Ligand source activities (1 row/activity)
| Ligands (move mouse cursor over ligand name to see structure) | Receptor | Assay information | Chemical information | ||||||||||||||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Sel. page | Common name |
GPCRdb ID |
#Vendors |
Reference ligand |
Fold selectivity |
# Tested GPCRs |
Species |
p-value (-log) |
Activity Type |
Activity Relation |
Activity Value |
AssayType |
Assay Description |
Source |
Mol weight |
Rot Bonds |
H don |
H acc |
LogP |
Smiles |
DOI |
| 1023 | 8454 | 0 | None | -10000 | 5 | Human | 6.0 | pEC50 | = | 6 | Functional | Guide to Pharmacology | None | None | None | None | 16025565 | ||||
| 3935 | 8399 | 0 | None | 50 | 2 | Human | 8.1 | pEC50 | = | 8.1 | Functional | Guide to Pharmacology | None | None | None | None | 15623572 | ||||
| 1048 | 10857 | 0 | None | -11 | 4 | Human | 8.5 | pEC50 | = | 8.5 | Functional | Guide to Pharmacology | None | None | None | None | 11285256 | ||||
| 1046 | 8722 | 0 | None | - | 1 | Human | 5.0 | pEC50 | None | 5 | Functional | Guide to Pharmacology | None | None | None | None | 11602630 | ||||
| 155817387 | 8722 | 0 | None | - | 1 | Human | 5.0 | pEC50 | None | 5 | Functional | Guide to Pharmacology | None | None | None | None | 11602630 | ||||
| 16131967 | 8722 | 0 | None | - | 1 | Human | 5.0 | pEC50 | None | 5 | Functional | Guide to Pharmacology | None | None | None | None | 11602630 | ||||
| 1044 | 7213 | 0 | None | 1 | 3 | Human | 6.0 | pEC50 | None | 6 | Functional | Guide to Pharmacology | None | None | None | None | 15187149 | ||||
| 1047 | 8733 | 17 | None | 3 | 4 | Human | 9.0 | pEC50 | None | 9.0 | Functional | Guide to Pharmacology | None | None | None | None | 15465011 | ||||
| 16131438 | 8733 | 17 | None | 3 | 4 | Human | 9.0 | pEC50 | None | 9.0 | Functional | Guide to Pharmacology | None | None | None | None | 15465011 | ||||
| 56947109 | 8733 | 17 | None | 3 | 4 | Human | 9.0 | pEC50 | None | 9.0 | Functional | Guide to Pharmacology | None | None | None | None | 15465011 | ||||
| CHEMBL4447799 | 8733 | 17 | None | 3 | 4 | Human | 9.0 | pEC50 | None | 9.0 | Functional | Guide to Pharmacology | None | None | None | None | 15465011 | ||||
| 1040 | 10866 | 0 | None | -4 | 2 | Human | 6.0 | pIC50 | None | 6 | Functional | Guide to Pharmacology | None | None | None | None | 16476585 | ||||
| Ligands (move mouse cursor over ligand name to see structure) | Receptor | Assay information | Chemical information | |||||||||||||||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Sel. page | Similar- ity |
Common name |
GPCRdb ID |
#Vendors |
Reference ligand |
Fold selectivity |
# Tested GPCRs |
Species |
p-value (-log) |
Activity Type |
Activity Relation |
Activity Value |
Assay Type |
Assay Description |
Source |
Mol weight |
Rot Bonds |
H don |
H acc |
LogP |
Smiles |
DOI |