Biased Signaling Atlas

Ligand source activities (1 row/activity)

Potency
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Ligands					Receptor			Assay information							Chemical information
Sel. page	Common name	GPCRdb ID	#Vendors	Reference ligand	Fold selectivity (Potency)	# tested GPCRs (Potency)	Species	p-value (-log)	Type	Activity Relation	Activity Value	Assay Type	Assay Description	Source	Mol weight	Rot Bonds	H don	H acc	LogP	Smiles	DOI
	1902746	31853	7	None	-	1	Human	4.3	pEC50	=	4.3	Functional	PUBCHEM_BIOASSAY: Dose Response cell-based high-throughput screening assay to identify agonists of galanin receptor 2 (GALR2). (Class of assay: confirmatory) [Related pubchem assays: 864 ]PUBCHEM_BIOASSAY: Dose Response cell-based high-throughput screening assay to identify agonists of galanin receptor 2 (GALR2). (Class of assay: confirmatory) [Related pubchem assays: 864 ]	ChEMBL	360	6	1	5	3.8	C=CCNC(=O)/C(C#N)=C/c1cn(-c2ccccc2)nc1-c1cccs1	nan
	CHEMBL1408432	31853	7	None	-	1	Human	4.3	pEC50	=	4.3	Functional	PUBCHEM_BIOASSAY: Dose Response cell-based high-throughput screening assay to identify agonists of galanin receptor 2 (GALR2). (Class of assay: confirmatory) [Related pubchem assays: 864 ]PUBCHEM_BIOASSAY: Dose Response cell-based high-throughput screening assay to identify agonists of galanin receptor 2 (GALR2). (Class of assay: confirmatory) [Related pubchem assays: 864 ]	ChEMBL	360	6	1	5	3.8	C=CCNC(=O)/C(C#N)=C/c1cn(-c2ccccc2)nc1-c1cccs1	nan
	4104905	36272	7	None	1	3	Human	5.0	pIC50	=	5.0	Functional	PUBCHEM_BIOASSAY: Dose Response cell-based high-throughput screening assay to identify antagonists of galanin receptor 2 (GALR2). (Class of assay: confirmatory) [Related pubchem assays: 828, 866 ]PUBCHEM_BIOASSAY: Dose Response cell-based high-throughput screening assay to identify antagonists of galanin receptor 2 (GALR2). (Class of assay: confirmatory) [Related pubchem assays: 828, 866 ]	ChEMBL	297	5	1	7	1.6	CCOC(=O)c1cc([N+](=O)[O-])c([N+](=O)[O-])cc1NC(C)=O	nan
	CHEMBL1447697	36272	7	None	1	3	Human	5.0	pIC50	=	5.0	Functional	PUBCHEM_BIOASSAY: Dose Response cell-based high-throughput screening assay to identify antagonists of galanin receptor 2 (GALR2). (Class of assay: confirmatory) [Related pubchem assays: 828, 866 ]PUBCHEM_BIOASSAY: Dose Response cell-based high-throughput screening assay to identify antagonists of galanin receptor 2 (GALR2). (Class of assay: confirmatory) [Related pubchem assays: 828, 866 ]	ChEMBL	297	5	1	7	1.6	CCOC(=O)c1cc([N+](=O)[O-])c([N+](=O)[O-])cc1NC(C)=O	nan
	1478923	51698	16	None	-1	2	Human	5.0	pIC50	=	5.0	Functional	PUBCHEM_BIOASSAY: Dose Response cell-based high-throughput screening assay to identify antagonists of galanin receptor 2 (GALR2). (Class of assay: confirmatory) [Related pubchem assays: 828, 866 ]PUBCHEM_BIOASSAY: Dose Response cell-based high-throughput screening assay to identify antagonists of galanin receptor 2 (GALR2). (Class of assay: confirmatory) [Related pubchem assays: 828, 866 ]	ChEMBL	265	4	1	4	2.9	O=C(/C=C/Sc1nc[nH]n1)c1ccc(Cl)cc1	nan
	CHEMBL1586531	51698	16	None	-1	2	Human	5.0	pIC50	=	5.0	Functional	PUBCHEM_BIOASSAY: Dose Response cell-based high-throughput screening assay to identify antagonists of galanin receptor 2 (GALR2). (Class of assay: confirmatory) [Related pubchem assays: 828, 866 ]PUBCHEM_BIOASSAY: Dose Response cell-based high-throughput screening assay to identify antagonists of galanin receptor 2 (GALR2). (Class of assay: confirmatory) [Related pubchem assays: 828, 866 ]	ChEMBL	265	4	1	4	2.9	O=C(/C=C/Sc1nc[nH]n1)c1ccc(Cl)cc1	nan
	638439	103322	69	None	2	2	Human	5.0	pIC50	=	5.0	Functional	PUBCHEM_BIOASSAY: Dose response counterscreen for antagonists of galanin receptor 2 (GalR2): a cell-based high-throughput screening assay for inhibitors of beta-lactamase activity. (Class of assay: confirmatory) [Related pubchem assays: 828, 1225, 866 ]PUBCHEM_BIOASSAY: Dose response counterscreen for antagonists of galanin receptor 2 (GalR2): a cell-based high-throughput screening assay for inhibitors of beta-lactamase activity. (Class of assay: confirmatory) [Related pubchem assays: 828, 1225, 866 ]	ChEMBL	195	3	1	4	1.6	COc1cc(/C=C/[N+](=O)[O-])ccc1O	nan
	CHEMBL309016	103322	69	None	2	2	Human	5.0	pIC50	=	5.0	Functional	PUBCHEM_BIOASSAY: Dose response counterscreen for antagonists of galanin receptor 2 (GalR2): a cell-based high-throughput screening assay for inhibitors of beta-lactamase activity. (Class of assay: confirmatory) [Related pubchem assays: 828, 1225, 866 ]PUBCHEM_BIOASSAY: Dose response counterscreen for antagonists of galanin receptor 2 (GalR2): a cell-based high-throughput screening assay for inhibitors of beta-lactamase activity. (Class of assay: confirmatory) [Related pubchem assays: 828, 1225, 866 ]	ChEMBL	195	3	1	4	1.6	COc1cc(/C=C/[N+](=O)[O-])ccc1O	nan
	4686258	51569	7	None	-	1	Human	5.9	pIC50	=	5.9	Functional	PUBCHEM_BIOASSAY: Dose Response cell-based high-throughput screening assay to identify antagonists of galanin receptor 2 (GALR2). (Class of assay: confirmatory) [Related pubchem assays: 828, 866 ]PUBCHEM_BIOASSAY: Dose Response cell-based high-throughput screening assay to identify antagonists of galanin receptor 2 (GALR2). (Class of assay: confirmatory) [Related pubchem assays: 828, 866 ]	ChEMBL	278	4	2	8	1.5	CNc1nc2cc([N+](=O)[O-])c([N+](=O)[O-])cc2nc1NC	nan
	CHEMBL1585420	51569	7	None	-	1	Human	5.9	pIC50	=	5.9	Functional	PUBCHEM_BIOASSAY: Dose Response cell-based high-throughput screening assay to identify antagonists of galanin receptor 2 (GALR2). (Class of assay: confirmatory) [Related pubchem assays: 828, 866 ]PUBCHEM_BIOASSAY: Dose Response cell-based high-throughput screening assay to identify antagonists of galanin receptor 2 (GALR2). (Class of assay: confirmatory) [Related pubchem assays: 828, 866 ]	ChEMBL	278	4	2	8	1.5	CNc1nc2cc([N+](=O)[O-])c([N+](=O)[O-])cc2nc1NC	nan
	3775080	37609	17	None	-1	2	Human	4.8	pIC50	=	4.8	Functional	PUBCHEM_BIOASSAY: Dose Response cell-based high-throughput screening assay to identify antagonists of galanin receptor 2 (GALR2). (Class of assay: confirmatory) [Related pubchem assays: 828, 866 ]PUBCHEM_BIOASSAY: Dose Response cell-based high-throughput screening assay to identify antagonists of galanin receptor 2 (GALR2). (Class of assay: confirmatory) [Related pubchem assays: 828, 866 ]	ChEMBL	306	4	0	6	2.9	CC(=O)SC(C[N+](=O)[O-])c1cn(C(C)=O)c2ccccc12	nan
	CHEMBL1458812	37609	17	None	-1	2	Human	4.8	pIC50	=	4.8	Functional	PUBCHEM_BIOASSAY: Dose Response cell-based high-throughput screening assay to identify antagonists of galanin receptor 2 (GALR2). (Class of assay: confirmatory) [Related pubchem assays: 828, 866 ]PUBCHEM_BIOASSAY: Dose Response cell-based high-throughput screening assay to identify antagonists of galanin receptor 2 (GALR2). (Class of assay: confirmatory) [Related pubchem assays: 828, 866 ]	ChEMBL	306	4	0	6	2.9	CC(=O)SC(C[N+](=O)[O-])c1cn(C(C)=O)c2ccccc12	nan
	1478923	51698	16	None	-1	2	Human	4.8	pIC50	=	4.8	Functional	PUBCHEM_BIOASSAY: Dose response counterscreen for antagonists of galanin receptor 2 (GalR2): a cell-based high-throughput screening assay for inhibitors of beta-lactamase activity. (Class of assay: confirmatory) [Related pubchem assays: 828, 1225, 866 ]PUBCHEM_BIOASSAY: Dose response counterscreen for antagonists of galanin receptor 2 (GalR2): a cell-based high-throughput screening assay for inhibitors of beta-lactamase activity. (Class of assay: confirmatory) [Related pubchem assays: 828, 1225, 866 ]	ChEMBL	265	4	1	4	2.9	O=C(/C=C/Sc1nc[nH]n1)c1ccc(Cl)cc1	nan
	CHEMBL1586531	51698	16	None	-1	2	Human	4.8	pIC50	=	4.8	Functional	PUBCHEM_BIOASSAY: Dose response counterscreen for antagonists of galanin receptor 2 (GalR2): a cell-based high-throughput screening assay for inhibitors of beta-lactamase activity. (Class of assay: confirmatory) [Related pubchem assays: 828, 1225, 866 ]PUBCHEM_BIOASSAY: Dose response counterscreen for antagonists of galanin receptor 2 (GalR2): a cell-based high-throughput screening assay for inhibitors of beta-lactamase activity. (Class of assay: confirmatory) [Related pubchem assays: 828, 1225, 866 ]	ChEMBL	265	4	1	4	2.9	O=C(/C=C/Sc1nc[nH]n1)c1ccc(Cl)cc1	nan
	3775080	37609	17	None	-1	2	Human	4.8	pIC50	=	4.8	Functional	PUBCHEM_BIOASSAY: Dose response counterscreen for antagonists of galanin receptor 2 (GalR2): a cell-based high-throughput screening assay for inhibitors of beta-lactamase activity. (Class of assay: confirmatory) [Related pubchem assays: 828, 1225, 866 ]PUBCHEM_BIOASSAY: Dose response counterscreen for antagonists of galanin receptor 2 (GalR2): a cell-based high-throughput screening assay for inhibitors of beta-lactamase activity. (Class of assay: confirmatory) [Related pubchem assays: 828, 1225, 866 ]	ChEMBL	306	4	0	6	2.9	CC(=O)SC(C[N+](=O)[O-])c1cn(C(C)=O)c2ccccc12	nan
	CHEMBL1458812	37609	17	None	-1	2	Human	4.8	pIC50	=	4.8	Functional	PUBCHEM_BIOASSAY: Dose response counterscreen for antagonists of galanin receptor 2 (GalR2): a cell-based high-throughput screening assay for inhibitors of beta-lactamase activity. (Class of assay: confirmatory) [Related pubchem assays: 828, 1225, 866 ]PUBCHEM_BIOASSAY: Dose response counterscreen for antagonists of galanin receptor 2 (GalR2): a cell-based high-throughput screening assay for inhibitors of beta-lactamase activity. (Class of assay: confirmatory) [Related pubchem assays: 828, 1225, 866 ]	ChEMBL	306	4	0	6	2.9	CC(=O)SC(C[N+](=O)[O-])c1cn(C(C)=O)c2ccccc12	nan
	2585250	28145	7	None	-5	3	Human	4.8	pIC50	=	4.8	Functional	PUBCHEM_BIOASSAY: Dose response counterscreen for antagonists of galanin receptor 2 (GalR2): a cell-based high-throughput screening assay for inhibitors of beta-lactamase activity. (Class of assay: confirmatory) [Related pubchem assays: 828, 1225, 866 ]PUBCHEM_BIOASSAY: Dose response counterscreen for antagonists of galanin receptor 2 (GalR2): a cell-based high-throughput screening assay for inhibitors of beta-lactamase activity. (Class of assay: confirmatory) [Related pubchem assays: 828, 1225, 866 ]	ChEMBL	396	6	1	5	2.2	CCc1ccccc1NC(=O)CN(C)C(=O)Cn1ncc(Cl)c(Cl)c1=O	nan
	CHEMBL1374788	28145	7	None	-5	3	Human	4.8	pIC50	=	4.8	Functional	PUBCHEM_BIOASSAY: Dose response counterscreen for antagonists of galanin receptor 2 (GalR2): a cell-based high-throughput screening assay for inhibitors of beta-lactamase activity. (Class of assay: confirmatory) [Related pubchem assays: 828, 1225, 866 ]PUBCHEM_BIOASSAY: Dose response counterscreen for antagonists of galanin receptor 2 (GalR2): a cell-based high-throughput screening assay for inhibitors of beta-lactamase activity. (Class of assay: confirmatory) [Related pubchem assays: 828, 1225, 866 ]	ChEMBL	396	6	1	5	2.2	CCc1ccccc1NC(=O)CN(C)C(=O)Cn1ncc(Cl)c(Cl)c1=O	nan
	5335764	45653	8	None	-	1	Human	4.8	pIC50	=	4.8	Functional	PUBCHEM_BIOASSAY: Dose response counterscreen for antagonists of galanin receptor 2 (GalR2): a cell-based high-throughput screening assay for inhibitors of beta-lactamase activity. (Class of assay: confirmatory) [Related pubchem assays: 828, 1225, 866 ]PUBCHEM_BIOASSAY: Dose response counterscreen for antagonists of galanin receptor 2 (GalR2): a cell-based high-throughput screening assay for inhibitors of beta-lactamase activity. (Class of assay: confirmatory) [Related pubchem assays: 828, 1225, 866 ]	ChEMBL	342	5	1	3	4.5	Cc1cccc(C(=O)Nc2ccc(C(=O)/C=C/c3cccnc3)cc2)c1	nan
	CHEMBL1531933	45653	8	None	-	1	Human	4.8	pIC50	=	4.8	Functional	PUBCHEM_BIOASSAY: Dose response counterscreen for antagonists of galanin receptor 2 (GalR2): a cell-based high-throughput screening assay for inhibitors of beta-lactamase activity. (Class of assay: confirmatory) [Related pubchem assays: 828, 1225, 866 ]PUBCHEM_BIOASSAY: Dose response counterscreen for antagonists of galanin receptor 2 (GalR2): a cell-based high-throughput screening assay for inhibitors of beta-lactamase activity. (Class of assay: confirmatory) [Related pubchem assays: 828, 1225, 866 ]	ChEMBL	342	5	1	3	4.5	Cc1cccc(C(=O)Nc2ccc(C(=O)/C=C/c3cccnc3)cc2)c1	nan
	5335764	45653	8	None	-	1	Human	4.7	pIC50	=	4.7	Functional	PUBCHEM_BIOASSAY: Dose Response cell-based high-throughput screening assay to identify antagonists of galanin receptor 2 (GALR2). (Class of assay: confirmatory) [Related pubchem assays: 828, 866 ]PUBCHEM_BIOASSAY: Dose Response cell-based high-throughput screening assay to identify antagonists of galanin receptor 2 (GALR2). (Class of assay: confirmatory) [Related pubchem assays: 828, 866 ]	ChEMBL	342	5	1	3	4.5	Cc1cccc(C(=O)Nc2ccc(C(=O)/C=C/c3cccnc3)cc2)c1	nan
	CHEMBL1531933	45653	8	None	-	1	Human	4.7	pIC50	=	4.7	Functional	PUBCHEM_BIOASSAY: Dose Response cell-based high-throughput screening assay to identify antagonists of galanin receptor 2 (GALR2). (Class of assay: confirmatory) [Related pubchem assays: 828, 866 ]PUBCHEM_BIOASSAY: Dose Response cell-based high-throughput screening assay to identify antagonists of galanin receptor 2 (GALR2). (Class of assay: confirmatory) [Related pubchem assays: 828, 866 ]	ChEMBL	342	5	1	3	4.5	Cc1cccc(C(=O)Nc2ccc(C(=O)/C=C/c3cccnc3)cc2)c1	nan
	5064340	40182	1	None	-	1	Human	4.3	pIC50	=	4.3	Functional	PUBCHEM_BIOASSAY: Dose Response cell-based high-throughput screening assay to identify antagonists of galanin receptor 2 (GALR2). (Class of assay: confirmatory) [Related pubchem assays: 828, 866 ]PUBCHEM_BIOASSAY: Dose Response cell-based high-throughput screening assay to identify antagonists of galanin receptor 2 (GALR2). (Class of assay: confirmatory) [Related pubchem assays: 828, 866 ]	ChEMBL	337	3	2	5	5.4	Nc1[nH]c(N=Nc2nc(-c3ccc(F)cc3)cs2)c2ccccc12	nan
	CHEMBL1482215	40182	1	None	-	1	Human	4.3	pIC50	=	4.3	Functional	PUBCHEM_BIOASSAY: Dose Response cell-based high-throughput screening assay to identify antagonists of galanin receptor 2 (GALR2). (Class of assay: confirmatory) [Related pubchem assays: 828, 866 ]PUBCHEM_BIOASSAY: Dose Response cell-based high-throughput screening assay to identify antagonists of galanin receptor 2 (GALR2). (Class of assay: confirmatory) [Related pubchem assays: 828, 866 ]	ChEMBL	337	3	2	5	5.4	Nc1[nH]c(N=Nc2nc(-c3ccc(F)cc3)cs2)c2ccccc12	nan
	919665	24376	7	None	-	1	Human	4.3	pIC50	=	4.3	Functional	PUBCHEM_BIOASSAY: Dose Response cell-based high-throughput screening assay to identify antagonists of galanin receptor 2 (GALR2). (Class of assay: confirmatory) [Related pubchem assays: 828, 866 ]PUBCHEM_BIOASSAY: Dose Response cell-based high-throughput screening assay to identify antagonists of galanin receptor 2 (GALR2). (Class of assay: confirmatory) [Related pubchem assays: 828, 866 ]	ChEMBL	343	2	1	5	2.5	CCOC(=O)N1CCN(c2[nH]cnc3c4cc(F)ccc4nc2-3)CC1	nan
	CHEMBL1342746	24376	7	None	-	1	Human	4.3	pIC50	=	4.3	Functional	PUBCHEM_BIOASSAY: Dose Response cell-based high-throughput screening assay to identify antagonists of galanin receptor 2 (GALR2). (Class of assay: confirmatory) [Related pubchem assays: 828, 866 ]PUBCHEM_BIOASSAY: Dose Response cell-based high-throughput screening assay to identify antagonists of galanin receptor 2 (GALR2). (Class of assay: confirmatory) [Related pubchem assays: 828, 866 ]	ChEMBL	343	2	1	5	2.5	CCOC(=O)N1CCN(c2[nH]cnc3c4cc(F)ccc4nc2-3)CC1	nan
	2585042	46582	7	None	-3	4	Human	5.3	pIC50	=	5.3	Functional	PUBCHEM_BIOASSAY: Dose Response cell-based high-throughput screening assay to identify antagonists of galanin receptor 2 (GALR2). (Class of assay: confirmatory) [Related pubchem assays: 828, 866 ]PUBCHEM_BIOASSAY: Dose Response cell-based high-throughput screening assay to identify antagonists of galanin receptor 2 (GALR2). (Class of assay: confirmatory) [Related pubchem assays: 828, 866 ]	ChEMBL	480	4	0	6	2.2	O=C(Cn1ncc(Cl)c(Cl)c1=O)N1CCN(S(=O)(=O)c2ccc3ccccc3c2)CC1	nan
	CHEMBL1540377	46582	7	None	-3	4	Human	5.3	pIC50	=	5.3	Functional	PUBCHEM_BIOASSAY: Dose Response cell-based high-throughput screening assay to identify antagonists of galanin receptor 2 (GALR2). (Class of assay: confirmatory) [Related pubchem assays: 828, 866 ]PUBCHEM_BIOASSAY: Dose Response cell-based high-throughput screening assay to identify antagonists of galanin receptor 2 (GALR2). (Class of assay: confirmatory) [Related pubchem assays: 828, 866 ]	ChEMBL	480	4	0	6	2.2	O=C(Cn1ncc(Cl)c(Cl)c1=O)N1CCN(S(=O)(=O)c2ccc3ccccc3c2)CC1	nan
	1345012	34763	9	None	-	1	Human	5.2	pIC50	=	5.2	Functional	PUBCHEM_BIOASSAY: Dose Response cell-based high-throughput screening assay to identify antagonists of galanin receptor 2 (GALR2). (Class of assay: confirmatory) [Related pubchem assays: 828, 866 ]PUBCHEM_BIOASSAY: Dose Response cell-based high-throughput screening assay to identify antagonists of galanin receptor 2 (GALR2). (Class of assay: confirmatory) [Related pubchem assays: 828, 866 ]	ChEMBL	425	5	3	4	4.7	O=C(/C=C/c1ccc(Cl)cc1)NC(=S)Nc1ccc(NC(=O)c2ccco2)cc1	nan
	CHEMBL1432794	34763	9	None	-	1	Human	5.2	pIC50	=	5.2	Functional	PUBCHEM_BIOASSAY: Dose Response cell-based high-throughput screening assay to identify antagonists of galanin receptor 2 (GALR2). (Class of assay: confirmatory) [Related pubchem assays: 828, 866 ]PUBCHEM_BIOASSAY: Dose Response cell-based high-throughput screening assay to identify antagonists of galanin receptor 2 (GALR2). (Class of assay: confirmatory) [Related pubchem assays: 828, 866 ]	ChEMBL	425	5	3	4	4.7	O=C(/C=C/c1ccc(Cl)cc1)NC(=S)Nc1ccc(NC(=O)c2ccco2)cc1	nan
	4104905	36272	7	None	1	3	Human	5.1	pIC50	=	5.1	Functional	PUBCHEM_BIOASSAY: Dose response counterscreen for antagonists of galanin receptor 2 (GalR2): a cell-based high-throughput screening assay for inhibitors of beta-lactamase activity. (Class of assay: confirmatory) [Related pubchem assays: 828, 1225, 866 ]PUBCHEM_BIOASSAY: Dose response counterscreen for antagonists of galanin receptor 2 (GalR2): a cell-based high-throughput screening assay for inhibitors of beta-lactamase activity. (Class of assay: confirmatory) [Related pubchem assays: 828, 1225, 866 ]	ChEMBL	297	5	1	7	1.6	CCOC(=O)c1cc([N+](=O)[O-])c([N+](=O)[O-])cc1NC(C)=O	nan
	CHEMBL1447697	36272	7	None	1	3	Human	5.1	pIC50	=	5.1	Functional	PUBCHEM_BIOASSAY: Dose response counterscreen for antagonists of galanin receptor 2 (GalR2): a cell-based high-throughput screening assay for inhibitors of beta-lactamase activity. (Class of assay: confirmatory) [Related pubchem assays: 828, 1225, 866 ]PUBCHEM_BIOASSAY: Dose response counterscreen for antagonists of galanin receptor 2 (GalR2): a cell-based high-throughput screening assay for inhibitors of beta-lactamase activity. (Class of assay: confirmatory) [Related pubchem assays: 828, 1225, 866 ]	ChEMBL	297	5	1	7	1.6	CCOC(=O)c1cc([N+](=O)[O-])c([N+](=O)[O-])cc1NC(C)=O	nan
	2585250	28145	7	None	-5	3	Human	5.1	pIC50	=	5.1	Functional	PUBCHEM_BIOASSAY: Dose Response cell-based high-throughput screening assay to identify antagonists of galanin receptor 2 (GALR2). (Class of assay: confirmatory) [Related pubchem assays: 828, 866 ]PUBCHEM_BIOASSAY: Dose Response cell-based high-throughput screening assay to identify antagonists of galanin receptor 2 (GALR2). (Class of assay: confirmatory) [Related pubchem assays: 828, 866 ]	ChEMBL	396	6	1	5	2.2	CCc1ccccc1NC(=O)CN(C)C(=O)Cn1ncc(Cl)c(Cl)c1=O	nan
	CHEMBL1374788	28145	7	None	-5	3	Human	5.1	pIC50	=	5.1	Functional	PUBCHEM_BIOASSAY: Dose Response cell-based high-throughput screening assay to identify antagonists of galanin receptor 2 (GALR2). (Class of assay: confirmatory) [Related pubchem assays: 828, 866 ]PUBCHEM_BIOASSAY: Dose Response cell-based high-throughput screening assay to identify antagonists of galanin receptor 2 (GALR2). (Class of assay: confirmatory) [Related pubchem assays: 828, 866 ]	ChEMBL	396	6	1	5	2.2	CCc1ccccc1NC(=O)CN(C)C(=O)Cn1ncc(Cl)c(Cl)c1=O	nan
	260557	36779	16	None	1	2	Human	5.1	pIC50	=	5.1	Functional	PUBCHEM_BIOASSAY: Dose Response cell-based high-throughput screening assay to identify antagonists of galanin receptor 2 (GALR2). (Class of assay: confirmatory) [Related pubchem assays: 828, 866 ]PUBCHEM_BIOASSAY: Dose Response cell-based high-throughput screening assay to identify antagonists of galanin receptor 2 (GALR2). (Class of assay: confirmatory) [Related pubchem assays: 828, 866 ]	ChEMBL	326	3	1	4	3.7	CN(C)c1ccc(NC2=C(Cl)C(=O)c3ccccc3C2=O)cc1	nan
	CHEMBL1451772	36779	16	None	1	2	Human	5.1	pIC50	=	5.1	Functional	PUBCHEM_BIOASSAY: Dose Response cell-based high-throughput screening assay to identify antagonists of galanin receptor 2 (GALR2). (Class of assay: confirmatory) [Related pubchem assays: 828, 866 ]PUBCHEM_BIOASSAY: Dose Response cell-based high-throughput screening assay to identify antagonists of galanin receptor 2 (GALR2). (Class of assay: confirmatory) [Related pubchem assays: 828, 866 ]	ChEMBL	326	3	1	4	3.7	CN(C)c1ccc(NC2=C(Cl)C(=O)c3ccccc3C2=O)cc1	nan
	3319616	30954	3	None	2	3	Human	5.1	pIC50	=	5.1	Functional	PUBCHEM_BIOASSAY: Dose Response cell-based high-throughput screening assay to identify antagonists of galanin receptor 2 (GALR2). (Class of assay: confirmatory) [Related pubchem assays: 828, 866 ]PUBCHEM_BIOASSAY: Dose Response cell-based high-throughput screening assay to identify antagonists of galanin receptor 2 (GALR2). (Class of assay: confirmatory) [Related pubchem assays: 828, 866 ]	ChEMBL	252	3	0	7	2.0	O=[N+]([O-])c1cc(-c2ncccn2)c([N+](=O)[O-])s1	nan
	CHEMBL1400481	30954	3	None	2	3	Human	5.1	pIC50	=	5.1	Functional	PUBCHEM_BIOASSAY: Dose Response cell-based high-throughput screening assay to identify antagonists of galanin receptor 2 (GALR2). (Class of assay: confirmatory) [Related pubchem assays: 828, 866 ]PUBCHEM_BIOASSAY: Dose Response cell-based high-throughput screening assay to identify antagonists of galanin receptor 2 (GALR2). (Class of assay: confirmatory) [Related pubchem assays: 828, 866 ]	ChEMBL	252	3	0	7	2.0	O=[N+]([O-])c1cc(-c2ncccn2)c([N+](=O)[O-])s1	nan
	3319616	30954	3	None	2	3	Human	5.0	pIC50	=	5.0	Functional	PUBCHEM_BIOASSAY: Dose response counterscreen for antagonists of galanin receptor 2 (GalR2): a cell-based high-throughput screening assay for inhibitors of beta-lactamase activity. (Class of assay: confirmatory) [Related pubchem assays: 828, 1225, 866 ]PUBCHEM_BIOASSAY: Dose response counterscreen for antagonists of galanin receptor 2 (GalR2): a cell-based high-throughput screening assay for inhibitors of beta-lactamase activity. (Class of assay: confirmatory) [Related pubchem assays: 828, 1225, 866 ]	ChEMBL	252	3	0	7	2.0	O=[N+]([O-])c1cc(-c2ncccn2)c([N+](=O)[O-])s1	nan
	CHEMBL1400481	30954	3	None	2	3	Human	5.0	pIC50	=	5.0	Functional	PUBCHEM_BIOASSAY: Dose response counterscreen for antagonists of galanin receptor 2 (GalR2): a cell-based high-throughput screening assay for inhibitors of beta-lactamase activity. (Class of assay: confirmatory) [Related pubchem assays: 828, 1225, 866 ]PUBCHEM_BIOASSAY: Dose response counterscreen for antagonists of galanin receptor 2 (GalR2): a cell-based high-throughput screening assay for inhibitors of beta-lactamase activity. (Class of assay: confirmatory) [Related pubchem assays: 828, 1225, 866 ]	ChEMBL	252	3	0	7	2.0	O=[N+]([O-])c1cc(-c2ncccn2)c([N+](=O)[O-])s1	nan
	11417	3591	0	None	3	2	Human	6.8	pEC50	=	6.8	Functional	Determined by measuring SRE-luc activity in HEK293-Gqi cells expressing hGALR2.Determined by measuring SRE-luc activity in HEK293-Gqi cells expressing hGALR2.	Guide to Pharmacology		None	None	None		None	24517231
	8547	1266	0	None	-	1	Rat	9.2	pEC50	=	9.2	Functional	Potentiation of galanin-induced IP1 accumulation <i>in vitro</i>.Potentiation of galanin-induced IP1 accumulation <i>in vitro</i>.	Guide to Pharmacology	765	13	5	7	7.3	O=C(N[C@H](C(=O)N[C@H](C(=O)Nc1ccc2c(c1)[nH]c(=O)cc2C)CCCNC(=O)OC(C)(C)C)CC1CCCCC1)OCC1C2C=CC=CC2c2c1cccc2	20660766
	91827369	1266	0	None	-	1	Rat	9.2	pEC50	=	9.2	Functional	Potentiation of galanin-induced IP1 accumulation <i>in vitro</i>.Potentiation of galanin-induced IP1 accumulation <i>in vitro</i>.	Guide to Pharmacology	765	13	5	7	7.3	O=C(N[C@H](C(=O)N[C@H](C(=O)Nc1ccc2c(c1)[nH]c(=O)cc2C)CCCNC(=O)OC(C)(C)C)CC1CCCCC1)OCC1C2C=CC=CC2c2c1cccc2	20660766
	11419	3213	0	None	-	1	Human	7.1	pEC50	=	7.1	Functional	SRE-luc reporter activation in HEK293 Gqi cells expressing hGAL<sub>3</sub> receptor.SRE-luc reporter activation in HEK293 Gqi cells expressing hGAL<sub>3</sub> receptor.	Guide to Pharmacology		None	None	None		None	32231393
	6095	1709	0	None	-2	2	Human	6.5	pEC50	=	6.5	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9880084
	3896	2410	0	None	-58	4	Rat	6.5	pEC50	=	6.5	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9305929
	6095	1709	0	None	2	2	Rat	6.8	pEC50	=	6.8	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9305929
	16132180	1694	14	None	-89	4	Rat	7.0	pEC50	=	7.0	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9305929
	16133822	1694	14	None	-89	4	Rat	7.0	pEC50	=	7.0	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9305929
	6087	1694	14	None	-89	4	Rat	7.0	pEC50	=	7.0	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9305929
	CHEMBL499980	1694	14	None	-89	4	Rat	7.0	pEC50	=	7.0	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9305929
	16131409	1693	0	None	-16	3	Rat	7.2	pEC50	=	7.2	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9305929
	6086	1693	0	None	-16	3	Rat	7.2	pEC50	=	7.2	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9305929
	155817479	1706	0	None	-	1	Human	7.5	pEC50	=	7.5	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9880084
	6083	1706	0	None	-	1	Human	7.5	pEC50	=	7.5	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9880084
	3898	2413	0	None	-562	4	Rat	7.5	pEC50	=	7.5	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9305929
	3899	2414	0	None	-15	4	Rat	7.6	pEC50	=	7.6	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9305929
	155817484	1686	0	None	-42	5	Rat	7.7	pEC50	=	7.7	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9305929
	6117	1686	0	None	-42	5	Rat	7.7	pEC50	=	7.7	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9305929
	6129	1686	0	None	-42	5	Rat	7.7	pEC50	=	7.7	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9305929
	3899	2414	0	None	-32	4	Human	7.8	pEC50	=	7.8	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9880084
	155817463	765	0	None	-3	4	Human	8.0	pEC50	=	8.0	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9880084
	3861	765	0	None	-3	4	Human	8.0	pEC50	=	8.0	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9880084
	155817484	1686	0	None	-25	5	Human	8.1	pEC50	=	8.1	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9880084
	6117	1686	0	None	-25	5	Human	8.1	pEC50	=	8.1	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9880084
	6129	1686	0	None	-25	5	Human	8.1	pEC50	=	8.1	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9880084
	3897	2412	0	None	-	1	Human	8.1	pEC50	=	8.1	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9685625
	3897	2412	0	None	-	1	Human	8.1	pEC50	=	8.1	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9880084
	155817487	1699	0	None	9	2	Human	8.3	pEC50	=	8.3	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9685625
	155817487	1699	0	None	9	2	Human	8.3	pEC50	=	8.3	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9880084
	6130	1699	0	None	9	2	Human	8.3	pEC50	=	8.3	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9685625
	6130	1699	0	None	9	2	Human	8.3	pEC50	=	8.3	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9880084
	16133243	1684	0	None	-17	5	Rat	8.3	pEC50	=	8.3	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	10601261
	3593	1684	0	None	-17	5	Rat	8.3	pEC50	=	8.3	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	10601261
	16132180	1694	14	None	-12	4	Human	8.3	pEC50	=	8.3	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9685625
	16132180	1694	14	None	-12	4	Human	8.3	pEC50	=	8.3	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9880084
	16133822	1694	14	None	-12	4	Human	8.3	pEC50	=	8.3	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9685625
	16133822	1694	14	None	-12	4	Human	8.3	pEC50	=	8.3	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9880084
	6087	1694	14	None	-12	4	Human	8.3	pEC50	=	8.3	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9685625
	6087	1694	14	None	-12	4	Human	8.3	pEC50	=	8.3	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9880084
	CHEMBL499980	1694	14	None	-12	4	Human	8.3	pEC50	=	8.3	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9685625
	CHEMBL499980	1694	14	None	-12	4	Human	8.3	pEC50	=	8.3	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9880084
	3898	2413	0	None	-316	4	Human	8.5	pEC50	=	8.5	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9685625
	3898	2413	0	None	-316	4	Human	8.5	pEC50	=	8.5	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9880084
	155817463	765	0	None	-2	4	Rat	8.5	pEC50	=	8.5	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9305929
	3861	765	0	None	-2	4	Rat	8.5	pEC50	=	8.5	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9305929
	101927062	1685	21	None	-24	5	Human	8.5	pEC50	=	8.5	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9685625
	101927062	1685	21	None	-24	5	Human	8.5	pEC50	=	8.5	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9880084
	155817445	1685	21	None	-24	5	Human	8.5	pEC50	=	8.5	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9685625
	155817445	1685	21	None	-24	5	Human	8.5	pEC50	=	8.5	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9880084
	16133823	1685	21	None	-24	5	Human	8.5	pEC50	=	8.5	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9685625
	16133823	1685	21	None	-24	5	Human	8.5	pEC50	=	8.5	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9880084
	3592	1685	21	None	-24	5	Human	8.5	pEC50	=	8.5	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9685625
	3592	1685	21	None	-24	5	Human	8.5	pEC50	=	8.5	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9880084
	44584852	1685	21	None	-24	5	Human	8.5	pEC50	=	8.5	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9685625
	44584852	1685	21	None	-24	5	Human	8.5	pEC50	=	8.5	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9880084
	6090	1685	21	None	-24	5	Human	8.5	pEC50	=	8.5	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9685625
	6090	1685	21	None	-24	5	Human	8.5	pEC50	=	8.5	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9880084
	91898917	1685	21	None	-24	5	Human	8.5	pEC50	=	8.5	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9685625
	91898917	1685	21	None	-24	5	Human	8.5	pEC50	=	8.5	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9880084
	CHEMBL506553	1685	21	None	-24	5	Human	8.5	pEC50	=	8.5	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9685625
	CHEMBL506553	1685	21	None	-24	5	Human	8.5	pEC50	=	8.5	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9880084
	3896	2410	0	None	-3	4	Human	8.6	pEC50	=	8.6	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9480833
	3896	2410	0	None	-3	4	Human	8.6	pEC50	=	8.6	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9685625
	3896	2410	0	None	-3	4	Human	8.6	pEC50	=	8.6	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9880084
	6120	1712	0	None	15	2	Rat	8.6	pEC50	=	8.6	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	10601261
	16131409	1693	0	None	1	3	Human	9.1	pEC50	=	9.1	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9685625
	6086	1693	0	None	1	3	Human	9.1	pEC50	=	9.1	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9685625
	155817483	1687	0	None	1	2	Human	6.0	pEC50	>	6	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9685625
	6094	1687	0	None	1	2	Human	6.0	pEC50	>	6	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9685625
	155817480	1701	0	None	-1	3	Human	6.0	pEC50	>	6	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9880084
	155817480	1701	0	None	-1	3	Rat	6.0	pEC50	>	6	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9305929
	6091	1701	0	None	-1	3	Human	6.0	pEC50	>	6	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9880084
	6091	1701	0	None	-1	3	Rat	6.0	pEC50	>	6	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9305929
	155817483	1687	0	None	-1	2	Rat	6.0	pIC50	=	6	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9427506
	6094	1687	0	None	-1	2	Rat	6.0	pIC50	=	6	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9427506
	155817475	1704	0	None	-	1	Rat	6.7	pIC50	=	6.7	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	7683428
	5359	1704	0	None	-	1	Rat	6.7	pIC50	=	6.7	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	7683428
	155817485	1727	0	None	1	2	Human	7.2	pIC50	=	7.2	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	15944009
	6121	1727	0	None	1	2	Human	7.2	pIC50	=	7.2	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	15944009
	3594	1711	0	None	-2	3	Human	7.6	pIC50	=	7.6	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	15944009
	3594	1711	0	None	-2	3	Human	7.6	pIC50	=	7.6	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	20880399
	134813891	1728	0	None	2	2	Human	7.8	pIC50	=	7.8	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	15944009
	6122	1728	0	None	2	2	Human	7.8	pIC50	=	7.8	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	15944009
	3896	2410	0	None	-58	4	Rat	7.9	pIC50	=	7.9	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9108306
	3896	2410	0	None	-58	4	Rat	7.9	pIC50	=	7.9	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9427506
	155817463	765	0	None	-2	4	Rat	8.0	pIC50	=	8.0	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9108306
	155817463	765	0	None	-2	4	Rat	8.0	pIC50	=	8.0	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9427506
	3861	765	0	None	-2	4	Rat	8.0	pIC50	=	8.0	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9108306
	3861	765	0	None	-2	4	Rat	8.0	pIC50	=	8.0	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9427506
	155817463	765	0	None	-3	4	Human	8.1	pIC50	=	8.1	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9685625
	3861	765	0	None	-3	4	Human	8.1	pIC50	=	8.1	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9685625
	16131409	1693	0	None	-16	3	Rat	8.1	pIC50	=	8.1	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9427506
	6086	1693	0	None	-16	3	Rat	8.1	pIC50	=	8.1	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9427506
	16132180	1694	14	None	-89	4	Rat	8.2	pIC50	=	8.2	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9108306
	16132180	1694	14	None	-89	4	Rat	8.2	pIC50	=	8.2	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9427506
	16133822	1694	14	None	-89	4	Rat	8.2	pIC50	=	8.2	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9108306
	16133822	1694	14	None	-89	4	Rat	8.2	pIC50	=	8.2	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9427506
	6087	1694	14	None	-89	4	Rat	8.2	pIC50	=	8.2	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9108306
	6087	1694	14	None	-89	4	Rat	8.2	pIC50	=	8.2	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9427506
	CHEMBL499980	1694	14	None	-89	4	Rat	8.2	pIC50	=	8.2	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9108306
	CHEMBL499980	1694	14	None	-89	4	Rat	8.2	pIC50	=	8.2	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9427506
	3896	2410	0	None	-3	4	Human	8.4	pIC50	=	8.4	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9685625
	16133243	1684	0	None	-7	5	Human	8.5	pIC50	=	8.5	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9685625
	16133243	1684	0	None	-7	5	Human	8.5	pIC50	=	8.5	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9880084
	3593	1684	0	None	-7	5	Human	8.5	pIC50	=	8.5	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9685625
	3593	1684	0	None	-7	5	Human	8.5	pIC50	=	8.5	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9880084
	155817465	1700	0	None	2	3	Rat	8.5	pIC50	=	8.5	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9108306
	3876	1700	0	None	2	3	Rat	8.5	pIC50	=	8.5	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9108306
	16131409	1693	0	None	1	3	Human	8.6	pIC50	=	8.6	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9685625
	6086	1693	0	None	1	3	Human	8.6	pIC50	=	8.6	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9685625
	3899	2414	0	None	-15	4	Rat	8.6	pIC50	=	8.6	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9108306
	3899	2414	0	None	-15	4	Rat	8.6	pIC50	=	8.6	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9427506
	16132180	1694	14	None	-12	4	Human	8.7	pIC50	=	8.7	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9685625
	16133822	1694	14	None	-12	4	Human	8.7	pIC50	=	8.7	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9685625
	6087	1694	14	None	-12	4	Human	8.7	pIC50	=	8.7	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9685625
	CHEMBL499980	1694	14	None	-12	4	Human	8.7	pIC50	=	8.7	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9685625
	155817487	1699	0	None	9	2	Human	8.7	pIC50	=	8.7	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9427506
	155817487	1699	0	None	9	2	Human	8.7	pIC50	=	8.7	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9685625
	6130	1699	0	None	9	2	Human	8.7	pIC50	=	8.7	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9427506
	6130	1699	0	None	9	2	Human	8.7	pIC50	=	8.7	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9685625
	155817474	1698	0	None	489	2	Rat	8.8	pIC50	=	8.8	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	11481429
	5357	1698	0	None	489	2	Rat	8.8	pIC50	=	8.8	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	11481429
	6082	3426	0	None	-4	2	Rat	8.8	pIC50	=	8.8	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	11481429
	155817473	1690	0	None	-1	2	Rat	8.8	pIC50	=	8.8	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	11481429
	5356	1690	0	None	-1	2	Rat	8.8	pIC50	=	8.8	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	11481429
	6084	1690	0	None	-1	2	Rat	8.8	pIC50	=	8.8	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	11481429
	101927062	1685	21	None	-24	5	Rat	8.8	pIC50	=	8.8	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	11481429
	101927062	1685	21	None	-24	5	Rat	8.8	pIC50	=	8.8	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9108306
	101927062	1685	21	None	-24	5	Rat	8.8	pIC50	=	8.8	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9427506
	155817445	1685	21	None	-24	5	Rat	8.8	pIC50	=	8.8	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	11481429
	155817445	1685	21	None	-24	5	Rat	8.8	pIC50	=	8.8	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9108306
	155817445	1685	21	None	-24	5	Rat	8.8	pIC50	=	8.8	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9427506
	16133823	1685	21	None	-24	5	Rat	8.8	pIC50	=	8.8	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	11481429
	16133823	1685	21	None	-24	5	Rat	8.8	pIC50	=	8.8	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9108306
	16133823	1685	21	None	-24	5	Rat	8.8	pIC50	=	8.8	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9427506
	3592	1685	21	None	-24	5	Rat	8.8	pIC50	=	8.8	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	11481429
	3592	1685	21	None	-24	5	Rat	8.8	pIC50	=	8.8	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9108306
	3592	1685	21	None	-24	5	Rat	8.8	pIC50	=	8.8	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9427506
	44584852	1685	21	None	-24	5	Rat	8.8	pIC50	=	8.8	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	11481429
	44584852	1685	21	None	-24	5	Rat	8.8	pIC50	=	8.8	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9108306
	44584852	1685	21	None	-24	5	Rat	8.8	pIC50	=	8.8	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9427506
	6090	1685	21	None	-24	5	Rat	8.8	pIC50	=	8.8	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	11481429
	6090	1685	21	None	-24	5	Rat	8.8	pIC50	=	8.8	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9108306
	6090	1685	21	None	-24	5	Rat	8.8	pIC50	=	8.8	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9427506
	91898917	1685	21	None	-24	5	Rat	8.8	pIC50	=	8.8	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	11481429
	91898917	1685	21	None	-24	5	Rat	8.8	pIC50	=	8.8	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9108306
	91898917	1685	21	None	-24	5	Rat	8.8	pIC50	=	8.8	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9427506
	CHEMBL506553	1685	21	None	-24	5	Rat	8.8	pIC50	=	8.8	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	11481429
	CHEMBL506553	1685	21	None	-24	5	Rat	8.8	pIC50	=	8.8	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9108306
	CHEMBL506553	1685	21	None	-24	5	Rat	8.8	pIC50	=	8.8	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9427506
	3898	2413	0	None	-562	4	Rat	9.0	pIC50	=	9.0	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9108306
	3898	2413	0	None	-562	4	Rat	9.0	pIC50	=	9.0	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9427506
	16133243	1684	0	None	-17	5	Rat	9.0	pIC50	=	9.0	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	10601261
	16133243	1684	0	None	-17	5	Rat	9.0	pIC50	=	9.0	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	20880399
	16133243	1684	0	None	-17	5	Rat	9.0	pIC50	=	9.0	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9427506
	3593	1684	0	None	-17	5	Rat	9.0	pIC50	=	9.0	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	10601261
	3593	1684	0	None	-17	5	Rat	9.0	pIC50	=	9.0	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	20880399
	3593	1684	0	None	-17	5	Rat	9.0	pIC50	=	9.0	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9427506
	101927062	1685	21	None	-24	5	Human	9.3	pIC50	=	9.3	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9685625
	155817445	1685	21	None	-24	5	Human	9.3	pIC50	=	9.3	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9685625
	16133823	1685	21	None	-24	5	Human	9.3	pIC50	=	9.3	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9685625
	3592	1685	21	None	-24	5	Human	9.3	pIC50	=	9.3	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9685625
	44584852	1685	21	None	-24	5	Human	9.3	pIC50	=	9.3	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9685625
	6090	1685	21	None	-24	5	Human	9.3	pIC50	=	9.3	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9685625
	91898917	1685	21	None	-24	5	Human	9.3	pIC50	=	9.3	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9685625
	CHEMBL506553	1685	21	None	-24	5	Human	9.3	pIC50	=	9.3	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9685625
	155817484	1686	0	None	-42	5	Rat	9.4	pIC50	=	9.4	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9108306
	155817484	1686	0	None	-42	5	Rat	9.4	pIC50	=	9.4	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9427506
	6117	1686	0	None	-42	5	Rat	9.4	pIC50	=	9.4	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9108306
	6117	1686	0	None	-42	5	Rat	9.4	pIC50	=	9.4	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9427506
	6129	1686	0	None	-42	5	Rat	9.4	pIC50	=	9.4	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9108306
	6129	1686	0	None	-42	5	Rat	9.4	pIC50	=	9.4	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9427506
	155817484	1686	0	None	-25	5	Human	9.5	pIC50	=	9.5	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9685625
	6117	1686	0	None	-25	5	Human	9.5	pIC50	=	9.5	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9685625
	6129	1686	0	None	-25	5	Human	9.5	pIC50	=	9.5	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9685625
	16133243	1684	0	None	-7	5	Human	9.5	pIC50	=	9.5	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9685625
	3593	1684	0	None	-7	5	Human	9.5	pIC50	=	9.5	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9685625
	6120	1712	0	None	15	2	Rat	9.6	pIC50	=	9.6	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	10601261
	6124	1411	1	None	-158	2	Human	4.5	pIC50	>	4.5	Functional	UnclassifiedUnclassified	Guide to Pharmacology	286	1	0	4	1.5	Cc1ccc(cc1)C1=CS(=O)(=O)CCCS1(=O)=O	10896115
	9947811	1411	1	None	-158	2	Human	4.5	pIC50	>	4.5	Functional	UnclassifiedUnclassified	Guide to Pharmacology	286	1	0	4	1.5	Cc1ccc(cc1)C1=CS(=O)(=O)CCCS1(=O)=O	10896115
	CHEMBL3906195	1411	1	None	-158	2	Human	4.5	pIC50	>	4.5	Functional	UnclassifiedUnclassified	Guide to Pharmacology	286	1	0	4	1.5	Cc1ccc(cc1)C1=CS(=O)(=O)CCCS1(=O)=O	10896115
	131863305	324	0	None	-1	3	Rat	6.0	pIC50	>	6	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	20880399
	155817486	324	0	None	-1	3	Rat	6.0	pIC50	>	6	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	20880399
	6123	324	0	None	-1	3	Rat	6.0	pIC50	>	6	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	20880399
	155817480	1701	0	None	-1	3	Human	6.0	pIC50	>	6	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9427506
	155817480	1701	0	None	-1	3	Human	6.0	pIC50	>	6	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9685625
	6091	1701	0	None	-1	3	Human	6.0	pIC50	>	6	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9427506
	6091	1701	0	None	-1	3	Human	6.0	pIC50	>	6	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9685625
	155817481	1702	0	None	-1	3	Rat	6.0	pIC50	>	6	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9108306
	6092	1702	0	None	-1	3	Rat	6.0	pIC50	>	6	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9108306

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Ligands					Receptor			Assay information							Chemical information
Sel. page	Common name	GPCRdb ID	#Vendors	Reference ligand	Fold selectivity (Affinity)	# tested GPCRs (Affinity)	Species	p-value (-log)	Type	Activity Relation	Activity Value	Assay Type	Assay Description	Source	Mol weight	Rot Bonds	H don	H acc	LogP	Smiles	DOI
	72548703	161019	0	None	-	0	Human	9.7	pIC50	=	9.7	Binding	Displacement of [125I]-endothelin-1 from human recombinant GAL2 receptor after 120 mins by scintillation counting analysisDisplacement of [125I]-endothelin-1 from human recombinant GAL2 receptor after 120 mins by scintillation counting analysis	ChEMBL	583	8	3	6	5.8	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(C(=O)N[C@H]3C[C@H](C(=O)O)C3)nc2CC2CCCCC2)c2ccccc12	10.1016/j.bmcl.2018.03.093
	CHEMBL4128926	161019	0	None	-	0	Human	9.7	pIC50	=	9.7	Binding	Displacement of [125I]-endothelin-1 from human recombinant GAL2 receptor after 120 mins by scintillation counting analysisDisplacement of [125I]-endothelin-1 from human recombinant GAL2 receptor after 120 mins by scintillation counting analysis	ChEMBL	583	8	3	6	5.8	CC(C)(C)NS(=O)(=O)c1ccc(-c2sc(C(=O)N[C@H]3C[C@H](C(=O)O)C3)nc2CC2CCCCC2)c2ccccc12	10.1016/j.bmcl.2018.03.093
	CHEMBL501079	212359	10	None	-11	2	Human	9.1	pIC50	=	9.1	Binding	Binding affinity to human GAL2 receptor by radioligand displacement assayBinding affinity to human GAL2 receptor by radioligand displacement assay	ChEMBL		None	None	None		CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](Cc1c[nH]cn1)NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)CN)[C@@H](C)O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](Cc1c[nH]cn1)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](Cc1c[nH]cn1)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)NCC(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C)C(N)=O	10.1016/j.bmc.2013.03.016
	57392517	68462	0	None	-	0	Human	6.0	pIC50	=	6.0	Binding	Displacement of [125I]galanin from GalR2 by gamma countingDisplacement of [125I]galanin from GalR2 by gamma counting	ChEMBL	473	8	3	7	6.6	COc1ccc(Nc2cc(Nc3ccc(OC(F)(F)F)cc3)nc(NC3CCCCC3)n2)cc1	10.1016/j.bmcl.2011.09.033
	CHEMBL1921997	68462	0	None	-	0	Human	6.0	pIC50	=	6.0	Binding	Displacement of [125I]galanin from GalR2 by gamma countingDisplacement of [125I]galanin from GalR2 by gamma counting	ChEMBL	473	8	3	7	6.6	COc1ccc(Nc2cc(Nc3ccc(OC(F)(F)F)cc3)nc(NC3CCCCC3)n2)cc1	10.1016/j.bmcl.2011.09.033
	57396058	68401	0	None	-	0	Human	6.0	pIC50	=	6.0	Binding	Displacement of [125I]galanin from GalR2 by gamma countingDisplacement of [125I]galanin from GalR2 by gamma counting	ChEMBL	375	6	2	6	5.0	COc1ccc(Nc2cc(Nc3ccccc3)nc(N3CCCCC3)n2)cc1	10.1016/j.bmcl.2011.09.033
	CHEMBL1921902	68401	0	None	-	0	Human	6.0	pIC50	=	6.0	Binding	Displacement of [125I]galanin from GalR2 by gamma countingDisplacement of [125I]galanin from GalR2 by gamma counting	ChEMBL	375	6	2	6	5.0	COc1ccc(Nc2cc(Nc3ccccc3)nc(N3CCCCC3)n2)cc1	10.1016/j.bmcl.2011.09.033
	57401222	68470	0	None	-	0	Human	5.9	pIC50	=	5.9	Binding	Displacement of [125I]galanin from GalR2 by gamma countingDisplacement of [125I]galanin from GalR2 by gamma counting	ChEMBL	403	6	2	6	5.6	COc1ccc(Nc2nc(Nc3ccc(C)cc3C)cc(N3CCCCC3)n2)cc1	10.1016/j.bmcl.2011.09.033
	CHEMBL1922004	68470	0	None	-	0	Human	5.9	pIC50	=	5.9	Binding	Displacement of [125I]galanin from GalR2 by gamma countingDisplacement of [125I]galanin from GalR2 by gamma counting	ChEMBL	403	6	2	6	5.6	COc1ccc(Nc2nc(Nc3ccc(C)cc3C)cc(N3CCCCC3)n2)cc1	10.1016/j.bmcl.2011.09.033
	57395993	68460	0	None	-	0	Human	4.9	pIC50	=	4.9	Binding	Displacement of [125I]galanin from GalR2 by gamma countingDisplacement of [125I]galanin from GalR2 by gamma counting	ChEMBL	455	9	3	7	6.3	COc1ccc(Nc2cc(Nc3ccc(OC(F)F)cc3)nc(NC3CCCCC3)n2)cc1	10.1016/j.bmcl.2011.09.033
	CHEMBL1921995	68460	0	None	-	0	Human	4.9	pIC50	=	4.9	Binding	Displacement of [125I]galanin from GalR2 by gamma countingDisplacement of [125I]galanin from GalR2 by gamma counting	ChEMBL	455	9	3	7	6.3	COc1ccc(Nc2cc(Nc3ccc(OC(F)F)cc3)nc(NC3CCCCC3)n2)cc1	10.1016/j.bmcl.2011.09.033
	57401225	68483	0	None	-	0	Human	5.9	pIC50	=	5.9	Binding	Displacement of [125I]galanin from GalR2 by gamma countingDisplacement of [125I]galanin from GalR2 by gamma counting	ChEMBL	437	7	2	7	5.4	COc1ccc(Nc2nc(Nc3ccc(OC)c(F)c3)cc(N3CCCC(C)C3)n2)cc1	10.1016/j.bmcl.2011.09.033
	CHEMBL1922019	68483	0	None	-	0	Human	5.9	pIC50	=	5.9	Binding	Displacement of [125I]galanin from GalR2 by gamma countingDisplacement of [125I]galanin from GalR2 by gamma counting	ChEMBL	437	7	2	7	5.4	COc1ccc(Nc2nc(Nc3ccc(OC)c(F)c3)cc(N3CCCC(C)C3)n2)cc1	10.1016/j.bmcl.2011.09.033
	57394237	68463	0	None	-	0	Human	5.8	pIC50	=	5.8	Binding	Displacement of [125I]galanin from GalR2 by gamma countingDisplacement of [125I]galanin from GalR2 by gamma counting	ChEMBL	419	8	3	7	5.7	COc1ccc(Nc2cc(Nc3cccc(OC)c3)nc(NC3CCCCC3)n2)cc1	10.1016/j.bmcl.2011.09.033
	CHEMBL1921998	68463	0	None	-	0	Human	5.8	pIC50	=	5.8	Binding	Displacement of [125I]galanin from GalR2 by gamma countingDisplacement of [125I]galanin from GalR2 by gamma counting	ChEMBL	419	8	3	7	5.7	COc1ccc(Nc2cc(Nc3cccc(OC)c3)nc(NC3CCCCC3)n2)cc1	10.1016/j.bmcl.2011.09.033
	57397798	68466	0	None	-	0	Human	5.7	pIC50	=	5.7	Binding	Displacement of [125I]galanin from GalR2 by gamma countingDisplacement of [125I]galanin from GalR2 by gamma counting	ChEMBL	527	6	1	8	5.4	COc1ccc(Nc2cc(N3CCCCC3)nc(N3CCCN(c4ncccc4C(F)(F)F)CC3)n2)cc1	10.1016/j.bmcl.2011.09.033
	CHEMBL1922000	68466	0	None	-	0	Human	5.7	pIC50	=	5.7	Binding	Displacement of [125I]galanin from GalR2 by gamma countingDisplacement of [125I]galanin from GalR2 by gamma counting	ChEMBL	527	6	1	8	5.4	COc1ccc(Nc2cc(N3CCCCC3)nc(N3CCCN(c4ncccc4C(F)(F)F)CC3)n2)cc1	10.1016/j.bmcl.2011.09.033
	57392518	68477	0	None	-	0	Human	5.7	pIC50	=	5.7	Binding	Displacement of [125I]galanin from GalR2 by gamma countingDisplacement of [125I]galanin from GalR2 by gamma counting	ChEMBL	457	7	2	6	5.9	COc1ccc(Nc2nc(NCc3cccc(C(F)(F)F)c3)cc(N3CCCCC3)n2)cc1	10.1016/j.bmcl.2011.09.033
	CHEMBL1922011	68477	0	None	-	0	Human	5.7	pIC50	=	5.7	Binding	Displacement of [125I]galanin from GalR2 by gamma countingDisplacement of [125I]galanin from GalR2 by gamma counting	ChEMBL	457	7	2	6	5.9	COc1ccc(Nc2nc(NCc3cccc(C(F)(F)F)c3)cc(N3CCCCC3)n2)cc1	10.1016/j.bmcl.2011.09.033
	CHEMBL501079	212359	10	None	-11	2	Human	8.6	pIC50	=	8.6	Binding	Binding affinity to human GAL2 receptor by radioligand displacement assayBinding affinity to human GAL2 receptor by radioligand displacement assay	ChEMBL		None	None	None		CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](Cc1c[nH]cn1)NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)CN)[C@@H](C)O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](Cc1c[nH]cn1)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](Cc1c[nH]cn1)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)NCC(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C)C(N)=O	10.1016/j.ejmech.2013.01.044
	101927062	1685	21	None	-8	6	Human	8.6	pIC50	=	8.6	Binding	Displacement of [125I]galanin from human recombinant GAL2 receptor expressed in CHO cells measured after 120 mins by scintillation counting methodDisplacement of [125I]galanin from human recombinant GAL2 receptor expressed in CHO cells measured after 120 mins by scintillation counting method	ChEMBL		None	None	None		None	10.1016/j.bmc.2016.11.014
	155817445	1685	21	None	-8	6	Human	8.6	pIC50	=	8.6	Binding	Displacement of [125I]galanin from human recombinant GAL2 receptor expressed in CHO cells measured after 120 mins by scintillation counting methodDisplacement of [125I]galanin from human recombinant GAL2 receptor expressed in CHO cells measured after 120 mins by scintillation counting method	ChEMBL		None	None	None		None	10.1016/j.bmc.2016.11.014
	16133823	1685	21	None	-8	6	Human	8.6	pIC50	=	8.6	Binding	Displacement of [125I]galanin from human recombinant GAL2 receptor expressed in CHO cells measured after 120 mins by scintillation counting methodDisplacement of [125I]galanin from human recombinant GAL2 receptor expressed in CHO cells measured after 120 mins by scintillation counting method	ChEMBL		None	None	None		None	10.1016/j.bmc.2016.11.014
	3592	1685	21	None	-8	6	Human	8.6	pIC50	=	8.6	Binding	Displacement of [125I]galanin from human recombinant GAL2 receptor expressed in CHO cells measured after 120 mins by scintillation counting methodDisplacement of [125I]galanin from human recombinant GAL2 receptor expressed in CHO cells measured after 120 mins by scintillation counting method	ChEMBL		None	None	None		None	10.1016/j.bmc.2016.11.014
	44584852	1685	21	None	-8	6	Human	8.6	pIC50	=	8.6	Binding	Displacement of [125I]galanin from human recombinant GAL2 receptor expressed in CHO cells measured after 120 mins by scintillation counting methodDisplacement of [125I]galanin from human recombinant GAL2 receptor expressed in CHO cells measured after 120 mins by scintillation counting method	ChEMBL		None	None	None		None	10.1016/j.bmc.2016.11.014
	6090	1685	21	None	-8	6	Human	8.6	pIC50	=	8.6	Binding	Displacement of [125I]galanin from human recombinant GAL2 receptor expressed in CHO cells measured after 120 mins by scintillation counting methodDisplacement of [125I]galanin from human recombinant GAL2 receptor expressed in CHO cells measured after 120 mins by scintillation counting method	ChEMBL		None	None	None		None	10.1016/j.bmc.2016.11.014
	91898917	1685	21	None	-8	6	Human	8.6	pIC50	=	8.6	Binding	Displacement of [125I]galanin from human recombinant GAL2 receptor expressed in CHO cells measured after 120 mins by scintillation counting methodDisplacement of [125I]galanin from human recombinant GAL2 receptor expressed in CHO cells measured after 120 mins by scintillation counting method	ChEMBL		None	None	None		None	10.1016/j.bmc.2016.11.014
	CHEMBL506553	1685	21	None	-8	6	Human	8.6	pIC50	=	8.6	Binding	Displacement of [125I]galanin from human recombinant GAL2 receptor expressed in CHO cells measured after 120 mins by scintillation counting methodDisplacement of [125I]galanin from human recombinant GAL2 receptor expressed in CHO cells measured after 120 mins by scintillation counting method	ChEMBL		None	None	None		None	10.1016/j.bmc.2016.11.014
	57399458	68468	0	None	-	0	Human	5.7	pIC50	=	5.7	Binding	Displacement of [125I]galanin from GalR2 by gamma countingDisplacement of [125I]galanin from GalR2 by gamma counting	ChEMBL	545	6	1	8	5.5	COc1ccc(Nc2cc(N3CCCCC3)nc(N3CCCN(c4ncccc4C(F)(F)F)CC3)n2)cc1F	10.1016/j.bmcl.2011.09.033
	CHEMBL1922002	68468	0	None	-	0	Human	5.7	pIC50	=	5.7	Binding	Displacement of [125I]galanin from GalR2 by gamma countingDisplacement of [125I]galanin from GalR2 by gamma counting	ChEMBL	545	6	1	8	5.5	COc1ccc(Nc2cc(N3CCCCC3)nc(N3CCCN(c4ncccc4C(F)(F)F)CC3)n2)cc1F	10.1016/j.bmcl.2011.09.033
	57395994	68467	0	None	-	0	Human	5.7	pIC50	=	5.7	Binding	Displacement of [125I]galanin from GalR2 by gamma countingDisplacement of [125I]galanin from GalR2 by gamma counting	ChEMBL	525	5	1	7	6.0	Cc1ccc(C)c(Nc2cc(N3CCCCC3)nc(N3CCCN(c4ncccc4C(F)(F)F)CC3)n2)c1	10.1016/j.bmcl.2011.09.033
	CHEMBL1922001	68467	0	None	-	0	Human	5.7	pIC50	=	5.7	Binding	Displacement of [125I]galanin from GalR2 by gamma countingDisplacement of [125I]galanin from GalR2 by gamma counting	ChEMBL	525	5	1	7	6.0	Cc1ccc(C)c(Nc2cc(N3CCCCC3)nc(N3CCCN(c4ncccc4C(F)(F)F)CC3)n2)c1	10.1016/j.bmcl.2011.09.033
	16078939	180130	15	None	-	0	Rat	7.7	pIC50	=	7.7	Binding	Inhibition of [3H]glycine uptake at rat glycine transporter 2 expressed in african green monkey COS7 cellsInhibition of [3H]glycine uptake at rat glycine transporter 2 expressed in african green monkey COS7 cells	ChEMBL	395	9	2	4	3.9	N[C@@H](COC(c1cccc(F)c1)c1ccccc1OCc1ccccc1)C(=O)O	10.1016/j.bmcl.2008.10.104
	CHEMBL475562	180130	15	None	-	0	Rat	7.7	pIC50	=	7.7	Binding	Inhibition of [3H]glycine uptake at rat glycine transporter 2 expressed in african green monkey COS7 cellsInhibition of [3H]glycine uptake at rat glycine transporter 2 expressed in african green monkey COS7 cells	ChEMBL	395	9	2	4	3.9	N[C@@H](COC(c1cccc(F)c1)c1ccccc1OCc1ccccc1)C(=O)O	10.1016/j.bmcl.2008.10.104
	CHEMBL514318	213819	0	None	-	0	Rat	6.7	pIC50	=	6.7	Binding	Inhibition of [3H]glycine uptake at rat glycine transporter 2 expressed in african green monkey COS7 cellsInhibition of [3H]glycine uptake at rat glycine transporter 2 expressed in african green monkey COS7 cells	ChEMBL		None	None	None		CC[C@H](C)[C@@H]1NC(=O)[C@H](Cc2ccccc2)NC(=O)[C@H]([C@@H](C)CC)NC(=O)[C@H]([C@@H](C)CC)NC1=O	10.1016/j.bmcl.2008.10.104
	CHEMBL475845	212284	0	None	-	0	Rat	5.7	pIC50	=	5.7	Binding	Inhibition of [3H]glycine uptake at rat glycine transporter 2 expressed in african green monkey COS7 cellsInhibition of [3H]glycine uptake at rat glycine transporter 2 expressed in african green monkey COS7 cells	ChEMBL		None	None	None		CC[C@H](C)[C@@H]1NC(=O)[C@H](Cc2ccccc2)NC(=O)[C@H]([C@H](CS(=O)(=O)O)C(C)=O)NC(=O)[C@H]([C@@H](C)CC)NC1=O	10.1016/j.bmcl.2008.10.104
	57390718	68486	0	None	-	0	Human	4.6	pIC50	=	4.6	Binding	Displacement of [125I]galanin from GalR2 by gamma countingDisplacement of [125I]galanin from GalR2 by gamma counting	ChEMBL	500	8	2	8	5.4	COc1ccc(Nc2nc(Nc3ccc(OC)c(F)c3)cc(N3CCN(c4ccccc4)CC3)n2)cc1	10.1016/j.bmcl.2011.09.033
	CHEMBL1922023	68486	0	None	-	0	Human	4.6	pIC50	=	4.6	Binding	Displacement of [125I]galanin from GalR2 by gamma countingDisplacement of [125I]galanin from GalR2 by gamma counting	ChEMBL	500	8	2	8	5.4	COc1ccc(Nc2nc(Nc3ccc(OC)c(F)c3)cc(N3CCN(c4ccccc4)CC3)n2)cc1	10.1016/j.bmcl.2011.09.033
	CHEMBL515145	213821	0	None	-	0	Rat	6.6	pIC50	=	6.6	Binding	Inhibition of [3H]glycine uptake at rat glycine transporter 2 expressed in african green monkey COS7 cellsInhibition of [3H]glycine uptake at rat glycine transporter 2 expressed in african green monkey COS7 cells	ChEMBL		None	None	None		CC[C@H](C)[C@@H]1NC(=O)[C@H](Cc2ccccc2)NC(=O)[C@H]([C@H](C)[C@@H](C)O)NC(=O)[C@H]([C@@H](C)CC)NC1=O	10.1016/j.bmcl.2008.10.104
	57401223	68482	0	None	-	0	Human	5.5	pIC50	=	5.5	Binding	Displacement of [125I]galanin from GalR2 by gamma countingDisplacement of [125I]galanin from GalR2 by gamma counting	ChEMBL	411	9	2	7	5.0	CCN(CC)c1cc(Nc2ccc(OC)c(F)c2)nc(Nc2ccc(OC)cc2)n1	10.1016/j.bmcl.2011.09.033
	CHEMBL1922017	68482	0	None	-	0	Human	5.5	pIC50	=	5.5	Binding	Displacement of [125I]galanin from GalR2 by gamma countingDisplacement of [125I]galanin from GalR2 by gamma counting	ChEMBL	411	9	2	7	5.0	CCN(CC)c1cc(Nc2ccc(OC)c(F)c2)nc(Nc2ccc(OC)cc2)n1	10.1016/j.bmcl.2011.09.033
	CHEMBL501079	212359	10	None	-11	2	Human	8.5	pIC50	=	8.5	Binding	Displacement of radiolabeled galanin from human galanin 2 receptorDisplacement of radiolabeled galanin from human galanin 2 receptor	ChEMBL		None	None	None		CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](Cc1c[nH]cn1)NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)CN)[C@@H](C)O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](Cc1c[nH]cn1)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](Cc1c[nH]cn1)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)NCC(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C)C(N)=O	10.1021/jm8007618
	CHEMBL501079	212359	10	None	-11	2	Human	8.5	pIC50	=	8.5	Binding	Inhibition of human GAL2 receptorInhibition of human GAL2 receptor	ChEMBL		None	None	None		CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](Cc1c[nH]cn1)NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)CN)[C@@H](C)O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](Cc1c[nH]cn1)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](Cc1c[nH]cn1)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)NCC(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C)C(N)=O	10.1021/jm701575k
	54764411	68473	0	None	-	0	Human	6.5	pIC50	=	6.5	Binding	Displacement of [125I]galanin from GalR2 by gamma countingDisplacement of [125I]galanin from GalR2 by gamma counting	ChEMBL	459	7	2	7	5.9	COc1ccc(Nc2nc(Nc3ccc(OC(F)(F)F)cc3)cc(N3CCCCC3)n2)cc1	10.1016/j.bmcl.2011.09.033
	CHEMBL1922007	68473	0	None	-	0	Human	6.5	pIC50	=	6.5	Binding	Displacement of [125I]galanin from GalR2 by gamma countingDisplacement of [125I]galanin from GalR2 by gamma counting	ChEMBL	459	7	2	7	5.9	COc1ccc(Nc2nc(Nc3ccc(OC(F)(F)F)cc3)cc(N3CCCCC3)n2)cc1	10.1016/j.bmcl.2011.09.033
	57394235	68453	0	None	-	0	Human	5.5	pIC50	=	5.5	Binding	Displacement of [125I]galanin from GalR2 by gamma countingDisplacement of [125I]galanin from GalR2 by gamma counting	ChEMBL	411	7	2	6	5.6	FC(F)Oc1ccc(Nc2cc(Nc3ccccc3)nc(N3CCCCC3)n2)cc1	10.1016/j.bmcl.2011.09.033
	CHEMBL1921988	68453	0	None	-	0	Human	5.5	pIC50	=	5.5	Binding	Displacement of [125I]galanin from GalR2 by gamma countingDisplacement of [125I]galanin from GalR2 by gamma counting	ChEMBL	411	7	2	6	5.6	FC(F)Oc1ccc(Nc2cc(Nc3ccccc3)nc(N3CCCCC3)n2)cc1	10.1016/j.bmcl.2011.09.033
	57399456	68457	0	None	-	0	Human	5.5	pIC50	=	5.5	Binding	Displacement of [125I]galanin from GalR2 by gamma countingDisplacement of [125I]galanin from GalR2 by gamma counting	ChEMBL	430	6	1	7	4.2	COc1ccc(Nc2cc(N3CCN(c4ccccc4)CC3)nc(N3CCCC3)n2)cc1	10.1016/j.bmcl.2011.09.033
	CHEMBL1921992	68457	0	None	-	0	Human	5.5	pIC50	=	5.5	Binding	Displacement of [125I]galanin from GalR2 by gamma countingDisplacement of [125I]galanin from GalR2 by gamma counting	ChEMBL	430	6	1	7	4.2	COc1ccc(Nc2cc(N3CCN(c4ccccc4)CC3)nc(N3CCCC3)n2)cc1	10.1016/j.bmcl.2011.09.033
	57397796	68455	0	None	-	0	Human	5.4	pIC50	=	5.4	Binding	Displacement of [125I]galanin from GalR2 by gamma countingDisplacement of [125I]galanin from GalR2 by gamma counting	ChEMBL	403	6	2	7	4.6	c1ccc(Nc2cc(NCc3ccc4c(c3)OCO4)nc(N3CCCCC3)n2)cc1	10.1016/j.bmcl.2011.09.033
	CHEMBL1921990	68455	0	None	-	0	Human	5.4	pIC50	=	5.4	Binding	Displacement of [125I]galanin from GalR2 by gamma countingDisplacement of [125I]galanin from GalR2 by gamma counting	ChEMBL	403	6	2	7	4.6	c1ccc(Nc2cc(NCc3ccc4c(c3)OCO4)nc(N3CCCCC3)n2)cc1	10.1016/j.bmcl.2011.09.033
	54764328	68472	0	None	-	0	Human	6.4	pIC50	=	6.4	Binding	Displacement of [125I]galanin from GalR2 by gamma countingDisplacement of [125I]galanin from GalR2 by gamma counting	ChEMBL	459	7	2	7	5.9	COc1ccc(Nc2nc(Nc3cccc(OC(F)(F)F)c3)cc(N3CCCCC3)n2)cc1	10.1016/j.bmcl.2011.09.033
	CHEMBL1922006	68472	0	None	-	0	Human	6.4	pIC50	=	6.4	Binding	Displacement of [125I]galanin from GalR2 by gamma countingDisplacement of [125I]galanin from GalR2 by gamma counting	ChEMBL	459	7	2	7	5.9	COc1ccc(Nc2nc(Nc3cccc(OC(F)(F)F)c3)cc(N3CCCCC3)n2)cc1	10.1016/j.bmcl.2011.09.033
	54764412	68479	0	None	-	0	Human	6.4	pIC50	=	6.4	Binding	Displacement of [125I]galanin from GalR2 by gamma countingDisplacement of [125I]galanin from GalR2 by gamma counting	ChEMBL	407	6	2	6	5.4	COc1ccc(Nc2nc(Nc3cccc(F)c3C)cc(N3CCCCC3)n2)cc1	10.1016/j.bmcl.2011.09.033
	CHEMBL1922013	68479	0	None	-	0	Human	6.4	pIC50	=	6.4	Binding	Displacement of [125I]galanin from GalR2 by gamma countingDisplacement of [125I]galanin from GalR2 by gamma counting	ChEMBL	407	6	2	6	5.4	COc1ccc(Nc2nc(Nc3cccc(F)c3C)cc(N3CCCCC3)n2)cc1	10.1016/j.bmcl.2011.09.033
	57401220	68454	0	None	-	0	Human	5.4	pIC50	=	5.4	Binding	Displacement of [125I]galanin from GalR2 by gamma countingDisplacement of [125I]galanin from GalR2 by gamma counting	ChEMBL	411	7	2	6	5.6	FC(F)Oc1cccc(Nc2cc(Nc3ccccc3)nc(N3CCCCC3)n2)c1	10.1016/j.bmcl.2011.09.033
	CHEMBL1921989	68454	0	None	-	0	Human	5.4	pIC50	=	5.4	Binding	Displacement of [125I]galanin from GalR2 by gamma countingDisplacement of [125I]galanin from GalR2 by gamma counting	ChEMBL	411	7	2	6	5.6	FC(F)Oc1cccc(Nc2cc(Nc3ccccc3)nc(N3CCCCC3)n2)c1	10.1016/j.bmcl.2011.09.033
	57394241	68480	0	None	-	0	Human	5.4	pIC50	=	5.4	Binding	Displacement of [125I]galanin from GalR2 by gamma countingDisplacement of [125I]galanin from GalR2 by gamma counting	ChEMBL	427	6	2	6	5.8	COc1ccc(Nc2nc(Nc3ccc(F)c(Cl)c3)cc(N3CCCCC3)n2)cc1	10.1016/j.bmcl.2011.09.033
	CHEMBL1922014	68480	0	None	-	0	Human	5.4	pIC50	=	5.4	Binding	Displacement of [125I]galanin from GalR2 by gamma countingDisplacement of [125I]galanin from GalR2 by gamma counting	ChEMBL	427	6	2	6	5.8	COc1ccc(Nc2nc(Nc3ccc(F)c(Cl)c3)cc(N3CCCCC3)n2)cc1	10.1016/j.bmcl.2011.09.033
	57394240	68476	0	None	-	0	Human	6.4	pIC50	=	6.4	Binding	Displacement of [125I]galanin from GalR2 by gamma countingDisplacement of [125I]galanin from GalR2 by gamma counting	ChEMBL	423	7	2	7	5.1	COc1ccc(Nc2nc(Nc3ccc(OC)c(F)c3)cc(N3CCCCC3)n2)cc1	10.1016/j.bmcl.2011.09.033
	CHEMBL1922010	68476	0	None	-	0	Human	6.4	pIC50	=	6.4	Binding	Displacement of [125I]galanin from GalR2 by gamma countingDisplacement of [125I]galanin from GalR2 by gamma counting	ChEMBL	423	7	2	7	5.1	COc1ccc(Nc2nc(Nc3ccc(OC)c(F)c3)cc(N3CCCCC3)n2)cc1	10.1016/j.bmcl.2011.09.033
	57397799	68471	0	None	-	0	Human	6.4	pIC50	=	6.4	Binding	Displacement of [125I]galanin from GalR2 by gamma countingDisplacement of [125I]galanin from GalR2 by gamma counting	ChEMBL	403	6	2	6	5.6	COc1ccc(Nc2nc(Nc3cc(C)ccc3C)cc(N3CCCCC3)n2)cc1	10.1016/j.bmcl.2011.09.033
	CHEMBL1922005	68471	0	None	-	0	Human	6.4	pIC50	=	6.4	Binding	Displacement of [125I]galanin from GalR2 by gamma countingDisplacement of [125I]galanin from GalR2 by gamma counting	ChEMBL	403	6	2	6	5.6	COc1ccc(Nc2nc(Nc3cc(C)ccc3C)cc(N3CCCCC3)n2)cc1	10.1016/j.bmcl.2011.09.033
	CHEMBL474037	212274	0	None	-	0	Rat	6.4	pIC50	=	6.4	Binding	Inhibition of [3H]glycine uptake at rat glycine transporter 2 expressed in african green monkey COS7 cellsInhibition of [3H]glycine uptake at rat glycine transporter 2 expressed in african green monkey COS7 cells	ChEMBL		None	None	None		CC[C@H](C)[C@@H]1NC(=O)[C@H](C(C)C)NC(=O)[C@H](Cc2ccccc2)NC(=O)[C@H]([C@H](C)[C@@H](C)O)NC1=O	10.1016/j.bmcl.2008.10.104
	57394303	68400	0	None	-	0	Human	5.3	pIC50	=	5.3	Binding	Displacement of [125I]galanin from GalR2 by gamma countingDisplacement of [125I]galanin from GalR2 by gamma counting	ChEMBL	373	5	2	5	5.6	Cc1ccc(C)c(Nc2cc(Nc3ccccc3)nc(N3CCCCC3)n2)c1	10.1016/j.bmcl.2011.09.033
	CHEMBL1921901	68400	0	None	-	0	Human	5.3	pIC50	=	5.3	Binding	Displacement of [125I]galanin from GalR2 by gamma countingDisplacement of [125I]galanin from GalR2 by gamma counting	ChEMBL	373	5	2	5	5.6	Cc1ccc(C)c(Nc2cc(Nc3ccccc3)nc(N3CCCCC3)n2)c1	10.1016/j.bmcl.2011.09.033
	57394239	68475	0	None	-	0	Human	6.3	pIC50	=	6.3	Binding	Displacement of [125I]galanin from GalR2 by gamma countingDisplacement of [125I]galanin from GalR2 by gamma counting	ChEMBL	441	8	2	7	5.6	COc1ccc(Nc2nc(Nc3cccc(OC(F)F)c3)cc(N3CCCCC3)n2)cc1	10.1016/j.bmcl.2011.09.033
	CHEMBL1922009	68475	0	None	-	0	Human	6.3	pIC50	=	6.3	Binding	Displacement of [125I]galanin from GalR2 by gamma countingDisplacement of [125I]galanin from GalR2 by gamma counting	ChEMBL	441	8	2	7	5.6	COc1ccc(Nc2nc(Nc3cccc(OC(F)F)c3)cc(N3CCCCC3)n2)cc1	10.1016/j.bmcl.2011.09.033
	CHEMBL474038	212275	0	None	-	0	Rat	6.3	pIC50	=	6.3	Binding	Inhibition of [3H]glycine uptake at rat glycine transporter 2 expressed in african green monkey COS7 cellsInhibition of [3H]glycine uptake at rat glycine transporter 2 expressed in african green monkey COS7 cells	ChEMBL		None	None	None		CC(C)[C@@H]1NC(=O)[C@H](Cc2ccccc2)NC(=O)[C@H]([C@H](C)[C@@H](C)O)NC(=O)[C@H](C(C)C)NC1=O	10.1016/j.bmcl.2008.10.104
	57399457	68464	0	None	-	0	Human	6.3	pIC50	=	6.3	Binding	Displacement of [125I]galanin from GalR2 by gamma countingDisplacement of [125I]galanin from GalR2 by gamma counting	ChEMBL	473	8	3	7	6.6	COc1ccc(Nc2cc(Nc3cccc(OC(F)(F)F)c3)nc(NC3CCCCC3)n2)cc1	10.1016/j.bmcl.2011.09.033
	CHEMBL1921999	68464	0	None	-	0	Human	6.3	pIC50	=	6.3	Binding	Displacement of [125I]galanin from GalR2 by gamma countingDisplacement of [125I]galanin from GalR2 by gamma counting	ChEMBL	473	8	3	7	6.6	COc1ccc(Nc2cc(Nc3cccc(OC(F)(F)F)c3)nc(NC3CCCCC3)n2)cc1	10.1016/j.bmcl.2011.09.033
	57394238	68469	0	None	-	0	Human	6.3	pIC50	=	6.3	Binding	Displacement of [125I]galanin from GalR2 by gamma countingDisplacement of [125I]galanin from GalR2 by gamma counting	ChEMBL	529	5	1	7	5.8	Cc1c(F)cccc1Nc1cc(N2CCCCC2)nc(N2CCCN(c3ncccc3C(F)(F)F)CC2)n1	10.1016/j.bmcl.2011.09.033
	CHEMBL1922003	68469	0	None	-	0	Human	6.3	pIC50	=	6.3	Binding	Displacement of [125I]galanin from GalR2 by gamma countingDisplacement of [125I]galanin from GalR2 by gamma counting	ChEMBL	529	5	1	7	5.8	Cc1c(F)cccc1Nc1cc(N2CCCCC2)nc(N2CCCN(c3ncccc3C(F)(F)F)CC2)n1	10.1016/j.bmcl.2011.09.033
	CHEMBL473840	212273	0	None	-	0	Rat	6.2	pIC50	=	6.2	Binding	Inhibition of [3H]glycine uptake at rat glycine transporter 2 expressed in african green monkey COS7 cellsInhibition of [3H]glycine uptake at rat glycine transporter 2 expressed in african green monkey COS7 cells	ChEMBL		None	None	None		CC[C@H](C)[C@@H]1NC(=O)[C@H](Cc2ccccc2)NC(=O)[C@H]([C@H](C)[C@@H](C)O)NC(=O)[C@H](C(C)C)NC1=O	10.1016/j.bmcl.2008.10.104
	57394304	68402	0	None	-	0	Human	5.2	pIC50	=	5.2	Binding	Displacement of [125I]galanin from GalR2 by gamma countingDisplacement of [125I]galanin from GalR2 by gamma counting	ChEMBL	429	6	2	6	5.9	FC(F)(F)Oc1cccc(Nc2cc(Nc3ccccc3)nc(N3CCCCC3)n2)c1	10.1016/j.bmcl.2011.09.033
	CHEMBL1921903	68402	0	None	-	0	Human	5.2	pIC50	=	5.2	Binding	Displacement of [125I]galanin from GalR2 by gamma countingDisplacement of [125I]galanin from GalR2 by gamma counting	ChEMBL	429	6	2	6	5.9	FC(F)(F)Oc1cccc(Nc2cc(Nc3ccccc3)nc(N3CCCCC3)n2)c1	10.1016/j.bmcl.2011.09.033
	57401221	68461	0	None	-	0	Human	6.1	pIC50	=	6.1	Binding	Displacement of [125I]galanin from GalR2 by gamma countingDisplacement of [125I]galanin from GalR2 by gamma counting	ChEMBL	455	9	3	7	6.3	COc1ccc(Nc2cc(Nc3cccc(OC(F)F)c3)nc(NC3CCCCC3)n2)cc1	10.1016/j.bmcl.2011.09.033
	CHEMBL1921996	68461	0	None	-	0	Human	6.1	pIC50	=	6.1	Binding	Displacement of [125I]galanin from GalR2 by gamma countingDisplacement of [125I]galanin from GalR2 by gamma counting	ChEMBL	455	9	3	7	6.3	COc1ccc(Nc2cc(Nc3cccc(OC(F)F)c3)nc(NC3CCCCC3)n2)cc1	10.1016/j.bmcl.2011.09.033
	57390716	68481	0	None	-	0	Human	6.1	pIC50	=	6.1	Binding	Displacement of [125I]galanin from GalR2 by gamma countingDisplacement of [125I]galanin from GalR2 by gamma counting	ChEMBL	437	7	2	7	5.5	COc1ccc(Nc2nc(Nc3ccc(OC)c(F)c3)cc(N3CCCCCC3)n2)cc1	10.1016/j.bmcl.2011.09.033
	CHEMBL1922016	68481	0	None	-	0	Human	6.1	pIC50	=	6.1	Binding	Displacement of [125I]galanin from GalR2 by gamma countingDisplacement of [125I]galanin from GalR2 by gamma counting	ChEMBL	437	7	2	7	5.5	COc1ccc(Nc2nc(Nc3ccc(OC)c(F)c3)cc(N3CCCCCC3)n2)cc1	10.1016/j.bmcl.2011.09.033
	57399459	68474	0	None	-	0	Human	6.1	pIC50	=	6.1	Binding	Displacement of [125I]galanin from GalR2 by gamma countingDisplacement of [125I]galanin from GalR2 by gamma counting	ChEMBL	443	6	2	6	6.0	COc1ccc(Nc2nc(Nc3ccc(C(F)(F)F)cc3)cc(N3CCCCC3)n2)cc1	10.1016/j.bmcl.2011.09.033
	CHEMBL1922008	68474	0	None	-	0	Human	6.1	pIC50	=	6.1	Binding	Displacement of [125I]galanin from GalR2 by gamma countingDisplacement of [125I]galanin from GalR2 by gamma counting	ChEMBL	443	6	2	6	6.0	COc1ccc(Nc2nc(Nc3ccc(C(F)(F)F)cc3)cc(N3CCCCC3)n2)cc1	10.1016/j.bmcl.2011.09.033
	57397797	68459	0	None	-	0	Human	5.1	pIC50	=	5.1	Binding	Displacement of [125I]galanin from GalR2 by gamma countingDisplacement of [125I]galanin from GalR2 by gamma counting	ChEMBL	391	7	2	7	4.6	COc1ccc(Nc2cc(Nc3ccc(OC)cc3)nc(N3CCCC3)n2)cc1	10.1016/j.bmcl.2011.09.033
	CHEMBL1921994	68459	0	None	-	0	Human	5.1	pIC50	=	5.1	Binding	Displacement of [125I]galanin from GalR2 by gamma countingDisplacement of [125I]galanin from GalR2 by gamma counting	ChEMBL	391	7	2	7	4.6	COc1ccc(Nc2cc(Nc3ccc(OC)cc3)nc(N3CCCC3)n2)cc1	10.1016/j.bmcl.2011.09.033
	57395992	68456	0	None	-	0	Human	5.1	pIC50	=	5.1	Binding	Displacement of [125I]galanin from GalR2 by gamma countingDisplacement of [125I]galanin from GalR2 by gamma counting	ChEMBL	393	6	2	6	5.1	COc1ccc(Nc2cc(Nc3ccccc3)nc(N3CCCCC3)n2)cc1F	10.1016/j.bmcl.2011.09.033
	CHEMBL1921991	68456	0	None	-	0	Human	5.1	pIC50	=	5.1	Binding	Displacement of [125I]galanin from GalR2 by gamma countingDisplacement of [125I]galanin from GalR2 by gamma counting	ChEMBL	393	6	2	6	5.1	COc1ccc(Nc2cc(Nc3ccccc3)nc(N3CCCCC3)n2)cc1F	10.1016/j.bmcl.2011.09.033
	CHEMBL451169	212216	0	None	-	0	Rat	7.1	pIC50	=	7.1	Binding	Inhibition of [3H]glycine uptake at rat glycine transporter 2 expressed in african green monkey COS7 cellsInhibition of [3H]glycine uptake at rat glycine transporter 2 expressed in african green monkey COS7 cells	ChEMBL		None	None	None		CC[C@H](C)[C@@H]1NC(=O)[C@H](Cc2cn(OC)c3ccccc23)NC(=O)[C@H](CCCCC(C)=O)NC(=O)[C@H]2CCCCN2C1=O	10.1016/j.bmcl.2008.10.104
	57401228	68488	0	None	-	0	Human	5.0	pIC50	=	5.0	Binding	Displacement of [125I]galanin from GalR2 by gamma countingDisplacement of [125I]galanin from GalR2 by gamma counting	ChEMBL	538	7	2	9	5.6	COc1ccc(Nc2nc(Nc3ccc(OC)c(F)c3)cc(N3CCCN(C(=O)OC(C)(C)C)CC3)n2)cc1	10.1016/j.bmcl.2011.09.033
	CHEMBL1922025	68488	0	None	-	0	Human	5.0	pIC50	=	5.0	Binding	Displacement of [125I]galanin from GalR2 by gamma countingDisplacement of [125I]galanin from GalR2 by gamma counting	ChEMBL	538	7	2	9	5.6	COc1ccc(Nc2nc(Nc3ccc(OC)c(F)c3)cc(N3CCCN(C(=O)OC(C)(C)C)CC3)n2)cc1	10.1016/j.bmcl.2011.09.033
	57394236	68458	0	None	-	0	Human	6.0	pIC50	=	6.0	Binding	Displacement of [125I]galanin from GalR2 by gamma countingDisplacement of [125I]galanin from GalR2 by gamma counting	ChEMBL	391	7	2	7	4.6	COc1ccc(Nc2cc(Nc3cccc(OC)c3)nc(N3CCCC3)n2)cc1	10.1016/j.bmcl.2011.09.033
	CHEMBL1921993	68458	0	None	-	0	Human	6.0	pIC50	=	6.0	Binding	Displacement of [125I]galanin from GalR2 by gamma countingDisplacement of [125I]galanin from GalR2 by gamma counting	ChEMBL	391	7	2	7	4.6	COc1ccc(Nc2cc(Nc3cccc(OC)c3)nc(N3CCCC3)n2)cc1	10.1016/j.bmcl.2011.09.033
	57395995	68478	0	None	-	0	Human	6.0	pIC50	=	6.0	Binding	Displacement of [125I]galanin from GalR2 by gamma countingDisplacement of [125I]galanin from GalR2 by gamma counting	ChEMBL	407	6	2	6	5.4	COc1ccc(Nc2nc(Nc3ccc(F)cc3C)cc(N3CCCCC3)n2)cc1	10.1016/j.bmcl.2011.09.033
	CHEMBL1922012	68478	0	None	-	0	Human	6.0	pIC50	=	6.0	Binding	Displacement of [125I]galanin from GalR2 by gamma countingDisplacement of [125I]galanin from GalR2 by gamma counting	ChEMBL	407	6	2	6	5.4	COc1ccc(Nc2nc(Nc3ccc(F)cc3C)cc(N3CCCCC3)n2)cc1	10.1016/j.bmcl.2011.09.033
	CHEMBL526003	213893	24	None	-10	3	Human	9.0	pKd	=	9	Binding	Binding affinity to human GalR2Binding affinity to human GalR2	ChEMBL		None	None	None		CSCC[C@H](NC(=O)[C@H](CC(C)C)NC(=O)CNC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)CN)[C@@H](C)O)C(N)=O	10.1021/jm801088x
	CHEMBL506210	212434	0	None	478	2	Human	8.7	pKd	=	8.7	Binding	Binding affinity to human GalR2Binding affinity to human GalR2	ChEMBL		None	None	None		None	10.1021/jm801088x
	CHEMBL503473	212396	13	None	-60	3	Human	8.7	pKd	=	8.7	Binding	Binding affinity to human GalR2Binding affinity to human GalR2	ChEMBL		None	None	None		CC(C)C[C@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)CN)[C@@H](C)O)C(=O)NCC(=O)N1CCC[C@H]1C(=O)N1CCC[C@H]1C(=O)N1CCC[C@H]1C(=O)NCC(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](CO)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](CCCNC(=N)N)C(N)=O	10.1021/jm801088x
	155817464	1471	0	None	-5	4	Human	8.6	pKd	=	8.6	Binding	Binding affinity to human GalR2Binding affinity to human GalR2	ChEMBL		None	None	None		None	10.1021/jm801088x
	3866	1471	0	None	-5	4	Human	8.6	pKd	=	8.6	Binding	Binding affinity to human GalR2Binding affinity to human GalR2	ChEMBL		None	None	None		None	10.1021/jm801088x
	44587986	1471	0	None	-5	4	Human	8.6	pKd	=	8.6	Binding	Binding affinity to human GalR2Binding affinity to human GalR2	ChEMBL		None	None	None		None	10.1021/jm801088x
	91934870	1471	0	None	-5	4	Human	8.6	pKd	=	8.6	Binding	Binding affinity to human GalR2Binding affinity to human GalR2	ChEMBL		None	None	None		None	10.1021/jm801088x
	CHEMBL499179	1471	0	None	-5	4	Human	8.6	pKd	=	8.6	Binding	Binding affinity to human GalR2Binding affinity to human GalR2	ChEMBL		None	None	None		None	10.1021/jm801088x
	71717271	85663	1	None	-1	3	Human	4.6	pKd	=	4.6	Binding	Binding affinity to human GalR2Binding affinity to human GalR2	ChEMBL	678	13	4	7	6.5	Cc1cc(=O)oc2cc(NC(=O)[C@@H](CCCCN)NC(=O)[C@H](CC3CCCCC3)NC(=O)OCC3c4ccccc4-c4ccccc43)ccc12	10.1021/jm801088x
	CHEMBL2309599	85663	1	None	-1	3	Human	4.6	pKd	=	4.6	Binding	Binding affinity to human GalR2Binding affinity to human GalR2	ChEMBL	678	13	4	7	6.5	Cc1cc(=O)oc2cc(NC(=O)[C@@H](CCCCN)NC(=O)[C@H](CC3CCCCC3)NC(=O)OCC3c4ccccc4-c4ccccc43)ccc12	10.1021/jm801088x
	16132180	1694	14	None	-3	8	Human	8.3	pKd	=	8.3	Binding	Binding affinity to human GalR2Binding affinity to human GalR2	ChEMBL		None	None	None		None	10.1021/jm801088x
	16133822	1694	14	None	-3	8	Human	8.3	pKd	=	8.3	Binding	Binding affinity to human GalR2Binding affinity to human GalR2	ChEMBL		None	None	None		None	10.1021/jm801088x
	6087	1694	14	None	-3	8	Human	8.3	pKd	=	8.3	Binding	Binding affinity to human GalR2Binding affinity to human GalR2	ChEMBL		None	None	None		None	10.1021/jm801088x
	CHEMBL499980	1694	14	None	-3	8	Human	8.3	pKd	=	8.3	Binding	Binding affinity to human GalR2Binding affinity to human GalR2	ChEMBL		None	None	None		None	10.1021/jm801088x
	CHEMBL604373	214045	3	None	-7	2	Human	9.2	pKi	=	9.2	Binding	Binding affinity to human GalR2Binding affinity to human GalR2	ChEMBL		None	None	None		CC(C)C[C@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@@H]1CCCN1C(=O)[C@H](CCCCN)NC(=O)[C@@H]1CCCN1C(=O)[C@@H](CCCNC(=N)N)NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)CN)[C@@H](C)O)C(N)=O	10.1021/jm9018349
	CHEMBL501079	212359	10	None	-11	2	Human	9.1	pKi	=	9.1	Binding	Binding affinity to human GalR2Binding affinity to human GalR2	ChEMBL		None	None	None		CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](Cc1c[nH]cn1)NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)CN)[C@@H](C)O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](Cc1c[nH]cn1)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](Cc1c[nH]cn1)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)NCC(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C)C(N)=O	10.1021/jm9018349
	CHEMBL526003	213893	24	None	-10	3	Human	9.0	pKi	=	9.0	Binding	Binding affinity to human GalR2Binding affinity to human GalR2	ChEMBL		None	None	None		CSCC[C@H](NC(=O)[C@H](CC(C)C)NC(=O)CNC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)CN)[C@@H](C)O)C(N)=O	10.1021/jm9018349
	CHEMBL592413	214032	0	None	-4	2	Human	8.9	pKi	=	8.9	Binding	Binding affinity to human GalR2Binding affinity to human GalR2	ChEMBL		None	None	None		CC[C@H](C)[C@H](NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)CN)[C@@H](C)O)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@H](C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](Cc1ccc(O)cc1)C(N)=O)[C@@H](C)O	10.1021/jm9018349
	CHEMBL604990	214047	20	None	-15	2	Human	8.8	pKi	=	8.8	Binding	Binding affinity to human GalR2Binding affinity to human GalR2	ChEMBL		None	None	None		CC(C)C[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](C)NC(=O)[C@@H]1CCCN1C(=O)[C@@H]1CCCN1C(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)CN)[C@@H](C)O)C(=O)N[C@@H](C)C(N)=O	10.1021/jm9018349
	CHEMBL578710	214001	20	None	501	2	Human	8.8	pKi	=	8.8	Binding	Binding affinity to human GalR2Binding affinity to human GalR2	ChEMBL		None	None	None		CC(C)C[C@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@@H](N)Cc1c[nH]c2ccccc12)[C@@H](C)O)C(N)=O	10.1021/jm9018349
	CHEMBL503473	212396	13	None	-60	3	Human	8.7	pKi	=	8.7	Binding	Binding affinity to human GalR2Binding affinity to human GalR2	ChEMBL		None	None	None		CC(C)C[C@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)CN)[C@@H](C)O)C(=O)NCC(=O)N1CCC[C@H]1C(=O)N1CCC[C@H]1C(=O)N1CCC[C@H]1C(=O)NCC(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](CO)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](CCCNC(=N)N)C(N)=O	10.1021/jm9018349
	25180488	187782	0	None	-4	2	Human	7.0	pKi	=	7.0	Binding	Displacement of europium-labeled galanin from human GalR2 expressed in CHO-K1 cellsDisplacement of europium-labeled galanin from human GalR2 expressed in CHO-K1 cells	ChEMBL	2111	78	26	26	-0.5	CCCCCCCCCCCCCCCC(=O)NCCCC[C@H](NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)CNC)[C@@H](C)O)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O	10.1021/jm801088x
	CHEMBL501306	187782	0	None	-4	2	Human	7.0	pKi	=	7.0	Binding	Displacement of europium-labeled galanin from human GalR2 expressed in CHO-K1 cellsDisplacement of europium-labeled galanin from human GalR2 expressed in CHO-K1 cells	ChEMBL	2111	78	26	26	-0.5	CCCCCCCCCCCCCCCC(=O)NCCCC[C@H](NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)CNC)[C@@H](C)O)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O	10.1021/jm801088x
	CHEMBL2324949	207782	0	None	-3	2	Human	6.9	pKi	=	6.9	Binding	Displacement of euporium-galanin from human GalR2 after 1.5 hrs by DELFIA assayDisplacement of euporium-galanin from human GalR2 after 1.5 hrs by DELFIA assay	ChEMBL		None	None	None		CNCC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@]1(C)CCC/C=C/CCC[C@@](C)(C(=O)NCC(=O)N2CCC[C@H]2C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc2ccc(O)cc2)NC(=O)CNC1=O)[C@@H](C)O	10.1016/j.bmc.2012.10.026
	CHEMBL508083	212936	0	None	-25	2	Human	7.9	pKi	=	7.9	Binding	Displacement of europium-labeled galanin from human GalR2 expressed in CHO-K1 cellsDisplacement of europium-labeled galanin from human GalR2 expressed in CHO-K1 cells	ChEMBL		None	None	None		CC(C)C[C@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)CN)[C@@H](C)O)C(=O)NCC(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1cnc[nH]1)C(=O)N[C@@H](C)C(=O)N[C@H](C(N)=O)C(C)C	10.1021/jm801088x
	25180498	192753	0	None	-4	2	Human	5.9	pKi	=	5.9	Binding	Displacement of europium-labeled galanin from human GalR2 expressed in CHO-K1 cellsDisplacement of europium-labeled galanin from human GalR2 expressed in CHO-K1 cells	ChEMBL	1957	75	25	24	0.3	CCCCCCCCCCCCCCCC(=O)NCCCC[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)CNC)[C@@H](C)O)C(=O)N[C@@H](CCCCN)C(N)=O	10.1021/jm801088x
	CHEMBL524892	192753	0	None	-4	2	Human	5.9	pKi	=	5.9	Binding	Displacement of europium-labeled galanin from human GalR2 expressed in CHO-K1 cellsDisplacement of europium-labeled galanin from human GalR2 expressed in CHO-K1 cells	ChEMBL	1957	75	25	24	0.3	CCCCCCCCCCCCCCCC(=O)NCCCC[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)CNC)[C@@H](C)O)C(=O)N[C@@H](CCCCN)C(N)=O	10.1021/jm801088x
	44563953	176226	0	None	-11	2	Human	7.8	pKi	=	7.8	Binding	Displacement of europium labeled galanin from human recombinant GalR2 receptor by time-resolved fluorescence binding assayDisplacement of europium labeled galanin from human recombinant GalR2 receptor by time-resolved fluorescence binding assay	ChEMBL	2028	72	25	27	-2.5	CCCCCCCCCC(=O)NCCCC[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)OC(=O)CNC)[C@@H](C)O)C(=O)N[C@@H](CCCCN)C(N)=O	10.1021/jm801397w
	CHEMBL460706	176226	0	None	-11	2	Human	7.8	pKi	=	7.8	Binding	Displacement of europium labeled galanin from human recombinant GalR2 receptor by time-resolved fluorescence binding assayDisplacement of europium labeled galanin from human recombinant GalR2 receptor by time-resolved fluorescence binding assay	ChEMBL	2028	72	25	27	-2.5	CCCCCCCCCC(=O)NCCCC[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)OC(=O)CNC)[C@@H](C)O)C(=O)N[C@@H](CCCCN)C(N)=O	10.1021/jm801397w
	44563952	188093	0	None	-20	2	Human	7.8	pKi	=	7.8	Binding	Displacement of europium labeled galanin from human recombinant GalR2 receptor by time-resolved fluorescence binding assayDisplacement of europium labeled galanin from human recombinant GalR2 receptor by time-resolved fluorescence binding assay	ChEMBL	2000	70	25	27	-3.2	CCCCCCCC(=O)NCCCC[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)OC(=O)CNC)[C@@H](C)O)C(=O)N[C@@H](CCCCN)C(N)=O	10.1021/jm801397w
	CHEMBL503900	188093	0	None	-20	2	Human	7.8	pKi	=	7.8	Binding	Displacement of europium labeled galanin from human recombinant GalR2 receptor by time-resolved fluorescence binding assayDisplacement of europium labeled galanin from human recombinant GalR2 receptor by time-resolved fluorescence binding assay	ChEMBL	2000	70	25	27	-3.2	CCCCCCCC(=O)NCCCC[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)OC(=O)CNC)[C@@H](C)O)C(=O)N[C@@H](CCCCN)C(N)=O	10.1021/jm801397w
	44563957	172173	0	None	-3	2	Human	7.8	pKi	=	7.8	Binding	Displacement of europium labeled galanin from human recombinant GalR2 receptor by time-resolved fluorescence binding assayDisplacement of europium labeled galanin from human recombinant GalR2 receptor by time-resolved fluorescence binding assay	ChEMBL	2140	80	25	27	0.7	CCCCCCCCCCCCCCCCCC(=O)NCCCC[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)OC(=O)CNC)[C@@H](C)O)C(=O)N[C@@H](CCCCN)C(N)=O	10.1021/jm801397w
	CHEMBL450827	172173	0	None	-3	2	Human	7.8	pKi	=	7.8	Binding	Displacement of europium labeled galanin from human recombinant GalR2 receptor by time-resolved fluorescence binding assayDisplacement of europium labeled galanin from human recombinant GalR2 receptor by time-resolved fluorescence binding assay	ChEMBL	2140	80	25	27	0.7	CCCCCCCCCCCCCCCCCC(=O)NCCCC[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)OC(=O)CNC)[C@@H](C)O)C(=O)N[C@@H](CCCCN)C(N)=O	10.1021/jm801397w
	25180491	192848	0	None	-16	2	Human	7.8	pKi	=	7.8	Binding	Displacement of europium-labeled galanin from human GalR2 expressed in CHO-K1 cellsDisplacement of europium-labeled galanin from human GalR2 expressed in CHO-K1 cells	ChEMBL	2111	78	26	26	-0.5	CCCCCCCCCCCCCCCC(=O)NCCCC[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@@H](CCCCN)NC(=O)[C@H]1CCCN1C(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)CNC)[C@@H](C)O)C(=O)N[C@@H](CCCCN)C(N)=O	10.1021/jm801088x
	CHEMBL526500	192848	0	None	-16	2	Human	7.8	pKi	=	7.8	Binding	Displacement of europium-labeled galanin from human GalR2 expressed in CHO-K1 cellsDisplacement of europium-labeled galanin from human GalR2 expressed in CHO-K1 cells	ChEMBL	2111	78	26	26	-0.5	CCCCCCCCCCCCCCCC(=O)NCCCC[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@@H](CCCCN)NC(=O)[C@H]1CCCN1C(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)CNC)[C@@H](C)O)C(=O)N[C@@H](CCCCN)C(N)=O	10.1021/jm801088x
	CHEMBL2324950	207783	0	None	-4	2	Human	7.8	pKi	=	7.8	Binding	Displacement of euporium-galanin from human GalR2 after 1.5 hrs by DELFIA assayDisplacement of euporium-galanin from human GalR2 after 1.5 hrs by DELFIA assay	ChEMBL		None	None	None		CNCC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)NCC(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N1CCC[C@H]1C(=O)N[C@@]1(C)CCC/C=C\CCC[C@@](C)(C(=O)N[C@@H](CCCCN)C(N)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC1=O)[C@@H](C)O	10.1016/j.bmc.2012.10.026
	45104656	196895	0	None	-9	2	Human	7.8	pKi	=	7.8	Binding	Displacement of Eu-labeled galanin from human GalR2 by DELFIA competitive assayDisplacement of Eu-labeled galanin from human GalR2 by DELFIA competitive assay	ChEMBL	2082	76	25	25	0.3	CCCCCCCCCCCCCCCC(=O)NCCCC[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(C)=O)[C@@H](C)O)C(=O)N[C@@H](CCCCN)C(N)=O	10.1021/jm9018349
	CHEMBL578317	196895	0	None	-9	2	Human	7.8	pKi	=	7.8	Binding	Displacement of Eu-labeled galanin from human GalR2 by DELFIA competitive assayDisplacement of Eu-labeled galanin from human GalR2 by DELFIA competitive assay	ChEMBL	2082	76	25	25	0.3	CCCCCCCCCCCCCCCC(=O)NCCCC[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(C)=O)[C@@H](C)O)C(=O)N[C@@H](CCCCN)C(N)=O	10.1021/jm9018349
	44563954	188325	0	None	-11	2	Human	7.8	pKi	=	7.8	Binding	Displacement of europium labeled galanin from human recombinant GalR2 receptor by time-resolved fluorescence binding assayDisplacement of europium labeled galanin from human recombinant GalR2 receptor by time-resolved fluorescence binding assay	ChEMBL	2056	74	25	27	-1.7	CCCCCCCCCCCC(=O)NCCCC[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)OC(=O)CNC)[C@@H](C)O)C(=O)N[C@@H](CCCCN)C(N)=O	10.1021/jm801397w
	CHEMBL507733	188325	0	None	-11	2	Human	7.8	pKi	=	7.8	Binding	Displacement of europium labeled galanin from human recombinant GalR2 receptor by time-resolved fluorescence binding assayDisplacement of europium labeled galanin from human recombinant GalR2 receptor by time-resolved fluorescence binding assay	ChEMBL	2056	74	25	27	-1.7	CCCCCCCCCCCC(=O)NCCCC[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)OC(=O)CNC)[C@@H](C)O)C(=O)N[C@@H](CCCCN)C(N)=O	10.1021/jm801397w
	25180486	192867	0	None	-1	2	Human	6.8	pKi	=	6.8	Binding	Displacement of europium-labeled galanin from human GalR2 expressed in CHO-K1 cellsDisplacement of europium-labeled galanin from human GalR2 expressed in CHO-K1 cells	ChEMBL	1935	66	23	23	-0.4	CCCCCCCCCCCCCCCC(=O)NCCCC[C@H](NC(=O)[C@H](C)NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)CNC)[C@@H](C)O)C(N)=O	10.1021/jm801088x
	44587983	192867	0	None	-1	2	Human	6.8	pKi	=	6.8	Binding	Displacement of europium-labeled galanin from human GalR2 expressed in CHO-K1 cellsDisplacement of europium-labeled galanin from human GalR2 expressed in CHO-K1 cells	ChEMBL	1935	66	23	23	-0.4	CCCCCCCCCCCCCCCC(=O)NCCCC[C@H](NC(=O)[C@H](C)NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)CNC)[C@@H](C)O)C(N)=O	10.1021/jm801088x
	CHEMBL526862	192867	0	None	-1	2	Human	6.8	pKi	=	6.8	Binding	Displacement of europium-labeled galanin from human GalR2 expressed in CHO-K1 cellsDisplacement of europium-labeled galanin from human GalR2 expressed in CHO-K1 cells	ChEMBL	1935	66	23	23	-0.4	CCCCCCCCCCCCCCCC(=O)NCCCC[C@H](NC(=O)[C@H](C)NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)CNC)[C@@H](C)O)C(N)=O	10.1021/jm801088x
	25180489	187677	0	None	-5	2	Human	7.8	pKi	=	7.8	Binding	Displacement of Eu-labeled galanin from human GalR2 by DELFIA competitive assayDisplacement of Eu-labeled galanin from human GalR2 by DELFIA competitive assay	ChEMBL	2097	77	26	26	-0.8	CCCCCCCCCCCCCCCC(=O)NCCCC[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)CN)[C@@H](C)O)C(=O)N[C@@H](CCCCN)C(N)=O	10.1021/jm9018349
	CHEMBL499807	187677	0	None	-5	2	Human	7.8	pKi	=	7.8	Binding	Displacement of Eu-labeled galanin from human GalR2 by DELFIA competitive assayDisplacement of Eu-labeled galanin from human GalR2 by DELFIA competitive assay	ChEMBL	2097	77	26	26	-0.8	CCCCCCCCCCCCCCCC(=O)NCCCC[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)CN)[C@@H](C)O)C(=O)N[C@@H](CCCCN)C(N)=O	10.1021/jm9018349
	44563955	192739	0	None	-7	2	Human	7.7	pKi	=	7.7	Binding	Displacement of europium labeled galanin from human recombinant GalR2 receptor by time-resolved fluorescence binding assayDisplacement of europium labeled galanin from human recombinant GalR2 receptor by time-resolved fluorescence binding assay	ChEMBL	2084	76	25	27	-0.9	CCCCCCCCCCCCCC(=O)NCCCC[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)OC(=O)CNC)[C@@H](C)O)C(=O)N[C@@H](CCCCN)C(N)=O	10.1021/jm801397w
	CHEMBL524678	192739	0	None	-7	2	Human	7.7	pKi	=	7.7	Binding	Displacement of europium labeled galanin from human recombinant GalR2 receptor by time-resolved fluorescence binding assayDisplacement of europium labeled galanin from human recombinant GalR2 receptor by time-resolved fluorescence binding assay	ChEMBL	2084	76	25	27	-0.9	CCCCCCCCCCCCCC(=O)NCCCC[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)OC(=O)CNC)[C@@H](C)O)C(=O)N[C@@H](CCCCN)C(N)=O	10.1021/jm801397w
	CHEMBL501079	212359	10	None	-11	2	Human	8.6	pKi	=	8.6	Binding	Binding affinity to human GAL2 receptor by radioligand displacement assayBinding affinity to human GAL2 receptor by radioligand displacement assay	ChEMBL		None	None	None		CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](Cc1c[nH]cn1)NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)CN)[C@@H](C)O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](Cc1c[nH]cn1)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](Cc1c[nH]cn1)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)NCC(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C)C(N)=O	10.1016/j.ejmech.2013.01.044
	45104657	199776	0	None	18	2	Human	7.7	pKi	=	7.7	Binding	Displacement of Eu-labeled galanin from human GalR2 by DELFIA competitive assayDisplacement of Eu-labeled galanin from human GalR2 by DELFIA competitive assay	ChEMBL	2054	76	25	25	0.3	CCCCCCCCCCCCCCCC(=O)NCCCC[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC)[C@@H](C)O)C(=O)N[C@@H](CCCCN)C(N)=O	10.1021/jm9018349
	CHEMBL604991	199776	0	None	18	2	Human	7.7	pKi	=	7.7	Binding	Displacement of Eu-labeled galanin from human GalR2 by DELFIA competitive assayDisplacement of Eu-labeled galanin from human GalR2 by DELFIA competitive assay	ChEMBL	2054	76	25	25	0.3	CCCCCCCCCCCCCCCC(=O)NCCCC[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC)[C@@H](C)O)C(=O)N[C@@H](CCCCN)C(N)=O	10.1021/jm9018349
	44563958	188167	0	None	-40	2	Human	7.7	pKi	=	7.7	Binding	Displacement of europium labeled galanin from human recombinant GalR2 receptor by time-resolved fluorescence binding assayDisplacement of europium labeled galanin from human recombinant GalR2 receptor by time-resolved fluorescence binding assay	ChEMBL	2122	78	25	32	-5.9	CNCC(=O)O[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)NCC(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N1CCC[C@H]1C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCNC(=O)COCCOCCOCCOCCOC)C(=O)N[C@@H](CCCCN)C(N)=O)[C@@H](C)O	10.1021/jm801397w
	CHEMBL505299	188167	0	None	-40	2	Human	7.7	pKi	=	7.7	Binding	Displacement of europium labeled galanin from human recombinant GalR2 receptor by time-resolved fluorescence binding assayDisplacement of europium labeled galanin from human recombinant GalR2 receptor by time-resolved fluorescence binding assay	ChEMBL	2122	78	25	32	-5.9	CNCC(=O)O[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)NCC(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N1CCC[C@H]1C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCNC(=O)COCCOCCOCCOCCOC)C(=O)N[C@@H](CCCCN)C(N)=O)[C@@H](C)O	10.1021/jm801397w
	25180497	192869	0	None	-5	2	Human	6.7	pKi	=	6.7	Binding	Displacement of europium-labeled galanin from human GalR2 expressed in CHO-K1 cellsDisplacement of europium-labeled galanin from human GalR2 expressed in CHO-K1 cells	ChEMBL	2213	87	29	28	-0.4	CCCCCCCCCCCCCCCC(=O)NCCCC[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)CNC)[C@@H](C)O)C(=O)N[C@@H](CCCCN)C(N)=O	10.1021/jm801088x
	CHEMBL526889	192869	0	None	-5	2	Human	6.7	pKi	=	6.7	Binding	Displacement of europium-labeled galanin from human GalR2 expressed in CHO-K1 cellsDisplacement of europium-labeled galanin from human GalR2 expressed in CHO-K1 cells	ChEMBL	2213	87	29	28	-0.4	CCCCCCCCCCCCCCCC(=O)NCCCC[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)CNC)[C@@H](C)O)C(=O)N[C@@H](CCCCN)C(N)=O	10.1021/jm801088x
	CHEMBL592170	214031	0	None	2	2	Human	6.7	pKi	=	6.7	Binding	Binding affinity to human GalR2Binding affinity to human GalR2	ChEMBL		None	None	None		CC(C)C[C@H](NC(=O)CNC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](CO)NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](CO)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@H](CC(N)=O)NC(=O)CNC(=O)[C@@H](NC(=O)[C@H](C)NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)CN)[C@@H](C)O)C(C)C)C(=O)N[C@H](C(=O)N[C@@H](CO)C(N)=O)[C@@H](C)O	10.1021/jm9018349
	25180487	192799	0	None	-11	2	Human	7.7	pKi	=	7.7	Binding	Displacement of europium-labeled galanin from human GalR2 expressed in CHO-K1 cellsDisplacement of europium-labeled galanin from human GalR2 expressed in CHO-K1 cells	ChEMBL	2111	78	26	26	-0.5	CCCCCCCCCCCCCCCC(=O)NCCCC[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)CNC)[C@@H](C)O)C(N)=O	10.1021/jm801088x
	CHEMBL525755	192799	0	None	-11	2	Human	7.7	pKi	=	7.7	Binding	Displacement of europium-labeled galanin from human GalR2 expressed in CHO-K1 cellsDisplacement of europium-labeled galanin from human GalR2 expressed in CHO-K1 cells	ChEMBL	2111	78	26	26	-0.5	CCCCCCCCCCCCCCCC(=O)NCCCC[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)CNC)[C@@H](C)O)C(N)=O	10.1021/jm801088x
	25180489	187677	0	None	-5	2	Human	7.7	pKi	=	7.7	Binding	Displacement of europium-labeled galanin from human GalR2 expressed in CHO-K1 cellsDisplacement of europium-labeled galanin from human GalR2 expressed in CHO-K1 cells	ChEMBL	2097	77	26	26	-0.8	CCCCCCCCCCCCCCCC(=O)NCCCC[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)CN)[C@@H](C)O)C(=O)N[C@@H](CCCCN)C(N)=O	10.1021/jm801088x
	CHEMBL499807	187677	0	None	-5	2	Human	7.7	pKi	=	7.7	Binding	Displacement of europium-labeled galanin from human GalR2 expressed in CHO-K1 cellsDisplacement of europium-labeled galanin from human GalR2 expressed in CHO-K1 cells	ChEMBL	2097	77	26	26	-0.8	CCCCCCCCCCCCCCCC(=O)NCCCC[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)CN)[C@@H](C)O)C(=O)N[C@@H](CCCCN)C(N)=O	10.1021/jm801088x
	44563951	188350	0	None	-60	2	Human	7.6	pKi	=	7.6	Binding	Displacement of europium labeled galanin from human recombinant GalR2 receptor by time-resolved fluorescence binding assayDisplacement of europium labeled galanin from human recombinant GalR2 receptor by time-resolved fluorescence binding assay	ChEMBL	1874	63	25	27	-5.8	CNCC(=O)O[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)NCC(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N1CCC[C@H]1C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O)[C@@H](C)O	10.1021/jm801397w
	CHEMBL508036	188350	0	None	-60	2	Human	7.6	pKi	=	7.6	Binding	Displacement of europium labeled galanin from human recombinant GalR2 receptor by time-resolved fluorescence binding assayDisplacement of europium labeled galanin from human recombinant GalR2 receptor by time-resolved fluorescence binding assay	ChEMBL	1874	63	25	27	-5.8	CNCC(=O)O[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)NCC(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N1CCC[C@H]1C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O)[C@@H](C)O	10.1021/jm801397w
	CHEMBL525055	213858	0	None	-60	2	Human	7.6	pKi	=	7.6	Binding	Displacement of europium-labeled galanin from human GalR2 expressed in CHO-K1 cellsDisplacement of europium-labeled galanin from human GalR2 expressed in CHO-K1 cells	ChEMBL		None	None	None		CNCC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)NCC(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N1CCC[C@H]1C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O)[C@@H](C)O	10.1021/jm801088x
	25180494	188144	0	None	-4	2	Human	7.6	pKi	=	7.6	Binding	Displacement of europium-labeled galanin from human GalR2 expressed in CHO-K1 cellsDisplacement of europium-labeled galanin from human GalR2 expressed in CHO-K1 cells	ChEMBL	2111	78	26	26	-0.5	CCCCCCCCCCCCCCCC(=O)NCCCC[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)CNC)[C@@H](C)O)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O	10.1021/jm801088x
	CHEMBL504914	188144	0	None	-4	2	Human	7.6	pKi	=	7.6	Binding	Displacement of europium-labeled galanin from human GalR2 expressed in CHO-K1 cellsDisplacement of europium-labeled galanin from human GalR2 expressed in CHO-K1 cells	ChEMBL	2111	78	26	26	-0.5	CCCCCCCCCCCCCCCC(=O)NCCCC[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)CNC)[C@@H](C)O)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O	10.1021/jm801088x
	CHEMBL501079	212359	10	None	-11	2	Human	8.5	pKi	=	8.5	Binding	Displacement of radiolabeled galanin from human galanin 2 receptorDisplacement of radiolabeled galanin from human galanin 2 receptor	ChEMBL		None	None	None		CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](Cc1c[nH]cn1)NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)CN)[C@@H](C)O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](Cc1c[nH]cn1)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](Cc1c[nH]cn1)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)NCC(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C)C(N)=O	10.1021/jm8007618
	71717271	85663	1	None	-2	3	Rat	4.5	pKi	=	4.5	Binding	Binding affinity to rat GalR2Binding affinity to rat GalR2	ChEMBL	678	13	4	7	6.5	Cc1cc(=O)oc2cc(NC(=O)[C@@H](CCCCN)NC(=O)[C@H](CC3CCCCC3)NC(=O)OCC3c4ccccc4-c4ccccc43)ccc12	10.1021/jm9018349
	CHEMBL2309599	85663	1	None	-2	3	Rat	4.5	pKi	=	4.5	Binding	Binding affinity to rat GalR2Binding affinity to rat GalR2	ChEMBL	678	13	4	7	6.5	Cc1cc(=O)oc2cc(NC(=O)[C@@H](CCCCN)NC(=O)[C@H](CC3CCCCC3)NC(=O)OCC3c4ccccc4-c4ccccc43)ccc12	10.1021/jm9018349
	45104655	196950	0	None	-3	2	Human	7.5	pKi	=	7.5	Binding	Displacement of Eu-labeled galanin from human GalR2 by DELFIA competitive assayDisplacement of Eu-labeled galanin from human GalR2 by DELFIA competitive assay	ChEMBL	2111	77	26	26	-0.4	CCCCCCCCCCCCCCCC(=O)NCCCC[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@H](C)N)[C@@H](C)O)C(=O)N[C@@H](CCCCN)C(N)=O	10.1021/jm9018349
	CHEMBL578910	196950	0	None	-3	2	Human	7.5	pKi	=	7.5	Binding	Displacement of Eu-labeled galanin from human GalR2 by DELFIA competitive assayDisplacement of Eu-labeled galanin from human GalR2 by DELFIA competitive assay	ChEMBL	2111	77	26	26	-0.4	CCCCCCCCCCCCCCCC(=O)NCCCC[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@H](C)N)[C@@H](C)O)C(=O)N[C@@H](CCCCN)C(N)=O	10.1021/jm9018349
	25180495	188245	0	None	8	2	Human	7.3	pKi	=	7.3	Binding	Displacement of Eu-labeled galanin from human GalR2 by DELFIA competitive assayDisplacement of Eu-labeled galanin from human GalR2 by DELFIA competitive assay	ChEMBL	2040	75	25	25	0.1	CCCCCCCCCCCCCCCC(=O)NCCCC[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@@H](N)Cc1c[nH]c2ccccc12)[C@@H](C)O)C(=O)N[C@@H](CCCCN)C(N)=O	10.1021/jm9018349
	CHEMBL506495	188245	0	None	8	2	Human	7.3	pKi	=	7.3	Binding	Displacement of Eu-labeled galanin from human GalR2 by DELFIA competitive assayDisplacement of Eu-labeled galanin from human GalR2 by DELFIA competitive assay	ChEMBL	2040	75	25	25	0.1	CCCCCCCCCCCCCCCC(=O)NCCCC[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@@H](N)Cc1c[nH]c2ccccc12)[C@@H](C)O)C(=O)N[C@@H](CCCCN)C(N)=O	10.1021/jm9018349
	25180495	188245	0	None	8	2	Human	7.3	pKi	=	7.3	Binding	Displacement of europium-labeled galanin from human GalR2 expressed in CHO-K1 cellsDisplacement of europium-labeled galanin from human GalR2 expressed in CHO-K1 cells	ChEMBL	2040	75	25	25	0.1	CCCCCCCCCCCCCCCC(=O)NCCCC[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@@H](N)Cc1c[nH]c2ccccc12)[C@@H](C)O)C(=O)N[C@@H](CCCCN)C(N)=O	10.1021/jm801088x
	CHEMBL506495	188245	0	None	8	2	Human	7.3	pKi	=	7.3	Binding	Displacement of europium-labeled galanin from human GalR2 expressed in CHO-K1 cellsDisplacement of europium-labeled galanin from human GalR2 expressed in CHO-K1 cells	ChEMBL	2040	75	25	25	0.1	CCCCCCCCCCCCCCCC(=O)NCCCC[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@@H](N)Cc1c[nH]c2ccccc12)[C@@H](C)O)C(=O)N[C@@H](CCCCN)C(N)=O	10.1021/jm801088x
	25180496	188135	0	None	-2	2	Human	7.3	pKi	=	7.3	Binding	Displacement of europium-labeled galanin from human GalR2 expressed in CHO-K1 cellsDisplacement of europium-labeled galanin from human GalR2 expressed in CHO-K1 cells	ChEMBL	2153	81	26	26	0.8	CCCCCCCCCCCCCCCC(=O)NCCCC[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)CCCCCN)[C@@H](C)O)C(=O)N[C@@H](CCCCN)C(N)=O	10.1021/jm801088x
	CHEMBL504758	188135	0	None	-2	2	Human	7.3	pKi	=	7.3	Binding	Displacement of europium-labeled galanin from human GalR2 expressed in CHO-K1 cellsDisplacement of europium-labeled galanin from human GalR2 expressed in CHO-K1 cells	ChEMBL	2153	81	26	26	0.8	CCCCCCCCCCCCCCCC(=O)NCCCC[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)CCCCCN)[C@@H](C)O)C(=O)N[C@@H](CCCCN)C(N)=O	10.1021/jm801088x
	24760995	196910	0	None	-14	2	Human	7.3	pKi	=	7.3	Binding	Displacement of Eu-labeled galanin from human GalR2 by DELFIA competitive assayDisplacement of Eu-labeled galanin from human GalR2 by DELFIA competitive assay	ChEMBL	2112	78	26	26	0.1	CCCCCCCCCCCCCCCC(=O)NCCCC[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)CNC)[C@@H](C)O)C(=O)N[C@@H](CCCCN)C(=O)O	10.1021/jm9018349
	CHEMBL578514	196910	0	None	-14	2	Human	7.3	pKi	=	7.3	Binding	Displacement of Eu-labeled galanin from human GalR2 by DELFIA competitive assayDisplacement of Eu-labeled galanin from human GalR2 by DELFIA competitive assay	ChEMBL	2112	78	26	26	0.1	CCCCCCCCCCCCCCCC(=O)NCCCC[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)CNC)[C@@H](C)O)C(=O)N[C@@H](CCCCN)C(=O)O	10.1021/jm9018349
	44563956	188302	0	None	-14	2	Human	7.3	pKi	=	7.3	Binding	Displacement of europium labeled galanin from human recombinant GalR2 receptor by time-resolved fluorescence binding assayDisplacement of europium labeled galanin from human recombinant GalR2 receptor by time-resolved fluorescence binding assay	ChEMBL	2112	78	25	27	-0.1	CCCCCCCCCCCCCCCC(=O)NCCCC[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)OC(=O)CNC)[C@@H](C)O)C(=O)N[C@@H](CCCCN)C(N)=O	10.1021/jm801397w
	CHEMBL507353	188302	0	None	-14	2	Human	7.3	pKi	=	7.3	Binding	Displacement of europium labeled galanin from human recombinant GalR2 receptor by time-resolved fluorescence binding assayDisplacement of europium labeled galanin from human recombinant GalR2 receptor by time-resolved fluorescence binding assay	ChEMBL	2112	78	25	27	-0.1	CCCCCCCCCCCCCCCC(=O)NCCCC[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)OC(=O)CNC)[C@@H](C)O)C(=O)N[C@@H](CCCCN)C(N)=O	10.1021/jm801397w
	44587984	192761	1	None	-14	2	Human	7.3	pKi	=	7.3	Binding	Displacement of europium-labeled galanin from human GalR2 expressed in CHO-K1 cellsDisplacement of europium-labeled galanin from human GalR2 expressed in CHO-K1 cells	ChEMBL	2111	78	26	26	-0.5	CCCCCCCCCCCCCCCC(=O)NCCCC[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)CNC)[C@@H](C)O)C(=O)N[C@@H](CCCCN)C(N)=O	10.1021/jm801088x
	CHEMBL525023	192761	1	None	-14	2	Human	7.3	pKi	=	7.3	Binding	Displacement of europium-labeled galanin from human GalR2 expressed in CHO-K1 cellsDisplacement of europium-labeled galanin from human GalR2 expressed in CHO-K1 cells	ChEMBL	2111	78	26	26	-0.5	CCCCCCCCCCCCCCCC(=O)NCCCC[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)CNC)[C@@H](C)O)C(=O)N[C@@H](CCCCN)C(N)=O	10.1021/jm801088x
	24760995	196910	0	None	-14	2	Human	7.3	pKi	=	7.3	Binding	Binding affinity to human GalR2Binding affinity to human GalR2	ChEMBL	2112	78	26	26	0.1	CCCCCCCCCCCCCCCC(=O)NCCCC[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)CNC)[C@@H](C)O)C(=O)N[C@@H](CCCCN)C(=O)O	10.1021/jm9018349
	CHEMBL578514	196910	0	None	-14	2	Human	7.3	pKi	=	7.3	Binding	Binding affinity to human GalR2Binding affinity to human GalR2	ChEMBL	2112	78	26	26	0.1	CCCCCCCCCCCCCCCC(=O)NCCCC[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)CNC)[C@@H](C)O)C(=O)N[C@@H](CCCCN)C(=O)O	10.1021/jm9018349
	25180490	62855	0	None	-19	2	Human	7.2	pKi	=	7.2	Binding	Displacement of europium-labeled galanin from human GalR2 expressed in CHO-K1 cellsDisplacement of europium-labeled galanin from human GalR2 expressed in CHO-K1 cells	ChEMBL	2195	78	32	26	-3.1	CCCCCCCCCCCCCCCC(=O)NCCCC[C@H](NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)CNC)[C@@H](C)O)C(=O)N[C@@H](CCCNC(=N)N)C(N)=O	10.1021/jm801088x
	91934869	62855	0	None	-19	2	Human	7.2	pKi	=	7.2	Binding	Displacement of europium-labeled galanin from human GalR2 expressed in CHO-K1 cellsDisplacement of europium-labeled galanin from human GalR2 expressed in CHO-K1 cells	ChEMBL	2195	78	32	26	-3.1	CCCCCCCCCCCCCCCC(=O)NCCCC[C@H](NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)CNC)[C@@H](C)O)C(=O)N[C@@H](CCCNC(=N)N)C(N)=O	10.1021/jm801088x
	CHEMBL1790054	62855	0	None	-19	2	Human	7.2	pKi	=	7.2	Binding	Displacement of europium-labeled galanin from human GalR2 expressed in CHO-K1 cellsDisplacement of europium-labeled galanin from human GalR2 expressed in CHO-K1 cells	ChEMBL	2195	78	32	26	-3.1	CCCCCCCCCCCCCCCC(=O)NCCCC[C@H](NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)CNC)[C@@H](C)O)C(=O)N[C@@H](CCCNC(=N)N)C(N)=O	10.1021/jm801088x
	25180492	188304	0	None	-2	2	Human	7.1	pKi	=	7.1	Binding	Displacement of europium-labeled galanin from human GalR2 expressed in CHO-K1 cellsDisplacement of europium-labeled galanin from human GalR2 expressed in CHO-K1 cells	ChEMBL	2014	77	26	25	-0.5	CCCCCCCCCCCCCCCC(=O)NCCCC[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)CNC)[C@@H](C)O)C(=O)N[C@@H](CCCCN)C(N)=O	10.1021/jm801088x
	CHEMBL507373	188304	0	None	-2	2	Human	7.1	pKi	=	7.1	Binding	Displacement of europium-labeled galanin from human GalR2 expressed in CHO-K1 cellsDisplacement of europium-labeled galanin from human GalR2 expressed in CHO-K1 cells	ChEMBL	2014	77	26	25	-0.5	CCCCCCCCCCCCCCCC(=O)NCCCC[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)CNC)[C@@H](C)O)C(=O)N[C@@H](CCCCN)C(N)=O	10.1021/jm801088x
	CHEMBL592415	214033	0	None	5	2	Human	8.0	pKi	=	8.0	Binding	Binding affinity to human GalR2Binding affinity to human GalR2	ChEMBL		None	None	None		None	10.1021/jm9018349
	155817484	1686	0	None	-3	6	Rat	9.1	pKd	=	9.1	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9281594
	155817484	1686	0	None	-3	6	Rat	9.1	pKd	=	9.1	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9427506
	155817484	1686	0	None	-3	6	Rat	9.1	pKd	=	9.1	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9578584
	155817484	1686	0	None	-3	6	Rat	9.1	pKd	=	9.1	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9722565
	6117	1686	0	None	-3	6	Rat	9.1	pKd	=	9.1	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9281594
	6117	1686	0	None	-3	6	Rat	9.1	pKd	=	9.1	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9427506
	6117	1686	0	None	-3	6	Rat	9.1	pKd	=	9.1	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9578584
	6117	1686	0	None	-3	6	Rat	9.1	pKd	=	9.1	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9722565
	6129	1686	0	None	-3	6	Rat	9.1	pKd	=	9.1	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9281594
	6129	1686	0	None	-3	6	Rat	9.1	pKd	=	9.1	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9427506
	6129	1686	0	None	-3	6	Rat	9.1	pKd	=	9.1	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9578584
	6129	1686	0	None	-3	6	Rat	9.1	pKd	=	9.1	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9722565
	155817484	1686	0	None	-1	6	Human	9.5	pKd	=	9.5	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9880084
	6117	1686	0	None	-1	6	Human	9.5	pKd	=	9.5	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9880084
	6129	1686	0	None	-1	6	Human	9.5	pKd	=	9.5	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9880084
	155817484	1686	0	None	-1	6	Human	9.9	pKd	=	9.9	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9685625
	6117	1686	0	None	-1	6	Human	9.9	pKd	=	9.9	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9685625
	6129	1686	0	None	-1	6	Human	9.9	pKd	=	9.9	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9685625
	24748735	1725	1	None	3	2	Rat	5.0	pKd	>	5	Binding	UnclassifiedUnclassified	Guide to Pharmacology	988	12	7	15	4.2	NCCCC[C@@H](C(=O)OC)NC(=O)[C@]1(C)NC(=O)c2nc(oc2C)[C@@](C)(NC(=O)c2nc([C@](NC(=O)c3nc1oc3C)(C)C(=O)NCC1CCCCC1)oc2C)C(=O)NC1c2ccccc2c2c1cccc2	15240875
	24748735	1725	1	None	3	2	Rat	5.0	pKd	>	5	Binding	UnclassifiedUnclassified	Guide to Pharmacology	988	12	7	15	4.2	NCCCC[C@@H](C(=O)OC)NC(=O)[C@]1(C)NC(=O)c2nc(oc2C)[C@@](C)(NC(=O)c2nc([C@](NC(=O)c3nc1oc3C)(C)C(=O)NCC1CCCCC1)oc2C)C(=O)NC1c2ccccc2c2c1cccc2	15944002
	6119	1725	1	None	3	2	Rat	5.0	pKd	>	5	Binding	UnclassifiedUnclassified	Guide to Pharmacology	988	12	7	15	4.2	NCCCC[C@@H](C(=O)OC)NC(=O)[C@]1(C)NC(=O)c2nc(oc2C)[C@@](C)(NC(=O)c2nc([C@](NC(=O)c3nc1oc3C)(C)C(=O)NCC1CCCCC1)oc2C)C(=O)NC1c2ccccc2c2c1cccc2	15240875
	6119	1725	1	None	3	2	Rat	5.0	pKd	>	5	Binding	UnclassifiedUnclassified	Guide to Pharmacology	988	12	7	15	4.2	NCCCC[C@@H](C(=O)OC)NC(=O)[C@]1(C)NC(=O)c2nc(oc2C)[C@@](C)(NC(=O)c2nc([C@](NC(=O)c3nc1oc3C)(C)C(=O)NCC1CCCCC1)oc2C)C(=O)NC1c2ccccc2c2c1cccc2	15944002
	CHEMBL1187471	1725	1	None	3	2	Rat	5.0	pKd	>	5	Binding	UnclassifiedUnclassified	Guide to Pharmacology	988	12	7	15	4.2	NCCCC[C@@H](C(=O)OC)NC(=O)[C@]1(C)NC(=O)c2nc(oc2C)[C@@](C)(NC(=O)c2nc([C@](NC(=O)c3nc1oc3C)(C)C(=O)NCC1CCCCC1)oc2C)C(=O)NC1c2ccccc2c2c1cccc2	15240875
	CHEMBL1187471	1725	1	None	3	2	Rat	5.0	pKd	>	5	Binding	UnclassifiedUnclassified	Guide to Pharmacology	988	12	7	15	4.2	NCCCC[C@@H](C(=O)OC)NC(=O)[C@]1(C)NC(=O)c2nc(oc2C)[C@@](C)(NC(=O)c2nc([C@](NC(=O)c3nc1oc3C)(C)C(=O)NCC1CCCCC1)oc2C)C(=O)NC1c2ccccc2c2c1cccc2	15944002
	16131409	1693	0	125I-GALANIN	4	3	Rat	9.2	pKi	=	9.2	Binding	NoneNone	PDSP KiDatabase		None	None	None		None	None
	6086	1693	0	125I-GALANIN	4	3	Rat	9.2	pKi	=	9.2	Binding	NoneNone	PDSP KiDatabase		None	None	None		None	None
	None	214290	0	125I-h Galanin	-1	6	Rat	9.1	pKi	=	9.1	Binding	NoneNone	PDSP KiDatabase	418	8	0	4	4.3	CC1=CC=C(C=C1)OCCN(C2=CC=CC=C2OC)C(=O)CN3CCCCC3.Cl	None
	None	214290	0	125I-GALANIN	-1	6	Rat	9.0	pKi	=	9	Binding	NoneNone	PDSP KiDatabase	418	8	0	4	4.3	CC1=CC=C(C=C1)OCCN(C2=CC=CC=C2OC)C(=O)CN3CCCCC3.Cl	None
	None	214290	0	125I-GALANIN	1	6	Human	9.0	pKi	=	9.0	Binding	NoneNone	PDSP KiDatabase	418	8	0	4	4.3	CC1=CC=C(C=C1)OCCN(C2=CC=CC=C2OC)C(=O)CN3CCCCC3.Cl	None
	None	214290	0	125I-p Galanin	-1	6	Rat	9.0	pKi	=	9.0	Binding	NoneNone	PDSP KiDatabase	418	8	0	4	4.3	CC1=CC=C(C=C1)OCCN(C2=CC=CC=C2OC)C(=O)CN3CCCCC3.Cl	None
	None	214290	0	125I-h Galanin	-1	6	Rat	8.9	pKi	=	8.9	Binding	NoneNone	PDSP KiDatabase	418	8	0	4	4.3	CC1=CC=C(C=C1)OCCN(C2=CC=CC=C2OC)C(=O)CN3CCCCC3.Cl	None
	None	214290	0	125I-GALANIN	-1	6	Rat	8.7	pKi	=	8.7	Binding	NoneNone	PDSP KiDatabase	418	8	0	4	4.3	CC1=CC=C(C=C1)OCCN(C2=CC=CC=C2OC)C(=O)CN3CCCCC3.Cl	None
	None	214290	0	125I-GALANIN	-1	6	Rat	7.6	pKi	=	7.6	Binding	NoneNone	PDSP KiDatabase	418	8	0	4	4.3	CC1=CC=C(C=C1)OCCN(C2=CC=CC=C2OC)C(=O)CN3CCCCC3.Cl	None
	5311268	1726	0	None	-2	2	Rat	4.5	pKi	=	4.5	Binding	UnclassifiedUnclassified	Guide to Pharmacology	678	13	4	7	6.5	NCCCC[C@@H](C(=O)Nc1ccc2c(c1)oc(=O)cc2C)NC(=O)[C@@H](NC(=O)OCC1c2ccccc2c2c1cccc2)CC1CCCCC1	15240875
	5311268	1726	0	None	-2	2	Rat	4.5	pKi	=	4.5	Binding	UnclassifiedUnclassified	Guide to Pharmacology	678	13	4	7	6.5	NCCCC[C@@H](C(=O)Nc1ccc2c(c1)oc(=O)cc2C)NC(=O)[C@@H](NC(=O)OCC1c2ccccc2c2c1cccc2)CC1CCCCC1	15944002
	6118	1726	0	None	-2	2	Rat	4.5	pKi	=	4.5	Binding	UnclassifiedUnclassified	Guide to Pharmacology	678	13	4	7	6.5	NCCCC[C@@H](C(=O)Nc1ccc2c(c1)oc(=O)cc2C)NC(=O)[C@@H](NC(=O)OCC1c2ccccc2c2c1cccc2)CC1CCCCC1	15240875
	6118	1726	0	None	-2	2	Rat	4.5	pKi	=	4.5	Binding	UnclassifiedUnclassified	Guide to Pharmacology	678	13	4	7	6.5	NCCCC[C@@H](C(=O)Nc1ccc2c(c1)oc(=O)cc2C)NC(=O)[C@@H](NC(=O)OCC1c2ccccc2c2c1cccc2)CC1CCCCC1	15944002
	CHEMBL592414	1726	0	None	-2	2	Rat	4.5	pKi	=	4.5	Binding	UnclassifiedUnclassified	Guide to Pharmacology	678	13	4	7	6.5	NCCCC[C@@H](C(=O)Nc1ccc2c(c1)oc(=O)cc2C)NC(=O)[C@@H](NC(=O)OCC1c2ccccc2c2c1cccc2)CC1CCCCC1	15240875
	CHEMBL592414	1726	0	None	-2	2	Rat	4.5	pKi	=	4.5	Binding	UnclassifiedUnclassified	Guide to Pharmacology	678	13	4	7	6.5	NCCCC[C@@H](C(=O)Nc1ccc2c(c1)oc(=O)cc2C)NC(=O)[C@@H](NC(=O)OCC1c2ccccc2c2c1cccc2)CC1CCCCC1	15944002
	155817481	1702	0	None	-2	6	Rat	5.8	pKi	=	5.8	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9405385
	155817481	1702	0	None	-2	6	Rat	5.8	pKi	=	5.8	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9742938
	155817481	1702	0	None	-2	6	Rat	5.8	pKi	=	5.8	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9832122
	6092	1702	0	None	-2	6	Rat	5.8	pKi	=	5.8	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9405385
	6092	1702	0	None	-2	6	Rat	5.8	pKi	=	5.8	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9742938
	6092	1702	0	None	-2	6	Rat	5.8	pKi	=	5.8	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9832122
	6095	1709	0	None	-14	6	Human	6.7	pKi	=	6.7	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9880084
	155817474	1698	0	None	-5	5	Rat	7.1	pKi	=	7.1	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	15944007
	5357	1698	0	None	-5	5	Rat	7.1	pKi	=	7.1	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	15944007
	6108	1730	0	None	-	1	Human	7.2	pKi	=	7.2	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	23259957
	6105	1714	0	None	-14	2	Human	7.3	pKi	=	7.3	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	19053761
	6107	1722	0	None	8	2	Human	7.3	pKi	=	7.3	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	19053761
	6103	2407	0	None	18	3	Human	7.4	pKi	=	7.4	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	21333705
	6074	2409	0	None	301	3	Human	7.5	pKi	=	7.5	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	23192661
	6102	2406	0	None	3	3	Human	7.5	pKi	=	7.5	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	21333705
	6110	1723	0	None	-60	2	Human	7.6	pKi	=	7.6	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	19199479
	6116	1721	0	None	-40	2	Human	7.7	pKi	=	7.7	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	19199479
	6109	2790	0	None	17	2	Human	7.7	pKi	=	7.7	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	20121116
	6075	2077	0	None	5	3	Human	7.7	pKi	=	7.7	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	23600864
	6114	1717	0	None	-7	2	Human	7.7	pKi	=	7.7	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	19199479
	155817474	1698	0	None	5	5	Human	7.8	pKi	=	7.8	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	19467704
	5357	1698	0	None	5	5	Human	7.8	pKi	=	7.8	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	19467704
	6113	1716	0	None	-11	2	Human	7.8	pKi	=	7.8	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	19199479
	6115	1718	0	None	-3	2	Human	7.8	pKi	=	7.8	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	19199479
	6111	1719	0	None	-20	2	Human	7.8	pKi	=	7.8	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	19199479
	6112	1715	0	None	-11	2	Human	7.8	pKi	=	7.8	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	19199479
	155817463	765	0	None	-58	8	Mouse	7.9	pKi	=	7.9	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9832122
	3861	765	0	None	-58	8	Mouse	7.9	pKi	=	7.9	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9832122
	6095	1709	0	None	14	6	Rat	7.9	pKi	=	7.9	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9305929
	6095	1709	0	None	14	6	Rat	7.9	pKi	=	7.9	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9722565
	6106	1720	0	None	-10	2	Human	7.9	pKi	=	7.9	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	23259957
	3900	2418	0	None	31	3	Human	7.9	pKi	=	7.9	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	None
	3897	2412	0	None	-13	6	Rat	7.9	pKi	=	7.9	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9305929
	16132180	1694	14	None	-7	8	Mouse	7.9	pKi	=	7.9	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9832122
	16133822	1694	14	None	-7	8	Mouse	7.9	pKi	=	7.9	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9832122
	6087	1694	14	None	-7	8	Mouse	7.9	pKi	=	7.9	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9832122
	CHEMBL499980	1694	14	None	-7	8	Mouse	7.9	pKi	=	7.9	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9832122
	155817465	1700	0	None	-11	6	Rat	8.0	pKi	=	8.0	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9281594
	155817465	1700	0	None	-11	6	Rat	8.0	pKi	=	8.0	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9405385
	155817465	1700	0	None	-11	6	Rat	8.0	pKi	=	8.0	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9742938
	155817465	1700	0	None	-11	6	Rat	8.0	pKi	=	8.0	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9832122
	3876	1700	0	None	-11	6	Rat	8.0	pKi	=	8.0	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9281594
	3876	1700	0	None	-11	6	Rat	8.0	pKi	=	8.0	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9405385
	3876	1700	0	None	-11	6	Rat	8.0	pKi	=	8.0	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9742938
	3876	1700	0	None	-11	6	Rat	8.0	pKi	=	8.0	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9832122
	155817464	1471	0	None	-17	4	Rat	8.2	pKi	=	8.2	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9305929
	3866	1471	0	None	-17	4	Rat	8.2	pKi	=	8.2	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9305929
	44587986	1471	0	None	-17	4	Rat	8.2	pKi	=	8.2	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9305929
	91934870	1471	0	None	-17	4	Rat	8.2	pKi	=	8.2	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9305929
	CHEMBL499179	1471	0	None	-17	4	Rat	8.2	pKi	=	8.2	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9305929
	155817465	1700	0	None	-7	6	Mouse	8.2	pKi	=	8.2	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9832122
	3876	1700	0	None	-7	6	Mouse	8.2	pKi	=	8.2	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9832122
	6101	2405	0	None	75	3	Human	8.2	pKi	=	8.2	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	19467704
	6141	1691	0	None	-	1	Human	8.2	pKi	=	8.2	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9480833
	6099	2411	0	None	-23	2	Human	8.2	pKi	=	8.2	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	11600206
	6100	2416	0	None	-25	3	Human	8.2	pKi	=	8.2	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	None
	6104	2408	0	None	45	3	Human	8.3	pKi	=	8.3	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	21333705
	16132180	1694	14	None	-3	8	Rat	8.3	pKi	=	8.3	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9281594
	16132180	1694	14	None	-3	8	Rat	8.3	pKi	=	8.3	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9305929
	16132180	1694	14	None	-3	8	Rat	8.3	pKi	=	8.3	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9405385
	16132180	1694	14	None	-3	8	Rat	8.3	pKi	=	8.3	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9722565
	16132180	1694	14	None	-3	8	Rat	8.3	pKi	=	8.3	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9742938
	16132180	1694	14	None	-3	8	Rat	8.3	pKi	=	8.3	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9832122
	16133822	1694	14	None	-3	8	Rat	8.3	pKi	=	8.3	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9281594
	16133822	1694	14	None	-3	8	Rat	8.3	pKi	=	8.3	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9305929
	16133822	1694	14	None	-3	8	Rat	8.3	pKi	=	8.3	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9405385
	16133822	1694	14	None	-3	8	Rat	8.3	pKi	=	8.3	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9722565
	16133822	1694	14	None	-3	8	Rat	8.3	pKi	=	8.3	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9742938
	16133822	1694	14	None	-3	8	Rat	8.3	pKi	=	8.3	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9832122
	6087	1694	14	None	-3	8	Rat	8.3	pKi	=	8.3	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9281594
	6087	1694	14	None	-3	8	Rat	8.3	pKi	=	8.3	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9305929
	6087	1694	14	None	-3	8	Rat	8.3	pKi	=	8.3	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9405385
	6087	1694	14	None	-3	8	Rat	8.3	pKi	=	8.3	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9722565
	6087	1694	14	None	-3	8	Rat	8.3	pKi	=	8.3	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9742938
	6087	1694	14	None	-3	8	Rat	8.3	pKi	=	8.3	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9832122
	CHEMBL499980	1694	14	None	-3	8	Rat	8.3	pKi	=	8.3	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9281594
	CHEMBL499980	1694	14	None	-3	8	Rat	8.3	pKi	=	8.3	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9305929
	CHEMBL499980	1694	14	None	-3	8	Rat	8.3	pKi	=	8.3	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9405385
	CHEMBL499980	1694	14	None	-3	8	Rat	8.3	pKi	=	8.3	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9722565
	CHEMBL499980	1694	14	None	-3	8	Rat	8.3	pKi	=	8.3	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9742938
	CHEMBL499980	1694	14	None	-3	8	Rat	8.3	pKi	=	8.3	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9832122
	155817479	1706	0	None	-1	6	Human	8.3	pKi	=	8.3	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9880084
	6083	1706	0	None	-1	6	Human	8.3	pKi	=	8.3	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9880084
	6076	2078	0	None	2	3	Human	8.3	pKi	=	8.3	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	23600864
	3898	2413	0	None	-20	7	Mouse	8.3	pKi	=	8.3	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9832122
	6139	1696	0	None	1	2	Rat	8.3	pKi	=	8.3	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9405385
	16132180	1694	14	None	-3	8	Human	8.4	pKi	=	8.4	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	19053761
	16132180	1694	14	None	-3	8	Human	8.4	pKi	=	8.4	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9480833
	16132180	1694	14	None	-3	8	Human	8.4	pKi	=	8.4	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9880084
	16133822	1694	14	None	-3	8	Human	8.4	pKi	=	8.4	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	19053761
	16133822	1694	14	None	-3	8	Human	8.4	pKi	=	8.4	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9480833
	16133822	1694	14	None	-3	8	Human	8.4	pKi	=	8.4	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9880084
	6087	1694	14	None	-3	8	Human	8.4	pKi	=	8.4	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	19053761
	6087	1694	14	None	-3	8	Human	8.4	pKi	=	8.4	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9480833
	6087	1694	14	None	-3	8	Human	8.4	pKi	=	8.4	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9880084
	CHEMBL499980	1694	14	None	-3	8	Human	8.4	pKi	=	8.4	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	19053761
	CHEMBL499980	1694	14	None	-3	8	Human	8.4	pKi	=	8.4	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9480833
	CHEMBL499980	1694	14	None	-3	8	Human	8.4	pKi	=	8.4	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9880084
	101927062	1685	21	None	-8	6	Human	8.4	pKi	=	8.4	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	11983932
	101927062	1685	21	None	-8	6	Human	8.4	pKi	=	8.4	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9480833
	155817445	1685	21	None	-8	6	Human	8.4	pKi	=	8.4	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	11983932
	155817445	1685	21	None	-8	6	Human	8.4	pKi	=	8.4	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9480833
	16133823	1685	21	None	-8	6	Human	8.4	pKi	=	8.4	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	11983932
	16133823	1685	21	None	-8	6	Human	8.4	pKi	=	8.4	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9480833
	3592	1685	21	None	-8	6	Human	8.4	pKi	=	8.4	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	11983932
	3592	1685	21	None	-8	6	Human	8.4	pKi	=	8.4	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9480833
	44584852	1685	21	None	-8	6	Human	8.4	pKi	=	8.4	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	11983932
	44584852	1685	21	None	-8	6	Human	8.4	pKi	=	8.4	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9480833
	6090	1685	21	None	-8	6	Human	8.4	pKi	=	8.4	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	11983932
	6090	1685	21	None	-8	6	Human	8.4	pKi	=	8.4	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9480833
	91898917	1685	21	None	-8	6	Human	8.4	pKi	=	8.4	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	11983932
	91898917	1685	21	None	-8	6	Human	8.4	pKi	=	8.4	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9480833
	CHEMBL506553	1685	21	None	-8	6	Human	8.4	pKi	=	8.4	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	11983932
	CHEMBL506553	1685	21	None	-8	6	Human	8.4	pKi	=	8.4	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9480833
	3896	2410	0	None	-38	7	Rat	8.4	pKi	=	8.4	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	15944002
	3896	2410	0	None	-38	7	Rat	8.4	pKi	=	8.4	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9281594
	3896	2410	0	None	-38	7	Rat	8.4	pKi	=	8.4	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9305929
	3896	2410	0	None	-38	7	Rat	8.4	pKi	=	8.4	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9405385
	3896	2410	0	None	-38	7	Rat	8.4	pKi	=	8.4	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9722565
	3896	2410	0	None	-38	7	Rat	8.4	pKi	=	8.4	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9832122
	16133243	1684	0	None	-26	8	Mouse	8.4	pKi	=	8.4	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9832122
	3593	1684	0	None	-26	8	Mouse	8.4	pKi	=	8.4	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9832122
	3899	2414	0	None	-26	8	Rat	8.5	pKi	=	8.5	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	15944002
	3899	2414	0	None	-26	8	Rat	8.5	pKi	=	8.5	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9281594
	3899	2414	0	None	-26	8	Rat	8.5	pKi	=	8.5	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9305929
	3899	2414	0	None	-26	8	Rat	8.5	pKi	=	8.5	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9405385
	3899	2414	0	None	-26	8	Rat	8.5	pKi	=	8.5	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9722565
	3899	2414	0	None	-26	8	Rat	8.5	pKi	=	8.5	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9832122
	16131409	1693	0	None	-4	3	Human	8.5	pKi	=	8.5	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9480833
	6086	1693	0	None	-4	3	Human	8.5	pKi	=	8.5	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9480833
	155817463	765	0	None	-13	8	Rat	8.5	pKi	=	8.5	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9281594
	155817463	765	0	None	-13	8	Rat	8.5	pKi	=	8.5	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9305929
	155817463	765	0	None	-13	8	Rat	8.5	pKi	=	8.5	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9722565
	155817463	765	0	None	-13	8	Rat	8.5	pKi	=	8.5	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9832122
	3861	765	0	None	-13	8	Rat	8.5	pKi	=	8.5	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9281594
	3861	765	0	None	-13	8	Rat	8.5	pKi	=	8.5	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9305929
	3861	765	0	None	-13	8	Rat	8.5	pKi	=	8.5	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9722565
	3861	765	0	None	-13	8	Rat	8.5	pKi	=	8.5	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9832122
	155817487	1699	0	None	8	4	Human	8.5	pKi	=	8.5	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9880084
	6130	1699	0	None	8	4	Human	8.5	pKi	=	8.5	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9880084
	3899	2414	0	None	-21	8	Mouse	8.6	pKi	=	8.6	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9832122
	101927062	1685	21	None	-8	6	Rat	8.6	pKi	=	8.6	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9722565
	155817445	1685	21	None	-8	6	Rat	8.6	pKi	=	8.6	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9722565
	16133823	1685	21	None	-8	6	Rat	8.6	pKi	=	8.6	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9722565
	3592	1685	21	None	-8	6	Rat	8.6	pKi	=	8.6	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9722565
	44584852	1685	21	None	-8	6	Rat	8.6	pKi	=	8.6	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9722565
	6090	1685	21	None	-8	6	Rat	8.6	pKi	=	8.6	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9722565
	91898917	1685	21	None	-8	6	Rat	8.6	pKi	=	8.6	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9722565
	CHEMBL506553	1685	21	None	-8	6	Rat	8.6	pKi	=	8.6	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9722565
	155817479	1706	0	None	1	6	Rat	8.6	pKi	=	8.6	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9480833
	6083	1706	0	None	1	6	Rat	8.6	pKi	=	8.6	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9480833
	3899	2414	0	None	-18	8	Human	8.6	pKi	=	8.6	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9480833
	3899	2414	0	None	-18	8	Human	8.6	pKi	=	8.6	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9880084
	3898	2413	0	None	-9	7	Rat	8.7	pKi	=	8.7	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	15944002
	3898	2413	0	None	-9	7	Rat	8.7	pKi	=	8.7	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9281594
	3898	2413	0	None	-9	7	Rat	8.7	pKi	=	8.7	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9305929
	3898	2413	0	None	-9	7	Rat	8.7	pKi	=	8.7	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9722565
	3898	2413	0	None	-9	7	Rat	8.7	pKi	=	8.7	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9832122
	16133243	1684	0	None	-14	8	Human	8.7	pKi	=	8.7	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	19467704
	16133243	1684	0	None	-14	8	Human	8.7	pKi	=	8.7	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	21333705
	16133243	1684	0	None	-14	8	Human	8.7	pKi	=	8.7	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9480833
	16133243	1684	0	None	-14	8	Human	8.7	pKi	=	8.7	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9880084
	3593	1684	0	None	-14	8	Human	8.7	pKi	=	8.7	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	19467704
	3593	1684	0	None	-14	8	Human	8.7	pKi	=	8.7	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	21333705
	3593	1684	0	None	-14	8	Human	8.7	pKi	=	8.7	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9480833
	3593	1684	0	None	-14	8	Human	8.7	pKi	=	8.7	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9880084
	3898	2413	0	None	-7	7	Human	8.7	pKi	=	8.7	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9480833
	3898	2413	0	None	-7	7	Human	8.7	pKi	=	8.7	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9880084
	16133243	1684	0	None	-12	8	Rat	8.8	pKi	=	8.8	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	15944002
	16133243	1684	0	None	-12	8	Rat	8.8	pKi	=	8.8	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9281594
	16133243	1684	0	None	-12	8	Rat	8.8	pKi	=	8.8	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9405385
	16133243	1684	0	None	-12	8	Rat	8.8	pKi	=	8.8	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9722565
	16133243	1684	0	None	-12	8	Rat	8.8	pKi	=	8.8	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9742938
	16133243	1684	0	None	-12	8	Rat	8.8	pKi	=	8.8	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9832122
	3593	1684	0	None	-12	8	Rat	8.8	pKi	=	8.8	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	15944002
	3593	1684	0	None	-12	8	Rat	8.8	pKi	=	8.8	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9281594
	3593	1684	0	None	-12	8	Rat	8.8	pKi	=	8.8	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9405385
	3593	1684	0	None	-12	8	Rat	8.8	pKi	=	8.8	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9722565
	3593	1684	0	None	-12	8	Rat	8.8	pKi	=	8.8	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9742938
	3593	1684	0	None	-12	8	Rat	8.8	pKi	=	8.8	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9832122
	3897	2412	0	None	-8	6	Human	8.8	pKi	=	8.8	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	11600206
	3897	2412	0	None	-8	6	Human	8.8	pKi	=	8.8	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9880084
	101927062	1685	21	None	-8	6	Human	8.9	pKi	=	8.9	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	11600206
	101927062	1685	21	None	-8	6	Human	8.9	pKi	=	8.9	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9480833
	101927062	1685	21	None	-8	6	Human	8.9	pKi	=	8.9	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9880084
	155817445	1685	21	None	-8	6	Human	8.9	pKi	=	8.9	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	11600206
	155817445	1685	21	None	-8	6	Human	8.9	pKi	=	8.9	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9480833
	155817445	1685	21	None	-8	6	Human	8.9	pKi	=	8.9	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9880084
	16133823	1685	21	None	-8	6	Human	8.9	pKi	=	8.9	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	11600206
	16133823	1685	21	None	-8	6	Human	8.9	pKi	=	8.9	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9480833
	16133823	1685	21	None	-8	6	Human	8.9	pKi	=	8.9	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9880084
	3592	1685	21	None	-8	6	Human	8.9	pKi	=	8.9	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	11600206
	3592	1685	21	None	-8	6	Human	8.9	pKi	=	8.9	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9480833
	3592	1685	21	None	-8	6	Human	8.9	pKi	=	8.9	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9880084
	44584852	1685	21	None	-8	6	Human	8.9	pKi	=	8.9	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	11600206
	44584852	1685	21	None	-8	6	Human	8.9	pKi	=	8.9	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9480833
	44584852	1685	21	None	-8	6	Human	8.9	pKi	=	8.9	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9880084
	6090	1685	21	None	-8	6	Human	8.9	pKi	=	8.9	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	11600206
	6090	1685	21	None	-8	6	Human	8.9	pKi	=	8.9	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9480833
	6090	1685	21	None	-8	6	Human	8.9	pKi	=	8.9	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9880084
	91898917	1685	21	None	-8	6	Human	8.9	pKi	=	8.9	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	11600206
	91898917	1685	21	None	-8	6	Human	8.9	pKi	=	8.9	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9480833
	91898917	1685	21	None	-8	6	Human	8.9	pKi	=	8.9	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9880084
	CHEMBL506553	1685	21	None	-8	6	Human	8.9	pKi	=	8.9	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	11600206
	CHEMBL506553	1685	21	None	-8	6	Human	8.9	pKi	=	8.9	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9480833
	CHEMBL506553	1685	21	None	-8	6	Human	8.9	pKi	=	8.9	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9880084
	3896	2410	0	None	-13	7	Mouse	8.9	pKi	=	8.9	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9832122
	155817463	765	0	None	-4	8	Human	9.0	pKi	=	9.0	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9480833
	155817463	765	0	None	-4	8	Human	9.0	pKi	=	9.0	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9880084
	3861	765	0	None	-4	8	Human	9.0	pKi	=	9.0	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9480833
	3861	765	0	None	-4	8	Human	9.0	pKi	=	9.0	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9880084
	155817484	1686	0	None	-1	6	Human	9.0	pKi	=	9.0	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9880084
	6117	1686	0	None	-1	6	Human	9.0	pKi	=	9.0	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9880084
	6129	1686	0	None	-1	6	Human	9.0	pKi	=	9.0	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9880084
	155817465	1700	0	None	7	6	Human	9.0	pKi	=	9.0	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9480833
	3876	1700	0	None	7	6	Human	9.0	pKi	=	9.0	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9480833
	6137	1697	0	None	-	1	Human	9.1	pKi	=	9.1	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9480833
	155817484	1686	0	None	-3	6	Rat	9.1	pKi	=	9.1	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9305929
	155817484	1686	0	None	-3	6	Rat	9.1	pKi	=	9.1	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9722565
	6117	1686	0	None	-3	6	Rat	9.1	pKi	=	9.1	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9305929
	6117	1686	0	None	-3	6	Rat	9.1	pKi	=	9.1	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9722565
	6129	1686	0	None	-3	6	Rat	9.1	pKi	=	9.1	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9305929
	6129	1686	0	None	-3	6	Rat	9.1	pKi	=	9.1	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9722565
	16131409	1693	0	None	4	3	Rat	9.2	pKi	=	9.2	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9305929
	6086	1693	0	None	4	3	Rat	9.2	pKi	=	9.2	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9305929
	3897	2412	0	None	-13	6	Rat	9.2	pKi	=	9.2	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9305929
	3897	2412	0	None	-13	6	Rat	9.2	pKi	=	9.2	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9722565
	6127	1731	0	None	-575	3	Rat	5.0	pKi	>	5	Binding	UnclassifiedUnclassified	Guide to Pharmacology	397	3	0	4	5.2	COc1ccc(cn1)N1C(=O)/C(=N/c2ccc(c(c2)Cl)Cl)/c2c1cccc2	15944002
	9800980	1731	0	None	-575	3	Rat	5.0	pKi	>	5	Binding	UnclassifiedUnclassified	Guide to Pharmacology	397	3	0	4	5.2	COc1ccc(cn1)N1C(=O)/C(=N/c2ccc(c(c2)Cl)Cl)/c2c1cccc2	15944002
	1471834	3572	36	None	-588	3	Human	5.0	pKi	>	5	Binding	UnclassifiedUnclassified	Guide to Pharmacology	366	2	0	2	5.5	O=C1C(=Nc2cccc(c2)C(F)(F)F)c2c(N1c1ccccc1)cccc2	16287967
	6126	3572	36	None	-588	3	Human	5.0	pKi	>	5	Binding	UnclassifiedUnclassified	Guide to Pharmacology	366	2	0	2	5.5	O=C1C(=Nc2cccc(c2)C(F)(F)F)c2c(N1c1ccccc1)cccc2	16287967
	CHEMBL210288	3572	36	None	-588	3	Human	5.0	pKi	>	5	Binding	UnclassifiedUnclassified	Guide to Pharmacology	366	2	0	2	5.5	O=C1C(=Nc2cccc(c2)C(F)(F)F)c2c(N1c1ccccc1)cccc2	16287967
	155817481	1702	0	None	-3	6	Mouse	5.7	pKi	>	5.7	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9832122
	6092	1702	0	None	-3	6	Mouse	5.7	pKi	>	5.7	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9832122
	155817482	1688	0	None	-2	3	Mouse	5.7	pKi	>	5.7	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9832122
	6093	1688	0	None	-2	3	Mouse	5.7	pKi	>	5.7	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9832122
	6133	1466	0	None	-1	2	Rat	5.9	pKi	>	5.9	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9281594
	155817480	1701	0	None	1	6	Human	6.0	pKi	>	6	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9880084
	155817480	1701	0	None	-1	6	Rat	6.0	pKi	>	6	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9305929
	155817480	1701	0	None	-1	6	Rat	6.0	pKi	>	6	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9722565
	6091	1701	0	None	1	6	Human	6.0	pKi	>	6	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9880084
	6091	1701	0	None	-1	6	Rat	6.0	pKi	>	6	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9305929
	6091	1701	0	None	-1	6	Rat	6.0	pKi	>	6	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9722565
	6132	1800	0	None	-	1	Rat	6.0	pKi	>	6	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9405385
	11698643	3573	8	None	-194	4	Human	6.0	pKi	>	6	Binding	UnclassifiedUnclassified	Guide to Pharmacology	479	6	0	4	6.0	O=C1C(=Nc2cccc(c2)C(F)(F)F)c2c(N1c1cccc(c1)OCCN1CCCC1)cccc2	16287967
	6125	3573	8	None	-194	4	Human	6.0	pKi	>	6	Binding	UnclassifiedUnclassified	Guide to Pharmacology	479	6	0	4	6.0	O=C1C(=Nc2cccc(c2)C(F)(F)F)c2c(N1c1cccc(c1)OCCN1CCCC1)cccc2	16287967
	CHEMBL209497	3573	8	None	-194	4	Human	6.0	pKi	>	6	Binding	UnclassifiedUnclassified	Guide to Pharmacology	479	6	0	4	6.0	O=C1C(=Nc2cccc(c2)C(F)(F)F)c2c(N1c1cccc(c1)OCCN1CCCC1)cccc2	16287967
	6131	1799	0	None	-	1	Rat	6.1	pKi	>	6.1	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9281594
	155817482	1688	0	None	2	3	Human	6.2	pKi	>	6.2	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9480833
	6093	1688	0	None	2	3	Human	6.2	pKi	>	6.2	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9480833
	6140	1689	0	None	-	1	Human	6.2	pKi	>	6.2	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9480833
	155817481	1702	0	None	1	6	Human	6.2	pKi	>	6.2	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9480833
	6092	1702	0	None	1	6	Human	6.2	pKi	>	6.2	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9480833
	6138	1703	0	None	-	1	Human	6.2	pKi	>	6.2	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9480833
	6134	1705	0	None	-	1	Human	6.2	pKi	>	6.2	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9480833
	6136	1707	0	None	-	1	Human	6.2	pKi	>	6.2	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9480833
	6135	1708	0	None	-	1	Human	6.2	pKi	>	6.2	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9480833

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