SRIF-28


SMILES None
InChIKey GGYTXJNZMFRSLX-DFTNLTQTSA-N
Sequence SANSNPAMAPRERKAGCKNFFWKTFTSC

Chemical properties

Hydrogen bond acceptors None
Hydrogen bond donors None
Rotatable bonds None
Molecular weight (Da)

Drug properties

Molecular type Peptide
Physiological/Surrogate Endogenous
Approved drug No

Database connections

Bioactivities

Receptor Activity Source
GTP Uniprot Species Family Class Type Min Avg Max Database
SST1 SSR1 Human Somatostatin A pKi 8.6 9.0 9.4 Guide to Pharmacology
SST3 SSR3 Human Somatostatin A pKi 8.1 9.0 9.9 Guide to Pharmacology
SST4 SSR4 Human Somatostatin A pKi 8.1 8.65 9.2 Guide to Pharmacology
SST5 SSR5 Human Somatostatin A pKi 9.2 9.75 10.3 Guide to Pharmacology
SST5 SSR5 Rat Somatostatin A pKi 9.0 9.0 9.0 Guide to Pharmacology
SST2 SSR2 Rat Somatostatin A pKi 8.8 8.8 8.8 Guide to Pharmacology
SST5 SSR5 Mouse Somatostatin A pKi 9.8 9.85 9.9 Guide to Pharmacology
SST3 SSR3 Rat Somatostatin A pKi 9.1 9.1 9.1 Guide to Pharmacology
SST2 SSR2 Human Somatostatin A pKi 8.4 9.3 10.2 Guide to Pharmacology
Receptor Activity Source
GTP Uniprot Species Family Class Type Min Avg Max Database
MRGPRX2 MRGX2 Human A orphans A pEC50 5.38 5.38 5.38 Guide to Pharmacology
SST3 SSR3 Mouse Somatostatin A pIC50 10.2 10.2 10.2 Guide to Pharmacology
SST2 SSR2 Human Somatostatin A pEC50 8.64 8.64 8.64 ChEMBL
SST2 SSR2 Mouse Somatostatin A pIC50 9.0 9.25 9.5 Guide to Pharmacology