[Lys15,Arg16,Leu27]VIP-(1-7)/GRF-(8-27)-NH2
SMILES | None |
InChIKey | None |
Sequence | HSDAVFTNSYRKVLKRLSARKLLQDIL |
Chemical properties
Hydrogen bond acceptors | None |
Hydrogen bond donors | None |
Rotatable bonds | None |
Molecular weight (Da) |
Drug properties
Molecular type | Peptide |
Physiological/Surrogate | Surrogate |
Approved drug | No |
Database connections
Ligand site mutations | VPAC1 |
Bioactivities
Receptor | Activity | Source | |||||||
---|---|---|---|---|---|---|---|---|---|
GTP | Uniprot | Species | Family | Class | Type | Min | Avg | Max | Database |
Receptor | Activity | Source | |||||||
---|---|---|---|---|---|---|---|---|---|
GTP | Uniprot | Species | Family | Class | Type | Min | Avg | Max | Database |
VPAC1 | VIPR1 | Human | VIP and PACAP | B1 | pIC50 | 8.35 | 8.35 | 8.35 | Guide to Pharmacology |
VPAC1 | VIPR1 | Human | VIP and PACAP | B1 | pEC50 | 8.3 | 8.3 | 8.3 | Guide to Pharmacology |
VPAC2 | VIPR2 | Human | VIP and PACAP | B1 | pIC50 | 5.25 | 5.25 | 5.25 | Guide to Pharmacology |
VPAC2 | VIPR2 | Human | VIP and PACAP | B1 | pEC50 | 6.0 | 6.0 | 6.0 | Guide to Pharmacology |
VPAC1 | VIPR1 | Rat | VIP and PACAP | B1 | pIC50 | 8.7 | 8.7 | 8.7 | Guide to Pharmacology |
VPAC2 | VIPR2 | Rat | VIP and PACAP | B1 | pIC50 | 4.5 | 4.5 | 4.5 | Guide to Pharmacology |
PAC1 | PACR | Human | VIP and PACAP | B1 | pIC50 | 6.0 | 6.0 | 6.0 | Guide to Pharmacology |
PAC1 | PACR | Human | VIP and PACAP | B1 | pEC50 | 6.0 | 6.0 | 6.0 | Guide to Pharmacology |