PDB
Resolution
3.1 Å
Released
July 1, 2026
Receptor
Class
A
Species
Homo sapiens
Ligand
Function
3-OH-PCP
Agonist (partial)
Reference
—

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Ligand Amino Acid Generic Number Segment Interaction Type
3-OH-PCP D149 3.32x32 TM3 Van der Waals
3-OH-PCP Y150 3.33x33 TM3 hydrophobic
3-OH-PCP M153 3.36x36 TM3 hydrophobic
3-OH-PCP K235 5.39x40 TM5 Van der Waals
3-OH-PCP I298 6.51x51 TM6 hydrophobic
3-OH-PCP H299 6.52x52 TM6 Van der Waals
3-OH-PCP V302 6.55x55 TM6 hydrophobic
3-OH-PCP W320 7.35x34 TM7 hydrophobic
3-OH-PCP I324 7.39x38 TM7 Van der Waals

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Snake plot — Download: PNG | SVG
ICL1 T K M K ICL1ECL1 T W P F ECL1ICL2 P V K A L D F R ICL2ECL2 T T K Y R Q G S I D C T L T F S H ECL2ICL3 R M L S G ICL3ECL3 T I P E ECL3N-term M D S S A A P T N A S N C T D A L A Y S S C S P A P S P G S W V N L S H L D G N L S D P C G P N R T D L G G R D S L C P P T G S P S N-termC-term P T S S N I E Q Q N S T R I R Q N T R D H P S T A N T V D R T N H Q L E N L E A E T A P L P C-term M I T A I T I M A L Y S I V C V V G L F G N F L V M Y V I V R Y T A T N I Y I F N L A L A D A L A T S T L P F Q S V N Y L M G G T I L C K I V I S I D Y Y N M F T S I F T L C T M S V D R Y I A V C H T P R N A K I I N V C N W I L S S A I G L P V M F M A P T W Y W E N L L K I C V F I F A F I M P V L I I T V C Y G L M I L R L K S V S K E K D R N L R R I T R M V L V V V A V F I V C W T P I H I Y V I I K A L V T T F Q T V S W H F C I A L G Y T N S C L N P V L Y A F L D E N F R E F K R C F C I
Helix box plot — Download: PNG | SVG F N G F L G V V C V I S Y L A M I T I A 1 F N L A L A D A L A T S T L P F Q S V N 2 T C L T F I S T F M N Y Y D I S I V I K 3 A K I I N V C N W I L S S A I G L P V M 4 Y C V T I I L V P M I F A F I F V C I K L 5 L V V V A V F I V C W T P I H I Y V I I 6 V P N L C S N T Y G L A I C F H W S V 7

GPCRdb(A)
GPCRdb(A)
μ receptor
TM3
3x32 3.32x32 D149
3x33 3.33x33 Y150
3x36 3.36x36 M153
TM5
5x40 5.39x40 K235
TM6
6x51 6.51x51 I298
6x52 6.52x52 H299
6x55 6.55x55 V302
TM7
7x34 7.35x34 W320
7x38 7.39x38 I324