R L T S V G V S V F T L T I L S A D R Y K A V V K A I L K T C V K A G C V W I V S M I F A L P E A I F S K K L L Q E I H S L L C F L V F Y I I P L S I I S V Y Y S L I A R T L Y K S T L N I H A R K Q I E S R K R I A R T V L V L V A L F A L C W L P N H L L Y L Y H S F T S S A M H F I F T I F S R V L A F S N S C V N P F A L Y W L S K S F K A F Q K H Q L F
Helix box plot — Download: PNG | SVG A N G L I G V S I I V A Y T I Y I A C L 1 T S L A F G D L L L L T L C V P V D A T H 2 I T L T F V S V G V S T L R I F S L V K 3 T C V K A G C V W I V S M I F A L P E 4 Y Y V S I I S L P I I Y F V L F C L L S H 5 L V L V A L F A L C W L P N H L L Y L Y 6 F P N V C S N S F A L V R S F I T F I 7

GPCRdb(A)
GPCRdb(A)
BB3 receptor
TM5
5x43 5.42x43 C221
TM6
6x51 6.51x51 N287
6x52 6.52x52 H288
6x55 6.55x55 Y291
TM7
7x38 7.39x38 R316