PDB
Resolution
3.2 Å
Released
Feb. 12, 2025
Receptor
Class
A
Species
Homo sapiens
Ligand
#020_E1
Function
Antagonist
Reference
—

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Ligand Amino Acid Generic Number Segment Interaction Type
#020_E1 Y150 3.33x33 TM3 hydrophobic
#020_E1 M153 3.36x36 TM3 hydrophobic
#020_E1 W295 6.48x48 TM6 hydrophobic
#020_E1 I298 6.51x51 TM6 hydrophobic
#020_E1 H299 6.52x52 TM6 aromatic (face-to-edge)
#020_E1 V302 6.55x55 TM6 hydrophobic
#020_E1 I324 7.39x38 TM7 hydrophobic
#020_E1 Y328 7.43x42 TM7 hydrophobic

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Snake plot — Download: PNG | SVG
ICL1 T K M K ICL1ECL1 T W P F ECL1ICL2 P V K A L D F R ICL2ECL2 T T K Y R Q G S I D C T L T F S H ECL2ICL3 R M L S G ICL3ECL3 T I P E ECL3N-term M D S S A A P T N A S N C T D A L A Y S S C S P A P S P G S W V N L S H L D G N L S D P C G P N R T D L G G R D S L C P P T G S P S N-termC-term P T S S N I E Q Q N S T R I R Q N T R D H P S T A N T V D R T N H Q L E N L E A E T A P L P C-term M I T A I T I M A L Y S I V C V V G L F G N F L V M Y V I V R Y T A T N I Y I F N L A L A D A L A T S T L P F Q S V N Y L M G G T I L C K I V I S I D Y Y N M F T S I F T L C T M S V D R Y I A V C H T P R N A K I I N V C N W I L S S A I G L P V M F M A P T W Y W E N L L K I C V F I F A F I M P V L I I T V C Y G L M I L R L K S V S K E K D R N L R R I T R M V L V V V A V F I V C W T P I H I Y V I I K A L V T T F Q T V S W H F C I A L G Y T N S C L N P V L Y A F L D E N F R E F K R C F C I
Helix box plot — Download: PNG | SVG F N G F L G V V C V I S Y L A M I T I A 1 F N L A L A D A L A T S T L P F Q S V N 2 T C L T F I S T F M N Y Y D I S I V I K 3 A K I I N V C N W I L S S A I G L P V M 4 Y C V T I I L V P M I F A F I F V C I K L 5 L V V V A V F I V C W T P I H I Y V I I 6 V P N L C S N T Y G L A I C F H W S V 7

GPCRdb(A)
GPCRdb(A)
μ receptor
TM3
3x33 3.33x33 Y150
3x36 3.36x36 M153
TM6
6x48 6.48x48 W295
6x51 6.51x51 I298
6x52 6.52x52 H299
6x55 6.55x55 V302
TM7
7x38 7.39x38 I324
7x42 7.43x42 Y328