relaxin-3
SMILES | None |
InChIKey | None |
Sequence | None |
Chemical properties
Hydrogen bond acceptors | None |
Hydrogen bond donors | None |
Rotatable bonds | None |
Molecular weight (Da) |
Drug properties
Molecular type | Peptide |
Physiological/Surrogate | Endogenous |
Approved drug | No |
Database connections
Bioactivities
Receptor | Activity | Source | |||||||
---|---|---|---|---|---|---|---|---|---|
GTP | Uniprot | Species | Family | Class | Type | Min | Avg | Max | Database |
RXFP1 | RXFP1 | Human | Relaxin family peptide | A | pKi | 7.5 | 7.75 | 8.0 | Guide to Pharmacology |
RXFP2 | RXFP2 | Human | Relaxin family peptide | A | pKi | 7.0 | 7.0 | 7.0 | Guide to Pharmacology |
RXFP3 | RL3R1 | Human | Relaxin family peptide | A | pKi | 7.78 | 8.35 | 8.92 | Guide to Pharmacology |
RXFP4 | RL3R2 | Human | Relaxin family peptide | A | pKi | 8.81 | 8.91 | 8.83 | Guide to Pharmacology |
Receptor | Activity | Source | |||||||
---|---|---|---|---|---|---|---|---|---|
GTP | Uniprot | Species | Family | Class | Type | Min | Avg | Max | Database |
RXFP3 | RL3R1 | Human | Relaxin family peptide | A | pIC50 | 9.4 | 9.5 | 9.6 | Guide to Pharmacology |
RXFP3 | RL3R1 | Human | Relaxin family peptide | A | pEC50 | 8.26 | 9.1 | 9.93 | Guide to Pharmacology |
RXFP4 | RL3R2 | Human | Relaxin family peptide | A | pIC50 | 8.8 | 8.9 | 9.0 | Guide to Pharmacology |
RXFP4 | RL3R2 | Human | Relaxin family peptide | A | pEC50 | 8.7 | 9.2 | 9.7 | Guide to Pharmacology |