PDB
Resolution
3.1 Å
Released
May 20, 2026
Receptor
Class
A
Species
Homo sapiens
Ligand
Function
AR234958
Agonist
Reference
—

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Ligand Amino Acid Generic Number Segment Interaction Type
AR234958 H36 1.36x36 TM1 Van der Waals
AR234958 I84 2.57x57 TM2 hydrophobic
AR234958 L87 2.60x60 TM2 hydrophobic
AR234958 S88 2.61x61 TM2 Van der Waals
AR234958 Y91 2.64x64 TM2 Van der Waals
AR234958 Y95 ECL1 polar (hydrogen bond)
AR234958 Y102 3.22x22 TM3 Van der Waals
AR234958 V106 3.26x26 TM3 Van der Waals
AR234958 S109 3.29x29 TM3 Van der Waals
AR234958 Y168 4.61x61 TM4 Van der Waals
AR234958 Y248 6.55x55 TM6 Van der Waals
AR234958 H262 7.35x34 TM7 aromatic (edge-to-face)
AR234958 H263 7.36x35 TM7 Van der Waals
AR234958 L266 7.39x38 TM7 hydrophobic

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Snake plot — Download: PNG | SVG
ICL1 R R ICL1ECL1 Y E L ECL1ICL2 P I W Y R C H R ICL2ECL2 I D R E E E S H S R N ECL2ICL3 A S H ICL3ECL3 W S T F ECL3N-term M D G S N V T S F V V E E P T N I S T G R N A S V G N A H R Q N-termC-term L T R A F K D E M Q P R R Q K D N C N T V T V E T V V C-term I P I V H W V I M S I S P V G F V E N G I L L W F L C F R M N P F T V Y I T H L S I A D I S L L F C I F I L S I D Y A L D S S G H Y Y T I V T L S V T F L F G Y N T G L Y L L T A I S V E R C L S V L Y P K Y Q S A L V C A L L W A L S C L V T T M E Y V M C D C R A V I I F I A I L S F L V F T P L M L V S S T I L V V K I R K N T W S S K L Y I V I M V T I I I F L I F A M P M R L L Y L L Y Y E Y G N L H H I S L L F S T I N S S A N P F I Y F F V G S S F K E V K K K R S L K V
Helix box plot — Download: PNG | SVG G N E V F G V P S I S M I V W H V I P I 1 T H L S I A D I S L L F C I F I L S I D 2 A T L L Y L G T N Y G F L F T V S L T V 3 S A L V C A L L W A L S C L V T T M E Y 4 I T S S V L M L P T F V L F S L I A I F I 5 M V T I I I F L I F A M P M R L L Y L L 6 F P N A S S N I T S F L L S I H H L N 7

GPCRdb(A)
GPCRdb(A)
MAS1
TM1
1x36 1.36x36 H36
TM2
2x57 2.57x57 I84
2x60 2.60x60 L87
2x61 2.61x61 S88
2x64 2.64x64 Y91
TM3
3x22 3.22x22 Y102
3x26 3.26x26 V106
3x29 3.29x29 S109
TM4
4x61 4.61x61 Y168
TM6
6x55 6.55x55 Y248
TM7
7x34 7.35x34 H262
7x35 7.36x35 H263
7x38 7.39x38 L266