[Leu9,des-Arg10]kallidin
SMILES | None |
InChIKey | AGTPZUQKOYEAOH-MDKUUQCZSA-N |
Sequence | KRPPGFSPL |
Chemical properties
Hydrogen bond acceptors | None |
Hydrogen bond donors | None |
Rotatable bonds | None |
Molecular weight (Da) |
Drug properties
Molecular type | Peptide |
Physiological/Surrogate | Surrogate |
Approved drug | No |
Database connections
Bioactivities
Receptor | Activity | Source | |||||||
---|---|---|---|---|---|---|---|---|---|
GTP | Uniprot | Species | Family | Class | Type | Min | Avg | Max | Database |
B1 | BKRB1 | Human | Bradykinin | A | pKi | 9.1 | 9.2 | 9.3 | Guide to Pharmacology |
B1 | BKRB1 | Mouse | Bradykinin | A | pKi | 8.1 | 8.1 | 8.1 | Guide to Pharmacology |
Receptor | Activity | Source | |||||||
---|---|---|---|---|---|---|---|---|---|
GTP | Uniprot | Species | Family | Class | Type | Min | Avg | Max | Database |
B1 | BKRB1 | Human | Bradykinin | A | pIC50 | 8.9 | 8.9 | 8.9 | Guide to Pharmacology |
B1 | BKRB1 | Mouse | Bradykinin | A | pA2 | 7.0 | 7.0 | 7.0 | Guide to Pharmacology |
B1 | BKRB1 | Human | Bradykinin | A | pIC50 | 6.0 | 6.0 | 6.0 | ChEMBL |