Biased Signaling Atlas

Ligand source activities (1 row/activity)

Potency
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Ligands					Receptor			Assay information							Chemical information
Sel. page	Common name	GPCRdb ID	#Vendors	Reference ligand	Fold selectivity (Potency)	# tested GPCRs (Potency)	Species	p-value (-log)	Type	Activity Relation	Activity Value	Assay Type	Assay Description	Source	Mol weight	Rot Bonds	H don	H acc	LogP	Smiles	DOI
	90012275	133128	0	None	-	1	Human	6.0	pAC50	=	6.0	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	416	6	2	3	5.9	CCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(C(C)(C)C)c1	nan
	CHEMBL3714858	133128	0	None	-	1	Human	6.0	pAC50	=	6.0	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	416	6	2	3	5.9	CCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(C(C)(C)C)c1	nan
	56593334	133598	0	None	-	1	Human	6.0	pAC50	=	6.0	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	454	5	2	4	4.8	O=C(Nc1cccc(S(=O)(=O)C(F)(F)F)c1)c1ccccc1NC(=O)C1CCCCC1	nan
	CHEMBL3716462	133598	0	None	-	1	Human	6.0	pAC50	=	6.0	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	454	5	2	4	4.8	O=C(Nc1cccc(S(=O)(=O)C(F)(F)F)c1)c1ccccc1NC(=O)C1CCCCC1	nan
	90011833	133778	0	None	-	1	Human	6.0	pAC50	=	6.0	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	429	5	2	4	5.1	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1cccc([N+](=O)[O-])c1	nan
	CHEMBL3717071	133778	0	None	-	1	Human	6.0	pAC50	=	6.0	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	429	5	2	4	5.1	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1cccc([N+](=O)[O-])c1	nan
	56593330	133863	0	None	-	1	Human	6.9	pAC50	=	6.9	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	492	7	2	5	4.9	CCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	nan
	CHEMBL3717389	133863	0	None	-	1	Human	6.9	pAC50	=	6.9	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	492	7	2	5	4.9	CCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	nan
	56593346	133808	0	None	-	1	Human	5.9	pAC50	=	5.9	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	468	5	2	3	6.1	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NC(=O)c1ccccc1OC(F)(F)F	nan
	CHEMBL3717178	133808	0	None	-	1	Human	5.9	pAC50	=	5.9	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	468	5	2	3	6.1	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NC(=O)c1ccccc1OC(F)(F)F	nan
	90010727	133291	0	None	-	1	Human	4.9	pAC50	=	4.9	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	487	6	2	4	4.6	CCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cncc(I)c1	nan
	CHEMBL3715451	133291	0	None	-	1	Human	4.9	pAC50	=	4.9	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	487	6	2	4	4.6	CCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cncc(I)c1	nan
	118037864	133359	0	None	-	1	Human	4.9	pAC50	=	4.9	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	424	4	3	3	5.1	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NC(=O)c1cccc2nc[nH]c12	nan
	CHEMBL3715676	133359	0	None	-	1	Human	4.9	pAC50	=	4.9	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	424	4	3	3	5.1	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NC(=O)c1cccc2nc[nH]c12	nan
	2806493	133595	4	None	-	1	Human	5.9	pAC50	=	5.9	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	384	4	2	2	5.2	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1ccccc1	nan
	CHEMBL3716450	133595	4	None	-	1	Human	5.9	pAC50	=	5.9	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	384	4	2	2	5.2	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1ccccc1	nan
	118037922	134163	0	None	-	1	Human	5.9	pAC50	=	5.9	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	612	8	2	6	6.1	CC(C)(C)OC(=O)N1CCN(CCOc2ccccc2C(=O)Nc2ccccc2C(=O)Nc2cccc(C(F)(F)F)c2)CC1	nan
	CHEMBL3718384	134163	0	None	-	1	Human	5.9	pAC50	=	5.9	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	612	8	2	6	6.1	CC(C)(C)OC(=O)N1CCN(CCOc2ccccc2C(=O)Nc2ccccc2C(=O)Nc2cccc(C(F)(F)F)c2)CC1	nan
	90010869	134342	0	None	-	1	Human	5.9	pAC50	=	5.9	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	392	6	2	4	4.9	COc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(SC)c1	nan
	CHEMBL3718995	134342	0	None	-	1	Human	5.9	pAC50	=	5.9	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	392	6	2	4	4.9	COc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(SC)c1	nan
	38269206	134157	0	None	-	1	Human	4.9	pAC50	=	4.9	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	340	4	2	2	4.6	O=C(Nc1cccc(F)c1)c1ccccc1NC(=O)C1CCCCC1	nan
	CHEMBL3718363	134157	0	None	-	1	Human	4.9	pAC50	=	4.9	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	340	4	2	2	4.6	O=C(Nc1cccc(F)c1)c1ccccc1NC(=O)C1CCCCC1	nan
	90010751	133849	0	None	-	1	Human	5.8	pAC50	=	5.8	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	400	7	2	3	5.6	C/C=C\c1cccc(NC(=O)c2ccccc2NC(=O)c2ccccc2OCC)c1	nan
	CHEMBL3717338	133849	0	None	-	1	Human	5.8	pAC50	=	5.8	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	400	7	2	3	5.6	C/C=C\c1cccc(NC(=O)c2ccccc2NC(=O)c2ccccc2OCC)c1	nan
	90012348	134063	0	None	-	1	Human	5.8	pAC50	=	5.8	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	429	5	2	4	5.1	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1ccc([N+](=O)[O-])cc1	nan
	CHEMBL3718077	134063	0	None	-	1	Human	5.8	pAC50	=	5.8	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	429	5	2	4	5.1	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1ccc([N+](=O)[O-])cc1	nan
	90010773	133388	0	None	-1	2	Human	4.8	pAC50	=	4.8	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	375	4	2	4	4.2	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1ccno1	nan
	CHEMBL3715750	133388	0	None	-1	2	Human	4.8	pAC50	=	4.8	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	375	4	2	4	4.2	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1ccno1	nan
	90011033	134350	0	None	-	1	Human	4.8	pAC50	=	4.8	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	434	4	2	2	6.4	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1ccc2ccccc2c1	nan
	CHEMBL3719015	134350	0	None	-	1	Human	4.8	pAC50	=	4.8	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	434	4	2	2	6.4	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1ccc2ccccc2c1	nan
	56593309	133239	0	None	-	1	Human	5.8	pAC50	=	5.8	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	493	7	2	6	4.3	CCOc1ccccc1C(=O)Nc1ncccc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	nan
	CHEMBL3715203	133239	0	None	-	1	Human	5.8	pAC50	=	5.8	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	493	7	2	6	4.3	CCOc1ccccc1C(=O)Nc1ncccc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	nan
	90011788	133303	0	None	-	1	Human	5.8	pAC50	=	5.8	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	409	4	2	3	5.1	N#Cc1ccc(C(=O)Nc2ccccc2C(=O)Nc2cccc(C(F)(F)F)c2)cc1	nan
	CHEMBL3715489	133303	0	None	-	1	Human	5.8	pAC50	=	5.8	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	409	4	2	3	5.1	N#Cc1ccc(C(=O)Nc2ccccc2C(=O)Nc2cccc(C(F)(F)F)c2)cc1	nan
	90012098	134057	0	None	-	1	Human	5.8	pAC50	=	5.8	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	462	4	2	2	6.0	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1cccc(Br)c1	nan
	CHEMBL3718061	134057	0	None	-	1	Human	5.8	pAC50	=	5.8	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	462	4	2	2	6.0	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1cccc(Br)c1	nan
	56593314	133817	0	None	-	1	Human	6.7	pAC50	=	6.7	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	478	6	2	5	4.5	COc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	nan
	CHEMBL3717211	133817	0	None	-	1	Human	6.7	pAC50	=	6.7	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	478	6	2	5	4.5	COc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	nan
	56593340	133577	0	None	-	1	Human	5.7	pAC50	=	5.7	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	414	5	2	3	5.2	COc1cccc(C(=O)Nc2ccccc2C(=O)Nc2cccc(C(F)(F)F)c2)c1	nan
	CHEMBL3716394	133577	0	None	-	1	Human	5.7	pAC50	=	5.7	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	414	5	2	3	5.2	COc1cccc(C(=O)Nc2ccccc2C(=O)Nc2cccc(C(F)(F)F)c2)c1	nan
	1313624	133925	8	None	-	1	Human	5.7	pAC50	=	5.7	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	418	4	2	2	5.9	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1cccc(Cl)c1	nan
	CHEMBL3717590	133925	8	None	-	1	Human	5.7	pAC50	=	5.7	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	418	4	2	2	5.9	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1cccc(Cl)c1	nan
	56593311	133964	0	None	-	1	Human	5.7	pAC50	=	5.7	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	422	5	2	3	6.1	O=C(Nc1cccc(SC(F)(F)F)c1)c1ccccc1NC(=O)C1CCCCC1	nan
	CHEMBL3717723	133964	0	None	-	1	Human	5.7	pAC50	=	5.7	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	422	5	2	3	6.1	O=C(Nc1cccc(SC(F)(F)F)c1)c1ccccc1NC(=O)C1CCCCC1	nan
	24671974	134269	2	None	-	1	Human	5.7	pAC50	=	5.7	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	390	4	2	3	5.3	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1cccs1	nan
	CHEMBL3718728	134269	2	None	-	1	Human	5.7	pAC50	=	5.7	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	390	4	2	3	5.3	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1cccs1	nan
	90012130	133162	0	None	-	1	Human	5.7	pAC50	=	5.7	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	409	4	2	3	5.1	N#Cc1cccc(C(=O)Nc2ccccc2C(=O)Nc2cccc(C(F)(F)F)c2)c1	nan
	CHEMBL3714976	133162	0	None	-	1	Human	5.7	pAC50	=	5.7	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	409	4	2	3	5.1	N#Cc1cccc(C(=O)Nc2ccccc2C(=O)Nc2cccc(C(F)(F)F)c2)c1	nan
	90010778	133690	0	None	-	1	Human	5.7	pAC50	=	5.7	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	400	7	2	3	5.6	C/C=C/c1cccc(NC(=O)c2ccccc2NC(=O)c2ccccc2OCC)c1	nan
	CHEMBL3716808	133690	0	None	-	1	Human	5.7	pAC50	=	5.7	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	400	7	2	3	5.6	C/C=C/c1cccc(NC(=O)c2ccccc2NC(=O)c2ccccc2OCC)c1	nan
	56593317	134425	0	None	-	1	Human	5.7	pAC50	=	5.7	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	404	4	2	2	5.9	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NC(=O)C1CCCCCC1	nan
	CHEMBL3719257	134425	0	None	-	1	Human	5.7	pAC50	=	5.7	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	404	4	2	2	5.9	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NC(=O)C1CCCCCC1	nan
	40622265	133357	2	None	-	1	Human	5.6	pAC50	=	5.6	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	374	4	2	3	4.8	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1ccco1	nan
	CHEMBL3715664	133357	2	None	-	1	Human	5.6	pAC50	=	5.6	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	374	4	2	3	4.8	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1ccco1	nan
	127024729	133953	0	None	-	1	Human	5.6	pAC50	=	5.6	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	500	7	2	6	4.0	CCOc1ccccc1C(=O)NC1SC=CC1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	nan
	CHEMBL3717683	133953	0	None	-	1	Human	5.6	pAC50	=	5.6	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	500	7	2	6	4.0	CCOc1ccccc1C(=O)NC1SC=CC1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	nan
	90010630	134274	0	None	-	1	Human	5.6	pAC50	=	5.6	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	404	4	2	2	5.7	CC1CCC(C(=O)Nc2ccccc2C(=O)Nc2cccc(C(F)(F)F)c2)CC1	nan
	CHEMBL3718740	134274	0	None	-	1	Human	5.6	pAC50	=	5.6	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	404	4	2	2	5.7	CC1CCC(C(=O)Nc2ccccc2C(=O)Nc2cccc(C(F)(F)F)c2)CC1	nan
	5298634	134435	10	None	-	1	Human	5.6	pAC50	=	5.6	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	376	4	2	2	5.1	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NC(=O)C1CCCC1	nan
	CHEMBL3719295	134435	10	None	-	1	Human	5.6	pAC50	=	5.6	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	376	4	2	2	5.1	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NC(=O)C1CCCC1	nan
	56593335	133782	0	None	-	1	Human	6.6	pAC50	=	6.6	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	428	6	2	3	5.6	CCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	nan
	CHEMBL3717089	133782	0	None	-	1	Human	6.6	pAC50	=	6.6	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	428	6	2	3	5.6	CCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	nan
	90011775	133149	0	None	-	1	Human	5.6	pAC50	=	5.6	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	418	4	2	2	5.9	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1ccc(Cl)cc1	nan
	CHEMBL3714926	133149	0	None	-	1	Human	5.6	pAC50	=	5.6	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	418	4	2	2	5.9	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1ccc(Cl)cc1	nan
	90011735	133247	0	None	-	1	Human	5.6	pAC50	=	5.6	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	511	8	2	4	6.1	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NC(=O)c1ccccc1OCCN1CCCCC1	nan
	CHEMBL3715244	133247	0	None	-	1	Human	5.6	pAC50	=	5.6	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	511	8	2	4	6.1	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NC(=O)c1ccccc1OCCN1CCCCC1	nan
	56593308	133636	0	None	-	1	Human	5.6	pAC50	=	5.6	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	466	5	2	2	7.1	O=C(Nc1cccc(-c2ccccc2C(F)(F)F)c1)c1ccccc1NC(=O)C1CCCCC1	nan
	CHEMBL3716596	133636	0	None	-	1	Human	5.6	pAC50	=	5.6	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	466	5	2	2	7.1	O=C(Nc1cccc(-c2ccccc2C(F)(F)F)c1)c1ccccc1NC(=O)C1CCCCC1	nan
	56593324	133693	0	None	-	1	Human	5.6	pAC50	=	5.6	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	478	8	2	5	5.2	CCOc1ccccc1C(=O)Nc1ccccc1CNc1cccc(S(=O)(=O)C(F)(F)F)c1	nan
	CHEMBL3716811	133693	0	None	-	1	Human	5.6	pAC50	=	5.6	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	478	8	2	5	5.2	CCOc1ccccc1C(=O)Nc1ccccc1CNc1cccc(S(=O)(=O)C(F)(F)F)c1	nan
	56593333	133712	0	None	-	1	Human	5.6	pAC50	=	5.6	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	400	4	2	2	5.2	O=C(Nc1cccc(Br)c1)c1ccccc1NC(=O)C1CCCCC1	nan
	CHEMBL3716871	133712	0	None	-	1	Human	5.6	pAC50	=	5.6	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	400	4	2	2	5.2	O=C(Nc1cccc(Br)c1)c1ccccc1NC(=O)C1CCCCC1	nan
	56593350	134124	0	None	-	1	Human	5.6	pAC50	=	5.6	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	378	4	2	2	5.8	CC(C)(C)c1cccc(NC(=O)c2ccccc2NC(=O)C2CCCCC2)c1	nan
	CHEMBL3718273	134124	0	None	-	1	Human	5.6	pAC50	=	5.6	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	378	4	2	2	5.8	CC(C)(C)c1cccc(NC(=O)c2ccccc2NC(=O)C2CCCCC2)c1	nan
	56593315	133789	0	None	-	1	Human	6.5	pAC50	=	6.5	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	446	6	2	4	5.8	COc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(SC(F)(F)F)c1	nan
	CHEMBL3717103	133789	0	None	-	1	Human	6.5	pAC50	=	6.5	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	446	6	2	4	5.8	COc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(SC(F)(F)F)c1	nan
	90010752	133172	0	None	-	1	Human	5.5	pAC50	=	5.5	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	448	4	2	2	5.1	O=C(Nc1cccc(I)c1)c1ccccc1NC(=O)C1CCCCC1	nan
	CHEMBL3714999	133172	0	None	-	1	Human	5.5	pAC50	=	5.5	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	448	4	2	2	5.1	O=C(Nc1cccc(I)c1)c1ccccc1NC(=O)C1CCCCC1	nan
	90011874	133189	0	None	-	1	Human	5.5	pAC50	=	5.5	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	452	4	2	2	6.2	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1cccc(C(F)(F)F)c1	nan
	CHEMBL3715040	133189	0	None	-	1	Human	5.5	pAC50	=	5.5	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	452	4	2	2	6.2	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1cccc(C(F)(F)F)c1	nan
	56593323	133213	0	None	-	1	Human	5.5	pAC50	=	5.5	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	493	7	2	6	4.3	CCOc1ccccc1C(=O)Nc1cnccc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	nan
	CHEMBL3715105	133213	0	None	-	1	Human	5.5	pAC50	=	5.5	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	493	7	2	6	4.3	CCOc1ccccc1C(=O)Nc1cnccc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	nan
	56593318	133609	0	None	-	1	Human	5.5	pAC50	=	5.5	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	362	4	2	2	4.7	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NC(=O)C1CCC1	nan
	CHEMBL3716512	133609	0	None	-	1	Human	5.5	pAC50	=	5.5	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	362	4	2	2	4.7	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NC(=O)C1CCC1	nan
	90010791	133749	0	None	-	1	Human	4.5	pAC50	=	4.5	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	361	6	2	4	4.0	CCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1ccccn1	nan
	CHEMBL3716987	133749	0	None	-	1	Human	4.5	pAC50	=	4.5	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	361	6	2	4	4.0	CCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1ccccn1	nan
	56593313	134328	0	None	-	1	Human	4.5	pAC50	=	4.5	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	428	5	1	3	5.2	COc1ccccc1C(=O)Nc1ccccc1C(=O)N(C)c1cccc(C(F)(F)F)c1	nan
	CHEMBL3718895	134328	0	None	-	1	Human	4.5	pAC50	=	4.5	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	428	5	1	3	5.2	COc1ccccc1C(=O)Nc1ccccc1C(=O)N(C)c1cccc(C(F)(F)F)c1	nan
	56593329	133910	0	None	-	1	Human	6.5	pAC50	=	6.5	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	414	5	2	3	5.2	COc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	nan
	CHEMBL3717553	133910	0	None	-	1	Human	6.5	pAC50	=	6.5	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	414	5	2	3	5.2	COc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	nan
	56593336	133320	0	None	-	1	Human	5.5	pAC50	=	5.5	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	356	4	2	2	5.1	O=C(Nc1cccc(Cl)c1)c1ccccc1NC(=O)C1CCCCC1	nan
	CHEMBL3715551	133320	0	None	-	1	Human	5.5	pAC50	=	5.5	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	356	4	2	2	5.1	O=C(Nc1cccc(Cl)c1)c1ccccc1NC(=O)C1CCCCC1	nan
	56593337	133209	0	None	-	1	Human	5.4	pAC50	=	5.4	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	418	4	2	2	5.9	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1ccccc1Cl	nan
	CHEMBL3715097	133209	0	None	-	1	Human	5.4	pAC50	=	5.4	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	418	4	2	2	5.9	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1ccccc1Cl	nan
	127024591	133220	0	None	-	1	Human	5.4	pAC50	=	5.4	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	457	8	3	4	4.8	CNCCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	nan
	CHEMBL3715139	133220	0	None	-	1	Human	5.4	pAC50	=	5.4	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	457	8	3	4	4.8	CNCCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	nan
	2233108	133946	9	None	-	1	Human	5.4	pAC50	=	5.4	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	398	4	2	2	5.5	Cc1cccc(C(=O)Nc2ccccc2C(=O)Nc2cccc(C(F)(F)F)c2)c1	nan
	CHEMBL3717655	133946	9	None	-	1	Human	5.4	pAC50	=	5.4	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	398	4	2	2	5.5	Cc1cccc(C(=O)Nc2ccccc2C(=O)Nc2cccc(C(F)(F)F)c2)c1	nan
	1511185	133314	12	None	-	1	Human	4.4	pAC50	=	4.4	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	336	4	2	2	4.8	Cc1cccc(NC(=O)c2ccccc2NC(=O)C2CCCCC2)c1	nan
	CHEMBL3715535	133314	12	None	-	1	Human	4.4	pAC50	=	4.4	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	336	4	2	2	4.8	Cc1cccc(NC(=O)c2ccccc2NC(=O)C2CCCCC2)c1	nan
	4795548	133714	6	None	-	1	Human	4.4	pAC50	=	4.4	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	352	5	2	3	4.5	COc1cccc(NC(=O)c2ccccc2NC(=O)C2CCCCC2)c1	nan
	CHEMBL3716878	133714	6	None	-	1	Human	4.4	pAC50	=	4.4	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	352	5	2	3	4.5	COc1cccc(NC(=O)c2ccccc2NC(=O)C2CCCCC2)c1	nan
	32157880	133720	5	None	-	1	Human	4.4	pAC50	=	4.4	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	340	4	2	2	4.6	O=C(Nc1ccc(F)cc1)c1ccccc1NC(=O)C1CCCCC1	nan
	CHEMBL3716901	133720	5	None	-	1	Human	4.4	pAC50	=	4.4	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	340	4	2	2	4.6	O=C(Nc1ccc(F)cc1)c1ccccc1NC(=O)C1CCCCC1	nan
	90010785	133164	0	None	-	1	Human	5.4	pAC50	=	5.4	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	574	5	2	4	5.1	O=C(Nc1ccccc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1)c1ccccc1I	nan
	CHEMBL3714984	133164	0	None	-	1	Human	5.4	pAC50	=	5.4	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	574	5	2	4	5.1	O=C(Nc1ccccc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1)c1ccccc1I	nan
	118043134	133212	0	None	-	1	Human	5.4	pAC50	=	5.4	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	520	4	2	2	7.2	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1cc(C(F)(F)F)cc(C(F)(F)F)c1	nan
	CHEMBL3715104	133212	0	None	-	1	Human	5.4	pAC50	=	5.4	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	520	4	2	2	7.2	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1cc(C(F)(F)F)cc(C(F)(F)F)c1	nan
	21179517	133426	0	None	-	1	Human	5.4	pAC50	=	5.4	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	424	4	2	2	6.7	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1Nc1cccc(C(F)(F)F)c1	nan
	CHEMBL3715901	133426	0	None	-	1	Human	5.4	pAC50	=	5.4	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	424	4	2	2	6.7	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1Nc1cccc(C(F)(F)F)c1	nan
	56593306	133771	0	None	-	1	Human	5.4	pAC50	=	5.4	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	398	4	2	2	5.5	Cc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	nan
	CHEMBL3717045	133771	0	None	-	1	Human	5.4	pAC50	=	5.4	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	398	4	2	2	5.5	Cc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	nan
	90012794	133989	0	None	-	1	Human	5.4	pAC50	=	5.4	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	462	4	2	2	6.0	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1ccc(Br)cc1	nan
	CHEMBL3717803	133989	0	None	-	1	Human	5.4	pAC50	=	5.4	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	462	4	2	2	6.0	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1ccc(Br)cc1	nan
	54784887	134159	2	None	-	1	Human	5.4	pAC50	=	5.4	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	356	4	2	2	5.7	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1Nc1ccccc1	nan
	CHEMBL3718373	134159	2	None	-	1	Human	5.4	pAC50	=	5.4	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	356	4	2	2	5.7	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1Nc1ccccc1	nan
	1313916	39856	8	None	-	1	Human	7.3	pAC50	=	7.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	390	4	2	2	5.5	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NC(=O)C1CCCCC1	nan
	CHEMBL1479446	39856	8	None	-	1	Human	7.3	pAC50	=	7.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	390	4	2	2	5.5	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NC(=O)C1CCCCC1	nan
	56593322	133202	0	None	-	1	Human	7.3	pAC50	=	7.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	520	9	2	5	5.7	CCCCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	nan
	CHEMBL3715081	133202	0	None	-	1	Human	7.3	pAC50	=	7.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	520	9	2	5	5.7	CCCCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	nan
	56593331	134203	0	None	-	1	Human	6.3	pAC50	=	6.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	442	6	2	3	6.0	CC(C)Oc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	nan
	CHEMBL3718541	134203	0	None	-	1	Human	6.3	pAC50	=	6.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	442	6	2	3	6.0	CC(C)Oc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	nan
	90011206	133286	0	None	-	1	Human	5.3	pAC50	=	5.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	513	8	2	5	4.9	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NC(=O)c1ccccc1OCCN1CCOCC1	nan
	CHEMBL3715429	133286	0	None	-	1	Human	5.3	pAC50	=	5.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	513	8	2	5	4.9	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NC(=O)c1ccccc1OCCN1CCOCC1	nan
	56593347	133316	0	None	-	1	Human	5.3	pAC50	=	5.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	493	7	2	6	4.3	CCOc1ccccc1C(=O)Nc1cccnc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	nan
	CHEMBL3715539	133316	0	None	-	1	Human	5.3	pAC50	=	5.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	493	7	2	6	4.3	CCOc1ccccc1C(=O)Nc1cccnc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	nan
	90010797	133342	0	None	-	1	Human	5.3	pAC50	=	5.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	442	4	2	2	6.1	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NC(=O)C12CC3CC(CC(C3)C1)C2	nan
	CHEMBL3715615	133342	0	None	-	1	Human	5.3	pAC50	=	5.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	442	4	2	2	6.1	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NC(=O)C12CC3CC(CC(C3)C1)C2	nan
	4484023	133746	6	None	-	1	Human	5.3	pAC50	=	5.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	398	4	2	2	5.5	Cc1ccc(C(=O)Nc2ccccc2C(=O)Nc2cccc(C(F)(F)F)c2)cc1	nan
	CHEMBL3716976	133746	6	None	-	1	Human	5.3	pAC50	=	5.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	398	4	2	2	5.5	Cc1ccc(C(=O)Nc2ccccc2C(=O)Nc2cccc(C(F)(F)F)c2)cc1	nan
	56593338	134208	0	None	-	1	Human	5.3	pAC50	=	5.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	444	8	2	5	3.1	CCOc1ccccc1C(=O)NCCC(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	nan
	CHEMBL3718557	134208	0	None	-	1	Human	5.3	pAC50	=	5.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	444	8	2	5	3.1	CCOc1ccccc1C(=O)NCCC(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	nan
	56593307	134298	0	None	-	1	Human	5.3	pAC50	=	5.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	386	5	2	3	5.7	COc1ccccc1Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	nan
	CHEMBL3718811	134298	0	None	-	1	Human	5.3	pAC50	=	5.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	386	5	2	3	5.7	COc1ccccc1Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	nan
	90011315	133682	0	None	-	1	Human	4.3	pAC50	=	4.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	370	5	2	2	5.6	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NCc1ccccc1	nan
	CHEMBL3716765	133682	0	None	-	1	Human	4.3	pAC50	=	4.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	370	5	2	2	5.6	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NCc1ccccc1	nan
	127024076	133966	0	None	-	1	Human	4.3	pAC50	=	4.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	308	4	2	2	3.5	O=CNc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	nan
	CHEMBL3717734	133966	0	None	-	1	Human	4.3	pAC50	=	4.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	308	4	2	2	3.5	O=CNc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	nan
	90010896	134006	0	None	-	1	Human	4.3	pAC50	=	4.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	438	5	2	2	6.6	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NCc1cccc(C(F)(F)F)c1	nan
	CHEMBL3717869	134006	0	None	-	1	Human	4.3	pAC50	=	4.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	438	5	2	2	6.6	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NCc1cccc(C(F)(F)F)c1	nan
	56593316	133245	0	None	-	1	Human	7.3	pAC50	=	7.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	506	8	2	5	5.3	CCCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	nan
	CHEMBL3715235	133245	0	None	-	1	Human	7.3	pAC50	=	7.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	506	8	2	5	5.3	CCCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	nan
	56593341	133312	0	None	-	1	Human	6.3	pAC50	=	6.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	508	7	2	5	5.6	CCSc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	nan
	CHEMBL3715526	133312	0	None	-	1	Human	6.3	pAC50	=	6.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	508	7	2	5	5.6	CCSc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	nan
	90010758	133294	0	None	-	1	Human	5.3	pAC50	=	5.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	460	5	2	2	6.9	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1cccc(-c2ccccc2)c1	nan
	CHEMBL3715462	133294	0	None	-	1	Human	5.3	pAC50	=	5.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	460	5	2	2	6.9	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1cccc(-c2ccccc2)c1	nan
	56593299	133490	0	None	-	1	Human	5.3	pAC50	=	5.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	368	5	2	3	5.2	CSc1cccc(NC(=O)c2ccccc2NC(=O)C2CCCCC2)c1	nan
	CHEMBL3716127	133490	0	None	-	1	Human	5.3	pAC50	=	5.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	368	5	2	3	5.2	CSc1cccc(NC(=O)c2ccccc2NC(=O)C2CCCCC2)c1	nan
	56593339	133602	0	None	-	1	Human	5.3	pAC50	=	5.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	378	6	2	2	5.3	CCC(CC)C(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	nan
	CHEMBL3716488	133602	0	None	-	1	Human	5.3	pAC50	=	5.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	378	6	2	2	5.3	CCC(CC)C(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	nan
	56593319	133694	0	None	-	1	Human	5.3	pAC50	=	5.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	364	6	2	2	5.1	CCCCC(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	nan
	CHEMBL3716813	133694	0	None	-	1	Human	5.3	pAC50	=	5.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	364	6	2	2	5.1	CCCCC(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	nan
	90010729	133700	0	None	-	1	Human	5.3	pAC50	=	5.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	429	6	2	4	5.2	COc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(N2CCCCC2)c1	nan
	CHEMBL3716829	133700	0	None	-	1	Human	5.3	pAC50	=	5.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	429	6	2	4	5.2	COc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(N2CCCCC2)c1	nan
	90010865	134199	0	None	-	1	Human	5.3	pAC50	=	5.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	380	3	2	3	5.3	CC(C)(C)OC(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	nan
	CHEMBL3718514	134199	0	None	-	1	Human	5.3	pAC50	=	5.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	380	3	2	3	5.3	CC(C)(C)OC(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	nan
	90010599	134439	0	None	-	1	Human	5.3	pAC50	=	5.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	364	5	2	2	5.6	CC(C)c1cccc(NC(=O)c2ccccc2NC(=O)C2CCCCC2)c1	nan
	CHEMBL3719301	134439	0	None	-	1	Human	5.3	pAC50	=	5.3	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	364	5	2	2	5.6	CC(C)c1cccc(NC(=O)c2ccccc2NC(=O)C2CCCCC2)c1	nan
	90011364	133536	0	None	-	1	Human	5.2	pAC50	=	5.2	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	376	5	2	2	6.0	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NCC1CCCCC1	nan
	CHEMBL3716260	133536	0	None	-	1	Human	5.2	pAC50	=	5.2	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	376	5	2	2	6.0	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NCC1CCCCC1	nan
	90011496	133626	0	None	-	1	Human	5.2	pAC50	=	5.2	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	434	4	2	2	6.4	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NC(=O)c1cccc2ccccc12	nan
	CHEMBL3716563	133626	0	None	-	1	Human	5.2	pAC50	=	5.2	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	434	4	2	2	6.4	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NC(=O)c1cccc2ccccc12	nan
	90011579	133747	0	None	-	1	Human	5.2	pAC50	=	5.2	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	452	4	2	2	6.2	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1ccc(C(F)(F)F)cc1	nan
	CHEMBL3716978	133747	0	None	-	1	Human	5.2	pAC50	=	5.2	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	452	4	2	2	6.2	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1ccc(C(F)(F)F)cc1	nan
	56593303	134094	1	None	-	1	Human	5.2	pAC50	=	5.2	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	385	4	2	3	4.6	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1cccnc1	nan
	CHEMBL3718178	134094	1	None	-	1	Human	5.2	pAC50	=	5.2	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	385	4	2	3	4.6	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1cccnc1	nan
	60288826	134125	1	None	-	1	Human	5.2	pAC50	=	5.2	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	426	5	2	3	5.4	CC(=O)c1ccc(C(=O)Nc2ccccc2C(=O)Nc2cccc(C(F)(F)F)c2)cc1	nan
	CHEMBL3718279	134125	1	None	-	1	Human	5.2	pAC50	=	5.2	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	426	5	2	3	5.4	CC(=O)c1ccc(C(=O)Nc2ccccc2C(=O)Nc2cccc(C(F)(F)F)c2)cc1	nan
	56593326	134224	0	None	-	1	Human	5.2	pAC50	=	5.2	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	367	5	2	4	4.4	O=C(Nc1cccc([N+](=O)[O-])c1)c1ccccc1NC(=O)C1CCCCC1	nan
	CHEMBL3718612	134224	0	None	-	1	Human	5.2	pAC50	=	5.2	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	367	5	2	4	4.4	O=C(Nc1cccc([N+](=O)[O-])c1)c1ccccc1NC(=O)C1CCCCC1	nan
	56593302	133253	0	None	-	1	Human	4.2	pAC50	=	4.2	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	338	6	2	3	4.0	COCCNc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	nan
	CHEMBL3715266	133253	0	None	-	1	Human	4.2	pAC50	=	4.2	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	338	6	2	3	4.0	COCCNc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	nan
	90011338	133269	0	None	-	1	Human	4.2	pAC50	=	4.2	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	485	9	2	4	5.5	CN(C)CCCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	nan
	CHEMBL3715346	133269	0	None	-	1	Human	4.2	pAC50	=	4.2	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	485	9	2	4	5.5	CN(C)CCCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	nan
	56593298	133959	0	None	-	1	Human	4.2	pAC50	=	4.2	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	400	6	2	3	5.6	COc1ccccc1CNc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	nan
	CHEMBL3717700	133959	0	None	-	1	Human	4.2	pAC50	=	4.2	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	400	6	2	3	5.6	COc1ccccc1CNc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	nan
	90010708	133772	0	None	-	1	Human	6.2	pAC50	=	6.2	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	385	6	2	4	4.5	CCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(C#N)c1	nan
	CHEMBL3717047	133772	0	None	-	1	Human	6.2	pAC50	=	6.2	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	385	6	2	4	4.5	CCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(C#N)c1	nan
	118043136	134402	0	None	-	1	Human	6.2	pAC50	=	6.2	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	460	7	2	4	6.2	CCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(SC(F)(F)F)c1	nan
	CHEMBL3719197	134402	0	None	-	1	Human	6.2	pAC50	=	6.2	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	460	7	2	4	6.2	CCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(SC(F)(F)F)c1	nan
	90010848	133211	0	None	-	1	Human	5.2	pAC50	=	5.2	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	424	6	2	5	3.6	COc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(S(C)(=O)=O)c1	nan
	CHEMBL3715101	133211	0	None	-	1	Human	5.2	pAC50	=	5.2	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	424	6	2	5	3.6	COc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(S(C)(=O)=O)c1	nan
	90010777	134054	0	None	-	1	Human	5.2	pAC50	=	5.2	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	346	4	2	2	4.4	C#Cc1cccc(NC(=O)c2ccccc2NC(=O)C2CCCCC2)c1	nan
	CHEMBL3718054	134054	0	None	-	1	Human	5.2	pAC50	=	5.2	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	346	4	2	2	4.4	C#Cc1cccc(NC(=O)c2ccccc2NC(=O)C2CCCCC2)c1	nan
	118037818	134186	0	None	-1	2	Human	5.2	pAC50	=	5.2	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	428	4	2	4	4.9	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1ccc2c(c1)OCO2	nan
	CHEMBL3718470	134186	0	None	-1	2	Human	5.2	pAC50	=	5.2	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	428	4	2	4	4.9	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1ccc2c(c1)OCO2	nan
	56593305	134167	0	None	-	1	Human	7.2	pAC50	=	7.2	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	546	7	2	5	5.4	O=C(Nc1cccc(S(=O)(=O)C(F)(F)F)c1)c1ccccc1NC(=O)c1ccccc1OCC(F)(F)F	nan
	CHEMBL3718400	134167	0	None	-	1	Human	7.2	pAC50	=	7.2	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	546	7	2	5	5.4	O=C(Nc1cccc(S(=O)(=O)C(F)(F)F)c1)c1ccccc1NC(=O)c1ccccc1OCC(F)(F)F	nan
	90010645	133268	0	None	-	1	Human	6.1	pAC50	=	6.1	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	486	6	2	3	5.2	CCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(I)c1	nan
	CHEMBL3715345	133268	0	None	-	1	Human	6.1	pAC50	=	6.1	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	486	6	2	3	5.2	CCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(I)c1	nan
	56593345	133384	0	None	-	1	Human	6.1	pAC50	=	6.1	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	493	7	2	6	4.3	CCOc1ccccc1C(=O)Nc1ccncc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	nan
	CHEMBL3715743	133384	0	None	-	1	Human	6.1	pAC50	=	6.1	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	493	7	2	6	4.3	CCOc1ccccc1C(=O)Nc1ccncc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	nan
	56593320	133619	0	None	-	1	Human	6.1	pAC50	=	6.1	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	458	8	2	4	5.2	COCCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	nan
	CHEMBL3716540	133619	0	None	-	1	Human	6.1	pAC50	=	6.1	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	458	8	2	4	5.2	COCCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	nan
	90011367	134251	0	None	-	1	Human	6.1	pAC50	=	6.1	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	476	6	2	3	7.0	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NC(=O)c1ccccc1Oc1ccccc1	nan
	CHEMBL3718664	134251	0	None	-	1	Human	6.1	pAC50	=	6.1	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	476	6	2	3	7.0	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NC(=O)c1ccccc1Oc1ccccc1	nan
	56593296	133634	0	None	-	1	Human	5.1	pAC50	=	5.1	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	444	6	2	4	5.2	COc1cccc(OC)c1C(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	nan
	CHEMBL3716581	133634	0	None	-	1	Human	5.1	pAC50	=	5.1	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	444	6	2	4	5.2	COc1cccc(OC)c1C(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	nan
	90011087	133750	0	None	-	1	Human	5.1	pAC50	=	5.1	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	452	4	2	2	6.2	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NC(=O)c1ccccc1C(F)(F)F	nan
	CHEMBL3716990	133750	0	None	-	1	Human	5.1	pAC50	=	5.1	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	452	4	2	2	6.2	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NC(=O)c1ccccc1C(F)(F)F	nan
	90011219	134135	0	None	-	1	Human	5.1	pAC50	=	5.1	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	510	4	2	2	5.8	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1ccccc1I	nan
	CHEMBL3718291	134135	0	None	-	1	Human	5.1	pAC50	=	5.1	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	510	4	2	2	5.8	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1ccccc1I	nan
	90011247	134193	0	None	-	1	Human	5.1	pAC50	=	5.1	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	462	4	2	2	6.0	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1ccccc1Br	nan
	CHEMBL3718498	134193	0	None	-	1	Human	5.1	pAC50	=	5.1	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	462	4	2	2	6.0	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1ccccc1Br	nan
	52764307	134345	0	None	-	1	Human	5.1	pAC50	=	5.1	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	385	4	2	3	4.6	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1ccncc1	nan
	CHEMBL3719005	134345	0	None	-	1	Human	5.1	pAC50	=	5.1	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	385	4	2	3	4.6	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1ccncc1	nan
	90010748	133214	0	None	-	1	Human	4.1	pAC50	=	4.1	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	367	5	2	4	4.4	O=C(Nc1ccc([N+](=O)[O-])cc1)c1ccccc1NC(=O)C1CCCCC1	nan
	CHEMBL3715107	133214	0	None	-	1	Human	4.1	pAC50	=	4.1	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	367	5	2	4	4.4	O=C(Nc1ccc([N+](=O)[O-])cc1)c1ccccc1NC(=O)C1CCCCC1	nan
	90010731	133371	0	None	-	1	Human	4.1	pAC50	=	4.1	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	361	6	2	4	4.0	CCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1ccncc1	nan
	CHEMBL3715708	133371	0	None	-	1	Human	4.1	pAC50	=	4.1	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	361	6	2	4	4.0	CCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1ccncc1	nan
	3348337	133926	1	None	-	1	Human	4.1	pAC50	=	4.1	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	322	3	2	2	3.9	CC(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	nan
	CHEMBL3717591	133926	1	None	-	1	Human	4.1	pAC50	=	4.1	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	322	3	2	2	3.9	CC(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	nan
	29448220	134339	0	None	-	1	Human	4.1	pAC50	=	4.1	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	366	4	2	4	4.2	O=C(Nc1ccc2c(c1)OCO2)c1ccccc1NC(=O)C1CCCCC1	nan
	CHEMBL3718975	134339	0	None	-	1	Human	4.1	pAC50	=	4.1	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	366	4	2	4	4.2	O=C(Nc1ccc2c(c1)OCO2)c1ccccc1NC(=O)C1CCCCC1	nan
	56593344	133174	0	None	-	1	Human	5.1	pAC50	=	5.1	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	398	5	2	2	5.1	O=C(Cc1ccccc1)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	nan
	CHEMBL3715001	133174	0	None	-	1	Human	5.1	pAC50	=	5.1	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	398	5	2	2	5.1	O=C(Cc1ccccc1)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	nan
	56593325	134244	0	None	-	1	Human	5.1	pAC50	=	5.1	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	348	4	2	2	4.3	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NC(=O)C1CC1	nan
	CHEMBL3718643	134244	0	None	-	1	Human	5.1	pAC50	=	5.1	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	348	4	2	2	4.3	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NC(=O)C1CC1	nan
	56593349	2534	25	None	-	1	Human	7.0	pAC50	=	7.0	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	506	7	2	5	5.3	CC(Oc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(c1)S(=O)(=O)C(F)(F)F)C	nan
	8322	2534	25	None	-	1	Human	7.0	pAC50	=	7.0	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	506	7	2	5	5.3	CC(Oc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(c1)S(=O)(=O)C(F)(F)F)C	nan
	CHEMBL3716980	2534	25	None	-	1	Human	7.0	pAC50	=	7.0	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	506	7	2	5	5.3	CC(Oc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(c1)S(=O)(=O)C(F)(F)F)C	nan
	90011702	133229	0	None	-	1	Human	5.0	pAC50	=	5.0	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	362	4	2	2	4.9	O=C(Nc1ccc2c(c1)CCC2)c1ccccc1NC(=O)C1CCCCC1	nan
	CHEMBL3715166	133229	0	None	-	1	Human	5.0	pAC50	=	5.0	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	362	4	2	2	4.9	O=C(Nc1ccc2c(c1)CCC2)c1ccccc1NC(=O)C1CCCCC1	nan
	56593321	133963	0	None	-	1	Human	5.0	pAC50	=	5.0	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	445	7	3	4	5.0	O=C(NCc1ccco1)c1ccccc1NC(=O)c1ccccc1NC(=O)C1CCCCC1	nan
	CHEMBL3717718	133963	0	None	-	1	Human	5.0	pAC50	=	5.0	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	445	7	3	4	5.0	O=C(NCc1ccco1)c1ccccc1NC(=O)c1ccccc1NC(=O)C1CCCCC1	nan
	90011489	134076	0	None	-	1	Human	5.0	pAC50	=	5.0	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	384	6	2	2	5.6	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NCCc1ccccc1	nan
	CHEMBL3718114	134076	0	None	-	1	Human	5.0	pAC50	=	5.0	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	384	6	2	2	5.6	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NCCc1ccccc1	nan
	60589025	134272	1	None	-	1	Human	5.0	pAC50	=	5.0	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	462	5	2	4	4.6	CS(=O)(=O)c1cccc(C(=O)Nc2ccccc2C(=O)Nc2cccc(C(F)(F)F)c2)c1	nan
	CHEMBL3718735	134272	1	None	-	1	Human	5.0	pAC50	=	5.0	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	462	5	2	4	4.6	CS(=O)(=O)c1cccc(C(=O)Nc2ccccc2C(=O)Nc2cccc(C(F)(F)F)c2)c1	nan
	1320335	134299	9	None	-	1	Human	5.0	pAC50	=	5.0	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	414	5	2	3	5.2	COc1ccc(C(=O)Nc2ccccc2C(=O)Nc2cccc(C(F)(F)F)c2)cc1	nan
	CHEMBL3718813	134299	9	None	-	1	Human	5.0	pAC50	=	5.0	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	414	5	2	3	5.2	COc1ccc(C(=O)Nc2ccccc2C(=O)Nc2cccc(C(F)(F)F)c2)cc1	nan
	730108	41298	15	None	-	1	Human	4.0	pAC50	=	4.0	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	322	4	2	2	4.5	O=C(Nc1ccccc1)c1ccccc1NC(=O)C1CCCCC1	nan
	CHEMBL1491180	41298	15	None	-	1	Human	4.0	pAC50	=	4.0	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	322	4	2	2	4.5	O=C(Nc1ccccc1)c1ccccc1NC(=O)C1CCCCC1	nan
	56593342	133894	0	None	-	1	Human	4.0	pAC50	=	4.0	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	390	4	2	2	5.5	O=C(Nc1ccc(C(F)(F)F)cc1)c1ccccc1NC(=O)C1CCCCC1	nan
	CHEMBL3717485	133894	0	None	-	1	Human	4.0	pAC50	=	4.0	Functional	Agonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assayAgonist activity at RXFP1 receptor (unknown origin) expressed in HEK293 cells assessed as stimulation of cAMP production incubated for 30 mins by TR-FRET based HTRF assay	ChEMBL	390	4	2	2	5.5	O=C(Nc1ccc(C(F)(F)F)cc1)c1ccccc1NC(=O)C1CCCCC1	nan
	162654489	180053	0	None	4	2	Human	10.5	pEC50	=	10.5	Functional	Agonist activity at human RXFP1 expressed in human HEK-293T cells co-transfected with pCRE beta-galactosidase reporter plasmid assessed as inhibition of IBMX-induced cAMP accumulation incubated for 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in human HEK-293T cells co-transfected with pCRE beta-galactosidase reporter plasmid assessed as inhibition of IBMX-induced cAMP accumulation incubated for 30 mins by HTRF assay	ChEMBL	5876	136	86	84	-20.9	CC[C@H](C)[C@@H]1NC(=O)[C@H](C)NC(=O)[C@H]([C@@H](C)CC)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](C(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCSC)NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](CO)NC(=O)[C@@H](N)CC(=O)O)C(C)C)[C@@H](C)CC)CSSC[C@@H]2NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](Cc3ccc(O)cc3)NC(=O)[C@@H](N)CC(C)C)CSCCSC[C@H](NC(=O)CNC(=O)[C@H](C(C)C)NC(=O)[C@H](Cc3cnc[nH]3)NC2=O)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CO)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](Cc2ccccc2)C(=O)NC(C(=O)O)CSSC[C@@H](C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)N[C@@H](CO)C(=O)O)[C@@H](C)O)NC1=O	10.1021/acs.jmedchem.0c01533
	CHEMBL4754949	180053	0	None	4	2	Human	10.5	pEC50	=	10.5	Functional	Agonist activity at human RXFP1 expressed in human HEK-293T cells co-transfected with pCRE beta-galactosidase reporter plasmid assessed as inhibition of IBMX-induced cAMP accumulation incubated for 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in human HEK-293T cells co-transfected with pCRE beta-galactosidase reporter plasmid assessed as inhibition of IBMX-induced cAMP accumulation incubated for 30 mins by HTRF assay	ChEMBL	5876	136	86	84	-20.9	CC[C@H](C)[C@@H]1NC(=O)[C@H](C)NC(=O)[C@H]([C@@H](C)CC)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](C(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCSC)NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](CO)NC(=O)[C@@H](N)CC(=O)O)C(C)C)[C@@H](C)CC)CSSC[C@@H]2NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](Cc3ccc(O)cc3)NC(=O)[C@@H](N)CC(C)C)CSCCSC[C@H](NC(=O)CNC(=O)[C@H](C(C)C)NC(=O)[C@H](Cc3cnc[nH]3)NC2=O)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CO)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](Cc2ccccc2)C(=O)NC(C(=O)O)CSSC[C@@H](C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)N[C@@H](CO)C(=O)O)[C@@H](C)O)NC1=O	10.1021/acs.jmedchem.0c01533
	162648163	179293	0	None	-	1	Human	10.0	pEC50	=	10	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	4895	203	66	67	-9.3	CCCCCCCCCCCCCCCCCCC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCCN)NC(=O)COCCOCCNC(=O)COCCOCCNC(=O)COCCOCCNC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](C)CNC(=O)[C@H](CO)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H](NC(=O)[C@H](CO)NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCC)NC(=O)[C@H](CCSC)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCC(=O)O)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4745611	179293	0	None	-	1	Human	10.0	pEC50	=	10	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	4895	203	66	67	-9.3	CCCCCCCCCCCCCCCCCCC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCCN)NC(=O)COCCOCCNC(=O)COCCOCCNC(=O)COCCOCCNC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](C)CNC(=O)[C@H](CO)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H](NC(=O)[C@H](CO)NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCC)NC(=O)[C@H](CCSC)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCC(=O)O)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	162672427	182617	0	None	-	1	Human	9.7	pEC50	=	9.7	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	4880	202	66	67	-10.3	CCCCCCCCCCCCCCCCCC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCCN)NC(=O)COCCOCCNC(=O)COCCOCCNC(=O)COCCOCCNC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](C)CNC(=O)[C@H](CO)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H](NC(=O)[C@H](CO)NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCC)NC(=O)[C@H](CCSC)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCC(=O)O)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4795810	182617	0	None	-	1	Human	9.7	pEC50	=	9.7	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	4880	202	66	67	-10.3	CCCCCCCCCCCCCCCCCC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCCN)NC(=O)COCCOCCNC(=O)COCCOCCNC(=O)COCCOCCNC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](C)CNC(=O)[C@H](CO)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H](NC(=O)[C@H](CO)NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCC)NC(=O)[C@H](CCSC)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCC(=O)O)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	162667576	181902	0	None	-	1	Human	9.4	pEC50	=	9.4	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	5414	233	69	76	-9.5	CCCCCCCCCCCCCCCCCCC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCCN)NC(=O)COCC(=O)NCCCOCCOCCOCCCNC(=O)COCC(=O)NCCCOCCOCCOCCCNC(=O)COCC(=O)NCCCOCCOCCOCCCNC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](C)CNC(=O)[C@H](CO)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H](NC(=O)[C@H](CO)NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCC)NC(=O)[C@H](CCSC)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCC(=O)O)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4786789	181902	0	None	-	1	Human	9.4	pEC50	=	9.4	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	5414	233	69	76	-9.5	CCCCCCCCCCCCCCCCCCC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCCN)NC(=O)COCC(=O)NCCCOCCOCCOCCCNC(=O)COCC(=O)NCCCOCCOCCOCCCNC(=O)COCC(=O)NCCCOCCOCCOCCCNC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](C)CNC(=O)[C@H](CO)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H](NC(=O)[C@H](CO)NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCC)NC(=O)[C@H](CCSC)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCC(=O)O)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	162654489	180053	0	None	4	2	Human	9.4	pEC50	=	9.4	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	5876	136	86	84	-20.9	CC[C@H](C)[C@@H]1NC(=O)[C@H](C)NC(=O)[C@H]([C@@H](C)CC)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](C(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCSC)NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](CO)NC(=O)[C@@H](N)CC(=O)O)C(C)C)[C@@H](C)CC)CSSC[C@@H]2NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](Cc3ccc(O)cc3)NC(=O)[C@@H](N)CC(C)C)CSCCSC[C@H](NC(=O)CNC(=O)[C@H](C(C)C)NC(=O)[C@H](Cc3cnc[nH]3)NC2=O)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CO)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](Cc2ccccc2)C(=O)NC(C(=O)O)CSSC[C@@H](C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)N[C@@H](CO)C(=O)O)[C@@H](C)O)NC1=O	10.1021/acs.jmedchem.0c01533
	CHEMBL4754949	180053	0	None	4	2	Human	9.4	pEC50	=	9.4	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	5876	136	86	84	-20.9	CC[C@H](C)[C@@H]1NC(=O)[C@H](C)NC(=O)[C@H]([C@@H](C)CC)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](C(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCSC)NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](CO)NC(=O)[C@@H](N)CC(=O)O)C(C)C)[C@@H](C)CC)CSSC[C@@H]2NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](Cc3ccc(O)cc3)NC(=O)[C@@H](N)CC(C)C)CSCCSC[C@H](NC(=O)CNC(=O)[C@H](C(C)C)NC(=O)[C@H](Cc3cnc[nH]3)NC2=O)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CO)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](Cc2ccccc2)C(=O)NC(C(=O)O)CSSC[C@@H](C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)N[C@@H](CO)C(=O)O)[C@@H](C)O)NC1=O	10.1021/acs.jmedchem.0c01533
	162677247	182948	0	None	-	1	Human	9.2	pEC50	=	9.2	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3441	156	40	48	-1.9	CCCCCCCCCCCCCCCCCCC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCCN)NC(=O)CCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCNC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCC(=O)O)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC	10.1021/acs.jmedchem.0c01533
	CHEMBL4799907	182948	0	None	-	1	Human	9.2	pEC50	=	9.2	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3441	156	40	48	-1.9	CCCCCCCCCCCCCCCCCCC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCCN)NC(=O)CCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCNC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCC(=O)O)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC	10.1021/acs.jmedchem.0c01533
	162661030	180867	0	None	-	1	Human	9.0	pEC50	=	9	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	4866	201	66	67	-10.6	CCCCCCCCCCCCCCCCC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCCN)NC(=O)COCCOCCNC(=O)COCCOCCNC(=O)COCCOCCNC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](C)CNC(=O)[C@H](CO)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H](NC(=O)[C@H](CO)NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCC)NC(=O)[C@H](CCSC)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCC(=O)O)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4764326	180867	0	None	-	1	Human	9.0	pEC50	=	9	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	4866	201	66	67	-10.6	CCCCCCCCCCCCCCCCC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCCN)NC(=O)COCCOCCNC(=O)COCCOCCNC(=O)COCCOCCNC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](C)CNC(=O)[C@H](CO)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H](NC(=O)[C@H](CO)NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCC)NC(=O)[C@H](CCSC)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCC(=O)O)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	162674882	182770	0	None	-	1	Human	9.0	pEC50	=	9	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	4191	177	54	60	-8.7	CCCCCCCCCCCCCCCCCC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCCN)NC(=O)CCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCNC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](C)CNC(=O)[C@H](CO)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H](NC(=O)[C@H](CO)NC(=O)[C@H](CCCC)NC(=O)[C@H](CCSC)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCC(=O)O)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4797641	182770	0	None	-	1	Human	9.0	pEC50	=	9	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	4191	177	54	60	-8.7	CCCCCCCCCCCCCCCCCC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCCN)NC(=O)CCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCNC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](C)CNC(=O)[C@H](CO)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H](NC(=O)[C@H](CO)NC(=O)[C@H](CCCC)NC(=O)[C@H](CCSC)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCC(=O)O)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	56593316	133245	0	None	-	1	Human	7.0	pEC50	=	7.0	Functional	Agonist activity at RXFP1 receptor in human THP1 cells assessed as stimulation of cAMP production incubated for 30 mins by HTRF assayAgonist activity at RXFP1 receptor in human THP1 cells assessed as stimulation of cAMP production incubated for 30 mins by HTRF assay	ChEMBL	506	8	2	5	5.3	CCCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	nan
	CHEMBL3715235	133245	0	None	-	1	Human	7.0	pEC50	=	7.0	Functional	Agonist activity at RXFP1 receptor in human THP1 cells assessed as stimulation of cAMP production incubated for 30 mins by HTRF assayAgonist activity at RXFP1 receptor in human THP1 cells assessed as stimulation of cAMP production incubated for 30 mins by HTRF assay	ChEMBL	506	8	2	5	5.3	CCCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	nan
	56593334	133598	0	None	-	1	Human	6.0	pEC50	=	6.0	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	454	5	2	4	4.8	O=C(Nc1cccc(S(=O)(=O)C(F)(F)F)c1)c1ccccc1NC(=O)C1CCCCC1	10.1016/j.ejmech.2018.06.008
	CHEMBL3716462	133598	0	None	-	1	Human	6.0	pEC50	=	6.0	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	454	5	2	4	4.8	O=C(Nc1cccc(S(=O)(=O)C(F)(F)F)c1)c1ccccc1NC(=O)C1CCCCC1	10.1016/j.ejmech.2018.06.008
	56593305	134167	0	None	-	1	Human	7.0	pEC50	=	7.0	Functional	Agonist activity at RXFP1 receptor in human THP1 cells assessed as stimulation of cAMP production incubated for 30 mins by HTRF assayAgonist activity at RXFP1 receptor in human THP1 cells assessed as stimulation of cAMP production incubated for 30 mins by HTRF assay	ChEMBL	546	7	2	5	5.4	O=C(Nc1cccc(S(=O)(=O)C(F)(F)F)c1)c1ccccc1NC(=O)c1ccccc1OCC(F)(F)F	nan
	CHEMBL3718400	134167	0	None	-	1	Human	7.0	pEC50	=	7.0	Functional	Agonist activity at RXFP1 receptor in human THP1 cells assessed as stimulation of cAMP production incubated for 30 mins by HTRF assayAgonist activity at RXFP1 receptor in human THP1 cells assessed as stimulation of cAMP production incubated for 30 mins by HTRF assay	ChEMBL	546	7	2	5	5.4	O=C(Nc1cccc(S(=O)(=O)C(F)(F)F)c1)c1ccccc1NC(=O)c1ccccc1OCC(F)(F)F	nan
	56593346	133808	0	None	-	1	Human	5.9	pEC50	=	5.9	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	468	5	2	3	6.1	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NC(=O)c1ccccc1OC(F)(F)F	10.1016/j.ejmech.2018.06.008
	CHEMBL3717178	133808	0	None	-	1	Human	5.9	pEC50	=	5.9	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	468	5	2	3	6.1	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NC(=O)c1ccccc1OC(F)(F)F	10.1016/j.ejmech.2018.06.008
	162664297	181499	0	None	-2	2	Human	7.9	pEC50	=	7.9	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	2767	100	45	38	-12.7	CCCC[C@H](NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)NC[C@H](C)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4781560	181499	0	None	-2	2	Human	7.9	pEC50	=	7.9	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	2767	100	45	38	-12.7	CCCC[C@H](NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)NC[C@H](C)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	56593322	133202	0	None	-	1	Human	6.9	pEC50	=	6.9	Functional	Agonist activity at RXFP1 receptor in human THP1 cells assessed as stimulation of cAMP production incubated for 30 mins by HTRF assayAgonist activity at RXFP1 receptor in human THP1 cells assessed as stimulation of cAMP production incubated for 30 mins by HTRF assay	ChEMBL	520	9	2	5	5.7	CCCCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	nan
	CHEMBL3715081	133202	0	None	-	1	Human	6.9	pEC50	=	6.9	Functional	Agonist activity at RXFP1 receptor in human THP1 cells assessed as stimulation of cAMP production incubated for 30 mins by HTRF assayAgonist activity at RXFP1 receptor in human THP1 cells assessed as stimulation of cAMP production incubated for 30 mins by HTRF assay	ChEMBL	520	9	2	5	5.7	CCCCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	nan
	162649438	179472	0	None	-	1	Human	6.9	pEC50	=	6.9	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3412	125	54	48	-14.4	CC[C@H](C)[C@H](NC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4747756	179472	0	None	-	1	Human	6.9	pEC50	=	6.9	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3412	125	54	48	-14.4	CC[C@H](C)[C@H](NC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	2806493	133595	4	None	-	1	Human	5.9	pEC50	=	5.9	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	384	4	2	2	5.2	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1ccccc1	10.1016/j.ejmech.2018.06.008
	CHEMBL3716450	133595	4	None	-	1	Human	5.9	pEC50	=	5.9	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	384	4	2	2	5.2	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1ccccc1	10.1016/j.ejmech.2018.06.008
	38269206	134157	0	None	-	1	Human	4.9	pEC50	=	4.9	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	340	4	2	2	4.6	O=C(Nc1cccc(F)c1)c1ccccc1NC(=O)C1CCCCC1	10.1016/j.ejmech.2018.06.008
	CHEMBL3718363	134157	0	None	-	1	Human	4.9	pEC50	=	4.9	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	340	4	2	2	4.6	O=C(Nc1cccc(F)c1)c1ccccc1NC(=O)C1CCCCC1	10.1016/j.ejmech.2018.06.008
	162659815	180618	0	None	-	1	Human	7.9	pEC50	=	7.9	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	2785	100	45	39	-13.2	CC[C@H](C)[C@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)C(=O)NC[C@H](C)C(=O)NC[C@H](C)C(=O)N[C@@H](CCC(=O)O)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)NC[C@H](C)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4761130	180618	0	None	-	1	Human	7.9	pEC50	=	7.9	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	2785	100	45	39	-13.2	CC[C@H](C)[C@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)C(=O)NC[C@H](C)C(=O)NC[C@H](C)C(=O)N[C@@H](CCC(=O)O)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)NC[C@H](C)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	162666079	181731	0	None	-	1	Human	7.9	pEC50	=	7.9	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	2855	106	46	40	-12.6	CC[C@H](C)[C@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)C(=O)NC[C@H](C)C(=O)NC[C@H](C)C(=O)N[C@@H](CCC(=O)O)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O	10.1021/acs.jmedchem.0c01533
	CHEMBL4784237	181731	0	None	-	1	Human	7.9	pEC50	=	7.9	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	2855	106	46	40	-12.6	CC[C@H](C)[C@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)C(=O)NC[C@H](C)C(=O)NC[C@H](C)C(=O)N[C@@H](CCC(=O)O)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O	10.1021/acs.jmedchem.0c01533
	162656358	180307	0	None	-	1	Human	6.8	pEC50	=	6.8	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3355	121	53	47	-14.4	CC[C@H](C)[C@H](NC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CO)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4757578	180307	0	None	-	1	Human	6.8	pEC50	=	6.8	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3355	121	53	47	-14.4	CC[C@H](C)[C@H](NC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CO)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	162677445	182961	0	None	-	1	Human	6.8	pEC50	=	6.8	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3139	113	49	43	-12.2	CC[C@H](C)[C@H](NC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(C)=O)C(C)C)[C@@H](C)CC)[C@@H](C)CC)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4800116	182961	0	None	-	1	Human	6.8	pEC50	=	6.8	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3139	113	49	43	-12.2	CC[C@H](C)[C@H](NC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(C)=O)C(C)C)[C@@H](C)CC)[C@@H](C)CC)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	56593309	133239	0	None	-	1	Human	5.8	pEC50	=	5.8	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	493	7	2	6	4.3	CCOc1ccccc1C(=O)Nc1ncccc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	CHEMBL3715203	133239	0	None	-	1	Human	5.8	pEC50	=	5.8	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	493	7	2	6	4.3	CCOc1ccccc1C(=O)Nc1ncccc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	162646950	179099	0	None	-	1	Human	7.8	pEC50	=	7.8	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3195	119	50	44	-12.3	CC[C@H](C)[C@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)C(=O)NC[C@H](C)C(=O)NC[C@H](C)C(=O)N[C@@H](CCC(=O)O)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O	10.1021/acs.jmedchem.0c01533
	CHEMBL4743539	179099	0	None	-	1	Human	7.8	pEC50	=	7.8	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3195	119	50	44	-12.3	CC[C@H](C)[C@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)C(=O)NC[C@H](C)C(=O)NC[C@H](C)C(=O)N[C@@H](CCC(=O)O)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O	10.1021/acs.jmedchem.0c01533
	162643258	181160	0	None	-	1	Human	7.8	pEC50	=	7.8	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3411	126	53	47	-12.8	CC[C@H](C)[C@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)C(=O)NCC(C)C(=O)NCC(C)C(=O)N[C@@H](CCC(=O)O)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)NC[C@H](C)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(=O)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4777259	181160	0	None	-	1	Human	7.8	pEC50	=	7.8	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3411	126	53	47	-12.8	CC[C@H](C)[C@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)C(=O)NCC(C)C(=O)NCC(C)C(=O)N[C@@H](CCC(=O)O)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)NC[C@H](C)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(=O)O	10.1021/acs.jmedchem.0c01533
	162674863	182731	0	None	-	1	Human	7.8	pEC50	=	7.8	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3509	135	52	47	-9.4	CCCCCCCCCCCCCCCCC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](C)CNC(=O)[C@H](CO)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H](NC(=O)[C@H](CO)NC(=O)[C@H](CCSC)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCC(=O)O)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4797258	182731	0	None	-	1	Human	7.8	pEC50	=	7.8	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3509	135	52	47	-9.4	CCCCCCCCCCCCCCCCC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](C)CNC(=O)[C@H](CO)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H](NC(=O)[C@H](CO)NC(=O)[C@H](CCSC)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCC(=O)O)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	162662427	181376	0	None	-	1	Human	7.8	pEC50	=	7.8	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3383	123	53	47	-14.2	CC[C@H](C)[C@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)C(=O)NC[C@H](C)C(=O)NC[C@H](C)C(=O)N[C@@H](CCC(=O)O)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)NC[C@H](C)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4779982	181376	0	None	-	1	Human	7.8	pEC50	=	7.8	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3383	123	53	47	-14.2	CC[C@H](C)[C@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)C(=O)NC[C@H](C)C(=O)NC[C@H](C)C(=O)N[C@@H](CCC(=O)O)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)NC[C@H](C)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	162648609	179235	0	None	-	1	Human	7.8	pEC50	=	7.8	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3292	122	50	45	-12.0	CCCC[C@H](OC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@H](CCCCN)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)NC[C@H](C)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCN)C(=O)N[C@@H](CCCCCNC(C)=O)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4744987	179235	0	None	-	1	Human	7.8	pEC50	=	7.8	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3292	122	50	45	-12.0	CCCC[C@H](OC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@H](CCCCN)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)NC[C@H](C)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCN)C(=O)N[C@@H](CCCCCNC(C)=O)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	162672427	182617	0	None	-	1	Human	7.7	pEC50	=	7.7	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins in presence of 2 % HSA by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins in presence of 2 % HSA by HTRF assay	ChEMBL	4880	202	66	67	-10.3	CCCCCCCCCCCCCCCCCC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCCN)NC(=O)COCCOCCNC(=O)COCCOCCNC(=O)COCCOCCNC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](C)CNC(=O)[C@H](CO)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H](NC(=O)[C@H](CO)NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCC)NC(=O)[C@H](CCSC)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCC(=O)O)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4795810	182617	0	None	-	1	Human	7.7	pEC50	=	7.7	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins in presence of 2 % HSA by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins in presence of 2 % HSA by HTRF assay	ChEMBL	4880	202	66	67	-10.3	CCCCCCCCCCCCCCCCCC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCCN)NC(=O)COCCOCCNC(=O)COCCOCCNC(=O)COCCOCCNC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](C)CNC(=O)[C@H](CO)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H](NC(=O)[C@H](CO)NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCC)NC(=O)[C@H](CCSC)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCC(=O)O)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	56593314	133817	0	None	-	1	Human	6.7	pEC50	=	6.7	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	478	6	2	5	4.5	COc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	CHEMBL3717211	133817	0	None	-	1	Human	6.7	pEC50	=	6.7	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	478	6	2	5	4.5	COc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	56593330	133863	0	None	-	1	Human	6.7	pEC50	=	6.7	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	492	7	2	5	4.9	CCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	CHEMBL3717389	133863	0	None	-	1	Human	6.7	pEC50	=	6.7	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	492	7	2	5	4.9	CCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	1313916	39856	8	None	-	1	Human	5.7	pEC50	=	5.7	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	390	4	2	2	5.5	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NC(=O)C1CCCCC1	10.1016/j.ejmech.2018.06.008
	CHEMBL1479446	39856	8	None	-	1	Human	5.7	pEC50	=	5.7	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	390	4	2	2	5.5	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NC(=O)C1CCCCC1	10.1016/j.ejmech.2018.06.008
	56593340	133577	0	None	-	1	Human	5.7	pEC50	=	5.7	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	414	5	2	3	5.2	COc1cccc(C(=O)Nc2ccccc2C(=O)Nc2cccc(C(F)(F)F)c2)c1	10.1016/j.ejmech.2018.06.008
	CHEMBL3716394	133577	0	None	-	1	Human	5.7	pEC50	=	5.7	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	414	5	2	3	5.2	COc1cccc(C(=O)Nc2ccccc2C(=O)Nc2cccc(C(F)(F)F)c2)c1	10.1016/j.ejmech.2018.06.008
	56593311	133964	0	None	-	1	Human	5.7	pEC50	=	5.7	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	422	5	2	3	6.1	O=C(Nc1cccc(SC(F)(F)F)c1)c1ccccc1NC(=O)C1CCCCC1	10.1016/j.ejmech.2018.06.008
	CHEMBL3717723	133964	0	None	-	1	Human	5.7	pEC50	=	5.7	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	422	5	2	3	6.1	O=C(Nc1cccc(SC(F)(F)F)c1)c1ccccc1NC(=O)C1CCCCC1	10.1016/j.ejmech.2018.06.008
	162650672	179576	0	None	-	1	Human	7.7	pEC50	=	7.7	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3152	116	49	43	-12.1	CC[C@H](C)[C@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)C(=O)NC[C@H](C)C(=O)NC[C@H](C)C(=O)N[C@@H](CCC(=O)O)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)NC[C@H](C)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O	10.1021/acs.jmedchem.0c01533
	CHEMBL4748931	179576	0	None	-	1	Human	7.7	pEC50	=	7.7	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3152	116	49	43	-12.1	CC[C@H](C)[C@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)C(=O)NC[C@H](C)C(=O)NC[C@H](C)C(=O)N[C@@H](CCC(=O)O)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)NC[C@H](C)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O	10.1021/acs.jmedchem.0c01533
	162648163	179293	0	None	-	1	Human	7.7	pEC50	=	7.7	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins in presence of 2 % HSA by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins in presence of 2 % HSA by HTRF assay	ChEMBL	4895	203	66	67	-9.3	CCCCCCCCCCCCCCCCCCC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCCN)NC(=O)COCCOCCNC(=O)COCCOCCNC(=O)COCCOCCNC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](C)CNC(=O)[C@H](CO)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H](NC(=O)[C@H](CO)NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCC)NC(=O)[C@H](CCSC)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCC(=O)O)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4745611	179293	0	None	-	1	Human	7.7	pEC50	=	7.7	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins in presence of 2 % HSA by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins in presence of 2 % HSA by HTRF assay	ChEMBL	4895	203	66	67	-9.3	CCCCCCCCCCCCCCCCCCC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCCN)NC(=O)COCCOCCNC(=O)COCCOCCNC(=O)COCCOCCNC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](C)CNC(=O)[C@H](CO)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H](NC(=O)[C@H](CO)NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCC)NC(=O)[C@H](CCSC)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCC(=O)O)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	56593349	2534	25	None	-	1	Human	6.7	pEC50	=	6.7	Functional	Agonist activity at RXFP1 receptor in human THP1 cells assessed as stimulation of cAMP production incubated for 30 mins by HTRF assayAgonist activity at RXFP1 receptor in human THP1 cells assessed as stimulation of cAMP production incubated for 30 mins by HTRF assay	ChEMBL	506	7	2	5	5.3	CC(Oc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(c1)S(=O)(=O)C(F)(F)F)C	nan
	8322	2534	25	None	-	1	Human	6.7	pEC50	=	6.7	Functional	Agonist activity at RXFP1 receptor in human THP1 cells assessed as stimulation of cAMP production incubated for 30 mins by HTRF assayAgonist activity at RXFP1 receptor in human THP1 cells assessed as stimulation of cAMP production incubated for 30 mins by HTRF assay	ChEMBL	506	7	2	5	5.3	CC(Oc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(c1)S(=O)(=O)C(F)(F)F)C	nan
	CHEMBL3716980	2534	25	None	-	1	Human	6.7	pEC50	=	6.7	Functional	Agonist activity at RXFP1 receptor in human THP1 cells assessed as stimulation of cAMP production incubated for 30 mins by HTRF assayAgonist activity at RXFP1 receptor in human THP1 cells assessed as stimulation of cAMP production incubated for 30 mins by HTRF assay	ChEMBL	506	7	2	5	5.3	CC(Oc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(c1)S(=O)(=O)C(F)(F)F)C	nan
	162659417	180644	0	None	-	1	Human	6.7	pEC50	=	6.7	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3257	114	52	46	-15.6	CC[C@H](C)[C@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CO)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)C(=O)N[C@@H](C)C(=O)NC[C@H](C)C(=O)N[C@@H](CO)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CO)C(=O)N[C@@H](CC(C)C)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4761424	180644	0	None	-	1	Human	6.7	pEC50	=	6.7	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3257	114	52	46	-15.6	CC[C@H](C)[C@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CO)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)C(=O)N[C@@H](C)C(=O)NC[C@H](C)C(=O)N[C@@H](CO)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CO)C(=O)N[C@@H](CC(C)C)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	162670766	182370	0	None	-	1	Human	6.7	pEC50	=	6.7	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3097	111	49	43	-13.1	CC[C@H](C)[C@H](NC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CO)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4792874	182370	0	None	-	1	Human	6.7	pEC50	=	6.7	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3097	111	49	43	-13.1	CC[C@H](C)[C@H](NC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CO)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	56593317	134425	0	None	-	1	Human	5.7	pEC50	=	5.7	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	404	4	2	2	5.9	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NC(=O)C1CCCCCC1	10.1016/j.ejmech.2018.06.008
	CHEMBL3719257	134425	0	None	-	1	Human	5.7	pEC50	=	5.7	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	404	4	2	2	5.9	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NC(=O)C1CCCCCC1	10.1016/j.ejmech.2018.06.008
	162654519	180088	0	None	-	1	Human	7.6	pEC50	=	7.6	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	2828	103	46	40	-13.3	CC[C@H](C)[C@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)C(=O)NC[C@H](C)C(=O)NC[C@H](C)C(=O)N[C@@H](CCC(=O)O)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4755239	180088	0	None	-	1	Human	7.6	pEC50	=	7.6	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	2828	103	46	40	-13.3	CC[C@H](C)[C@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)C(=O)NC[C@H](C)C(=O)NC[C@H](C)C(=O)N[C@@H](CCC(=O)O)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	162654037	180092	0	None	-	1	Human	6.6	pEC50	=	6.6	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3424	126	53	47	-12.7	CC[C@H](C)[C@H](NC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CO)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CCC(=O)O)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O	10.1021/acs.jmedchem.0c01533
	CHEMBL4755289	180092	0	None	-	1	Human	6.6	pEC50	=	6.6	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3424	126	53	47	-12.7	CC[C@H](C)[C@H](NC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CO)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CCC(=O)O)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O	10.1021/acs.jmedchem.0c01533
	5298634	134435	10	None	-	1	Human	5.6	pEC50	=	5.6	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	376	4	2	2	5.1	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NC(=O)C1CCCC1	10.1016/j.ejmech.2018.06.008
	CHEMBL3719295	134435	10	None	-	1	Human	5.6	pEC50	=	5.6	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	376	4	2	2	5.1	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NC(=O)C1CCCC1	10.1016/j.ejmech.2018.06.008
	56593332	161701	0	None	-	1	Human	5.6	pEC50	=	5.6	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	498	7	2	6	4.9	CCOc1ccccc1C(=O)Nc1sccc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	CHEMBL4163593	161701	0	None	-	1	Human	5.6	pEC50	=	5.6	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	498	7	2	6	4.9	CCOc1ccccc1C(=O)Nc1sccc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	162667576	181902	0	None	-	1	Human	7.6	pEC50	=	7.6	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins in presence of 2 % HSA by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins in presence of 2 % HSA by HTRF assay	ChEMBL	5414	233	69	76	-9.5	CCCCCCCCCCCCCCCCCCC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCCN)NC(=O)COCC(=O)NCCCOCCOCCOCCCNC(=O)COCC(=O)NCCCOCCOCCOCCCNC(=O)COCC(=O)NCCCOCCOCCOCCCNC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](C)CNC(=O)[C@H](CO)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H](NC(=O)[C@H](CO)NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCC)NC(=O)[C@H](CCSC)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCC(=O)O)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4786789	181902	0	None	-	1	Human	7.6	pEC50	=	7.6	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins in presence of 2 % HSA by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins in presence of 2 % HSA by HTRF assay	ChEMBL	5414	233	69	76	-9.5	CCCCCCCCCCCCCCCCCCC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCCN)NC(=O)COCC(=O)NCCCOCCOCCOCCCNC(=O)COCC(=O)NCCCOCCOCCOCCCNC(=O)COCC(=O)NCCCOCCOCCOCCCNC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](C)CNC(=O)[C@H](CO)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H](NC(=O)[C@H](CO)NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCC)NC(=O)[C@H](CCSC)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCC(=O)O)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	56593335	133782	0	None	-	1	Human	6.6	pEC50	=	6.6	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	428	6	2	3	5.6	CCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	CHEMBL3717089	133782	0	None	-	1	Human	6.6	pEC50	=	6.6	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	428	6	2	3	5.6	CCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	56593308	133636	0	None	-	1	Human	5.6	pEC50	=	5.6	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	466	5	2	2	7.1	O=C(Nc1cccc(-c2ccccc2C(F)(F)F)c1)c1ccccc1NC(=O)C1CCCCC1	10.1016/j.ejmech.2018.06.008
	CHEMBL3716596	133636	0	None	-	1	Human	5.6	pEC50	=	5.6	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	466	5	2	2	7.1	O=C(Nc1cccc(-c2ccccc2C(F)(F)F)c1)c1ccccc1NC(=O)C1CCCCC1	10.1016/j.ejmech.2018.06.008
	56593333	133712	0	None	-	1	Human	5.6	pEC50	=	5.6	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	400	4	2	2	5.2	O=C(Nc1cccc(Br)c1)c1ccccc1NC(=O)C1CCCCC1	10.1016/j.ejmech.2018.06.008
	CHEMBL3716871	133712	0	None	-	1	Human	5.6	pEC50	=	5.6	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	400	4	2	2	5.2	O=C(Nc1cccc(Br)c1)c1ccccc1NC(=O)C1CCCCC1	10.1016/j.ejmech.2018.06.008
	56593350	134124	0	None	-	1	Human	5.6	pEC50	=	5.6	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	378	4	2	2	5.8	CC(C)(C)c1cccc(NC(=O)c2ccccc2NC(=O)C2CCCCC2)c1	10.1016/j.ejmech.2018.06.008
	CHEMBL3718273	134124	0	None	-	1	Human	5.6	pEC50	=	5.6	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	378	4	2	2	5.8	CC(C)(C)c1cccc(NC(=O)c2ccccc2NC(=O)C2CCCCC2)c1	10.1016/j.ejmech.2018.06.008
	162672610	182434	0	None	-35	2	Human	6.6	pEC50	=	6.6	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins in presence of 2 % HSA by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins in presence of 2 % HSA by HTRF assay	ChEMBL	4064	171	53	59	-9.7	CCCCCCCCCCCCCCCCC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCCN)NC(=O)CCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCNC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](C)CNC(=O)[C@H](CO)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H](NC(=O)[C@H](CO)NC(=O)[C@H](CCSC)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCC(=O)O)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4793799	182434	0	None	-35	2	Human	6.6	pEC50	=	6.6	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins in presence of 2 % HSA by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins in presence of 2 % HSA by HTRF assay	ChEMBL	4064	171	53	59	-9.7	CCCCCCCCCCCCCCCCC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCCN)NC(=O)CCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCNC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](C)CNC(=O)[C@H](CO)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H](NC(=O)[C@H](CO)NC(=O)[C@H](CCSC)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCC(=O)O)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	56593323	133213	0	None	-	1	Human	5.5	pEC50	=	5.5	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	493	7	2	6	4.3	CCOc1ccccc1C(=O)Nc1cnccc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	CHEMBL3715105	133213	0	None	-	1	Human	5.5	pEC50	=	5.5	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	493	7	2	6	4.3	CCOc1ccccc1C(=O)Nc1cnccc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	56593318	133609	0	None	-	1	Human	5.5	pEC50	=	5.5	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	362	4	2	2	4.7	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NC(=O)C1CCC1	10.1016/j.ejmech.2018.06.008
	CHEMBL3716512	133609	0	None	-	1	Human	5.5	pEC50	=	5.5	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	362	4	2	2	4.7	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NC(=O)C1CCC1	10.1016/j.ejmech.2018.06.008
	56593313	134328	0	None	-	1	Human	4.5	pEC50	=	4.5	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	428	5	1	3	5.2	COc1ccccc1C(=O)Nc1ccccc1C(=O)N(C)c1cccc(C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	CHEMBL3718895	134328	0	None	-	1	Human	4.5	pEC50	=	4.5	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	428	5	1	3	5.2	COc1ccccc1C(=O)Nc1ccccc1C(=O)N(C)c1cccc(C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	162652974	179836	0	None	-	1	Human	8.5	pEC50	=	8.5	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	4163	175	54	60	-9.4	CCCCCCCCCCCCCCCC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCCN)NC(=O)CCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCNC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](C)CNC(=O)[C@H](CO)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H](NC(=O)[C@H](CO)NC(=O)[C@H](CCCC)NC(=O)[C@H](CCSC)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCC(=O)O)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4752287	179836	0	None	-	1	Human	8.5	pEC50	=	8.5	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	4163	175	54	60	-9.4	CCCCCCCCCCCCCCCC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCCN)NC(=O)CCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCNC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](C)CNC(=O)[C@H](CO)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H](NC(=O)[C@H](CO)NC(=O)[C@H](CCCC)NC(=O)[C@H](CCSC)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCC(=O)O)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	162672610	182434	0	None	-35	2	Human	8.4	pEC50	=	8.4	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	4064	171	53	59	-9.7	CCCCCCCCCCCCCCCCC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCCN)NC(=O)CCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCNC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](C)CNC(=O)[C@H](CO)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H](NC(=O)[C@H](CO)NC(=O)[C@H](CCSC)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCC(=O)O)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4793799	182434	0	None	-35	2	Human	8.4	pEC50	=	8.4	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	4064	171	53	59	-9.7	CCCCCCCCCCCCCCCCC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCCN)NC(=O)CCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCNC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](C)CNC(=O)[C@H](CO)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H](NC(=O)[C@H](CO)NC(=O)[C@H](CCSC)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCC(=O)O)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	162674882	182770	0	None	-	1	Human	7.5	pEC50	=	7.5	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins in presence of 2 % HSA by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins in presence of 2 % HSA by HTRF assay	ChEMBL	4191	177	54	60	-8.7	CCCCCCCCCCCCCCCCCC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCCN)NC(=O)CCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCNC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](C)CNC(=O)[C@H](CO)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H](NC(=O)[C@H](CO)NC(=O)[C@H](CCCC)NC(=O)[C@H](CCSC)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCC(=O)O)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4797641	182770	0	None	-	1	Human	7.5	pEC50	=	7.5	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins in presence of 2 % HSA by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins in presence of 2 % HSA by HTRF assay	ChEMBL	4191	177	54	60	-8.7	CCCCCCCCCCCCCCCCCC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCCN)NC(=O)CCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCNC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](C)CNC(=O)[C@H](CO)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H](NC(=O)[C@H](CO)NC(=O)[C@H](CCCC)NC(=O)[C@H](CCSC)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCC(=O)O)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	162669540	182057	0	None	-	1	Human	7.5	pEC50	=	7.5	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	2867	105	45	40	-11.9	CCCC[C@H](OC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)NC[C@H](C)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCCNC(C)=O)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4788675	182057	0	None	-	1	Human	7.5	pEC50	=	7.5	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	2867	105	45	40	-11.9	CCCC[C@H](OC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)NC[C@H](C)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCCNC(C)=O)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	162670803	182254	0	None	-	1	Human	7.5	pEC50	=	7.5	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3314	119	53	47	-14.8	CC[C@H](C)[C@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CO)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)C(=O)N[C@@H](C)C(=O)NC[C@H](C)C(=O)N[C@@H](CO)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(=O)O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4791290	182254	0	None	-	1	Human	7.5	pEC50	=	7.5	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3314	119	53	47	-14.8	CC[C@H](C)[C@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CO)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)C(=O)N[C@@H](C)C(=O)NC[C@H](C)C(=O)N[C@@H](CO)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(=O)O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	56593329	133910	0	None	-	1	Human	6.5	pEC50	=	6.5	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	414	5	2	3	5.2	COc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	CHEMBL3717553	133910	0	None	-	1	Human	6.5	pEC50	=	6.5	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	414	5	2	3	5.2	COc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	56593336	133320	0	None	-	1	Human	5.5	pEC50	=	5.5	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	356	4	2	2	5.1	O=C(Nc1cccc(Cl)c1)c1ccccc1NC(=O)C1CCCCC1	10.1016/j.ejmech.2018.06.008
	CHEMBL3715551	133320	0	None	-	1	Human	5.5	pEC50	=	5.5	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	356	4	2	2	5.1	O=C(Nc1cccc(Cl)c1)c1ccccc1NC(=O)C1CCCCC1	10.1016/j.ejmech.2018.06.008
	56593314	133817	0	None	-	1	Human	6.5	pEC50	=	6.5	Functional	Agonist activity at RXFP1 receptor in human THP1 cells assessed as stimulation of cAMP production incubated for 30 mins by HTRF assayAgonist activity at RXFP1 receptor in human THP1 cells assessed as stimulation of cAMP production incubated for 30 mins by HTRF assay	ChEMBL	478	6	2	5	4.5	COc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	nan
	CHEMBL3717211	133817	0	None	-	1	Human	6.5	pEC50	=	6.5	Functional	Agonist activity at RXFP1 receptor in human THP1 cells assessed as stimulation of cAMP production incubated for 30 mins by HTRF assayAgonist activity at RXFP1 receptor in human THP1 cells assessed as stimulation of cAMP production incubated for 30 mins by HTRF assay	ChEMBL	478	6	2	5	4.5	COc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	nan
	56593330	133863	0	None	-	1	Human	6.4	pEC50	=	6.4	Functional	Agonist activity at RXFP1 receptor in human THP1 cells assessed as stimulation of cAMP production incubated for 30 mins by HTRF assayAgonist activity at RXFP1 receptor in human THP1 cells assessed as stimulation of cAMP production incubated for 30 mins by HTRF assay	ChEMBL	492	7	2	5	4.9	CCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	nan
	CHEMBL3717389	133863	0	None	-	1	Human	6.4	pEC50	=	6.4	Functional	Agonist activity at RXFP1 receptor in human THP1 cells assessed as stimulation of cAMP production incubated for 30 mins by HTRF assayAgonist activity at RXFP1 receptor in human THP1 cells assessed as stimulation of cAMP production incubated for 30 mins by HTRF assay	ChEMBL	492	7	2	5	4.9	CCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	nan
	162648114	179335	0	None	-	1	Human	6.4	pEC50	=	6.4	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	4489	180	64	59	-8.3	CCCC[C@H](NC(=O)[C@H](CCSC)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCC(=O)O)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCCNC(C)=O)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)NC[C@H](C)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCCNC(C)=O)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCC(=O)O)C(=O)N[C@@H](CCC(=O)O)C(=O)N[C@@H](CCC(N)=O)C(=O)CCCCCCCCCCCCCCCCCC(=O)O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4746080	179335	0	None	-	1	Human	6.4	pEC50	=	6.4	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	4489	180	64	59	-8.3	CCCC[C@H](NC(=O)[C@H](CCSC)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCC(=O)O)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCCNC(C)=O)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)NC[C@H](C)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCCNC(C)=O)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCC(=O)O)C(=O)N[C@@H](CCC(=O)O)C(=O)N[C@@H](CCC(N)=O)C(=O)CCCCCCCCCCCCCCCCCC(=O)O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	162649375	179540	0	None	-	1	Human	7.4	pEC50	=	7.4	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3327	120	53	47	-15.1	CC[C@H](C)[C@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CO)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)C(=O)NC[C@H](C)C(=O)NC[C@H](C)C(=O)N[C@@H](CO)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4748601	179540	0	None	-	1	Human	7.4	pEC50	=	7.4	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3327	120	53	47	-15.1	CC[C@H](C)[C@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CO)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)C(=O)NC[C@H](C)C(=O)NC[C@H](C)C(=O)N[C@@H](CO)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	56593337	133209	0	None	-	1	Human	5.4	pEC50	=	5.4	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	418	4	2	2	5.9	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1ccccc1Cl	10.1016/j.ejmech.2018.06.008
	CHEMBL3715097	133209	0	None	-	1	Human	5.4	pEC50	=	5.4	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	418	4	2	2	5.9	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1ccccc1Cl	10.1016/j.ejmech.2018.06.008
	56593300	161652	0	None	-	1	Human	5.4	pEC50	=	5.4	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	471	8	2	4	5.2	CN(C)CCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	CHEMBL4162685	161652	0	None	-	1	Human	5.4	pEC50	=	5.4	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	471	8	2	4	5.2	CN(C)CCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	1511185	133314	12	None	-	1	Human	4.4	pEC50	=	4.4	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	336	4	2	2	4.8	Cc1cccc(NC(=O)c2ccccc2NC(=O)C2CCCCC2)c1	10.1016/j.ejmech.2018.06.008
	CHEMBL3715535	133314	12	None	-	1	Human	4.4	pEC50	=	4.4	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	336	4	2	2	4.8	Cc1cccc(NC(=O)c2ccccc2NC(=O)C2CCCCC2)c1	10.1016/j.ejmech.2018.06.008
	4795548	133714	6	None	-	1	Human	4.4	pEC50	=	4.4	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	352	5	2	3	4.5	COc1cccc(NC(=O)c2ccccc2NC(=O)C2CCCCC2)c1	10.1016/j.ejmech.2018.06.008
	CHEMBL3716878	133714	6	None	-	1	Human	4.4	pEC50	=	4.4	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	352	5	2	3	4.5	COc1cccc(NC(=O)c2ccccc2NC(=O)C2CCCCC2)c1	10.1016/j.ejmech.2018.06.008
	162646638	179134	0	None	-	1	Human	6.4	pEC50	=	6.4	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3055	109	49	43	-14.1	CC[C@H](C)[C@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CO)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)C(=O)N[C@@H](C)C(=O)NC[C@H](C)C(=O)N[C@@H](CO)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4743958	179134	0	None	-	1	Human	6.4	pEC50	=	6.4	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3055	109	49	43	-14.1	CC[C@H](C)[C@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CO)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)C(=O)N[C@@H](C)C(=O)NC[C@H](C)C(=O)N[C@@H](CO)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	56593306	133771	0	None	-	1	Human	5.4	pEC50	=	5.4	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	398	4	2	2	5.5	Cc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	CHEMBL3717045	133771	0	None	-	1	Human	5.4	pEC50	=	5.4	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	398	4	2	2	5.5	Cc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	162644941	178820	0	None	-	1	Human	7.4	pEC50	=	7.4	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	2883	107	46	40	-11.8	CC[C@H](C)[C@H](NC(=O)C(C)CNC(=O)[C@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CCC(=O)O)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O	10.1021/acs.jmedchem.0c01533
	CHEMBL4739969	178820	0	None	-	1	Human	7.4	pEC50	=	7.4	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	2883	107	46	40	-11.8	CC[C@H](C)[C@H](NC(=O)C(C)CNC(=O)[C@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CCC(=O)O)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O	10.1021/acs.jmedchem.0c01533
	162649856	179559	0	None	-	1	Human	7.4	pEC50	=	7.4	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3481	130	54	48	-12.8	CC[C@H](C)[C@H](NC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CCC(=O)O)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O	10.1021/acs.jmedchem.0c01533
	CHEMBL4748830	179559	0	None	-	1	Human	7.4	pEC50	=	7.4	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3481	130	54	48	-12.8	CC[C@H](C)[C@H](NC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CCC(=O)O)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O	10.1021/acs.jmedchem.0c01533
	162663002	181466	0	None	-	1	Human	7.4	pEC50	=	7.4	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3122	115	48	43	-11.7	CCCC[C@H](OC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@H](CCCCN)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)NC[C@H](C)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4781139	181466	0	None	-	1	Human	7.4	pEC50	=	7.4	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3122	115	48	43	-11.7	CCCC[C@H](OC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@H](CCCCN)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)NC[C@H](C)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	162655145	180176	0	None	-	1	Human	7.3	pEC50	=	7.3	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3166	116	49	43	-11.4	CC[C@H](C)[C@H](NC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CO)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CCC(=O)O)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O	10.1021/acs.jmedchem.0c01533
	CHEMBL4756139	180176	0	None	-	1	Human	7.3	pEC50	=	7.3	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3166	116	49	43	-11.4	CC[C@H](C)[C@H](NC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CO)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CCC(=O)O)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O	10.1021/acs.jmedchem.0c01533
	56593322	133202	0	None	-	1	Human	7.3	pEC50	=	7.3	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	520	9	2	5	5.7	CCCCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	CHEMBL3715081	133202	0	None	-	1	Human	7.3	pEC50	=	7.3	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	520	9	2	5	5.7	CCCCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	47936	192819	82	None	-	1	Human	7.3	pEC50	=	7.3	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	410	2	3	7	1.5	C=C[C@@]1(C)CC(=O)[C@@]2(O)[C@](C)(O1)[C@@H](OC(C)=O)[C@@H](O)[C@H]1C(C)(C)CC[C@H](O)[C@@]12C	10.1016/j.ejmech.2018.06.008
	CHEMBL52606	192819	82	None	-	1	Human	7.3	pEC50	=	7.3	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	410	2	3	7	1.5	C=C[C@@]1(C)CC(=O)[C@@]2(O)[C@](C)(O1)[C@@H](OC(C)=O)[C@@H](O)[C@H]1C(C)(C)CC[C@H](O)[C@@]12C	10.1016/j.ejmech.2018.06.008
	56593331	134203	0	None	-	1	Human	6.3	pEC50	=	6.3	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	442	6	2	3	6.0	CC(C)Oc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	CHEMBL3718541	134203	0	None	-	1	Human	6.3	pEC50	=	6.3	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	442	6	2	3	6.0	CC(C)Oc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	56593335	133782	0	None	-	1	Human	6.3	pEC50	=	6.3	Functional	Agonist activity at RXFP1 receptor in human THP1 cells assessed as stimulation of cAMP production incubated for 30 mins by HTRF assayAgonist activity at RXFP1 receptor in human THP1 cells assessed as stimulation of cAMP production incubated for 30 mins by HTRF assay	ChEMBL	428	6	2	3	5.6	CCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	nan
	CHEMBL3717089	133782	0	None	-	1	Human	6.3	pEC50	=	6.3	Functional	Agonist activity at RXFP1 receptor in human THP1 cells assessed as stimulation of cAMP production incubated for 30 mins by HTRF assayAgonist activity at RXFP1 receptor in human THP1 cells assessed as stimulation of cAMP production incubated for 30 mins by HTRF assay	ChEMBL	428	6	2	3	5.6	CCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	nan
	56593347	133316	0	None	-	1	Human	5.3	pEC50	=	5.3	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	493	7	2	6	4.3	CCOc1ccccc1C(=O)Nc1cccnc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	CHEMBL3715539	133316	0	None	-	1	Human	5.3	pEC50	=	5.3	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	493	7	2	6	4.3	CCOc1ccccc1C(=O)Nc1cccnc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	162654330	179174	0	None	-	1	Human	6.3	pEC50	=	6.3	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3299	116	52	46	-14.6	CC[C@H](C)[C@H](NC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CO)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CO)C(=O)N[C@@H](CC(C)C)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4744303	179174	0	None	-	1	Human	6.3	pEC50	=	6.3	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3299	116	52	46	-14.6	CC[C@H](C)[C@H](NC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CO)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CO)C(=O)N[C@@H](CC(C)C)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	56593316	133245	0	None	-	1	Human	7.3	pEC50	=	7.3	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	506	8	2	5	5.3	CCCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	CHEMBL3715235	133245	0	None	-	1	Human	7.3	pEC50	=	7.3	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	506	8	2	5	5.3	CCCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	162654892	180038	0	None	-	1	Human	6.3	pEC50	=	6.3	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3083	110	49	43	-13.3	CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CO)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4754697	180038	0	None	-	1	Human	6.3	pEC50	=	6.3	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3083	110	49	43	-13.3	CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CO)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	56593315	133789	0	None	-	1	Human	6.3	pEC50	=	6.3	Functional	Agonist activity at RXFP1 receptor in human THP1 cells assessed as stimulation of cAMP production incubated for 30 mins by HTRF assayAgonist activity at RXFP1 receptor in human THP1 cells assessed as stimulation of cAMP production incubated for 30 mins by HTRF assay	ChEMBL	446	6	2	4	5.8	COc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(SC(F)(F)F)c1	nan
	CHEMBL3717103	133789	0	None	-	1	Human	6.3	pEC50	=	6.3	Functional	Agonist activity at RXFP1 receptor in human THP1 cells assessed as stimulation of cAMP production incubated for 30 mins by HTRF assayAgonist activity at RXFP1 receptor in human THP1 cells assessed as stimulation of cAMP production incubated for 30 mins by HTRF assay	ChEMBL	446	6	2	4	5.8	COc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(SC(F)(F)F)c1	nan
	56593299	133490	0	None	-	1	Human	5.3	pEC50	=	5.3	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	368	5	2	3	5.2	CSc1cccc(NC(=O)c2ccccc2NC(=O)C2CCCCC2)c1	10.1016/j.ejmech.2018.06.008
	CHEMBL3716127	133490	0	None	-	1	Human	5.3	pEC50	=	5.3	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	368	5	2	3	5.2	CSc1cccc(NC(=O)c2ccccc2NC(=O)C2CCCCC2)c1	10.1016/j.ejmech.2018.06.008
	56593339	133602	0	None	-	1	Human	5.3	pEC50	=	5.3	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	378	6	2	2	5.3	CCC(CC)C(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	CHEMBL3716488	133602	0	None	-	1	Human	5.3	pEC50	=	5.3	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	378	6	2	2	5.3	CCC(CC)C(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	56593319	133694	0	None	-	1	Human	5.3	pEC50	=	5.3	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	364	6	2	2	5.1	CCCCC(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	CHEMBL3716813	133694	0	None	-	1	Human	5.3	pEC50	=	5.3	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	364	6	2	2	5.1	CCCCC(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	162670817	182267	0	None	-	1	Human	7.3	pEC50	=	7.3	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3209	121	50	44	-11.0	CC[C@H](C)[C@H](NC[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CCC(=O)O)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O	10.1021/acs.jmedchem.0c01533
	CHEMBL4791486	182267	0	None	-	1	Human	7.3	pEC50	=	7.3	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3209	121	50	44	-11.0	CC[C@H](C)[C@H](NC[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CCC(=O)O)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O	10.1021/acs.jmedchem.0c01533
	56593303	134094	1	None	-	1	Human	5.2	pEC50	=	5.2	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	385	4	2	3	4.6	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1cccnc1	10.1016/j.ejmech.2018.06.008
	CHEMBL3718178	134094	1	None	-	1	Human	5.2	pEC50	=	5.2	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	385	4	2	3	4.6	O=C(Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1)c1cccnc1	10.1016/j.ejmech.2018.06.008
	56593326	134224	0	None	-	1	Human	5.2	pEC50	=	5.2	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	367	5	2	4	4.4	O=C(Nc1cccc([N+](=O)[O-])c1)c1ccccc1NC(=O)C1CCCCC1	10.1016/j.ejmech.2018.06.008
	CHEMBL3718612	134224	0	None	-	1	Human	5.2	pEC50	=	5.2	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	367	5	2	4	4.4	O=C(Nc1cccc([N+](=O)[O-])c1)c1ccccc1NC(=O)C1CCCCC1	10.1016/j.ejmech.2018.06.008
	56593302	133253	0	None	-	1	Human	4.2	pEC50	=	4.2	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	338	6	2	3	4.0	COCCNc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	CHEMBL3715266	133253	0	None	-	1	Human	4.2	pEC50	=	4.2	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	338	6	2	3	4.0	COCCNc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	56593305	134167	0	None	-	1	Human	7.2	pEC50	=	7.2	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	546	7	2	5	5.4	O=C(Nc1cccc(S(=O)(=O)C(F)(F)F)c1)c1ccccc1NC(=O)c1ccccc1OCC(F)(F)F	10.1016/j.ejmech.2018.06.008
	CHEMBL3718400	134167	0	None	-	1	Human	7.2	pEC50	=	7.2	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	546	7	2	5	5.4	O=C(Nc1cccc(S(=O)(=O)C(F)(F)F)c1)c1ccccc1NC(=O)c1ccccc1OCC(F)(F)F	10.1016/j.ejmech.2018.06.008
	162656612	180335	0	None	-	1	Human	6.2	pEC50	=	6.2	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3041	106	48	42	-13.3	CC[C@H](C)[C@H](NC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CO)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CO)C(=O)N[C@@H](CC(C)C)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4757890	180335	0	None	-	1	Human	6.2	pEC50	=	6.2	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3041	106	48	42	-13.3	CC[C@H](C)[C@H](NC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CO)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CO)C(=O)N[C@@H](CC(C)C)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	56593345	133384	0	None	-	1	Human	6.1	pEC50	=	6.1	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	493	7	2	6	4.3	CCOc1ccccc1C(=O)Nc1ccncc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	CHEMBL3715743	133384	0	None	-	1	Human	6.1	pEC50	=	6.1	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	493	7	2	6	4.3	CCOc1ccccc1C(=O)Nc1ccncc1C(=O)Nc1cccc(S(=O)(=O)C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	56593320	133619	0	None	-	1	Human	6.1	pEC50	=	6.1	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	458	8	2	4	5.2	COCCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	CHEMBL3716540	133619	0	None	-	1	Human	6.1	pEC50	=	6.1	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	458	8	2	4	5.2	COCCOc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	56593296	133634	0	None	-	1	Human	5.1	pEC50	=	5.1	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	444	6	2	4	5.2	COc1cccc(OC)c1C(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	CHEMBL3716581	133634	0	None	-	1	Human	5.1	pEC50	=	5.1	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	444	6	2	4	5.2	COc1cccc(OC)c1C(=O)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	162662592	181387	0	None	-	1	Human	5.1	pEC50	=	5.1	Functional	Agonist activity at human RXFP1 expressed in human HEK-293T cells co-transfected with pCRE beta-galactosidase reporter plasmid assessed as inhibition of IBMX-induced cAMP accumulation incubated for 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in human HEK-293T cells co-transfected with pCRE beta-galactosidase reporter plasmid assessed as inhibition of IBMX-induced cAMP accumulation incubated for 30 mins by HTRF assay	ChEMBL	2985	104	48	42	-13.7	CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CO)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](N)C(C)C)[C@@H](C)CC)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CO)C(=O)N[C@@H](CC(C)C)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4780098	181387	0	None	-	1	Human	5.1	pEC50	=	5.1	Functional	Agonist activity at human RXFP1 expressed in human HEK-293T cells co-transfected with pCRE beta-galactosidase reporter plasmid assessed as inhibition of IBMX-induced cAMP accumulation incubated for 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in human HEK-293T cells co-transfected with pCRE beta-galactosidase reporter plasmid assessed as inhibition of IBMX-induced cAMP accumulation incubated for 30 mins by HTRF assay	ChEMBL	2985	104	48	42	-13.7	CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CO)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](N)C(C)C)[C@@H](C)CC)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CO)C(=O)N[C@@H](CC(C)C)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	162675717	182695	0	None	-	1	Human	6.1	pEC50	=	6.1	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	4461	178	64	59	-9.0	CCCC[C@H](NC(=O)[C@H](CCSC)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCC(=O)O)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCCNC(C)=O)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)NC[C@H](C)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCCNC(C)=O)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCC(=O)O)C(=O)N[C@@H](CCC(=O)O)C(=O)N[C@@H](CCC(N)=O)C(=O)CCCCCCCCCCCCCCCC(=O)O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4796713	182695	0	None	-	1	Human	6.1	pEC50	=	6.1	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	4461	178	64	59	-9.0	CCCC[C@H](NC(=O)[C@H](CCSC)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCC(=O)O)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCCNC(C)=O)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)NC[C@H](C)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCCNC(C)=O)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCC(=O)O)C(=O)N[C@@H](CCC(=O)O)C(=O)N[C@@H](CCC(N)=O)C(=O)CCCCCCCCCCCCCCCC(=O)O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	56593344	133174	0	None	-	1	Human	5.1	pEC50	=	5.1	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	398	5	2	2	5.1	O=C(Cc1ccccc1)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	CHEMBL3715001	133174	0	None	-	1	Human	5.1	pEC50	=	5.1	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	398	5	2	2	5.1	O=C(Cc1ccccc1)Nc1ccccc1C(=O)Nc1cccc(C(F)(F)F)c1	10.1016/j.ejmech.2018.06.008
	56593325	134244	0	None	-	1	Human	5.1	pEC50	=	5.1	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	348	4	2	2	4.3	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NC(=O)C1CC1	10.1016/j.ejmech.2018.06.008
	CHEMBL3718643	134244	0	None	-	1	Human	5.1	pEC50	=	5.1	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	348	4	2	2	4.3	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NC(=O)C1CC1	10.1016/j.ejmech.2018.06.008
	162661030	180867	0	None	-	1	Human	7.1	pEC50	=	7.1	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins in presence of 2 % HSA by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins in presence of 2 % HSA by HTRF assay	ChEMBL	4866	201	66	67	-10.6	CCCCCCCCCCCCCCCCC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCCN)NC(=O)COCCOCCNC(=O)COCCOCCNC(=O)COCCOCCNC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](C)CNC(=O)[C@H](CO)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H](NC(=O)[C@H](CO)NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCC)NC(=O)[C@H](CCSC)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCC(=O)O)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4764326	180867	0	None	-	1	Human	7.1	pEC50	=	7.1	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins in presence of 2 % HSA by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins in presence of 2 % HSA by HTRF assay	ChEMBL	4866	201	66	67	-10.6	CCCCCCCCCCCCCCCCC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCCN)NC(=O)COCCOCCNC(=O)COCCOCCNC(=O)COCCOCCNC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](C)CNC(=O)[C@H](CO)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H](NC(=O)[C@H](CO)NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCC)NC(=O)[C@H](CCSC)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCC(=O)O)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	162661521	180948	0	None	-	1	Human	6.1	pEC50	=	6.1	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3341	120	53	47	-14.6	CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CO)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4765167	180948	0	None	-	1	Human	6.1	pEC50	=	6.1	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3341	120	53	47	-14.6	CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CO)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	162677247	182948	0	None	-	1	Human	8.1	pEC50	=	8.1	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins in presence of 2 % HSA by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins in presence of 2 % HSA by HTRF assay	ChEMBL	3441	156	40	48	-1.9	CCCCCCCCCCCCCCCCCCC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCCN)NC(=O)CCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCNC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCC(=O)O)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC	10.1021/acs.jmedchem.0c01533
	CHEMBL4799907	182948	0	None	-	1	Human	8.1	pEC50	=	8.1	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins in presence of 2 % HSA by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins in presence of 2 % HSA by HTRF assay	ChEMBL	3441	156	40	48	-1.9	CCCCCCCCCCCCCCCCCCC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCCN)NC(=O)CCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCNC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCCCCNC(C)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCC(=O)O)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC	10.1021/acs.jmedchem.0c01533
	162666829	181843	0	None	-	1	Human	7.0	pEC50	=	7.0	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3069	110	49	43	-13.8	CC[C@H](C)[C@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CO)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)C(=O)NC[C@H](C)C(=O)NC[C@H](C)C(=O)N[C@@H](CO)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4785899	181843	0	None	-	1	Human	7.0	pEC50	=	7.0	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3069	110	49	43	-13.8	CC[C@H](C)[C@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CO)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)C(=O)NC[C@H](C)C(=O)NC[C@H](C)C(=O)N[C@@H](CO)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	162664515	181493	0	None	-	1	Human	6.0	pEC50	=	6.0	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3027	105	48	42	-13.5	CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CO)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CO)C(=O)N[C@@H](CC(C)C)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4781482	181493	0	None	-	1	Human	6.0	pEC50	=	6.0	Functional	Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	3027	105	48	42	-13.5	CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CO)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(C)=O)C(C)C)[C@@H](C)CC)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CO)C(=O)N[C@@H](CC(C)C)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	56593349	2534	25	None	-	1	Human	7.0	pEC50	=	7.0	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	506	7	2	5	5.3	CC(Oc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(c1)S(=O)(=O)C(F)(F)F)C	10.1016/j.ejmech.2018.06.008
	8322	2534	25	None	-	1	Human	7.0	pEC50	=	7.0	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	506	7	2	5	5.3	CC(Oc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(c1)S(=O)(=O)C(F)(F)F)C	10.1016/j.ejmech.2018.06.008
	CHEMBL3716980	2534	25	None	-	1	Human	7.0	pEC50	=	7.0	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	506	7	2	5	5.3	CC(Oc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(c1)S(=O)(=O)C(F)(F)F)C	10.1016/j.ejmech.2018.06.008
	56593321	133963	0	None	-	1	Human	5.0	pEC50	=	5.0	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	445	7	3	4	5.0	O=C(NCc1ccco1)c1ccccc1NC(=O)c1ccccc1NC(=O)C1CCCCC1	10.1016/j.ejmech.2018.06.008
	CHEMBL3717718	133963	0	None	-	1	Human	5.0	pEC50	=	5.0	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	445	7	3	4	5.0	O=C(NCc1ccco1)c1ccccc1NC(=O)c1ccccc1NC(=O)C1CCCCC1	10.1016/j.ejmech.2018.06.008
	1320335	134299	9	None	-	1	Human	5.0	pEC50	=	5.0	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	414	5	2	3	5.2	COc1ccc(C(=O)Nc2ccccc2C(=O)Nc2cccc(C(F)(F)F)c2)cc1	10.1016/j.ejmech.2018.06.008
	CHEMBL3718813	134299	9	None	-	1	Human	5.0	pEC50	=	5.0	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	414	5	2	3	5.2	COc1ccc(C(=O)Nc2ccccc2C(=O)Nc2cccc(C(F)(F)F)c2)cc1	10.1016/j.ejmech.2018.06.008
	730108	41298	15	None	-	1	Human	4.0	pEC50	=	4.0	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	322	4	2	2	4.5	O=C(Nc1ccccc1)c1ccccc1NC(=O)C1CCCCC1	10.1016/j.ejmech.2018.06.008
	CHEMBL1491180	41298	15	None	-	1	Human	4.0	pEC50	=	4.0	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	322	4	2	2	4.5	O=C(Nc1ccccc1)c1ccccc1NC(=O)C1CCCCC1	10.1016/j.ejmech.2018.06.008
	56593342	133894	0	None	-	1	Human	4.0	pEC50	=	4.0	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	390	4	2	2	5.5	O=C(Nc1ccc(C(F)(F)F)cc1)c1ccccc1NC(=O)C1CCCCC1	10.1016/j.ejmech.2018.06.008
	CHEMBL3717485	133894	0	None	-	1	Human	4.0	pEC50	=	4.0	Functional	Agonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assayAgonist activity at human RXFP1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by HTRF assay	ChEMBL	390	4	2	2	5.5	O=C(Nc1ccc(C(F)(F)F)cc1)c1ccccc1NC(=O)C1CCCCC1	10.1016/j.ejmech.2018.06.008
	820020	21626	7	None	-	1	Human	7.0	pPotency	=	7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	232	2	2	3	1.6	O=C(NN=C1CCCC1)c1[nH]nc2c1CCC2	nan
	CHEMBL1319564	21626	7	None	-	1	Human	7.0	pPotency	=	7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	232	2	2	3	1.6	O=C(NN=C1CCCC1)c1[nH]nc2c1CCC2	nan
	2146184	44315	10	None	-	1	Human	7.0	pPotency	=	7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	4	0	4	2.4	CN(C)c1ccc(C(=S)N2CCN(S(=O)(=O)c3ccccc3)CC2)cc1	nan
	CHEMBL1519935	44315	10	None	-	1	Human	7.0	pPotency	=	7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	4	0	4	2.4	CN(C)c1ccc(C(=S)N2CCN(S(=O)(=O)c3ccccc3)CC2)cc1	nan
	1761	99215	9	None	-	1	Human	6.0	pPotency	=	6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	320	3	4	9	-1.7	Nc1ncnc2c1ncn2C1OC(C(=O)NC2CC2)C(O)C1O	nan
	CHEMBL28449	99215	9	None	-	1	Human	6.0	pPotency	=	6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	320	3	4	9	-1.7	Nc1ncnc2c1ncn2C1OC(C(=O)NC2CC2)C(O)C1O	nan
	16019574	10780	10	None	-14	2	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	5	1	8	3.9	O=S(=O)(c1ccccc1)c1nnn2c1nc(NCc1ccc(F)cc1)c1sccc12	nan
	CHEMBL1172596	10780	10	None	-14	2	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	5	1	8	3.9	O=S(=O)(c1ccccc1)c1nnn2c1nc(NCc1ccc(F)cc1)c1sccc12	nan
	4132952	19471	1	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	3	2	11	0.2	CCOP1(=O)OCC2OC(n3cnc4c(N)ncnc43)C(O)C2O1	nan
	CHEMBL1300691	19471	1	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	3	2	11	0.2	CCOP1(=O)OCC2OC(n3cnc4c(N)ncnc43)C(O)C2O1	nan
	54677759	20890	7	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	2	1	3	4.1	O=c1c(Cc2ccccc2)c(O)c2cccc3c4c(n1c23)CCCC4	nan
	CHEMBL1312172	20890	7	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	2	1	3	4.1	O=c1c(Cc2ccccc2)c(O)c2cccc3c4c(n1c23)CCCC4	nan
	16027480	21323	5	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	7	1	9	3.6	COc1cccc(C(=O)Nc2ccc(C(=O)OCc3cc(=O)n4nc(C5CC5)sc4n3)cc2)c1	nan
	CHEMBL1316197	21323	5	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	7	1	9	3.6	COc1cccc(C(=O)Nc2ccc(C(=O)OCc3cc(=O)n4nc(C5CC5)sc4n3)cc2)c1	nan
	941768	21891	8	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	288	2	3	7	-0.5	O=C1NC(=O)C(=NNc2ccc3c(c2)COC3=O)C(=O)N1	nan
	CHEMBL1321879	21891	8	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	288	2	3	7	-0.5	O=C1NC(=O)C(=NNc2ccc3c(c2)COC3=O)C(=O)N1	nan
	2764158	22446	30	None	-2	2	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	224	2	1	5	2.7	CSc1ccccc1-c1nnc(S)o1	nan
	CHEMBL1326901	22446	30	None	-2	2	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	224	2	1	5	2.7	CSc1ccccc1-c1nnc(S)o1	nan
	2810145	25731	6	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	4	1	6	3.6	COc1cc2nc(NC(=O)c3ccc(Cl)cc3)sc(=O)c2cc1OC	nan
	CHEMBL1354031	25731	6	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	4	1	6	3.6	COc1cc2nc(NC(=O)c3ccc(Cl)cc3)sc(=O)c2cc1OC	nan
	16010496	25905	2	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	5	2	6	0.6	Cc1ccc2ncc(C(=O)NCCc3ccc(S(N)(=O)=O)cc3)c(=O)n2c1	nan
	CHEMBL1356009	25905	2	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	5	2	6	0.6	Cc1ccc2ncc(C(=O)NCCc3ccc(S(N)(=O)=O)cc3)c(=O)n2c1	nan
	2140949	25906	12	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	7	1	7	4.8	COc1ccc(CCNc2nc3c(-c4cccc(F)c4)nnn3c3ccccc23)cc1OC	nan
	CHEMBL1356037	25906	12	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	7	1	7	4.8	COc1ccc(CCNc2nc3c(-c4cccc(F)c4)nnn3c3ccccc23)cc1OC	nan
	2137373	27049	15	None	-1	2	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	4	1	7	4.5	Cc1cccc(Nc2nc3c(S(=O)(=O)c4ccccc4)nnn3c3ccccc23)c1C	nan
	CHEMBL1366864	27049	15	None	-1	2	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	4	1	7	4.5	Cc1cccc(Nc2nc3c(S(=O)(=O)c4ccccc4)nnn3c3ccccc23)c1C	nan
	16027547	27337	5	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	7	1	8	4.5	CC(C)CC(=O)Nc1ccc(C(=O)OCc2cc(=O)n3nc(C4CCCCC4)sc3n2)cc1	nan
	CHEMBL1369113	27337	5	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	7	1	8	4.5	CC(C)CC(=O)Nc1ccc(C(=O)OCc2cc(=O)n3nc(C4CCCCC4)sc3n2)cc1	nan
	16009802	27670	6	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	5	1	5	4.9	CCCCNc1nc2c(-c3cccc(Br)c3)nnn2c2ccccc12	nan
	CHEMBL1371530	27670	6	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	5	1	5	4.9	CCCCNc1nc2c(-c3cccc(Br)c3)nnn2c2ccccc12	nan
	17581362	28621	8	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	436	5	1	8	3.1	COc1cccc(NC(=O)Cn2c3ccc(OC)cc3c3nc4n(c(=O)c32)CCS4)c1	nan
	CHEMBL1379032	28621	8	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	436	5	1	8	3.1	COc1cccc(NC(=O)Cn2c3ccc(OC)cc3c3nc4n(c(=O)c32)CCS4)c1	nan
	4875840	29424	6	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	6	2	4	2.5	COc1ccc(CNC(=O)CN2C(=O)NC(C)(c3cccc(Br)c3)C2=O)cc1	nan
	CHEMBL1386021	29424	6	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	6	2	4	2.5	COc1ccc(CNC(=O)CN2C(=O)NC(C)(c3cccc(Br)c3)C2=O)cc1	nan
	1486264	29791	13	None	-1	2	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	5	1	4	5.5	Cc1ccc(Sc2ccc(NC(=O)c3ccc(S(C)(=O)=O)cc3Cl)cc2)cc1	nan
	CHEMBL1388862	29791	13	None	-1	2	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	5	1	4	5.5	Cc1ccc(Sc2ccc(NC(=O)c3ccc(S(C)(=O)=O)cc3Cl)cc2)cc1	nan
	2810230	30221	6	None	2	2	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	2	1	4	3.9	O=C(Nc1nc2c(Br)cc(Br)cc2c(=O)s1)C1CCC1	nan
	CHEMBL1392489	30221	6	None	2	2	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	2	1	4	3.9	O=C(Nc1nc2c(Br)cc(Br)cc2c(=O)s1)C1CCC1	nan
	16012884	30700	6	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	356	4	0	7	3.1	COc1ccc(-n2ncc3c2ncn2nc(Cc4ccccc4)nc32)cc1	nan
	CHEMBL1397962	30700	6	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	356	4	0	7	3.1	COc1ccc(-n2ncc3c2ncn2nc(Cc4ccccc4)nc32)cc1	nan
	16021838	30730	5	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	4	1	4	5.1	CSc1ncc(C(=O)Nc2cccc(Cl)c2C)c(-c2ccccc2)n1	nan
	CHEMBL1398407	30730	5	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	4	1	4	5.1	CSc1ncc(C(=O)Nc2cccc(Cl)c2C)c(-c2ccccc2)n1	nan
	2135605	30907	13	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	351	4	1	5	4.6	c1ccc(CNc2nc3c(-c4ccccc4)nnn3c3ccccc23)cc1	nan
	CHEMBL1400053	30907	13	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	351	4	1	5	4.6	c1ccc(CNc2nc3c(-c4ccccc4)nnn3c3ccccc23)cc1	nan
	15990902	31630	6	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	373	4	2	3	5.7	Cc1cc(C)cc(Nc2cc(C(=O)NC3CCCCC3)c3ccccc3n2)c1	nan
	CHEMBL1406771	31630	6	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	373	4	2	3	5.7	Cc1cc(C)cc(Nc2cc(C(=O)NC3CCCCC3)c3ccccc3n2)c1	nan
	963186	32058	8	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	332	5	1	3	4.2	Cc1ccc(NC(=O)Cn2cc(C(=O)C3CC3)c3ccccc32)cc1	nan
	CHEMBL1410023	32058	8	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	332	5	1	3	4.2	Cc1ccc(NC(=O)Cn2cc(C(=O)C3CC3)c3ccccc32)cc1	nan
	15989908	32060	9	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	302	4	0	7	2.2	CCOC(=O)CSc1nc2ccccc2n2c(C)nnc12	nan
	CHEMBL1410062	32060	9	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	302	4	0	7	2.2	CCOC(=O)CSc1nc2ccccc2n2c(C)nnc12	nan
	15988850	32161	10	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	344	3	1	5	3.6	O=C(Nc1ccc(F)cc1F)c1cc(-c2ccc3c(c2)OCO3)on1	nan
	CHEMBL1410908	32161	10	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	344	3	1	5	3.6	O=C(Nc1ccc(F)cc1F)c1cc(-c2ccc3c(c2)OCO3)on1	nan
	1128972	32269	12	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	366	5	0	5	4.3	CCOC(=O)CSc1nc(-c2ccccc2)cc(C(F)(F)F)c1C#N	nan
	CHEMBL1411854	32269	12	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	366	5	0	5	4.3	CCOC(=O)CSc1nc(-c2ccccc2)cc(C(F)(F)F)c1C#N	nan
	3361436	34032	2	None	-1	2	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	4	4	4	4.2	Cc1ccc(NC(=S)NC(=O)c2ccccc2)cc1NC(=S)NC(=O)c1ccccc1	nan
	CHEMBL1426572	34032	2	None	-1	2	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	4	4	4	4.2	Cc1ccc(NC(=S)NC(=O)c2ccccc2)cc1NC(=S)NC(=O)c1ccccc1	nan
	1627636	34710	10	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	267	2	4	6	1.6	NN=C(S)Nc1cccc(-c2nnc(S)o2)c1	nan
	CHEMBL1432353	34710	10	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	267	2	4	6	1.6	NN=C(S)Nc1cccc(-c2nnc(S)o2)c1	nan
	8087251	34860	7	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	2	0	4	4.4	O=C(c1cc2c(s1)-c1ccccc1OC2)N1CCN(c2ccc(F)cc2)CC1	nan
	CHEMBL1433615	34860	7	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	2	0	4	4.4	O=C(c1cc2c(s1)-c1ccccc1OC2)N1CCN(c2ccc(F)cc2)CC1	nan
	16023146	35019	5	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	481	8	1	7	4.9	CCOc1ccc(CNC(=O)CSc2nnc(C)c3c(C)n(-c4ccc(Cl)cc4)nc23)cc1	nan
	CHEMBL1435835	35019	5	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	481	8	1	7	4.9	CCOc1ccc(CNC(=O)CSc2nnc(C)c3c(C)n(-c4ccc(Cl)cc4)nc23)cc1	nan
	1741544	37428	12	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	472	4	1	4	6.7	COc1ccccc1C(=O)Nc1ccc2oc(-c3cccc4c(Br)cccc34)nc2c1	nan
	CHEMBL1457270	37428	12	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	472	4	1	4	6.7	COc1ccccc1C(=O)Nc1ccc2oc(-c3cccc4c(Br)cccc34)nc2c1	nan
	2136370	37913	4	None	-1	2	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	6	1	7	3.3	CCCCNc1nc2c(S(=O)(=O)c3ccccc3)nnn2c2ccccc12	nan
	CHEMBL1461369	37913	4	None	-1	2	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	6	1	7	3.3	CCCCNc1nc2c(S(=O)(=O)c3ccccc3)nnn2c2ccccc12	nan
	3594053	39332	11	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	5	1	5	6.1	N#Cc1c(C(F)(F)F)cc(-c2cccs2)nc1SCC(=O)Nc1cccc(Cl)c1	nan
	CHEMBL1473447	39332	11	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	5	1	5	6.1	N#Cc1c(C(F)(F)F)cc(-c2cccs2)nc1SCC(=O)Nc1cccc(Cl)c1	nan
	16241285	40244	2	None	1	2	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	475	7	1	7	2.3	CN(C)C=O.CN(C)S(=O)(=O)c1cccc(NC(=O)CSc2ncnc3ccccc23)c1	nan
	CHEMBL1482781	40244	2	None	1	2	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	475	7	1	7	2.3	CN(C)C=O.CN(C)S(=O)(=O)c1cccc(NC(=O)CSc2ncnc3ccccc23)c1	nan
	1241177	41033	11	None	-1	3	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	6	0	8	2.4	c1ccc(COn2nnc3ccccc32)c(COn2nnc3ccccc32)c1	nan
	CHEMBL1489236	41033	11	None	-1	3	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	6	0	8	2.4	c1ccc(COn2nnc3ccccc32)c(COn2nnc3ccccc32)c1	nan
	16009541	41753	6	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	7	1	7	3.8	Cc1csc2nc(COc3ccc(NC(=O)COc4ccc(F)cc4)cc3)cc(=O)n12	nan
	CHEMBL1495115	41753	6	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	7	1	7	3.8	Cc1csc2nc(COc3ccc(NC(=O)COc4ccc(F)cc4)cc3)cc(=O)n12	nan
	2978485	42473	10	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	5	1	2	4.1	CCC(C)NC(=O)Cc1c(OC)ccc2cc(Br)ccc12	nan
	CHEMBL1501669	42473	10	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	5	1	2	4.1	CCC(C)NC(=O)Cc1c(OC)ccc2cc(Br)ccc12	nan
	7514097	42519	10	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	8	4	6	2.2	O=C(O)CCNc1ccc(NCCC(=O)O)c2c1C(=O)c1ccccc1C2=O	nan
	CHEMBL1502018	42519	10	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	8	4	6	2.2	O=C(O)CCNc1ccc(NCCC(=O)O)c2c1C(=O)c1ccccc1C2=O	nan
	5777938	42614	7	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	503	10	1	8	4.1	CCCOc1cccc(C2C(C(=O)c3ccc4c(c3)OCCO4)=C(O)C(=O)N2CCCn2ccnc2)c1	nan
	CHEMBL1502864	42614	7	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	503	10	1	8	4.1	CCCOc1cccc(C2C(C(=O)c3ccc4c(c3)OCCO4)=C(O)C(=O)N2CCCn2ccnc2)c1	nan
	1256983	43345	13	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	3	1	3	5.3	O=C(Nc1ccc(F)cc1)c1cc(-c2ccccn2)nc2c(Cl)cccc12	nan
	CHEMBL1509228	43345	13	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	3	1	3	5.3	O=C(Nc1ccc(F)cc1)c1cc(-c2ccccn2)nc2c(Cl)cccc12	nan
	16017574	43675	6	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	8	1	6	2.5	CCCCC(=O)Nc1nnc(S(=O)(=O)N(C)Cc2ccccc2)s1	nan
	CHEMBL1512435	43675	6	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	8	1	6	2.5	CCCCC(=O)Nc1nnc(S(=O)(=O)N(C)Cc2ccccc2)s1	nan
	15988274	43776	5	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	4	1	7	2.4	Cn1c(=O)c2sccc2n2c(CCC(=O)Nc3ccc(F)cc3)nnc12	nan
	CHEMBL1513838	43776	5	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	4	1	7	2.4	Cn1c(=O)c2sccc2n2c(CCC(=O)Nc3ccc(F)cc3)nnc12	nan
	4921215	43930	12	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	463	4	2	4	6.7	Cc1cc(C)c2c(NC(=O)c3ccccc3Cl)c(C(=O)Nc3ccc(C)c(C)c3)sc2n1	nan
	CHEMBL1516149	43930	12	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	463	4	2	4	6.7	Cc1cc(C)c2c(NC(=O)c3ccccc3Cl)c(C(=O)Nc3ccc(C)c(C)c3)sc2n1	nan
	135466071	45995	1	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	4	1	6	4.5	CCc1cc2c(s1)N1Cc3ccccc3C(C(=O)c3cccc([N+](=O)[O-])c3)=C1NC2=O	nan
	CHEMBL1535161	45995	1	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	4	1	6	4.5	CCc1cc2c(s1)N1Cc3ccccc3C(C(=O)c3cccc([N+](=O)[O-])c3)=C1NC2=O	nan
	16024942	47995	5	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	442	5	1	4	4.7	CCc1ccc(CNC(=O)C2CCN(c3nc4ccccc4nc3C(F)(F)F)CC2)cc1	nan
	CHEMBL1553067	47995	5	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	442	5	1	4	4.7	CCc1ccc(CNC(=O)C2CCN(c3nc4ccccc4nc3C(F)(F)F)CC2)cc1	nan
	16015892	48009	5	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	6	1	5	5.1	COc1ccc(-c2nc3cc(NC(=O)COc4ccc(C)c(C)c4)ccc3o2)cc1	nan
	CHEMBL1553238	48009	5	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	6	1	5	5.1	COc1ccc(-c2nc3cc(NC(=O)COc4ccc(C)c(C)c4)ccc3o2)cc1	nan
	16028168	48677	4	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	3	2	3	3.7	O=C1CC(c2ccccc2)Cc2[nH]c(=O)c(C(=O)Nc3cccc(F)c3)cc21	nan
	CHEMBL1560108	48677	4	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	3	2	3	3.7	O=C1CC(c2ccccc2)Cc2[nH]c(=O)c(C(=O)Nc3cccc(F)c3)cc21	nan
	16009056	49131	6	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	489	6	1	9	3.7	COC(=O)c1cc(NC(=O)CCc2c(C)nc3c4c(C)cc(C)nc4nn3c2C)cc(C(=O)OC)c1	nan
	CHEMBL1564251	49131	6	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	489	6	1	9	3.7	COC(=O)c1cc(NC(=O)CCc2c(C)nc3c4c(C)cc(C)nc4nn3c2C)cc(C(=O)OC)c1	nan
	626021	50073	12	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	292	3	2	4	3.0	CNC(=O)c1ccc(Nc2nnc(C)c3ccccc23)cc1	nan
	CHEMBL1572204	50073	12	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	292	3	2	4	3.0	CNC(=O)c1ccc(Nc2nnc(C)c3ccccc23)cc1	nan
	2462898	50494	7	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	308	5	0	5	3.4	COc1ccc(C(C)=O)cc1COc1ncnc2ccccc12	nan
	CHEMBL1576381	50494	7	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	308	5	0	5	3.4	COc1ccc(C(C)=O)cc1COc1ncnc2ccccc12	nan
	16024893	52134	5	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	6	1	6	4.2	COc1ccc(OC)c(CNC(=O)C2CCN(c3nc4ccccc4nc3C(F)(F)F)CC2)c1	nan
	CHEMBL1590399	52134	5	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	6	1	6	4.2	COc1ccc(OC)c(CNC(=O)C2CCN(c3nc4ccccc4nc3C(F)(F)F)CC2)c1	nan
	16010832	52165	6	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	5	1	6	3.0	Cc1ccc(NC(=O)Cn2c(=O)n(Cc3ccc(F)cc3)c(=O)c3cccnc32)cc1C	nan
	CHEMBL1590845	52165	6	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	5	1	6	3.0	Cc1ccc(NC(=O)Cn2c(=O)n(Cc3ccc(F)cc3)c(=O)c3cccnc32)cc1C	nan
	16019294	52248	11	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	4	1	8	5.2	Cc1cc(C)cc(Nc2nc3c(S(=O)(=O)c4cccc(Cl)c4)nnn3c3ccsc23)c1	nan
	CHEMBL1591857	52248	11	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	4	1	8	5.2	Cc1cc(C)cc(Nc2nc3c(S(=O)(=O)c4cccc(Cl)c4)nnn3c3ccsc23)c1	nan
	3854561	52325	15	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	5	1	4	5.5	N#Cc1c(C(F)(F)F)cc(-c2ccc(F)cc2)nc1SCC(=O)Nc1ccccc1	nan
	CHEMBL1592912	52325	15	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	5	1	4	5.5	N#Cc1c(C(F)(F)F)cc(-c2ccc(F)cc2)nc1SCC(=O)Nc1ccccc1	nan
	16018208	53227	5	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	6	1	5	3.5	Cc1c(C(=O)NCCN(C)C)oc2c1-c1nn(Cc3cccc(Cl)c3)cc1CC2	nan
	CHEMBL1601478	53227	5	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	6	1	5	3.5	Cc1c(C(=O)NCCN(C)C)oc2c1-c1nn(Cc3cccc(Cl)c3)cc1CC2	nan
	16025642	53378	5	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	550	6	1	6	5.9	Cc1cccc(C)c1NC(=O)CSc1ncc2c(n1)-c1ccc(Cl)cc1N(Cc1ccccc1)S2(=O)=O	nan
	CHEMBL1603009	53378	5	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	550	6	1	6	5.9	Cc1cccc(C)c1NC(=O)CSc1ncc2c(n1)-c1ccc(Cl)cc1N(Cc1ccccc1)S2(=O)=O	nan
	4402705	54450	11	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	4	1	8	-0.5	CN1C(=O)C(=NNc2cccc(S(=O)(=O)N3CCOCC3)c2)C(=O)N(C)C1=O	nan
	CHEMBL1611899	54450	11	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	4	1	8	-0.5	CN1C(=O)C(=NNc2cccc(S(=O)(=O)N3CCOCC3)c2)C(=O)N(C)C1=O	nan
	16018210	54464	3	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	4	1	4	5.8	Cc1ccccc1NC(=O)c1oc2c(c1C)-c1nn(Cc3cccc(Cl)c3)cc1CC2	nan
	CHEMBL1612043	54464	3	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	4	1	4	5.8	Cc1ccccc1NC(=O)c1oc2c(c1C)-c1nn(Cc3cccc(Cl)c3)cc1CC2	nan
	2795741	79470	5	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	4	1	5	5.4	Cc1nc(-c2ccc(S(=O)(=O)Nc3ccc(Br)cc3Cl)s2)cs1	nan
	CHEMBL212314	79470	5	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	4	1	5	5.4	Cc1nc(-c2ccc(S(=O)(=O)Nc3ccc(Br)cc3Cl)s2)cs1	nan
	3127110	107261	13	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	7	1	8	2.9	C/C(=N\CCCn1ccnc1)c1c(C)nn(-c2ccc([N+](=O)[O-])cc2)c1O	nan
	CHEMBL3191381	107261	13	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	7	1	8	2.9	C/C(=N\CCCn1ccnc1)c1c(C)nn(-c2ccc([N+](=O)[O-])cc2)c1O	nan
	1528721	107868	7	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	310	2	1	4	3.4	CC(=O)/N=c1\scc(-c2ccccc2)n1-c1cccc(O)c1	nan
	CHEMBL3198106	107868	7	None	-	1	Human	5.0	pPotency	=	5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	310	2	1	4	3.4	CC(=O)/N=c1\scc(-c2ccccc2)n1-c1cccc(O)c1	nan
	414	3330	29	None	-1445	5	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	6	4	9	0.5	OC[C@H]1O[C@H]([C@@H]([C@@H]1O)O)n1cnc2c1ncnc2N[C@@H](Cc1ccccc1)C	nan
	93205	3330	29	None	-1445	5	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	6	4	9	0.5	OC[C@H]1O[C@H]([C@@H]([C@@H]1O)O)n1cnc2c1ncnc2N[C@@H](Cc1ccccc1)C	nan
	CHEMBL139000	3330	29	None	-1445	5	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	6	4	9	0.5	OC[C@H]1O[C@H]([C@@H]([C@@H]1O)O)n1cnc2c1ncnc2N[C@@H](Cc1ccccc1)C	nan
	24818570	21003	0	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	5	3	4	3.8	COc1ccc(NC(=O)NNC(=O)COc2ccc3cc(Br)ccc3c2)cc1	nan
	CHEMBL1312949	21003	0	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	5	3	4	3.8	COc1ccc(NC(=O)NNC(=O)COc2ccc3cc(Br)ccc3c2)cc1	nan
	3138147	21472	14	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	6	0	5	5.7	O=C(CSc1nnc(-c2ccc(Br)cc2)n1-c1ccccc1)c1ccccc1	nan
	CHEMBL1318270	21472	14	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	6	0	5	5.7	O=C(CSc1nnc(-c2ccc(Br)cc2)n1-c1ccccc1)c1ccccc1	nan
	5428505	22863	24	None	-1	2	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	246	0	1	3	3.3	O=c1oc2cc(O)c(Cl)cc2c2ccccc12	nan
	CHEMBL1330383	22863	24	None	-1	2	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	246	0	1	3	3.3	O=c1oc2cc(O)c(Cl)cc2c2ccccc12	nan
	5913370	23805	8	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	269	6	1	5	2.8	COCCNc1oc(/C=C/c2ccccc2)nc1C#N	nan
	CHEMBL1337918	23805	8	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	269	6	1	5	2.8	COCCNc1oc(/C=C/c2ccccc2)nc1C#N	nan
	3694202	24153	19	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	4	1	6	5.2	Cc1cc(N2C(=O)C(O)=C(C(=O)c3cc4ccccc4o3)C2c2cccc(Cl)c2)no1	nan
	CHEMBL1341012	24153	19	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	4	1	6	5.2	Cc1cc(N2C(=O)C(O)=C(C(=O)c3cc4ccccc4o3)C2c2cccc(Cl)c2)no1	nan
	7190321	24528	12	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	345	4	0	7	2.6	O=C(CSc1ccc2nnc(-c3cccs3)n2n1)N1CCCC1	nan
	CHEMBL1344120	24528	12	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	345	4	0	7	2.6	O=C(CSc1ccc2nnc(-c3cccs3)n2n1)N1CCCC1	nan
	661441	24574	7	None	-2	2	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	233	3	1	3	2.8	CC(Sc1ccc2ccccc2n1)C(=O)O	nan
	CHEMBL1344527	24574	7	None	-2	2	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	233	3	1	3	2.8	CC(Sc1ccc2ccccc2n1)C(=O)O	nan
	CHEMBL1530959	24574	7	None	-2	2	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	233	3	1	3	2.8	CC(Sc1ccc2ccccc2n1)C(=O)O	nan
	16017580	25109	6	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	6	1	7	2.9	CN(Cc1ccco1)S(=O)(=O)c1nnc(NC(=O)c2ccccc2Cl)s1	nan
	CHEMBL1349094	25109	6	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	6	1	7	2.9	CN(Cc1ccco1)S(=O)(=O)c1nnc(NC(=O)c2ccccc2Cl)s1	nan
	3239502	26763	10	None	1	2	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	6	1	9	0.3	COc1ccc(-n2nnc3c(=O)n(CC(=O)NCC4CCCO4)cnc32)cc1	nan
	CHEMBL1364442	26763	10	None	1	2	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	6	1	9	0.3	COc1ccc(-n2nnc3c(=O)n(CC(=O)NCC4CCCO4)cnc32)cc1	nan
	7189863	29119	8	None	-1	2	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	3	1	7	2.9	O=C(Nc1nc2cc3c(cc2s1)OCO3)c1ccc(N2C(=O)CCC2=O)cc1	nan
	CHEMBL1383330	29119	8	None	-1	2	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	3	1	7	2.9	O=C(Nc1nc2cc3c(cc2s1)OCO3)c1ccc(N2C(=O)CCC2=O)cc1	nan
	16189478	29153	2	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	7	0	6	2.2	CCCCN(Cc1ccccc1)S(=O)(=O)c1ccc2c(c1)n(C)c(=O)c(=O)n2C	nan
	CHEMBL1383621	29153	2	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	7	0	6	2.2	CCCCN(Cc1ccccc1)S(=O)(=O)c1ccc2c(c1)n(C)c(=O)c(=O)n2C	nan
	2457625	30115	1	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	302	4	1	7	-0.0	CN(CC(=O)c1c(N)n(C)c(=O)n(C)c1=O)c1ccccc1	nan
	CHEMBL1391543	30115	1	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	302	4	1	7	-0.0	CN(CC(=O)c1c(N)n(C)c(=O)n(C)c1=O)c1ccccc1	nan
	686152	30290	38	None	-1	2	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	317	2	1	3	4.0	O=C(O)c1cc(-c2ccco2)nc2ccc(Br)cc12	nan
	CHEMBL1393131	30290	38	None	-1	2	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	317	2	1	3	4.0	O=C(O)c1cc(-c2ccco2)nc2ccc(Br)cc12	nan
	CHEMBL1576064	30290	38	None	-1	2	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	317	2	1	3	4.0	O=C(O)c1cc(-c2ccco2)nc2ccc(Br)cc12	nan
	16009717	30589	6	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	4	1	5	4.8	Fc1ccc(CNc2nc3c(-c4ccc(F)cc4)nnn3c3ccccc23)cc1	nan
	CHEMBL1396454	30589	6	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	4	1	5	4.8	Fc1ccc(CNc2nc3c(-c4ccc(F)cc4)nnn3c3ccccc23)cc1	nan
	24892133	30770	6	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	6	1	11	1.7	COc1ccccc1-c1nc(SCC(=O)Nc2cc(C)on2)c2c(=O)n(C)c(=O)n(C)c2n1	nan
	CHEMBL1398694	30770	6	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	6	1	11	1.7	COc1ccccc1-c1nc(SCC(=O)Nc2cc(C)on2)c2c(=O)n(C)c(=O)n(C)c2n1	nan
	1115170	32959	15	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	5	2	5	4.8	Cc1cccc(OCC(=O)Nc2ccc(-c3nc4cc(C)ccc4o3)c(O)c2)c1	nan
	CHEMBL1417596	32959	15	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	5	2	5	4.8	Cc1cccc(OCC(=O)Nc2ccc(-c3nc4cc(C)ccc4o3)c(O)c2)c1	nan
	15988646	35150	1	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	358	4	2	4	4.9	COc1ccccc1NC(=O)c1sc(-c2ccc(Cl)cc2)cc1N	nan
	CHEMBL1437533	35150	1	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	358	4	2	4	4.9	COc1ccccc1NC(=O)c1sc(-c2ccc(Cl)cc2)cc1N	nan
	1341231	35265	10	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	4	1	5	5.5	COc1ccc(-c2nc3cc(NC(=O)c4cc5ccccc5o4)ccc3o2)cc1	nan
	CHEMBL1438558	35265	10	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	4	1	5	5.5	COc1ccc(-c2nc3cc(NC(=O)c4cc5ccccc5o4)ccc3o2)cc1	nan
	2999623	36360	7	None	-1	3	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	9	0	8	2.9	CCN(CC)S(=O)(=O)c1ccc2c(c1)nc(CCC(=O)OCc1c(C)noc1C)n2C	nan
	CHEMBL1448461	36360	7	None	-1	3	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	9	0	8	2.9	CCN(CC)S(=O)(=O)c1ccc2c(c1)nc(CCC(=O)OCc1c(C)noc1C)n2C	nan
	2609971	38523	7	None	-1	2	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	7	1	7	3.2	CCCCn1c(SCC(=O)Nc2cc(C)on2)nc2ccccc2c1=O	nan
	CHEMBL1466287	38523	7	None	-1	2	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	7	1	7	3.2	CCCCn1c(SCC(=O)Nc2cc(C)on2)nc2ccccc2c1=O	nan
	16024828	41425	5	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	4	0	5	4.1	CC1CCN(S(=O)(=O)c2ccc3nc(N4CCN(c5ccccc5F)CC4)ccc3c2)CC1	nan
	CHEMBL1492051	41425	5	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	4	0	5	4.1	CC1CCN(S(=O)(=O)c2ccc3nc(N4CCN(c5ccccc5F)CC4)ccc3c2)CC1	nan
	3276076	42119	9	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	7	2	7	3.1	CCN(CC)S(=O)(=O)c1ccc(N2CCOCC2)c(NC(=O)c2cc(O)nc3ccccc23)c1	nan
	CHEMBL1498535	42119	9	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	7	2	7	3.1	CCN(CC)S(=O)(=O)c1ccc(N2CCOCC2)c(NC(=O)c2cc(O)nc3ccccc23)c1	nan
	3494087	43560	5	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	4	0	7	2.0	Cc1sc2ncnc(SCC(=O)N(C)C3CCS(=O)(=O)C3)c2c1C	nan
	CHEMBL1511159	43560	5	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	4	0	7	2.0	Cc1sc2ncnc(SCC(=O)N(C)C3CCS(=O)(=O)C3)c2c1C	nan
	22513173	43880	6	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	6	1	7	2.0	COc1ccc(-c2cc3c(=O)n(CC(=O)NCc4ccccc4F)ncn3n2)cc1	nan
	CHEMBL1515462	43880	6	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	6	1	7	2.0	COc1ccc(-c2cc3c(=O)n(CC(=O)NCc4ccccc4F)ncn3n2)cc1	nan
	16025349	44419	10	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	488	6	1	6	4.6	O=C(CSc1ncc2c(n1)-c1ccccc1N(Cc1ccccc1)S2(=O)=O)Nc1ccccc1	nan
	CHEMBL1520822	44419	10	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	488	6	1	6	4.6	O=C(CSc1ncc2c(n1)-c1ccccc1N(Cc1ccccc1)S2(=O)=O)Nc1ccccc1	nan
	16017252	45666	6	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	310	3	1	5	2.1	Cc1ccc(NC(=O)Cn2nc(C)n3cccc3c2=O)c(C)c1	nan
	CHEMBL1532051	45666	6	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	310	3	1	5	2.1	Cc1ccc(NC(=O)Cn2nc(C)n3cccc3c2=O)c(C)c1	nan
	659886	45970	13	None	1	3	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	6	1	5	5.4	CCc1ccccc1NC(=O)CSc1nc2c(c(-c3ccco3)c1C#N)CCCC2	nan
	CHEMBL1534846	45970	13	None	1	3	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	6	1	5	5.4	CCc1ccccc1NC(=O)CSc1nc2c(c(-c3ccco3)c1C#N)CCCC2	nan
	790785	46010	11	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	261	3	2	3	3.5	CCCc1c(C)nc2ccc(C(=O)O)cc2c1S	nan
	CHEMBL1535349	46010	11	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	261	3	2	3	3.5	CCCc1c(C)nc2ccc(C(=O)O)cc2c1S	nan
	3767937	46449	11	None	-3	2	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	5	1	6	5.6	N#Cc1c(N)nc(SCC(=O)C23CC4CC(CC(C4)C2)C3)c(C#N)c1-c1ccc(Cl)cc1	nan
	CHEMBL1539280	46449	11	None	-3	2	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	5	1	6	5.6	N#Cc1c(N)nc(SCC(=O)C23CC4CC(CC(C4)C2)C3)c(C#N)c1-c1ccc(Cl)cc1	nan
	24792845	50115	3	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	4	1	6	1.3	Cc1nn(CC(=O)NCC2CCCO2)c(=O)c2cc3ccccc3n12	nan
	CHEMBL1572639	50115	3	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	4	1	6	1.3	Cc1nn(CC(=O)NCC2CCCO2)c(=O)c2cc3ccccc3n12	nan
	319257	50133	3	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	218	4	2	2	3.0	C=C(C)C(=O)Nc1ccc(NC(C)C)cc1	nan
	CHEMBL1572793	50133	3	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	218	4	2	2	3.0	C=C(C)C(=O)Nc1ccc(NC(C)C)cc1	nan
	2100389	51421	7	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	7	1	8	2.5	O=C(COc1ncnc2scc(-c3ccccc3)c12)NCCN1C(=O)CSC1=O	nan
	CHEMBL1584231	51421	7	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	7	1	8	2.5	O=C(COc1ncnc2scc(-c3ccccc3)c12)NCCN1C(=O)CSC1=O	nan
	16019541	52163	5	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	463	4	1	8	5.1	Cc1ccc(C)c(S(=O)(=O)c2nnn3c2nc(Nc2ccc(C)c(C)c2)c2sccc23)c1	nan
	CHEMBL1590799	52163	5	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	463	4	1	8	5.1	Cc1ccc(C)c(S(=O)(=O)c2nnn3c2nc(Nc2ccc(C)c(C)c2)c2sccc23)c1	nan
	16025640	52220	5	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	566	8	1	7	5.6	CCOc1ccc(NC(=O)CSc2ncc3c(n2)-c2ccc(Cl)cc2N(Cc2ccccc2)S3(=O)=O)cc1	nan
	CHEMBL1591452	52220	5	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	566	8	1	7	5.6	CCOc1ccc(NC(=O)CSc2ncc3c(n2)-c2ccc(Cl)cc2N(Cc2ccccc2)S3(=O)=O)cc1	nan
	1189472	52675	12	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	6	1	6	2.9	CCOC(=O)c1cnc2ccc(Br)cc2c1NCCN1CCOCC1	nan
	CHEMBL1596394	52675	12	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	6	1	6	2.9	CCOC(=O)c1cnc2ccc(Br)cc2c1NCCN1CCOCC1	nan
	1115820	54414	22	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	6	1	6	5.4	COc1ccc(NC(=O)CSc2nc(-c3cccs3)cc(C(F)(F)F)c2C#N)cc1	nan
	CHEMBL1611566	54414	22	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	6	1	6	5.4	COc1ccc(NC(=O)CSc2nc(-c3cccs3)cc(C(F)(F)F)c2C#N)cc1	nan
	9581898	72242	8	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	2	1	5	2.0	Cc1cccc(C(=O)N/N=C2\CS(=O)(=O)N(C)c3ccsc32)c1	nan
	CHEMBL1992883	72242	8	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	2	1	5	2.0	Cc1cccc(C(=O)N/N=C2\CS(=O)(=O)N(C)c3ccsc32)c1	nan
	17584449	108625	7	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	5	0	7	2.6	COc1cc(C(=O)/N=C2\SC3CS(=O)(=O)CC3N2c2ccccc2)cc(OC)c1OC	nan
	CHEMBL3213657	108625	7	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	5	0	7	2.6	COc1cc(C(=O)/N=C2\SC3CS(=O)(=O)CC3N2c2ccccc2)cc(OC)c1OC	nan
	CHEMBL1411485	207022	0	None	-	1	Human	5.0	pPotency	=	5.0	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL		None	None	None		None	nan
	377	2717	47	None	-371	10	Human	5.9	pPotency	=	5.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	308	3	4	9	-1.8	CCNC(=O)[C@H]1O[C@H]([C@@H]([C@@H]1O)O)n1cnc2c1ncnc2N	nan
	425	2717	47	None	-371	10	Human	5.9	pPotency	=	5.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	308	3	4	9	-1.8	CCNC(=O)[C@H]1O[C@H]([C@@H]([C@@H]1O)O)n1cnc2c1ncnc2N	nan
	448222	2717	47	None	-371	10	Human	5.9	pPotency	=	5.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	308	3	4	9	-1.8	CCNC(=O)[C@H]1O[C@H]([C@@H]([C@@H]1O)O)n1cnc2c1ncnc2N	nan
	CHEMBL464859	2717	47	None	-371	10	Human	5.9	pPotency	=	5.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	308	3	4	9	-1.8	CCNC(=O)[C@H]1O[C@H]([C@@H]([C@@H]1O)O)n1cnc2c1ncnc2N	nan
	135415429	41065	7	None	2	3	Human	5.9	pPotency	=	5.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	477	8	1	9	4.1	CCN(CC)S(=O)(=O)c1ccc2c(c1)nc(SCc1nc(O)c3sccc3n1)n2CC	nan
	CHEMBL1489478	41065	7	None	2	3	Human	5.9	pPotency	=	5.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	477	8	1	9	4.1	CCN(CC)S(=O)(=O)c1ccc2c(c1)nc(SCc1nc(O)c3sccc3n1)n2CC	nan
	6076	106782	61	None	1	2	Human	5.9	pPotency	=	5.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	1	3	10	-0.8	Nc1ncnc2c1ncn2[C@@H]1O[C@@H]2COP(=O)(O)O[C@H]2[C@H]1O	nan
	CHEMBL1363683	106782	61	None	1	2	Human	5.9	pPotency	=	5.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	1	3	10	-0.8	Nc1ncnc2c1ncn2[C@@H]1O[C@@H]2COP(=O)(O)O[C@H]2[C@H]1O	nan
	CHEMBL316966	106782	61	None	1	2	Human	5.9	pPotency	=	5.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	1	3	10	-0.8	Nc1ncnc2c1ncn2[C@@H]1O[C@@H]2COP(=O)(O)O[C@H]2[C@H]1O	nan
	20923189	19594	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	5	0	6	2.1	COc1ccc(CN2C(=O)c3cccnc3C2=O)cc1S(=O)(=O)N1CCCCC1	nan
	CHEMBL1301594	19594	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	5	0	6	2.1	COc1ccc(CN2C(=O)c3cccnc3C2=O)cc1S(=O)(=O)N1CCCCC1	nan
	613860	20013	11	None	1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	4	1	6	2.9	Cc1noc(NS(=O)(=O)c2ccc(N3C(=O)c4ccccc4C3=O)cc2)c1C	nan
	CHEMBL1305078	20013	11	None	1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	4	1	6	2.9	Cc1noc(NS(=O)(=O)c2ccc(N3C(=O)c4ccccc4C3=O)cc2)c1C	nan
	2480606	20223	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	316	4	2	7	0.6	Cc1cccc(NCC(=O)c2c(N)n(C)c(=O)n(C)c2=O)c1C	nan
	CHEMBL1306773	20223	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	316	4	2	7	0.6	Cc1cccc(NCC(=O)c2c(N)n(C)c(=O)n(C)c2=O)c1C	nan
	224672	22507	44	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	253	3	1	3	3.1	O=C(O)CSc1ccnc2cc(Cl)ccc12	nan
	CHEMBL1327484	22507	44	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	253	3	1	3	3.1	O=C(O)CSc1ccnc2cc(Cl)ccc12	nan
	2384232	22575	27	None	-3	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	316	3	1	5	4.2	Cc1sc2ncnc(Sc3ccccc3C(=O)O)c2c1C	nan
	CHEMBL1327902	22575	27	None	-3	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	316	3	1	5	4.2	Cc1sc2ncnc(Sc3ccccc3C(=O)O)c2c1C	nan
	1442817	23049	4	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	5	1	7	3.6	Cc1nnc(NC(=O)CSc2nc(C(C)C)nc3ccccc23)s1	nan
	CHEMBL1331799	23049	4	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	5	1	7	3.6	Cc1nnc(NC(=O)CSc2nc(C(C)C)nc3ccccc23)s1	nan
	6103449	23669	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	361	2	0	3	4.0	CCN1/C(=C2\C(=O)N(C)C(=S)N2c2ccccc2)C=Cc2ccccc21	nan
	CHEMBL1336606	23669	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	361	2	0	3	4.0	CCN1/C(=C2\C(=O)N(C)C(=S)N2c2ccccc2)C=Cc2ccccc21	nan
	662886	23702	9	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	336	2	0	7	3.5	Brc1ccc(-c2nn3c(-c4ccco4)nnc3s2)o1	nan
	CHEMBL1336927	23702	9	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	336	2	0	7	3.5	Brc1ccc(-c2nn3c(-c4ccco4)nnc3s2)o1	nan
	16011044	26490	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	4	2	5	4.8	CCOC(=O)c1ccc(NC(=O)c2ccc3c(c2)NC(=O)c2ccccc2S3)cc1	nan
	CHEMBL1362040	26490	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	4	2	5	4.8	CCOC(=O)c1ccc(NC(=O)c2ccc3c(c2)NC(=O)c2ccccc2S3)cc1	nan
	826482	26611	11	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	250	1	2	6	1.8	CC1(C)Cc2c(sc3ncnc(NN)c23)CO1	nan
	CHEMBL1363060	26611	11	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	250	1	2	6	1.8	CC1(C)Cc2c(sc3ncnc(NN)c23)CO1	nan
	16024887	27018	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	6	1	5	4.6	CCOc1ccccc1CNC(=O)C1CCN(c2nc3ccccc3nc2C(F)(F)F)CC1	nan
	CHEMBL1366554	27018	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	6	1	5	4.6	CCOc1ccccc1CNC(=O)C1CCN(c2nc3ccccc3nc2C(F)(F)F)CC1	nan
	3207679	28940	4	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	5	1	5	3.9	Cc1cccc2cc(C#N)c(SCC(=O)NCc3cccs3)nc12	nan
	CHEMBL1381650	28940	4	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	5	1	5	3.9	Cc1cccc2cc(C#N)c(SCC(=O)NCc3cccs3)nc12	nan
	2445448	29431	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	4	0	7	1.4	COc1ccc(C(C)=O)cc1Cn1cnc2c(cnn2C)c1=O	nan
	CHEMBL1386075	29431	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	4	0	7	1.4	COc1ccc(C(C)=O)cc1Cn1cnc2c(cnn2C)c1=O	nan
	15988012	29789	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	6	1	8	2.6	COc1ccccc1NC(=O)CCCc1nnc2n(C)c(=O)c3sccc3n12	nan
	CHEMBL1388847	29789	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	6	1	8	2.6	COc1ccccc1NC(=O)CCCc1nnc2n(C)c(=O)c3sccc3n12	nan
	2917979	29869	13	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	5	1	9	4.0	COC(=O)c1sc(N2C(=O)C(O)=C(C(=O)c3ccc(C)o3)C2c2cccs2)nc1C	nan
	CHEMBL1389475	29869	13	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	5	1	9	4.0	COC(=O)c1sc(N2C(=O)C(O)=C(C(=O)c3ccc(C)o3)C2c2cccs2)nc1C	nan
	686152	30290	38	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	317	2	1	3	4.0	O=C(O)c1cc(-c2ccco2)nc2ccc(Br)cc12	nan
	CHEMBL1393131	30290	38	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	317	2	1	3	4.0	O=C(O)c1cc(-c2ccco2)nc2ccc(Br)cc12	nan
	CHEMBL1576064	30290	38	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	317	2	1	3	4.0	O=C(O)c1cc(-c2ccco2)nc2ccc(Br)cc12	nan
	15987889	32995	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	8	1	4	5.4	CCN(CC)CC(C)CNC(=O)c1cc(-c2ccc(Br)s2)nc2ccccc12	nan
	CHEMBL1417926	32995	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	8	1	4	5.4	CCN(CC)CC(C)CNC(=O)c1cc(-c2ccc(Br)s2)nc2ccccc12	nan
	20904552	33590	4	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	6	1	8	1.7	Cn1c(=O)c2sccc2n2c(CCCC(=O)NCc3cccnc3)nnc12	nan
	CHEMBL1422972	33590	4	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	6	1	8	1.7	Cn1c(=O)c2sccc2n2c(CCCC(=O)NCc3cccnc3)nnc12	nan
	2375468	34709	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	4	1	8	-0.2	Cn1c(N)c(C(=O)COc2ccc(C#N)cc2)c(=O)n(C)c1=O	nan
	CHEMBL1432350	34709	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	4	1	8	-0.2	Cn1c(N)c(C(=O)COc2ccc(C#N)cc2)c(=O)n(C)c1=O	nan
	16024881	34852	0	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	2	1	4	2.6	CNC(=O)C1CCN(c2nc3ccccc3nc2C(F)(F)F)CC1	nan
	CHEMBL1433473	34852	0	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	2	1	4	2.6	CNC(=O)C1CCN(c2nc3ccccc3nc2C(F)(F)F)CC1	nan
	15991045	34861	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	3	1	3	7.0	Cc1cccc(C(=O)Nc2ccc3oc(-c4cccc5c(Br)cccc45)nc3c2)c1	nan
	CHEMBL1433636	34861	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	3	1	3	7.0	Cc1cccc(C(=O)Nc2ccc3oc(-c4cccc5c(Br)cccc45)nc3c2)c1	nan
	16015278	34948	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	6	1	6	5.3	CC(=O)c1ccc(NC(=O)c2sc(-n3nc(C)c(Cc4ccccc4)c3C)nc2C)cc1	nan
	CHEMBL1434956	34948	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	6	1	6	5.3	CC(=O)c1ccc(NC(=O)c2sc(-n3nc(C)c(Cc4ccccc4)c3C)nc2C)cc1	nan
	5078950	35305	11	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	5	1	4	5.8	Cc1ccc(NC(=O)CSc2nc(-c3ccc(F)cc3)cc(C(F)(F)F)c2C#N)cc1	nan
	CHEMBL1438931	35305	11	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	5	1	4	5.8	Cc1ccc(NC(=O)CSc2nc(-c3ccc(F)cc3)cc(C(F)(F)F)c2C#N)cc1	nan
	5310383	35739	10	None	-1	3	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	5	1	8	0.3	O=C(Cn1cnc2c(nnn2-c2ccccc2)c1=O)NCC1CCCO1	nan
	CHEMBL1442757	35739	10	None	-1	3	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	5	1	8	0.3	O=C(Cn1cnc2c(nnn2-c2ccccc2)c1=O)NCC1CCCO1	nan
	948433	35752	11	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	6	1	4	3.7	COc1ccc(CNC(=O)CSc2cccc3cccnc23)cc1	nan
	CHEMBL1442938	35752	11	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	6	1	4	3.7	COc1ccc(CNC(=O)CSc2cccc3cccnc23)cc1	nan
	16019658	36013	8	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	5	1	7	3.2	Cc1ccc(NC(=O)CCCc2nnc3n(C)c(=O)c4sccc4n23)cc1C	nan
	CHEMBL1445403	36013	8	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	5	1	7	3.2	Cc1ccc(NC(=O)CCCc2nnc3n(C)c(=O)c4sccc4n23)cc1C	nan
	3208298	38590	4	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	373	5	1	7	3.7	CCc1cc2cc3c(cc2nc1SCC(=O)Nc1nccs1)OCO3	nan
	CHEMBL1466770	38590	4	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	373	5	1	7	3.7	CCc1cc2cc3c(cc2nc1SCC(=O)Nc1nccs1)OCO3	nan
	6623284	39242	10	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	5	0	7	3.0	CCS(=O)(=O)c1nc(S(=O)(=O)c2ccc(Cl)cc2)c(N2CCCC2)s1	nan
	CHEMBL1472373	39242	10	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	5	0	7	3.0	CCS(=O)(=O)c1nc(S(=O)(=O)c2ccc(Cl)cc2)c(N2CCCC2)s1	nan
	5302642	39370	12	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	463	5	2	4	6.6	CCc1ccc(NC(=O)c2sc3nc(C)c(Cl)c(C)c3c2NC(=O)c2ccccc2)cc1	nan
	CHEMBL1474011	39370	12	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	463	5	2	4	6.6	CCc1ccc(NC(=O)c2sc3nc(C)c(Cl)c(C)c3c2NC(=O)c2ccccc2)cc1	nan
	1203028	39395	11	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	4	2	8	0.0	CC(=O)Nc1cccc(NC(=O)Cn2cnc3c2c(=O)n(C)c(=O)n3C)c1	nan
	CHEMBL1474423	39395	11	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	4	2	8	0.0	CC(=O)Nc1cccc(NC(=O)Cn2cnc3c2c(=O)n(C)c(=O)n3C)c1	nan
	15988309	39726	10	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	440	4	0	8	2.1	Cn1c(=O)c2sccc2n2c(CCC(=O)N3CCN(c4ccc(F)cc4)CC3)nnc12	nan
	CHEMBL1478365	39726	10	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	440	4	0	8	2.1	Cn1c(=O)c2sccc2n2c(CCC(=O)N3CCN(c4ccc(F)cc4)CC3)nnc12	nan
	1387364	40562	10	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	4	1	7	2.2	CNS(=O)(=O)c1ccc(OC)c(-c2nnc3c4ccccc4c(C)nn23)c1	nan
	CHEMBL1485560	40562	10	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	4	1	7	2.2	CNS(=O)(=O)c1ccc(OC)c(-c2nnc3c4ccccc4c(C)nn23)c1	nan
	CHEMBL1576237	40562	10	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	4	1	7	2.2	CNS(=O)(=O)c1ccc(OC)c(-c2nnc3c4ccccc4c(C)nn23)c1	nan
	4238273	40616	8	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	4	1	6	2.9	Cn1c(SCC(=O)c2ccc3c(c2)NC(=O)CO3)nc2ccccc21	nan
	CHEMBL1485997	40616	8	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	4	1	6	2.9	Cn1c(SCC(=O)c2ccc3c(c2)NC(=O)CO3)nc2ccccc21	nan
	16025632	41513	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	4	1	6	4.3	Cc1ccc(C)c(NC(=O)CSc2ncc3c(n2)-c2ccc(Cl)cc2N(C)S3(=O)=O)c1	nan
	CHEMBL1492743	41513	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	4	1	6	4.3	Cc1ccc(C)c(NC(=O)CSc2ncc3c(n2)-c2ccc(Cl)cc2N(C)S3(=O)=O)c1	nan
	1252362	42282	15	None	-2	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	4	0	5	5.2	COc1ccc(-n2c(-c3cccc(OC)c3)nc(=S)c3c2CCCC3)cc1	nan
	CHEMBL1499911	42282	15	None	-2	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	4	0	5	5.2	COc1ccc(-n2c(-c3cccc(OC)c3)nc(=S)c3c2CCCC3)cc1	nan
	3173852	42374	6	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	5	2	4	3.8	CNC(=S)N(Cc1ccc(OC)cc1)Cc1cc2cc(C)ccc2nc1O	nan
	CHEMBL1500673	42374	6	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	5	2	4	3.8	CNC(=S)N(Cc1ccc(OC)cc1)Cc1cc2cc(C)ccc2nc1O	nan
	16189472	43009	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	7	1	6	2.1	CCN(CC)S(=O)(=O)c1ccc2c(c1)N(CC(=O)Nc1cccnc1Cl)C(=O)CO2	nan
	CHEMBL1506287	43009	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	7	1	6	2.1	CCN(CC)S(=O)(=O)c1ccc2c(c1)N(CC(=O)Nc1cccnc1Cl)C(=O)CO2	nan
	20953562	43346	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	5	1	7	2.9	COc1ccc(-c2cc3c(=O)n(CC(=O)Nc4cccc(Cl)c4)ncn3n2)cc1	nan
	CHEMBL1509249	43346	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	5	1	7	2.9	COc1ccc(-c2cc3c(=O)n(CC(=O)Nc4cccc(Cl)c4)ncn3n2)cc1	nan
	20923188	43513	4	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	7	1	6	2.4	COc1ccc(CN2C(=O)c3cccnc3C2=O)cc1S(=O)(=O)NCc1ccccc1	nan
	CHEMBL1510719	43513	4	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	7	1	6	2.4	COc1ccc(CN2C(=O)c3cccnc3C2=O)cc1S(=O)(=O)NCc1ccccc1	nan
	16025766	43785	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	491	5	1	4	5.8	Cc1cc2ccccc2n1-c1ccc(C(=O)N2CCC(C(=O)NCc3ccccc3Cl)CC2)s1	nan
	CHEMBL1514065	43785	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	491	5	1	4	5.8	Cc1cc2ccccc2n1-c1ccc(C(=O)N2CCC(C(=O)NCc3ccccc3Cl)CC2)s1	nan
	5206706	43795	13	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	4	1	4	4.8	CN(C)c1ccc(C(=O)Nc2ccc(-c3nc4ccccc4o3)cc2)cc1	nan
	CHEMBL1514233	43795	13	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	4	1	4	4.8	CN(C)c1ccc(C(=O)Nc2ccc(-c3nc4ccccc4o3)cc2)cc1	nan
	15988349	43911	0	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	463	6	1	5	4.0	Cc1ccc2c(=O)c(C(=O)c3cccc(Cl)c3)cn(CC(=O)NCc3ccc(F)cc3)c2n1	nan
	CHEMBL1515965	43911	0	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	463	6	1	5	4.0	Cc1ccc2c(=O)c(C(=O)c3cccc(Cl)c3)cn(CC(=O)NCc3ccc(F)cc3)c2n1	nan
	4458977	44137	10	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	6	1	11	0.7	CCc1nc(SCC(=O)Nc2nnc(CC)s2)c2c(=O)n(C)c(=O)n(C)c2n1	nan
	CHEMBL1518407	44137	10	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	6	1	11	0.7	CCc1nc(SCC(=O)Nc2nnc(CC)s2)c2c(=O)n(C)c(=O)n(C)c2n1	nan
	15989681	44235	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	507	7	1	7	4.1	COc1cc2c(=O)n(Cc3ccccc3Cl)c(=O)n(CC(=O)Nc3ccc(C)c(C)c3)c2cc1OC	nan
	CHEMBL1519224	44235	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	507	7	1	7	4.1	COc1cc2c(=O)n(Cc3ccccc3Cl)c(=O)n(CC(=O)Nc3ccc(C)c(C)c3)c2cc1OC	nan
	16019398	44943	8	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	3	0	9	2.6	CN1CCN(c2nc3c(S(=O)(=O)c4ccc(Cl)cc4)nnn3c3ccsc23)CC1	nan
	CHEMBL1525727	44943	8	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	3	0	9	2.6	CN1CCN(c2nc3c(S(=O)(=O)c4ccc(Cl)cc4)nnn3c3ccsc23)CC1	nan
	16009804	45292	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	5	1	7	4.3	Cc1ccc(NC(=O)Cn2c(=O)n(Cc3ccco3)c(=O)c3sc4ccccc4c32)cc1C	nan
	CHEMBL1528709	45292	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	5	1	7	4.3	Cc1ccc(NC(=O)Cn2c(=O)n(Cc3ccco3)c(=O)c3sc4ccccc4c32)cc1C	nan
	2808993	45406	5	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	4	0	5	3.4	CCc1nc2ccccc2nc1N1CCN(S(=O)(=O)c2ccc(Cl)cc2)CC1	nan
	CHEMBL1529717	45406	5	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	4	0	5	3.4	CCc1nc2ccccc2nc1N1CCN(S(=O)(=O)c2ccc(Cl)cc2)CC1	nan
	588806	46206	20	None	-1	3	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	248	4	1	4	2.5	Cc1nc(SCCC(=O)O)c2ccccc2n1	nan
	CHEMBL1537195	46206	20	None	-1	3	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	248	4	1	4	2.5	Cc1nc(SCCC(=O)O)c2ccccc2n1	nan
	2810142	46921	6	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	322	2	1	5	3.6	O=C(Nc1nc2ccsc2c(=O)s1)c1ccc(Cl)cc1	nan
	CHEMBL1543276	46921	6	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	322	2	1	5	3.6	O=C(Nc1nc2ccsc2c(=O)s1)c1ccc(Cl)cc1	nan
	2158355	47342	8	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	361	7	0	7	1.6	COCCN(CCOC)C(=O)c1cc2c(=O)n3ccccc3nc2s1	nan
	CHEMBL1546597	47342	8	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	361	7	0	7	1.6	COCCN(CCOC)C(=O)c1cc2c(=O)n3ccccc3nc2s1	nan
	1304353	48021	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	5	2	3	5.4	Cc1ccc(-c2sc(C(=O)Nc3ccc(Br)cc3)cc2CC(=O)O)cc1	nan
	CHEMBL1553391	48021	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	5	2	3	5.4	Cc1ccc(-c2sc(C(=O)Nc3ccc(Br)cc3)cc2CC(=O)O)cc1	nan
	3725217	48432	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	264	2	2	6	2.1	CC(C)C1Cc2c(sc3ncnc(NN)c23)CO1	nan
	CHEMBL1557963	48432	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	264	2	2	6	2.1	CC(C)C1Cc2c(sc3ncnc(NN)c23)CO1	nan
	16017731	49215	10	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	6	1	5	1.5	O=C(Cn1ccn(-c2ccc(F)cc2)c(=O)c1=O)NCCc1ccccc1	nan
	CHEMBL1565042	49215	10	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	6	1	5	1.5	O=C(Cn1ccn(-c2ccc(F)cc2)c(=O)c1=O)NCCc1ccccc1	nan
	7184630	51309	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	7	1	8	2.3	COc1ccccc1CNC(=O)CCCc1nnc2n(C)c(=O)c3sccc3n12	nan
	CHEMBL1583340	51309	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	7	1	8	2.3	COc1ccccc1CNC(=O)CCCc1nnc2n(C)c(=O)c3sccc3n12	nan
	24856176	51869	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	426	7	1	4	3.3	CN(CC(=O)Nc1ccccc1Cl)C(=O)COC(=O)Cc1c(F)cccc1Cl	nan
	CHEMBL1587934	51869	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	426	7	1	4	3.3	CN(CC(=O)Nc1ccccc1Cl)C(=O)COC(=O)Cc1c(F)cccc1Cl	nan
	16033298	52129	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	7	1	6	5.5	Cc1c(C(=O)NCc2ccc(OC(C)C)cc2)sc2ncnc(N(C)C3CCCCC3)c12	nan
	CHEMBL1590310	52129	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	7	1	6	5.5	Cc1c(C(=O)NCc2ccc(OC(C)C)cc2)sc2ncnc(N(C)C3CCCCC3)c12	nan
	16010771	52292	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	5	1	6	3.5	Cc1cccc(C)c1NC(=O)Cn1c(=O)n(Cc2ccccc2Cl)c(=O)c2cccnc21	nan
	CHEMBL1592455	52292	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	5	1	6	3.5	Cc1cccc(C)c1NC(=O)Cn1c(=O)n(Cc2ccccc2Cl)c(=O)c2cccnc21	nan
	16029563	52418	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	461	6	1	6	4.2	COc1ccc(NC(=O)Cn2cc(C(=O)c3ccncc3)c(=O)c3cc(C)ccc32)cc1Cl	nan
	CHEMBL1594200	52418	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	461	6	1	6	4.2	COc1ccc(NC(=O)Cn2cc(C(=O)c3ccncc3)c(=O)c3cc(C)ccc32)cc1Cl	nan
	18553656	52610	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	6	1	9	1.0	Cn1c(=O)c2c(SCC(=O)NCC3CCCO3)nc(CC(C)(C)C)nc2n(C)c1=O	nan
	CHEMBL1595812	52610	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	6	1	9	1.0	Cn1c(=O)c2c(SCC(=O)NCC3CCCO3)nc(CC(C)(C)C)nc2n(C)c1=O	nan
	773677	53241	27	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	1	1	4	3.9	Cc1ccc(-n2c(=S)[nH]c3sc4c(c3c2=O)CCC4)cc1	nan
	CHEMBL1601668	53241	27	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	1	1	4	3.9	Cc1ccc(-n2c(=S)[nH]c3sc4c(c3c2=O)CCC4)cc1	nan
	1414561	53609	28	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	306	3	1	5	4.0	C=CCn1c(=S)[nH]c2scc(-c3cccs3)c2c1=O	nan
	CHEMBL1604975	53609	28	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	306	3	1	5	4.0	C=CCn1c(=S)[nH]c2scc(-c3cccs3)c2c1=O	nan
	135693221	54695	0	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	4	2	4	4.7	Oc1ccc(-c2sc(Nc3ccccc3)n[n+]2-c2ccc(F)cc2)cc1	nan
	CHEMBL1359119	54695	0	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	4	2	4	4.7	Oc1ccc(-c2sc(Nc3ccccc3)n[n+]2-c2ccc(F)cc2)cc1	nan
	CHEMBL1615929	54695	0	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	4	2	4	4.7	Oc1ccc(-c2sc(Nc3ccccc3)n[n+]2-c2ccc(F)cc2)cc1	nan
	6476987	55060	2	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	538	3	2	4	5.3	CC1=C/C(=C(/c2cc(C)c(O)c(Br)c2)c2ccccc2S(=O)(=O)O)C=C(Br)C1=O	nan
	CHEMBL1385494	55060	2	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	538	3	2	4	5.3	CC1=C/C(=C(/c2cc(C)c(O)c(Br)c2)c2ccccc2S(=O)(=O)O)C=C(Br)C1=O	nan
	CHEMBL1618897	55060	2	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	538	3	2	4	5.3	CC1=C/C(=C(/c2cc(C)c(O)c(Br)c2)c2ccccc2S(=O)(=O)O)C=C(Br)C1=O	nan
	135502886	121162	23	None	-2	4	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	221	1	2	4	1.1	NC(=S)c1cc2ccc(O)cc2oc1=O	nan
	CHEMBL358644	121162	23	None	-2	4	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	221	1	2	4	1.1	NC(=S)c1cc2ccc(O)cc2oc1=O	nan
	24360	201653	101	None	-12	3	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	348	1	1	6	2.1	CC[C@@]1(O)C(=O)OCc2c1cc1n(c2=O)Cc2cc3ccccc3nc2-1	nan
	CHEMBL65	201653	101	None	-12	3	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	348	1	1	6	2.1	CC[C@@]1(O)C(=O)OCc2c1cc1n(c2=O)Cc2cc3ccccc3nc2-1	nan
	5359	205975	71	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	260	4	1	3	3.2	CC(C(=O)O)c1ccc(C(=O)c2cccs2)cc1	nan
	CHEMBL956	205975	71	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	260	4	1	3	3.2	CC(C(=O)O)c1ccc(C(=O)c2cccs2)cc1	nan
	2647611	52372	11	None	-	1	Human	3.9	pPotency	=	3.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	4	1	6	3.0	CC(=O)c1c(C)[nH]c(C(=O)OCc2cc(=O)n3cc(Br)ccc3n2)c1C	nan
	CHEMBL1593590	52372	11	None	-	1	Human	3.9	pPotency	=	3.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	4	1	6	3.0	CC(=O)c1c(C)[nH]c(C(=O)OCc2cc(=O)n3cc(Br)ccc3n2)c1C	nan
	126054	43687	34	None	-	1	Human	5.9	pPotency	=	5.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	576	11	7	12	-0.0	NCCNC(=O)Cc1ccc(NC(=O)Cc2ccc(Nc3ncnc4c3ncn4[C@@H]3O[C@H](CO)[C@@H](O)[C@H]3O)cc2)cc1	nan
	CHEMBL1512545	43687	34	None	-	1	Human	5.9	pPotency	=	5.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	576	11	7	12	-0.0	NCCNC(=O)Cc1ccc(NC(=O)Cc2ccc(Nc3ncnc4c3ncn4[C@@H]3O[C@H](CO)[C@@H](O)[C@H]3O)cc2)cc1	nan
	380	1261	49	None	-7413	5	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	335	4	4	9	-0.2	OC[C@H]1O[C@H]([C@@H]([C@@H]1O)O)n1cnc2c1ncnc2NC1CCCC1	nan
	657378	1261	49	None	-7413	5	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	335	4	4	9	-0.2	OC[C@H]1O[C@H]([C@@H]([C@@H]1O)O)n1cnc2c1ncnc2NC1CCCC1	nan
	CHEMBL68738	1261	49	None	-7413	5	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	335	4	4	9	-0.2	OC[C@H]1O[C@H]([C@@H]([C@@H]1O)O)n1cnc2c1ncnc2NC1CCCC1	nan
	191	13063	53	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	267	2	4	9	-2.0	Nc1ncnc2c1ncn2C1OC(CO)C(O)C1O	nan
	CHEMBL11909	13063	53	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	267	2	4	9	-2.0	Nc1ncnc2c1ncn2C1OC(CO)C(O)C1O	nan
	15988009	19511	9	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	9	1	9	2.3	COc1ccc(OC)c(CCNC(=O)CCCc2nnc3n(C)c(=O)c4sccc4n23)c1	nan
	CHEMBL1300978	19511	9	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	9	1	9	2.3	COc1ccc(OC)c(CCNC(=O)CCCc2nnc3n(C)c(=O)c4sccc4n23)c1	nan
	1246444	19558	13	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	8	2	8	2.6	COc1cc(OC)c(C(=O)Nc2ccc(S(=O)(=O)Nc3ncccn3)cc2)cc1OC	nan
	CHEMBL1301318	19558	13	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	8	2	8	2.6	COc1cc(OC)c(C(=O)Nc2ccc(S(=O)(=O)Nc3ncccn3)cc2)cc1OC	nan
	5733367	19596	15	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	482	9	1	6	3.8	CCOc1ccc(C(=O)C2=C(O)C(=O)N(CCCN3CCOCC3)C2c2ccc(F)cc2)cc1C	nan
	CHEMBL1301612	19596	15	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	482	9	1	6	3.8	CCOc1ccc(C(=O)C2=C(O)C(=O)N(CCCN3CCOCC3)C2c2ccc(F)cc2)cc1C	nan
	3207945	19636	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	346	7	1	5	2.9	CCOC(=O)CNC(=O)CSc1nc2c(C)cccc2cc1CC	nan
	CHEMBL1302034	19636	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	346	7	1	5	2.9	CCOC(=O)CNC(=O)CSc1nc2c(C)cccc2cc1CC	nan
	2978035	19862	8	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	366	4	1	4	1.3	O=C(CN1C(=O)c2ccc(Br)cc2C1=O)NCC1CCCO1	nan
	CHEMBL1303768	19862	8	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	366	4	1	4	1.3	O=C(CN1C(=O)c2ccc(Br)cc2C1=O)NCC1CCCO1	nan
	16194904	21027	9	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	5	0	9	1.6	CCOC(=O)N1CCN(C(=O)CSc2ccc3nnc(-c4ccccn4)n3n2)CC1	nan
	CHEMBL1313100	21027	9	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	5	0	9	1.6	CCOC(=O)N1CCN(C(=O)CSc2ccc3nnc(-c4ccccn4)n3n2)CC1	nan
	127136	21142	13	None	-5	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	335	5	0	2	5.0	CC[n+]1c(/C=C/C=C/c2ccc(N(C)C)cc2)sc2ccccc21	nan
	1549067	21142	13	None	-5	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	335	5	0	2	5.0	CC[n+]1c(/C=C/C=C/c2ccc(N(C)C)cc2)sc2ccccc21	nan
	1549068	21142	13	None	-5	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	335	5	0	2	5.0	CC[n+]1c(/C=C/C=C/c2ccc(N(C)C)cc2)sc2ccccc21	nan
	1549069	21142	13	None	-5	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	335	5	0	2	5.0	CC[n+]1c(/C=C/C=C/c2ccc(N(C)C)cc2)sc2ccccc21	nan
	CHEMBL1314043	21142	13	None	-5	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	335	5	0	2	5.0	CC[n+]1c(/C=C/C=C/c2ccc(N(C)C)cc2)sc2ccccc21	nan
	CHEMBL1556805	21142	13	None	-5	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	335	5	0	2	5.0	CC[n+]1c(/C=C/C=C/c2ccc(N(C)C)cc2)sc2ccccc21	nan
	3151367	21179	13	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	5	2	7	1.8	CCCn1c(=N)c(C(=O)NCC2CCCO2)cc2c(=O)n3cc(C)ccc3nc21	nan
	CHEMBL1314339	21179	13	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	5	2	7	1.8	CCCn1c(=N)c(C(=O)NCC2CCCO2)cc2c(=O)n3cc(C)ccc3nc21	nan
	16009645	21265	11	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	8	2	5	5.9	CCOc1ccc(C(=O)Nc2c(C(=O)Nc3ccccc3F)oc3ccccc23)cc1OCC	nan
	CHEMBL1315511	21265	11	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	8	2	5	5.9	CCOc1ccc(C(=O)Nc2c(C(=O)Nc3ccccc3F)oc3ccccc23)cc1OCC	nan
	16009682	21306	12	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	5	1	6	4.6	COc1cccc(CNc2nc3c(-c4ccccc4)nnn3c3ccccc23)c1	nan
	CHEMBL1315996	21306	12	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	5	1	6	4.6	COc1cccc(CNc2nc3c(-c4ccccc4)nnn3c3ccccc23)c1	nan
	16023134	21430	1	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	3	1	6	2.4	CNC(=O)C1CCCN(c2nnc(C)c3c(C)n(-c4ccccc4)nc23)C1	nan
	CHEMBL1317674	21430	1	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	3	1	6	2.4	CNC(=O)C1CCCN(c2nnc(C)c3c(C)n(-c4ccccc4)nc23)C1	nan
	16019581	21465	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	492	3	0	9	2.7	CN1CCN(c2nc3c(S(=O)(=O)c4ccc(Br)cc4)nnn3c3ccsc23)CC1	nan
	CHEMBL1318189	21465	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	492	3	0	9	2.7	CN1CCN(c2nc3c(S(=O)(=O)c4ccc(Br)cc4)nnn3c3ccsc23)CC1	nan
	16017720	21475	10	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	346	3	0	4	3.1	O=c1c(=O)n(-c2ccccc2)ccn1Cc1cccc(C(F)(F)F)c1	nan
	CHEMBL1318320	21475	10	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	346	3	0	4	3.1	O=c1c(=O)n(-c2ccccc2)ccn1Cc1cccc(C(F)(F)F)c1	nan
	2458272	21498	11	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	325	2	1	7	1.8	Cc1cc(C)n2nc(C(=O)Nc3ccc4c(c3)OCCO4)nc2n1	nan
	CHEMBL1318506	21498	11	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	325	2	1	7	1.8	Cc1cc(C)n2nc(C(=O)Nc3ccc4c(c3)OCCO4)nc2n1	nan
	15988341	21531	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	478	8	2	5	5.3	COc1ccc(-c2cc(C(=O)NCCc3ccccc3)c3c(-c4ccccc4)[nH]nc3n2)cc1OC	nan
	CHEMBL1318769	21531	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	478	8	2	5	5.3	COc1ccc(-c2cc(C(=O)NCCc3ccccc3)c3c(-c4ccccc4)[nH]nc3n2)cc1OC	nan
	3245692	21543	10	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	290	4	1	6	2.3	c1ccc(CCNc2nc3ccccc3n3nnnc23)cc1	nan
	CHEMBL1318873	21543	10	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	290	4	1	6	2.3	c1ccc(CCNc2nc3ccccc3n3nnnc23)cc1	nan
	16009520	21922	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	5	1	6	4.0	Cc1csc2nc(COc3ccc(NC(=O)c4ccccc4F)cc3)cc(=O)n12	nan
	CHEMBL1322132	21922	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	5	1	6	4.0	Cc1csc2nc(COc3ccc(NC(=O)c4ccccc4F)cc3)cc(=O)n12	nan
	1003845	21954	15	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	4	2	5	5.3	COc1cccc(-c2ccc3c(N)c(C(=O)Nc4ccc(C)c(F)c4)sc3n2)c1	nan
	CHEMBL1322400	21954	15	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	4	2	5	5.3	COc1cccc(-c2ccc3c(N)c(C(=O)Nc4ccc(C)c(F)c4)sc3n2)c1	nan
	1021427	22458	12	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	4	2	4	4.5	Cn1nc(C(=O)Nc2ccc(Br)cc2)cc1C(=O)Nc1ccc(Br)cc1	nan
	CHEMBL1327019	22458	12	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	4	2	4	4.5	Cn1nc(C(=O)Nc2ccc(Br)cc2)cc1C(=O)Nc1ccc(Br)cc1	nan
	1386649	23262	11	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	502	5	1	5	4.2	O=C(O)CCC(=O)N1CCN(c2nc(-c3ccccc3Cl)c3cc(Br)ccc3n2)CC1	nan
	1386650	23262	11	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	502	5	1	5	4.2	O=C(O)CCC(=O)N1CCN(c2nc(-c3ccccc3Cl)c3cc(Br)ccc3n2)CC1	nan
	CHEMBL1333441	23262	11	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	502	5	1	5	4.2	O=C(O)CCC(=O)N1CCN(c2nc(-c3ccccc3Cl)c3cc(Br)ccc3n2)CC1	nan
	24503354	23408	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	334	4	1	3	2.5	O=C(c1ccc(S(=O)(=O)Nc2ccccc2F)cc1)N1CCC1	nan
	CHEMBL1334480	23408	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	334	4	1	3	2.5	O=C(c1ccc(S(=O)(=O)Nc2ccccc2F)cc1)N1CCC1	nan
	15988003	23497	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	5	1	7	2.9	Cn1c(=O)c2sccc2n2c(CCCC(=O)Nc3ccc(F)c(F)c3)nnc12	nan
	CHEMBL1335235	23497	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	5	1	7	2.9	Cn1c(=O)c2sccc2n2c(CCCC(=O)Nc3ccc(F)c(F)c3)nnc12	nan
	135416637	23884	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	490	5	2	7	5.8	Cc1ccc(C)c(NC(=O)CSc2nc(O)c3c(C(F)(F)F)cc(-c4cccs4)nc3n2)c1	nan
	CHEMBL1338446	23884	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	490	5	2	7	5.8	Cc1ccc(C)c(NC(=O)CSc2nc(O)c3c(C(F)(F)F)cc(-c4cccs4)nc3n2)c1	nan
	1023823	24127	9	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	4	2	4	3.3	NS(=O)(=O)c1c(Sc2ccccc2C(=O)O)ccc2ccccc12	nan
	CHEMBL1340736	24127	9	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	4	2	4	3.3	NS(=O)(=O)c1c(Sc2ccccc2C(=O)O)ccc2ccccc12	nan
	3420063	24278	9	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	7	2	7	3.4	COc1ccc(C(=O)Nc2ccc(S(=O)(=O)Nc3onc(C)c3C)cc2)c(OC)c1	nan
	CHEMBL1342030	24278	9	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	7	2	7	3.4	COc1ccc(C(=O)Nc2ccc(S(=O)(=O)Nc3onc(C)c3C)cc2)c(OC)c1	nan
	2023917	24854	9	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	4	3	4	4.5	O=C(NC(=S)Nc1ccccc1C(=O)O)c1ccc(-c2ccc(Br)cc2)o1	nan
	CHEMBL1346887	24854	9	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	4	3	4	4.5	O=C(NC(=S)Nc1ccccc1C(=O)O)c1ccc(-c2ccc(Br)cc2)o1	nan
	6145649	24944	8	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	7	1	6	2.9	N#Cc1nc(/C=C/c2ccccc2)oc1NCCCN1CCOCC1	nan
	CHEMBL1347564	24944	8	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	7	1	6	2.9	N#Cc1nc(/C=C/c2ccccc2)oc1NCCCN1CCOCC1	nan
	3099832	25003	12	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	309	4	1	4	3.7	Cc1ccc(C(=O)Nc2nnc(Cc3ccccc3)s2)cc1	nan
	CHEMBL1348101	25003	12	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	309	4	1	4	3.7	Cc1ccc(C(=O)Nc2nnc(Cc3ccccc3)s2)cc1	nan
	16033268	25851	0	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	5	1	5	5.0	Cc1cccc(CNC(=O)c2sc3ncnc(N(C)C4CCCCC4)c3c2C)c1	nan
	CHEMBL1355268	25851	0	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	5	1	5	5.0	Cc1cccc(CNC(=O)c2sc3ncnc(N(C)C4CCCCC4)c3c2C)c1	nan
	16004219	25910	11	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	8	1	7	4.6	Brc1ccc(-c2ccc(CNCCSc3nnnn3-c3ccccc3)o2)cc1	nan
	CHEMBL1356105	25910	11	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	8	1	7	4.6	Brc1ccc(-c2ccc(CNCCSc3nnnn3-c3ccccc3)o2)cc1	nan
	16033294	25922	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	7	1	6	5.1	CCOc1ccc(CNC(=O)c2sc3ncnc(N(C)C4CCCCC4)c3c2C)cc1	nan
	CHEMBL1356206	25922	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	7	1	6	5.1	CCOc1ccc(CNC(=O)c2sc3ncnc(N(C)C4CCCCC4)c3c2C)cc1	nan
	16018776	25985	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	400	4	1	6	4.8	Cc1cc2c(cc3c(SCC(=O)Nc4cccc(Cl)c4C)nnc(C)n32)o1	nan
	CHEMBL1357046	25985	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	400	4	1	6	4.8	Cc1cc2c(cc3c(SCC(=O)Nc4cccc(Cl)c4C)nnc(C)n32)o1	nan
	16014983	26116	9	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	332	4	1	5	4.8	CSc1nc(Nc2cccc(C)c2)c(C#N)c(-c2ccccc2)n1	nan
	CHEMBL1358814	26116	9	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	332	4	1	5	4.8	CSc1nc(Nc2cccc(C)c2)c(C#N)c(-c2ccccc2)n1	nan
	7190674	26485	10	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	398	5	1	7	3.2	O=C(CSc1ccc2nnc(-c3cccnc3)n2n1)Nc1ccc(F)cc1F	nan
	CHEMBL1361981	26485	10	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	398	5	1	7	3.2	O=C(CSc1ccc2nnc(-c3cccnc3)n2n1)Nc1ccc(F)cc1F	nan
	2138626	26569	12	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	6	2	7	3.6	Cc1ccc(-c2nnn3c2nc(NCCc2ccc(S(N)(=O)=O)cc2)c2ccccc23)cc1	nan
	CHEMBL1362650	26569	12	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	6	2	7	3.6	Cc1ccc(-c2nnn3c2nc(NCCc2ccc(S(N)(=O)=O)cc2)c2ccccc23)cc1	nan
	4152428	26823	7	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	6	1	6	5.0	CCOc1ccc(NC(=O)CSc2ncnc3c2sc2ccccc23)cc1	nan
	CHEMBL1364957	26823	7	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	6	1	6	5.0	CCOc1ccc(NC(=O)CSc2ncnc3c2sc2ccccc23)cc1	nan
	15988005	26979	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	7	1	7	2.6	Cc1ccc(CCNC(=O)CCCc2nnc3n(C)c(=O)c4sccc4n23)cc1	nan
	CHEMBL1366276	26979	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	7	1	7	2.6	Cc1ccc(CCNC(=O)CCCc2nnc3n(C)c(=O)c4sccc4n23)cc1	nan
	15996111	27071	4	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	7	1	4	4.9	CCOCCCNC(=O)c1cc(-c2ccc(Br)s2)nc2ccccc12	nan
	CHEMBL1367087	27071	4	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	7	1	4	4.9	CCOCCCNC(=O)c1cc(-c2ccc(Br)s2)nc2ccccc12	nan
	659844	27157	14	None	-11	3	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	410	9	1	8	3.9	CCCCOC(=O)CSc1nc(N)c(C#N)c(-c2ccc(OCC)cc2)c1C#N	nan
	CHEMBL1367765	27157	14	None	-11	3	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	410	9	1	8	3.9	CCCCOC(=O)CSc1nc(N)c(C#N)c(-c2ccc(OCC)cc2)c1C#N	nan
	5287091	27185	12	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	2	1	2	4.7	Cc1ccc2nc(/C(C#N)=C/c3cccc(Br)c3)[nH]c2c1	nan
	CHEMBL1367954	27185	12	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	2	1	2	4.7	Cc1ccc2nc(/C(C#N)=C/c3cccc(Br)c3)[nH]c2c1	nan
	15991106	27215	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	447	5	1	5	6.0	Cc1cccc(NC(=O)CSc2nc(-c3cccs3)cc(C(F)(F)F)c2C#N)c1C	nan
	CHEMBL1368193	27215	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	447	5	1	5	6.0	Cc1cccc(NC(=O)CSc2nc(-c3cccs3)cc(C(F)(F)F)c2C#N)c1C	nan
	3544515	27245	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	6	1	9	2.2	O=C(O)CCn1c(SCc2cc(=O)n3ccccc3n2)nc2ccsc2c1=O	nan
	CHEMBL1368416	27245	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	6	1	9	2.2	O=C(O)CCn1c(SCc2cc(=O)n3ccccc3n2)nc2ccsc2c1=O	nan
	4191572	27314	8	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	316	3	1	4	3.3	COc1ccccc1Cn1c(=S)[nH]c2ccc(F)cc2c1=O	nan
	CHEMBL1368980	27314	8	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	316	3	1	4	3.3	COc1ccccc1Cn1c(=S)[nH]c2ccc(F)cc2c1=O	nan
	2743471	28251	20	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	276	2	1	4	3.7	CSc1cc(-c2ccc(Cl)cc2)nc(O)c1C#N	nan
	CHEMBL1375507	28251	20	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	276	2	1	4	3.7	CSc1cc(-c2ccc(Cl)cc2)nc(O)c1C#N	nan
	1175821	28255	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	5	0	10	0.7	CC(C)n1c(SCC(=O)N2CCN(C(=O)c3ccco3)CC2)nc2c1c(=O)n(C)c(=O)n2C	nan
	CHEMBL1375543	28255	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	5	0	10	0.7	CC(C)n1c(SCC(=O)N2CCN(C(=O)c3ccco3)CC2)nc2c1c(=O)n(C)c(=O)n2C	nan
	3241220	28293	7	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	4	1	6	1.4	O=C(Cn1cnc2c(oc3ccccc32)c1=O)NCC1CCCO1	nan
	CHEMBL1375857	28293	7	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	4	1	6	1.4	O=C(Cn1cnc2c(oc3ccccc32)c1=O)NCC1CCCO1	nan
	5733045	28549	12	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	5	1	5	4.5	COc1ccc(C(=O)C2=C(O)C(=O)N(c3ccccn3)C2c2cccc(Cl)c2)cc1	nan
	CHEMBL1378340	28549	12	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	5	1	5	4.5	COc1ccc(C(=O)C2=C(O)C(=O)N(c3ccccn3)C2c2cccc(Cl)c2)cc1	nan
	3746307	29072	25	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	280	1	1	5	3.4	Cn1c(=S)[nH]c2scc(-c3cccs3)c2c1=O	nan
	CHEMBL1382865	29072	25	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	280	1	1	5	3.4	Cn1c(=S)[nH]c2scc(-c3cccs3)c2c1=O	nan
	2939274	29131	14	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	5	1	7	4.5	CC(C)c1nnc(N2C(=O)C(O)=C(C(=O)c3cccs3)C2c2ccccc2)s1	nan
	CHEMBL1383461	29131	14	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	5	1	7	4.5	CC(C)c1nnc(N2C(=O)C(O)=C(C(=O)c3cccs3)C2c2ccccc2)s1	nan
	16194976	29204	9	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	5	0	9	1.6	CCOC(=O)N1CCN(C(=O)CSc2ccc3nnc(-c4cccnc4)n3n2)CC1	nan
	CHEMBL1384046	29204	9	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	5	0	9	1.6	CCOC(=O)N1CCN(C(=O)CSc2ccc3nnc(-c4cccnc4)n3n2)CC1	nan
	15987888	29247	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	7	1	4	4.8	CCN(CC)CCNC(=O)c1cc(-c2ccc(Br)s2)nc2ccccc12	nan
	CHEMBL1384448	29247	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	7	1	4	4.8	CCN(CC)CCNC(=O)c1cc(-c2ccc(Br)s2)nc2ccccc12	nan
	2944910	29322	10	None	-3	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	400	5	1	6	4.2	O=C(C1=C(O)C(=O)N(Cc2ccco2)C1c1cccnc1)c1cc2ccccc2o1	nan
	CHEMBL1385074	29322	10	None	-3	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	400	5	1	6	4.2	O=C(C1=C(O)C(=O)N(Cc2ccco2)C1c1cccnc1)c1cc2ccccc2o1	nan
	1928929	29573	12	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	3	2	7	5.5	Nc1c(C(=O)Nc2nc3ccccc3s2)sc2nc(-c3cccs3)ccc12	nan
	CHEMBL1387110	29573	12	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	3	2	7	5.5	Nc1c(C(=O)Nc2nc3ccccc3s2)sc2nc(-c3cccs3)ccc12	nan
	2237376	29595	17	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	6	2	8	3.0	CSc1ncc(Cl)c(C(=O)Nc2ccc(S(=O)(=O)Nc3nccc(C)n3)cc2)n1	nan
	CHEMBL1387290	29595	17	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	6	2	8	3.0	CSc1ncc(Cl)c(C(=O)Nc2ccc(S(=O)(=O)Nc3nccc(C)n3)cc2)n1	nan
	2779879	29979	28	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	296	3	1	3	4.1	Cc1c(C(=O)c2ccccc2C(=O)O)sc2ccccc12	nan
	CHEMBL1390399	29979	28	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	296	3	1	3	4.1	Cc1c(C(=O)c2ccccc2C(=O)O)sc2ccccc12	nan
	5088202	30476	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	4	2	5	5.1	COc1ccc(-c2ccc3c(N)c(C(=O)Nc4cccc(C)c4)sc3n2)cc1	nan
	CHEMBL1394959	30476	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	4	2	5	5.1	COc1ccc(-c2ccc3c(N)c(C(=O)Nc4cccc(C)c4)sc3n2)cc1	nan
	16018778	30570	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	3	0	5	5.0	Cc1cc2c(cc3c(SCc4ccc(Cl)cc4)nnc(C)n32)o1	nan
	CHEMBL1396136	30570	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	3	0	5	5.0	Cc1cc2c(cc3c(SCc4ccc(Cl)cc4)nnc(C)n32)o1	nan
	15987656	30634	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	515	12	1	6	5.8	CCOc1ccc(CCNC(=O)CSc2nc3ccccc3nc2Cc2ccc(C)cc2)cc1OCC	nan
	CHEMBL1397047	30634	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	515	12	1	6	5.8	CCOc1ccc(CCNC(=O)CSc2nc3ccccc3nc2Cc2ccc(C)cc2)cc1OCC	nan
	16018052	30656	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	6	1	4	3.8	Cc1cccc(CNC(=O)CCCn2c(=O)c3cccn3c3ccc(F)cc32)c1	nan
	CHEMBL1397347	30656	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	6	1	4	3.8	Cc1cccc(CNC(=O)CCCn2c(=O)c3cccn3c3ccc(F)cc32)c1	nan
	15987604	30675	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	6	2	4	6.3	Cc1ccc(OCC(=O)Nc2ccc3nc(Nc4cccc(Cl)c4)cc(C)c3c2)cc1	nan
	CHEMBL1397611	30675	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	6	2	4	6.3	Cc1ccc(OCC(=O)Nc2ccc3nc(Nc4cccc(Cl)c4)cc(C)c3c2)cc1	nan
	866239	30728	10	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	1	1	4	2.9	Cc1ccc(-n2c(=O)[nH]c3sc4c(c3c2=O)CCCC4)cc1	nan
	CHEMBL1398397	30728	10	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	1	1	4	2.9	Cc1ccc(-n2c(=O)[nH]c3sc4c(c3c2=O)CCCC4)cc1	nan
	15990870	30885	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	4	2	3	5.3	Cc1ccc(C)c(Nc2cc(C(=O)NC3CCCC3)c3ccccc3n2)c1	nan
	CHEMBL1399859	30885	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	4	2	3	5.3	Cc1ccc(C)c(Nc2cc(C(=O)NC3CCCC3)c3ccccc3n2)c1	nan
	20904142	30988	4	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	6	0	9	1.3	COc1ccc(N2CCN(C(=O)CCc3nnc4ccc(N5CCOCC5)nn34)CC2)cc1	nan
	CHEMBL1400806	30988	4	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	6	0	9	1.3	COc1ccc(N2CCN(C(=O)CCc3nnc4ccc(N5CCOCC5)nn34)CC2)cc1	nan
	2859630	31791	19	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	5	1	5	0.9	O=C(CN1C(=O)c2cccc3cccc(c23)C1=O)NCCN1CCOCC1	nan
	CHEMBL1408014	31791	19	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	5	1	5	0.9	O=C(CN1C(=O)c2cccc3cccc(c23)C1=O)NCCN1CCOCC1	nan
	22553366	31840	0	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	4	0	7	1.5	CCOC(=O)C1CCN(C(=O)Cn2c(=O)c3cccn3c3cccnc32)CC1	nan
	CHEMBL1408318	31840	0	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	4	0	7	1.5	CCOC(=O)C1CCN(C(=O)Cn2c(=O)c3cccn3c3cccnc32)CC1	nan
	2911470	32512	15	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	423	7	1	8	3.8	C=CCOc1ccc(C2C(C(=O)c3ccco3)=C(O)C(=O)N2c2nnc(C)s2)cc1	nan
	CHEMBL1413736	32512	15	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	423	7	1	8	3.8	C=CCOc1ccc(C2C(C(=O)c3ccco3)=C(O)C(=O)N2c2nnc(C)s2)cc1	nan
	663378	32537	8	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	255	3	0	5	3.4	N#CCCSc1ncnc2c1oc1ccccc12	nan
	CHEMBL1413946	32537	8	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	255	3	0	5	3.4	N#CCCSc1ncnc2c1oc1ccccc12	nan
	1175547	32622	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	8	1	9	2.6	COc1cc(OC)cc(-n2nnnc2SCC(=O)Nc2ccc(C(C)=O)cc2)c1	nan
	CHEMBL1414657	32622	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	8	1	9	2.6	COc1cc(OC)cc(-n2nnnc2SCC(=O)Nc2ccc(C(C)=O)cc2)c1	nan
	2152512	32646	9	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	498	6	0	9	3.2	CCOC(=O)c1cc2c(=O)n3ccccc3nc2n(Cc2ccco2)/c1=N\C(=O)c1ccccc1OC	nan
	CHEMBL1414820	32646	9	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	498	6	0	9	3.2	CCOC(=O)c1cc2c(=O)n3ccccc3nc2n(Cc2ccco2)/c1=N\C(=O)c1ccccc1OC	nan
	16033750	32772	10	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	440	4	0	3	5.8	CC(C)c1ccc(N2C(=O)N(Cc3ccccc3Cl)c3ccccc3S2(=O)=O)cc1	nan
	CHEMBL1416012	32772	10	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	440	4	0	3	5.8	CC(C)c1ccc(N2C(=O)N(Cc3ccccc3Cl)c3ccccc3S2(=O)=O)cc1	nan
	1138440	32811	4	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	8	0	10	1.8	CCCn1c(SCC(=O)c2ccc(OC)c(OC)c2)nc2c1c(=O)n(C)c(=O)n2C	nan
	CHEMBL1416338	32811	4	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	8	0	10	1.8	CCCn1c(SCC(=O)c2ccc(OC)c(OC)c2)nc2c1c(=O)n(C)c(=O)n2C	nan
	135445597	32900	21	None	-5	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	249	2	1	6	2.5	CSc1nc(O)c(C#N)c(-c2cccs2)n1	nan
	CHEMBL1417116	32900	21	None	-5	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	249	2	1	6	2.5	CSc1nc(O)c(C#N)c(-c2cccs2)n1	nan
	24892379	33060	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	475	6	1	9	1.7	Cn1c(=O)c2c(SCC(=O)NCC3CCCO3)nc(-c3ccccc3Cl)nc2n(C)c1=O	nan
	CHEMBL1418535	33060	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	475	6	1	9	1.7	Cn1c(=O)c2c(SCC(=O)NCC3CCCO3)nc(-c3ccccc3Cl)nc2n(C)c1=O	nan
	24789790	33106	2	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	400	3	0	8	0.8	CCOC(=O)N1CCN(S(=O)(=O)c2c(C)nc3scc(C)n3c2=O)CC1	nan
	CHEMBL1418824	33106	2	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	400	3	0	8	0.8	CCOC(=O)N1CCN(S(=O)(=O)c2c(C)nc3scc(C)n3c2=O)CC1	nan
	5220580	33205	14	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	358	5	1	5	4.0	CC(=O)c1sc(NC(=O)COc2ccc(Cl)cc2Cl)nc1C	nan
	CHEMBL1419730	33205	14	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	358	5	1	5	4.0	CC(=O)c1sc(NC(=O)COc2ccc(Cl)cc2Cl)nc1C	nan
	3699048	33210	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	4	2	6	3.5	Cc1ccc[n+](C2C(c3cccs3)C(C#N)=C([C-](C#N)C#N)NC2(O)c2ccccc2)c1	nan
	CHEMBL1419826	33210	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	4	2	6	3.5	Cc1ccc[n+](C2C(c3cccs3)C(C#N)=C([C-](C#N)C#N)NC2(O)c2ccccc2)c1	nan
	5790281	33343	8	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	446	10	1	7	3.7	CCCOc1ccc(C(=O)C2=C(O)C(=O)N(CCCn3ccnc3)C2c2cccnc2)cc1	nan
	CHEMBL1420847	33343	8	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	446	10	1	7	3.7	CCCOc1ccc(C(=O)C2=C(O)C(=O)N(CCCn3ccnc3)C2c2cccnc2)cc1	nan
	2974740	33351	12	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	4	1	4	4.9	Cc1cc(Br)cc2c(C(=O)NCC3CCCO3)cc(-c3cccs3)nc12	nan
	CHEMBL1420938	33351	12	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	4	1	4	4.9	Cc1cc(Br)cc2c(C(=O)NCC3CCCO3)cc(-c3cccs3)nc12	nan
	824727	33382	12	None	1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	295	2	0	4	2.2	CCOC(=O)c1cc(Br)c(=O)n2ccccc12	nan
	CHEMBL1421240	33382	12	None	1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	295	2	0	4	2.2	CCOC(=O)c1cc(Br)c(=O)n2ccccc12	nan
	6411582	33485	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	546	10	2	10	4.3	CCOC(=O)CCCCC(=O)c1[nH]c(O)nc1CSc1nnc2c3cc(Br)ccc3n(C)c2n1	nan
	CHEMBL1422131	33485	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	546	10	2	10	4.3	CCOC(=O)CCCCC(=O)c1[nH]c(O)nc1CSc1nnc2c3cc(Br)ccc3n(C)c2n1	nan
	4910054	33530	8	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	442	5	1	9	1.1	Cc1nn2c(-c3ccc(S(=O)(=O)N4CCN(CCO)CC4)o3)nnc2c2ccccc12	nan
	CHEMBL1422462	33530	8	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	442	5	1	9	1.1	Cc1nn2c(-c3ccc(S(=O)(=O)N4CCN(CCO)CC4)o3)nnc2c2ccccc12	nan
	2945586	33661	10	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	6	1	5	4.6	O=C(C1=C(O)C(=O)N(CCc2ccccc2)C1c1ccncc1)c1cc2ccccc2o1	nan
	CHEMBL1423531	33661	10	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	6	1	5	4.6	O=C(C1=C(O)C(=O)N(CCc2ccccc2)C1c1ccncc1)c1cc2ccccc2o1	nan
	614539	33698	5	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	2	1	2	4.7	O=C(Nc1cccc(C(F)(F)F)c1)c1cc(Br)cc2c1OCC2	nan
	CHEMBL1423802	33698	5	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	2	1	2	4.7	O=C(Nc1cccc(C(F)(F)F)c1)c1cc(Br)cc2c1OCC2	nan
	5928009	34017	9	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	498	5	2	9	-0.1	Cc1cccn2c(=O)c(/C=C(\C#N)C(=O)NC3CCS(=O)(=O)C3)c(N3CCC(C(N)=O)CC3)nc12	nan
	CHEMBL1426470	34017	9	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	498	5	2	9	-0.1	Cc1cccn2c(=O)c(/C=C(\C#N)C(=O)NC3CCS(=O)(=O)C3)c(N3CCC(C(N)=O)CC3)nc12	nan
	20957179	34112	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	5	0	9	0.6	CCN1CCN(C(=O)CCc2nnc3ccc(N4CCC5(CC4)OCCO5)nn23)CC1	nan
	CHEMBL1427296	34112	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	5	0	9	0.6	CCN1CCN(C(=O)CCc2nnc3ccc(N4CCC5(CC4)OCCO5)nn23)CC1	nan
	2376694	34117	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	345	4	2	8	0.5	Cn1c(N)c(C(=O)CSc2nc3ccccc3[nH]2)c(=O)n(C)c1=O	nan
	CHEMBL1427343	34117	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	345	4	2	8	0.5	Cn1c(N)c(C(=O)CSc2nc3ccccc3[nH]2)c(=O)n(C)c1=O	nan
	20970067	34342	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	497	9	1	8	2.4	COc1ccc(OC)c(CNS(=O)(=O)c2cc(CN3C(=O)c4cccnc4C3=O)ccc2OC)c1	nan
	CHEMBL1429318	34342	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	497	9	1	8	2.4	COc1ccc(OC)c(CNS(=O)(=O)c2cc(CN3C(=O)c4cccnc4C3=O)ccc2OC)c1	nan
	2950264	34361	14	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	5	1	6	2.6	O=C(CSc1ncnc2sc3c(c12)CCC3)NCC1CCCO1	nan
	CHEMBL1429474	34361	14	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	5	1	6	2.6	O=C(CSc1ncnc2sc3c(c12)CCC3)NCC1CCCO1	nan
	135436945	34856	9	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	3	2	4	5.5	Cc1ccc(C(=O)Nc2ccc(-c3nc4ccccc4s3)c(O)c2)c(C)c1	nan
	CHEMBL1433539	34856	9	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	3	2	4	5.5	Cc1ccc(C(=O)Nc2ccc(-c3nc4ccccc4s3)c(O)c2)c(C)c1	nan
	16030485	34957	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	8	1	4	4.5	CC(C)CCNC(=O)CSc1nc2ccccc2nc1Cc1ccccc1	nan
	CHEMBL1435046	34957	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	8	1	4	4.5	CC(C)CCNC(=O)CSc1nc2ccccc2nc1Cc1ccccc1	nan
	1775325	35016	16	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	4	0	6	4.3	COc1ccc(CN2COc3ccc4c(oc(=O)c5ccccc54)c3C2)cc1OC	nan
	CHEMBL1435817	35016	16	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	4	0	6	4.3	COc1ccc(CN2COc3ccc4c(oc(=O)c5ccccc54)c3C2)cc1OC	nan
	135433305	35519	1	None	-4	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	4	3	8	1.3	CNC(=O)NC(=O)CSc1nc(O)c(C#N)c(-c2cccs2)n1	nan
	CHEMBL1440872	35519	1	None	-4	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	4	3	8	1.3	CNC(=O)NC(=O)CSc1nc(O)c(C#N)c(-c2cccs2)n1	nan
	2816654	36158	11	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	279	1	1	6	1.9	CCOC(=O)N1CCc2c(sc3ncnc(O)c23)C1	nan
	CHEMBL1446784	36158	11	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	279	1	1	6	1.9	CCOC(=O)N1CCc2c(sc3ncnc(O)c23)C1	nan
	749058	36222	27	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	2	1	5	4.8	O=c1c2c(-c3cccs3)csc2[nH]c(=S)n1-c1ccccc1	nan
	CHEMBL1447245	36222	27	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	2	1	5	4.8	O=c1c2c(-c3cccs3)csc2[nH]c(=S)n1-c1ccccc1	nan
	739884	36316	77	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	246	1	1	2	3.9	O=C(O)c1sc2cc(Cl)ccc2c1Cl	nan
	CHEMBL1448105	36316	77	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	246	1	1	2	3.9	O=C(O)c1sc2cc(Cl)ccc2c1Cl	nan
	16033236	36497	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	5	1	5	5.4	Cc1c(C(=O)NCc2ccccc2Cl)sc2ncnc(N(C)C3CCCCC3)c12	nan
	CHEMBL1449453	36497	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	5	1	5	5.4	Cc1c(C(=O)NCc2ccccc2Cl)sc2ncnc(N(C)C3CCCCC3)c12	nan
	2572725	36658	6	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	4	0	6	2.8	Cc1cc(C(=O)OCC(=O)c2ccc(Br)s2)no1	nan
	CHEMBL1450791	36658	6	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	4	0	6	2.8	Cc1cc(C(=O)OCC(=O)c2ccc(Br)s2)no1	nan
	2787753	36877	16	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	258	4	3	8	0.6	CC(C)OC(=O)C(C)Nc1nnc(S)nc1O	nan
	CHEMBL1452524	36877	16	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	258	4	3	8	0.6	CC(C)OC(=O)C(C)Nc1nnc(S)nc1O	nan
	4984225	37354	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	6	1	6	1.8	CN(C)S(=O)(=O)c1ccc(C(=O)OCC(=O)Nc2cccnc2Cl)cc1	nan
	CHEMBL1456558	37354	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	6	1	6	1.8	CN(C)S(=O)(=O)c1ccc(C(=O)OCC(=O)Nc2cccnc2Cl)cc1	nan
	764734	37726	27	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	290	3	1	5	3.6	C=CCn1c(=S)[nH]c2scc(-c3ccco3)c2c1=O	nan
	CHEMBL1459809	37726	27	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	290	3	1	5	3.6	C=CCn1c(=S)[nH]c2scc(-c3ccco3)c2c1=O	nan
	2822524	37826	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	297	3	1	5	3.5	CCOC(=O)c1c(SC)nc2c(Cl)cccc2c1O	nan
	CHEMBL1460605	37826	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	297	3	1	5	3.5	CCOC(=O)c1c(SC)nc2c(Cl)cccc2c1O	nan
	2973900	38145	12	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	4	1	3	4.9	Cc1cc(Br)cc2c(C(=O)NCC3CCCO3)cc(-c3ccccc3)nc12	nan
	CHEMBL1463377	38145	12	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	4	1	3	4.9	Cc1cc(Br)cc2c(C(=O)NCC3CCCO3)cc(-c3ccccc3)nc12	nan
	5637963	38225	5	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	335	4	0	5	3.7	CCOC(=O)/C(C#N)=C/c1cc2ccccc2nc1N1CCCCC1	nan
	CHEMBL1464025	38225	5	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	335	4	0	5	3.7	CCOC(=O)/C(C#N)=C/c1cc2ccccc2nc1N1CCCCC1	nan
	1005162	38269	13	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	5	1	6	4.9	N#Cc1ccc(-c2ccc(F)cc2)nc1SCC(=O)Nc1sc2c(c1C#N)CCC2	nan
	CHEMBL1464360	38269	13	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	5	1	6	4.9	N#Cc1ccc(-c2ccc(F)cc2)nc1SCC(=O)Nc1sc2c(c1C#N)CCC2	nan
	2087618	38283	9	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	6	0	6	2.8	CCOc1cc(C=O)ccc1OCc1cc(=O)n2cc(C)ccc2n1	nan
	CHEMBL1464466	38283	9	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	6	0	6	2.8	CCOc1cc(C=O)ccc1OCc1cc(=O)n2cc(C)ccc2n1	nan
	20904553	38494	0	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	6	1	7	2.8	CC(NC(=O)CCCc1nnc2n(C)c(=O)c3sccc3n12)c1ccccc1	nan
	CHEMBL1466036	38494	0	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	6	1	7	2.8	CC(NC(=O)CCCc1nnc2n(C)c(=O)c3sccc3n12)c1ccccc1	nan
	20923124	38496	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	467	8	1	7	2.4	COc1ccc(CNS(=O)(=O)c2cc(CN3C(=O)c4cccnc4C3=O)ccc2OC)cc1	nan
	CHEMBL1466048	38496	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	467	8	1	7	2.4	COc1ccc(CNS(=O)(=O)c2cc(CN3C(=O)c4cccnc4C3=O)ccc2OC)cc1	nan
	16681736	38664	1	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	3	2	5	3.1	C1COCCO1.O=C(Nc1cccc2ccccc12)C(=O)C1C(=O)Nc2ccccc21	nan
	CHEMBL1467358	38664	1	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	3	2	5	3.1	C1COCCO1.O=C(Nc1cccc2ccccc12)C(=O)C1C(=O)Nc2ccccc21	nan
	2788467	38706	14	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	6	2	6	3.4	COc1ccccc1C(=O)Nc1ccc(S(=O)(=O)Nc2onc(C)c2C)cc1	nan
	CHEMBL1467713	38706	14	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	6	2	6	3.4	COc1ccccc1C(=O)Nc1ccc(S(=O)(=O)Nc2onc(C)c2C)cc1	nan
	4224805	38734	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	6	1	6	2.0	Cc1sc2ncn(CC(=O)NCCCC(=O)N3CCCCC3)c(=O)c2c1C	nan
	CHEMBL1468056	38734	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	6	1	6	2.0	Cc1sc2ncn(CC(=O)NCCCC(=O)N3CCCCC3)c(=O)c2c1C	nan
	22334123	38881	4	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	509	10	2	9	1.0	COc1ccc(-n2nc(C(=O)NCC(=O)NCCCN3CCOCC3)c3ccccc3c2=O)cc1OC	nan
	CHEMBL1469191	38881	4	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	509	10	2	9	1.0	COc1ccc(-n2nc(C(=O)NCC(=O)NCCCN3CCOCC3)c3ccccc3c2=O)cc1OC	nan
	5016620	39336	11	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	319	4	1	5	3.5	COc1ccc(-c2cc(C(=O)Nc3ccc(C#N)cc3)no2)cc1	nan
	CHEMBL1473482	39336	11	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	319	4	1	5	3.5	COc1ccc(-c2cc(C(=O)Nc3ccc(C#N)cc3)no2)cc1	nan
	775363	39477	15	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	3	1	7	0.7	Cc1ccc(NC(=O)Cn2cnc3c2c(=O)n(C)c(=O)n3C)cc1C	nan
	CHEMBL1475499	39477	15	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	3	1	7	0.7	Cc1ccc(NC(=O)Cn2cnc3c2c(=O)n(C)c(=O)n3C)cc1C	nan
	16009659	39536	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	471	6	1	7	4.1	COc1ccc(NC(=O)Cn2c(=O)n(Cc3ccccc3)c(=O)c3sc4ccccc4c32)cc1	nan
	CHEMBL1476377	39536	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	471	6	1	7	4.1	COc1ccc(NC(=O)Cn2c(=O)n(Cc3ccccc3)c(=O)c3sc4ccccc4c32)cc1	nan
	5730013	39584	11	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	6	2	8	4.0	CCC(Sc1nnc2c(n1)[nH]c1ccccc12)C(=O)Nc1nnc(C(C)C)s1	nan
	CHEMBL1476964	39584	11	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	6	2	8	4.0	CCC(Sc1nnc2c(n1)[nH]c1ccccc12)C(=O)Nc1nnc(C(C)C)s1	nan
	1782877	39643	14	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	465	8	2	6	3.9	COc1ccc(-c2cc3ccc(OCC(=O)NCC4CCC(C(=O)O)CC4)cc3oc2=O)cc1	nan
	CHEMBL1477517	39643	14	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	465	8	2	6	3.9	COc1ccc(-c2cc3ccc(OCC(=O)NCC4CCC(C(=O)O)CC4)cc3oc2=O)cc1	nan
	20957466	39895	1	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	8	1	7	1.7	CC1CCN(C(=O)CCc2nnc3ccc(NCCCN4CCCC4=O)nn23)CC1	nan
	CHEMBL1479770	39895	1	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	8	1	7	1.7	CC1CCN(C(=O)CCc2nnc3ccc(NCCCN4CCCC4=O)nn23)CC1	nan
	5378436	39897	12	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	1	1	6	1.4	Cn1c(=O)[nH]c2nnc(-c3ccc(Cl)c(Cl)c3)nc2c1=O	nan
	CHEMBL1479779	39897	12	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	1	1	6	1.4	Cn1c(=O)[nH]c2nnc(-c3ccc(Cl)c(Cl)c3)nc2c1=O	nan
	7207545	40704	9	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	5	1	6	4.2	Cc1nc(C)c(-c2ccc(SCC(=O)Nc3ccc(F)cc3F)nn2)s1	nan
	CHEMBL1486756	40704	9	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	5	1	6	4.2	Cc1nc(C)c(-c2ccc(SCC(=O)Nc3ccc(F)cc3F)nn2)s1	nan
	974443	40924	13	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	300	3	0	7	0.5	COc1cccc(Cn2cnc3c2c(=O)n(C)c(=O)n3C)c1	nan
	CHEMBL1488414	40924	13	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	300	3	0	7	0.5	COc1cccc(Cn2cnc3c2c(=O)n(C)c(=O)n3C)c1	nan
	250222	40963	12	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	302	2	1	3	2.9	O=C1c2ccccc2C(O)(c2ccccc2)N1c1ccncc1	nan
	CHEMBL1488698	40963	12	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	302	2	1	3	2.9	O=C1c2ccccc2C(O)(c2ccccc2)N1c1ccncc1	nan
	2158358	41013	12	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	2	0	7	1.8	CCOC(=O)N1CCN(C(=O)c2cc3c(=O)n4ccccc4nc3s2)CC1	nan
	CHEMBL1489076	41013	12	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	2	0	7	1.8	CCOC(=O)N1CCN(C(=O)c2cc3c(=O)n4ccccc4nc3s2)CC1	nan
	4000951	41147	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	5	1	11	1.8	Cn1c(N)c(C(=O)CSc2nn(-c3ccc(F)cc3)c(=S)s2)c(=O)n(C)c1=O	nan
	CHEMBL1490219	41147	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	5	1	11	1.8	Cn1c(N)c(C(=O)CSc2nn(-c3ccc(F)cc3)c(=S)s2)c(=O)n(C)c1=O	nan
	5310114	41207	4	None	1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	315	5	1	7	2.1	CCC(Sc1ccc2nnc(-c3cccnc3)n2n1)C(=O)O	nan
	CHEMBL1490578	41207	4	None	1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	315	5	1	7	2.1	CCC(Sc1ccc2nnc(-c3cccnc3)n2n1)C(=O)O	nan
	135436946	41217	9	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	4	2	5	5.6	CSc1ccc(C(=O)Nc2ccc(-c3nc4ccccc4s3)c(O)c2)cc1	nan
	CHEMBL1490651	41217	9	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	4	2	5	5.6	CSc1ccc(C(=O)Nc2ccc(-c3nc4ccccc4s3)c(O)c2)cc1	nan
	2857238	41386	8	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	6	2	3	4.3	CC(Oc1ccccc1)C(=O)Nc1ccc(NC(=O)c2ccccc2)cc1	nan
	CHEMBL1491753	41386	8	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	6	2	3	4.3	CC(Oc1ccccc1)C(=O)Nc1ccc(NC(=O)c2ccccc2)cc1	nan
	3913191	41548	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	7	2	6	2.1	CCN(CC)S(=O)(=O)c1ccc(OC)c(NC(=O)c2ccc(O)nc2)c1	nan
	CHEMBL1493081	41548	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	7	2	6	2.1	CCN(CC)S(=O)(=O)c1ccc(OC)c(NC(=O)c2ccc(O)nc2)c1	nan
	16009715	41706	11	None	1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	4	1	5	4.7	Fc1ccc(-c2nnn3c2nc(NCc2ccccc2)c2ccccc23)cc1	nan
	CHEMBL1494680	41706	11	None	1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	4	1	5	4.7	Fc1ccc(-c2nnn3c2nc(NCc2ccccc2)c2ccccc23)cc1	nan
	252183	41878	17	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	277	3	3	7	-0.3	O=C1NC(=O)C(=NNc2ccc([N+](=O)[O-])cc2)C(=O)N1	nan
	CHEMBL1496411	41878	17	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	277	3	3	7	-0.3	O=C1NC(=O)C(=NNc2ccc([N+](=O)[O-])cc2)C(=O)N1	nan
	4023603	42362	10	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	7	1	6	3.5	CCN1C(=O)C2(C(C(=O)c3cc4ccccc4o3)=C(O)C(=O)N2CCCN(C)C)c2ccccc21	nan
	4921719	42362	10	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	7	1	6	3.5	CCN1C(=O)C2(C(C(=O)c3cc4ccccc4o3)=C(O)C(=O)N2CCCN(C)C)c2ccccc21	nan
	CHEMBL1500596	42362	10	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	7	1	6	3.5	CCN1C(=O)C2(C(C(=O)c3cc4ccccc4o3)=C(O)C(=O)N2CCCN(C)C)c2ccccc21	nan
	2100904	42875	4	None	-2	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	4	1	6	3.9	Cc1nn(CCc2nn[nH]n2)c2nc(-c3ccc(Br)cc3)cc(C(F)(F)F)c12	nan
	CHEMBL1505221	42875	4	None	-2	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	4	1	6	3.9	Cc1nn(CCc2nn[nH]n2)c2nc(-c3ccc(Br)cc3)cc(C(F)(F)F)c12	nan
	1103129	43305	8	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	2	1	3	4.1	O=C(O)c1cccc(N2C(=O)c3cc4cccc(Br)c4cc3C2=O)c1	nan
	CHEMBL1508887	43305	8	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	2	1	3	4.1	O=C(O)c1cccc(N2C(=O)c3cc4cccc(Br)c4cc3C2=O)c1	nan
	15990473	43722	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	5	1	5	5.6	CCOc1ccccc1NC(=O)c1cn(C2CCCCC2)c(=O)c2c1c1ccccc1n2C	nan
	CHEMBL1513016	43722	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	5	1	5	5.6	CCOc1ccccc1NC(=O)c1cn(C2CCCCC2)c(=O)c2c1c1ccccc1n2C	nan
	3858365	43742	12	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	503	7	1	6	5.7	CCOC(=O)c1ccc(NC(=O)CSc2nc(-c3ccc(F)cc3)cc(C(F)(F)F)c2C#N)cc1	nan
	CHEMBL1513368	43742	12	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	503	7	1	6	5.7	CCOC(=O)c1ccc(NC(=O)CSc2nc(-c3ccc(F)cc3)cc(C(F)(F)F)c2C#N)cc1	nan
	16018934	43767	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	4	0	5	5.9	CCc1nnc(SCc2ccc(F)cc2Cl)c2cc3sc(C)cc3n12	nan
	CHEMBL1513698	43767	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	4	0	5	5.9	CCc1nnc(SCc2ccc(F)cc2Cl)c2cc3sc(C)cc3n12	nan
	16025722	43918	3	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	477	5	1	6	6.2	COc1cccc2c1Oc1ncccc1N(c1ccc(C(=O)NCc3ccccc3Cl)s1)C2	nan
	CHEMBL1516031	43918	3	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	477	5	1	6	6.2	COc1cccc2c1Oc1ncccc1N(c1ccc(C(=O)NCc3ccccc3Cl)s1)C2	nan
	5110655	44288	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	6	1	6	3.8	Cc1ccc(S(=O)(=O)N2CCCCC2)cc1NC(=O)CSc1ncnc2ccccc12	nan
	CHEMBL1519696	44288	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	6	1	6	3.8	Cc1ccc(S(=O)(=O)N2CCCCC2)cc1NC(=O)CSc1ncnc2ccccc12	nan
	2161841	44632	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	3	1	5	2.5	Cc1nc(SCC(=O)N2CC(=O)Nc3ccccc32)nc(C)c1C	nan
	CHEMBL1522742	44632	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	3	1	5	2.5	Cc1nc(SCC(=O)N2CC(=O)Nc3ccccc32)nc(C)c1C	nan
	1238361	44764	14	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	487	5	1	5	6.5	N#Cc1c(C(F)(F)F)cc(-c2cccs2)nc1SCC(=O)Nc1cccc(C(F)(F)F)c1	nan
	CHEMBL1523965	44764	14	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	487	5	1	5	6.5	N#Cc1c(C(F)(F)F)cc(-c2cccs2)nc1SCC(=O)Nc1cccc(C(F)(F)F)c1	nan
	20904542	44899	3	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	6	1	8	1.9	Cn1c(=O)c2sccc2n2c(CCCC(=O)NCc3ccco3)nnc12	nan
	CHEMBL1525378	44899	3	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	6	1	8	1.9	Cn1c(=O)c2sccc2n2c(CCCC(=O)NCc3ccco3)nnc12	nan
	2592811	44942	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	305	4	0	7	2.5	O=[N+]([O-])c1cc2c(c(CSc3ncccn3)c1)OCOC2	nan
	CHEMBL1525704	44942	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	305	4	0	7	2.5	O=[N+]([O-])c1cc2c(c(CSc3ncccn3)c1)OCOC2	nan
	6078768	44955	11	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	6	1	5	4.9	CCOc1ccc(C(=O)C2=C(O)C(=O)N(c3ccccn3)C2c2ccc(C)cc2)c(C)c1	nan
	CHEMBL1525799	44955	11	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	6	1	5	4.9	CCOc1ccc(C(=O)C2=C(O)C(=O)N(c3ccccn3)C2c2ccc(C)cc2)c(C)c1	nan
	1147569	44963	17	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	7	2	7	3.6	COc1cc(SC)ccc1C(=O)Nc1ccc(S(=O)(=O)Nc2nccc(C)n2)cc1	nan
	CHEMBL1525877	44963	17	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	7	2	7	3.6	COc1cc(SC)ccc1C(=O)Nc1ccc(S(=O)(=O)Nc2nccc(C)n2)cc1	nan
	4181953	45085	3	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	1	0	3	3.9	Cn1/c(=N\C(=O)c2ccc(F)cc2)sc2cc(Br)ccc21	nan
	CHEMBL1526825	45085	3	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	1	0	3	3.9	Cn1/c(=N\C(=O)c2ccc(F)cc2)sc2cc(Br)ccc21	nan
	5380406	45101	77	None	-2	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	212	0	1	3	2.7	O=c1oc2cc(O)ccc2c2ccccc12	nan
	CHEMBL1526978	45101	77	None	-2	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	212	0	1	3	2.7	O=c1oc2cc(O)ccc2c2ccccc12	nan
	5641185	45312	8	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	4	2	8	0.1	Cc1c(C(=O)NNc2cc(=O)n(C)c(=O)n2C)cccc1[N+](=O)[O-]	nan
	CHEMBL1528897	45312	8	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	4	2	8	0.1	Cc1c(C(=O)NNc2cc(=O)n(C)c(=O)n2C)cccc1[N+](=O)[O-]	nan
	1016791	45365	13	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	5	2	3	5.0	CC(C)c1ccc(OCC(=O)NC(=S)Nc2ccc3c4c(cccc24)CC3)cc1	nan
	CHEMBL1529358	45365	13	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	5	2	3	5.0	CC(C)c1ccc(OCC(=O)NC(=S)Nc2ccc3c4c(cccc24)CC3)cc1	nan
	7411882	45513	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	3	0	5	4.5	CC(=O)c1ccc(N2CCN(C(=O)c3cc4c(s3)-c3ccccc3OC4)CC2)cc1	nan
	CHEMBL1530681	45513	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	3	0	5	4.5	CC(=O)c1ccc(N2CCN(C(=O)c3cc4c(s3)-c3ccccc3OC4)CC2)cc1	nan
	16017598	45632	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	6	1	7	2.5	Cc1cccc(C(=O)Nc2nnc(S(=O)(=O)N(C)Cc3ccco3)s2)c1	nan
	CHEMBL1531718	45632	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	6	1	7	2.5	Cc1cccc(C(=O)Nc2nnc(S(=O)(=O)N(C)Cc3ccco3)s2)c1	nan
	16025817	45724	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	487	7	1	5	5.3	CCOc1ccc(CNC(=O)C2CCN(C(=O)c3ccc(-n4ccc5ccccc54)s3)CC2)cc1	nan
	CHEMBL1532579	45724	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	487	7	1	5	5.3	CCOc1ccc(CNC(=O)C2CCN(C(=O)c3ccc(-n4ccc5ccccc54)s3)CC2)cc1	nan
	20939726	45803	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	465	5	0	7	2.5	COc1ccc(CN2C(=O)c3cccnc3C2=O)cc1S(=O)(=O)N1CCOc2ccccc21	nan
	CHEMBL1533261	45803	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	465	5	0	7	2.5	COc1ccc(CN2C(=O)c3cccnc3C2=O)cc1S(=O)(=O)N1CCOc2ccccc21	nan
	16033292	45952	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	440	6	1	6	5.4	CSc1ccc(CNC(=O)c2sc3ncnc(N(C)C4CCCCC4)c3c2C)cc1	nan
	CHEMBL1534658	45952	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	440	6	1	6	5.4	CSc1ccc(CNC(=O)c2sc3ncnc(N(C)C4CCCCC4)c3c2C)cc1	nan
	135521540	46087	8	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	6	2	6	4.5	O=C(CCS(=O)(=O)c1ccccc1)Nc1ccc(-c2nc3ccccc3s2)c(O)c1	nan
	CHEMBL1536204	46087	8	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	6	2	6	4.5	O=C(CCS(=O)(=O)c1ccccc1)Nc1ccc(-c2nc3ccccc3s2)c(O)c1	nan
	2729862	46668	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	5	2	8	0.2	Cc1ccc(NCC(O)Cn2cnc3c2c(=O)n(C)c(=O)n3C)cc1	nan
	CHEMBL1541137	46668	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	5	2	8	0.2	Cc1ccc(NCC(O)Cn2cnc3c2c(=O)n(C)c(=O)n3C)cc1	nan
	2487501	46714	29	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	218	0	2	6	1.3	Oc1nc2ccccc2n2c(S)nnc12	nan
	CHEMBL1541468	46714	29	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	218	0	2	6	1.3	Oc1nc2ccccc2n2c(S)nnc12	nan
	16194809	47059	3	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	6	1	8	1.6	O=C(CSc1nnc2ccc(-c3ccccn3)nn12)NCC1CCCO1	nan
	CHEMBL1544280	47059	3	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	6	1	8	1.6	O=C(CSc1nnc2ccc(-c3ccccn3)nn12)NCC1CCCO1	nan
	1866349	47179	10	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	233	4	1	3	2.8	O=C(O)CCSc1ccc2ccccc2n1	nan
	661670	47179	10	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	233	4	1	3	2.8	O=C(O)CCSc1ccc2ccccc2n1	nan
	CHEMBL1406059	47179	10	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	233	4	1	3	2.8	O=C(O)CCSc1ccc2ccccc2n1	nan
	CHEMBL1545185	47179	10	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	233	4	1	3	2.8	O=C(O)CCSc1ccc2ccccc2n1	nan
	15988305	47976	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	5	1	7	2.5	Cn1c(=O)c2sccc2n2c(CCC(=O)NCc3ccc(Cl)cc3)nnc12	nan
	CHEMBL1552888	47976	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	5	1	7	2.5	Cn1c(=O)c2sccc2n2c(CCC(=O)NCc3ccc(Cl)cc3)nnc12	nan
	1327631	48139	10	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	7	1	5	5.1	CCc1ccc(OCC(=O)Nc2ccc3oc(-c4ccc(OC)cc4)nc3c2)cc1	nan
	CHEMBL1555206	48139	10	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	7	1	5	5.1	CCc1ccc(OCC(=O)Nc2ccc3oc(-c4ccc(OC)cc4)nc3c2)cc1	nan
	16033300	48152	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	6	1	5	5.3	CCc1ccc(CNC(=O)c2sc3ncnc(N(C)C4CCCCC4)c3c2C)cc1	nan
	CHEMBL1555399	48152	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	6	1	5	5.3	CCc1ccc(CNC(=O)c2sc3ncnc(N(C)C4CCCCC4)c3c2C)cc1	nan
	20970028	48232	0	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	5	1	5	1.7	CC(C)NS(=O)(=O)c1cc(F)ccc1CN1C(=O)c2cccnc2C1=O	nan
	CHEMBL1556192	48232	0	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	5	1	5	1.7	CC(C)NS(=O)(=O)c1cc(F)ccc1CN1C(=O)c2cccnc2C1=O	nan
	5202629	48450	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	6	1	7	2.4	Cn1cnnc1SCC(=O)Nc1cc(S(=O)(=O)N2CCCCC2)ccc1Cl	nan
	CHEMBL1558116	48450	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	6	1	7	2.4	Cn1cnnc1SCC(=O)Nc1cc(S(=O)(=O)N2CCCCC2)ccc1Cl	nan
	7411867	48749	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	2	0	4	4.3	O=C(c1cc2c(s1)-c1ccccc1OC2)N1CCN(c2ccccc2)CC1	nan
	CHEMBL1560888	48749	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	2	0	4	4.3	O=C(c1cc2c(s1)-c1ccccc1OC2)N1CCN(c2ccccc2)CC1	nan
	20923142	48935	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	6	1	6	1.6	COc1ccc(CN2C(=O)c3cccnc3C2=O)cc1S(=O)(=O)NC(C)C	nan
	CHEMBL1562552	48935	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	6	1	6	1.6	COc1ccc(CN2C(=O)c3cccnc3C2=O)cc1S(=O)(=O)NC(C)C	nan
	3505859	48937	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	8	1	8	2.3	CCN(CC)S(=O)(=O)c1ccc(C)c(NC(=O)Cn2cnc3cc([N+](=O)[O-])ccc3c2=O)c1	nan
	CHEMBL1562557	48937	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	8	1	8	2.3	CCN(CC)S(=O)(=O)c1ccc(C)c(NC(=O)Cn2cnc3cc([N+](=O)[O-])ccc3c2=O)c1	nan
	7524261	49037	3	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	5	1	7	2.6	CCS(=O)(=O)Nc1cccc(-c2ccc3nnc(-c4cccnc4)n3n2)c1	nan
	CHEMBL1563485	49037	3	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	5	1	7	2.6	CCS(=O)(=O)Nc1cccc(-c2ccc3nnc(-c4cccnc4)n3n2)c1	nan
	5389817	49207	8	None	1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	464	9	1	6	3.2	CCCOc1ccc(C(=O)C2=C(O)C(=O)N(CCCOC)C23C(=O)N(C)c2ccccc23)cc1	nan
	CHEMBL1564945	49207	8	None	1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	464	9	1	6	3.2	CCCOc1ccc(C(=O)C2=C(O)C(=O)N(CCCOC)C23C(=O)N(C)c2ccccc23)cc1	nan
	1111955	49222	12	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	6	1	6	4.1	COc1ccc(-n2nc3ccc(NC(=O)COc4ccc(C)c(C)c4)cc3n2)cc1	nan
	CHEMBL1565140	49222	12	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	6	1	6	4.1	COc1ccc(-n2nc3ccc(NC(=O)COc4ccc(C)c(C)c4)cc3n2)cc1	nan
	15988272	49553	1	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	5	0	9	2.0	COC(=O)c1ccc(OC)c(Cn2c(=O)n(-c3ccc(C)cc3)c(=O)c3c2cnn3C)c1	nan
	CHEMBL1567650	49553	1	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	5	0	9	2.0	COC(=O)c1ccc(OC)c(Cn2c(=O)n(-c3ccc(C)cc3)c(=O)c3c2cnn3C)c1	nan
	15991345	49748	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	3	0	5	5.1	CSc1ccc(C2c3c(oc4ccc(F)cc4c3=O)C(=O)N2c2ccc(C)cn2)cc1	nan
	CHEMBL1569335	49748	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	3	0	5	5.1	CSc1ccc(C2c3c(oc4ccc(F)cc4c3=O)C(=O)N2c2ccc(C)cn2)cc1	nan
	15988962	50034	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	9	1	4	5.6	CCCN(CCC)CCNC(=O)c1cc(-c2ccc(Br)s2)nc2ccccc12	nan
	CHEMBL1571921	50034	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	9	1	4	5.6	CCCN(CCC)CCNC(=O)c1cc(-c2ccc(Br)s2)nc2ccccc12	nan
	2483422	50537	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	6	1	6	1.1	Cn1c(CCC(=O)OCC(=O)NCC(F)(F)F)nc(=O)c2ccccc21	nan
	CHEMBL1576699	50537	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	6	1	6	1.1	Cn1c(CCC(=O)OCC(=O)NCC(F)(F)F)nc(=O)c2ccccc21	nan
	5070065	51012	16	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	480	8	1	8	5.1	CCCOc1cccc(C2C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2c2nc(C)c(C(C)=O)s2)c1	nan
	CHEMBL1580853	51012	16	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	480	8	1	8	5.1	CCCOc1cccc(C2C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2c2nc(C)c(C(C)=O)s2)c1	nan
	4295307	51086	16	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	5	1	7	4.5	COc1ccccc1C1C(C(=O)c2cc3ccccc3o2)=C(O)C(=O)N1c1cc(C)on1	nan
	CHEMBL1581437	51086	16	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	5	1	7	4.5	COc1ccccc1C1C(C(=O)c2cc3ccccc3o2)=C(O)C(=O)N1c1cc(C)on1	nan
	4808157	51278	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	330	5	0	8	0.5	COc1ccc(OCCn2cnc3c2c(=O)n(C)c(=O)n3C)cc1	nan
	CHEMBL1583111	51278	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	330	5	0	8	0.5	COc1ccc(OCCn2cnc3c2c(=O)n(C)c(=O)n3C)cc1	nan
	6530035	51786	3	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	488	9	1	7	2.6	CCN(CC)S(=O)(=O)c1ccc(C(=O)NCCN2C(=O)S/C(=C\c3cccnc3)C2=O)cc1	nan
	CHEMBL1587266	51786	3	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	488	9	1	7	2.6	CCN(CC)S(=O)(=O)c1ccc(C(=O)NCCN2C(=O)S/C(=C\c3cccnc3)C2=O)cc1	nan
	15988968	52189	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	482	6	1	5	5.7	COc1ccc(CNC(=O)c2cc(-c3ccc(Br)s3)nc3ccccc23)c(OC)c1	nan
	CHEMBL1591154	52189	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	482	6	1	5	5.7	COc1ccc(CNC(=O)c2cc(-c3ccc(Br)s3)nc3ccccc23)c(OC)c1	nan
	16024517	52206	10	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	6	1	5	5.0	Cc1ccc(C(=O)c2cn(CC(=O)Nc3ccc(C(C)C)cc3)c3nc(C)ccc3c2=O)cc1	nan
	CHEMBL1591352	52206	10	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	6	1	5	5.0	Cc1ccc(C(=O)c2cn(CC(=O)Nc3ccc(C(C)C)cc3)c3nc(C)ccc3c2=O)cc1	nan
	16018826	52269	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	5	1	6	4.2	CCc1cccc(NC(=O)CSc2nncn3c2cc2sccc23)c1	nan
	CHEMBL1592153	52269	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	5	1	6	4.2	CCc1cccc(NC(=O)CSc2nncn3c2cc2sccc23)c1	nan
	16010502	52349	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	2	0	4	4.4	O=C(c1cc2c(s1)-c1ccccc1OC2)N1CCN(c2ccccc2F)CC1	nan
	CHEMBL1593224	52349	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	2	0	4	4.4	O=C(c1cc2c(s1)-c1ccccc1OC2)N1CCN(c2ccccc2F)CC1	nan
	1191851	52892	10	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	7	1	5	5.0	CCc1ccccc1NC(=O)COc1ccc2oc(-c3ccc(OC)cc3)cc(=O)c2c1	nan
	CHEMBL1598484	52892	10	None	-1	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	7	1	5	5.0	CCc1ccccc1NC(=O)COc1ccc2oc(-c3ccc(OC)cc3)cc(=O)c2c1	nan
	20888741	53082	13	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	400	5	0	7	2.7	CCS(=O)(=O)c1nc(S(=O)(=O)c2ccc(C)cc2)c(N2CCCC2)s1	nan
	CHEMBL1600180	53082	13	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	400	5	0	7	2.7	CCS(=O)(=O)c1nc(S(=O)(=O)c2ccc(C)cc2)c(N2CCCC2)s1	nan
	16018860	53288	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	4	1	6	4.6	Cc1ccc(NC(=O)CSc2nnc(C)n3c2cc2sccc23)c(C)c1	nan
	CHEMBL1602197	53288	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	4	1	6	4.6	Cc1ccc(NC(=O)CSc2nnc(C)n3c2cc2sccc23)c(C)c1	nan
	135460554	53526	7	None	-2	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	291	4	1	7	2.5	CC(=O)CSc1nc(O)c(C#N)c(-c2cccs2)n1	nan
	CHEMBL1604187	53526	7	None	-2	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	291	4	1	7	2.5	CC(=O)CSc1nc(O)c(C#N)c(-c2cccs2)n1	nan
	16194880	53605	8	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	5	0	8	2.2	CCC(Sc1ccc2nnc(-c3cccnc3)n2n1)C(=O)OC	nan
	CHEMBL1604935	53605	8	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	5	0	8	2.2	CCC(Sc1ccc2nnc(-c3cccnc3)n2n1)C(=O)OC	nan
	2939815	53878	12	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	356	5	1	6	2.6	Cc1cc2ccccc2n2c(SCC(=O)NCC3CCCO3)nnc12	nan
	CHEMBL1607085	53878	12	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	356	5	1	6	2.6	Cc1cc2ccccc2n2c(SCC(=O)NCC3CCCO3)nnc12	nan
	16017570	54242	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	6	1	6	3.3	CN(Cc1ccccc1)S(=O)(=O)c1nnc(NC(=O)c2cccc(Cl)c2)s1	nan
	CHEMBL1610070	54242	6	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	6	1	6	3.3	CN(Cc1ccccc1)S(=O)(=O)c1nnc(NC(=O)c2cccc(Cl)c2)s1	nan
	7184628	54346	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	7	1	7	2.3	Cn1c(=O)c2sccc2n2c(CCCC(=O)NCCc3ccccc3)nnc12	nan
	CHEMBL1611000	54346	7	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	7	1	7	2.3	Cn1c(=O)c2sccc2n2c(CCCC(=O)NCCc3ccccc3)nnc12	nan
	20957175	54638	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	400	4	0	8	1.4	O=C(CCc1nnc2ccc(N3CCC4(CC3)OCCO4)nn12)N1CCCCC1	nan
	CHEMBL1613668	54638	5	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	400	4	0	8	1.4	O=C(CCc1nnc2ccc(N3CCC4(CC3)OCCO4)nn12)N1CCCCC1	nan
	11077	54751	32	None	-4	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	229	0	1	4	1.2	O=c1ccc2[n+]([O-])c3ccc(O)cc3oc-2c1	nan
	CHEMBL1353221	54751	32	None	-4	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	229	0	1	4	1.2	O=c1ccc2[n+]([O-])c3ccc(O)cc3oc-2c1	nan
	CHEMBL1616414	54751	32	None	-4	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	229	0	1	4	1.2	O=c1ccc2[n+]([O-])c3ccc(O)cc3oc-2c1	nan
	686692	54771	10	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	334	4	1	8	-0.5	Cn1c(=O)c2c(ncn2CCCC(=N)N2CCOCC2)n(C)c1=O	nan
	CHEMBL1309275	54771	10	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	334	4	1	8	-0.5	Cn1c(=O)c2c(ncn2CCCC(=N)N2CCOCC2)n(C)c1=O	nan
	CHEMBL1616571	54771	10	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	334	4	1	8	-0.5	Cn1c(=O)c2c(ncn2CCCC(=N)N2CCOCC2)n(C)c1=O	nan
	694704	55057	51	None	-2	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	2	1	3	3.8	O=C(O)c1cc(-c2cccnc2)nc2ccc(Br)cc12	nan
	CHEMBL1373811	55057	51	None	-2	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	2	1	3	3.8	O=C(O)c1cc(-c2cccnc2)nc2ccc(Br)cc12	nan
	CHEMBL1618856	55057	51	None	-2	2	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	2	1	3	3.8	O=C(O)c1cc(-c2cccnc2)nc2ccc(Br)cc12	nan
	3246720	55375	2	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	3	3	8	1.0	CC[C@@]1(O)C(=O)OCc2c1cc1n(c2=O)Cc2cc3c(NC(=O)CN)cccc3nc2-1	nan
	CHEMBL1445386	55375	2	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	3	3	8	1.0	CC[C@@]1(O)C(=O)OCc2c1cc1n(c2=O)Cc2cc3c(NC(=O)CN)cccc3nc2-1	nan
	CHEMBL1621717	55375	2	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	3	3	8	1.0	CC[C@@]1(O)C(=O)OCc2c1cc1n(c2=O)Cc2cc3c(NC(=O)CN)cccc3nc2-1	nan
	135439671	71857	9	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	5	2	9	0.1	Cn1c(=O)c2c(ncn2CC(=O)N/N=C/c2c[nH]nc2-c2ccc(F)cc2)n(C)c1=O	nan
	CHEMBL1980641	71857	9	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	5	2	9	0.1	Cn1c(=O)c2c(ncn2CC(=O)N/N=C/c2c[nH]nc2-c2ccc(F)cc2)n(C)c1=O	nan
	6187702	72428	4	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	4	1	6	2.6	C/C(=N\NC(=O)c1c(C)nc2ccccn12)c1ccc(N2CCOCC2)cc1	nan
	CHEMBL1999641	72428	4	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	4	1	6	2.6	C/C(=N\NC(=O)c1c(C)nc2ccccn12)c1ccc(N2CCOCC2)cc1	nan
	2058613	107882	11	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	498	6	0	9	3.2	CCOC(=O)c1cc2c(=O)n3ccccc3nc2n(Cc2ccco2)/c1=N/C(=O)c1cccc(OC)c1	nan
	CHEMBL3198223	107882	11	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	498	6	0	9	3.2	CCOC(=O)c1cc2c(=O)n3ccccc3nc2n(Cc2ccco2)/c1=N/C(=O)c1cccc(OC)c1	nan
	2947382	175742	12	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	356	7	1	5	1.8	CCN(CC)S(=O)(=O)c1ccc(OC)c(NC(=O)C2CCCO2)c1	nan
	CHEMBL459529	175742	12	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	356	7	1	5	1.8	CCN(CC)S(=O)(=O)c1ccc(OC)c(NC(=O)C2CCCO2)c1	nan
	3151452	197903	16	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	7	2	8	1.8	COCCCn1c(=N)c(C(=O)NCc2cccnc2)cc2c(=O)n3cccc(C)c3nc21	nan
	CHEMBL592554	197903	16	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	7	2	8	1.8	COCCCn1c(=N)c(C(=O)NCc2cccnc2)cc2c(=O)n3cccc(C)c3nc21	nan
	3159270	199919	15	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	319	3	0	5	2.6	Cc1c2c(n3c(nc4ccccc43)c1C#N)N(CCN(C)C)CC2	nan
	CHEMBL605753	199919	15	None	-	1	Human	4.9	pPotency	=	4.9	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	319	3	0	5	2.6	Cc1c2c(n3c(nc4ccccc43)c1C#N)N(CCN(C)C)CC2	nan
	9687	184753	22	None	1	2	Human	6.8	pPotency	=	6.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	7	2	11	1.7	CCCC(=O)Nc1ncnc2c1ncn2[C@@H]1O[C@@H]2COP(=O)(O)O[C@H]2[C@H]1OC(=O)CCC	nan
	CHEMBL1522836	184753	22	None	1	2	Human	6.8	pPotency	=	6.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	7	2	11	1.7	CCCC(=O)Nc1ncnc2c1ncn2[C@@H]1O[C@@H]2COP(=O)(O)O[C@H]2[C@H]1OC(=O)CCC	nan
	CHEMBL485980	184753	22	None	1	2	Human	6.8	pPotency	=	6.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	7	2	11	1.7	CCCC(=O)Nc1ncnc2c1ncn2[C@@H]1O[C@@H]2COP(=O)(O)O[C@H]2[C@H]1OC(=O)CCC	nan
	16682183	25142	1	None	-	1	Human	5.8	pPotency	=	5.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	2	0	5	4.6	CC(C)C(=O)N1CCC2(CC1)Oc1ccc(F)cc1C(=O)C21CC(c2ccc(Cl)cc2)=NO1	nan
	CHEMBL1349353	25142	1	None	-	1	Human	5.8	pPotency	=	5.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	2	0	5	4.6	CC(C)C(=O)N1CCC2(CC1)Oc1ccc(F)cc1C(=O)C21CC(c2ccc(Cl)cc2)=NO1	nan
	123807	858	47	None	-2630	7	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	4	4	9	0.4	OC[C@H]1O[C@H]([C@@H]([C@@H]1O)O)n1cnc2c1nc(Cl)nc2NC1CCCC1	nan
	374	858	47	None	-2630	7	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	4	4	9	0.4	OC[C@H]1O[C@H]([C@@H]([C@@H]1O)O)n1cnc2c1nc(Cl)nc2NC1CCCC1	nan
	379	858	47	None	-2630	7	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	4	4	9	0.4	OC[C@H]1O[C@H]([C@@H]([C@@H]1O)O)n1cnc2c1nc(Cl)nc2NC1CCCC1	nan
	CHEMBL284969	858	47	None	-2630	7	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	4	4	9	0.4	OC[C@H]1O[C@H]([C@@H]([C@@H]1O)O)n1cnc2c1nc(Cl)nc2NC1CCCC1	nan
	2099	2997	77	None	-234	3	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	278	5	0	7	0.2	CC(=O)CCCCn1c(=O)c2n(C)cnc2n(c1=O)C	nan
	4740	2997	77	None	-234	3	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	278	5	0	7	0.2	CC(=O)CCCCn1c(=O)c2n(C)cnc2n(c1=O)C	nan
	7095	2997	77	None	-234	3	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	278	5	0	7	0.2	CC(=O)CCCCn1c(=O)c2n(C)cnc2n(c1=O)C	nan
	CHEMBL628	2997	77	None	-234	3	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	278	5	0	7	0.2	CC(=O)CCCCn1c(=O)c2n(C)cnc2n(c1=O)C	nan
	DB00806	2997	77	None	-234	3	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	278	5	0	7	0.2	CC(=O)CCCCn1c(=O)c2n(C)cnc2n(c1=O)C	nan
	123683	3072	58	None	-33884	5	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	510	5	4	9	0.4	CNC(=O)[C@H]1O[C@H]([C@@H]([C@@H]1O)O)n1cnc2c1ncnc2NCc1cccc(c1)I	nan
	422	3072	58	None	-33884	5	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	510	5	4	9	0.4	CNC(=O)[C@H]1O[C@H]([C@@H]([C@@H]1O)O)n1cnc2c1ncnc2NCc1cccc(c1)I	nan
	CHEMBL119709	3072	58	None	-33884	5	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	510	5	4	9	0.4	CNC(=O)[C@H]1O[C@H]([C@@H]([C@@H]1O)O)n1cnc2c1ncnc2NCc1cccc(c1)I	nan
	DB05511	3072	58	None	-33884	5	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	510	5	4	9	0.4	CNC(=O)[C@H]1O[C@H]([C@@H]([C@@H]1O)O)n1cnc2c1ncnc2NCc1cccc(c1)I	nan
	2808307	10287	5	None	-9	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	345	4	2	4	4.2	CC(=O)c1sc(C(C)(C)C)cc1NC(=O)c1ccccc1C(=O)O	nan
	CHEMBL1162415	10287	5	None	-9	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	345	4	2	4	4.2	CC(=O)c1sc(C(C)(C)C)cc1NC(=O)c1ccccc1C(=O)O	nan
	16019490	10897	4	None	-8	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	3	0	9	2.6	Cc1ccc(C)c(S(=O)(=O)c2nnn3c2nc(N2CCOCC2)c2sccc23)c1	nan
	CHEMBL1173709	10897	4	None	-8	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	3	0	9	2.6	Cc1ccc(C)c(S(=O)(=O)c2nnn3c2nc(N2CCOCC2)c2sccc23)c1	nan
	2729861	20206	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	347	5	2	8	0.0	Cn1c(=O)c2c(ncn2CC(O)CNc2ccc(F)cc2)n(C)c1=O	nan
	CHEMBL1306604	20206	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	347	5	2	8	0.0	Cn1c(=O)c2c(ncn2CC(O)CNc2ccc(F)cc2)n(C)c1=O	nan
	713572	20309	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	258	0	2	4	3.0	CC1(C)Cc2ccccc2-c2nc(S)nc(O)c21	nan
	CHEMBL1307433	20309	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	258	0	2	4	3.0	CC1(C)Cc2ccccc2-c2nc(S)nc(O)c21	nan
	20884214	20596	0	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	6	1	8	1.4	CCC(C(=O)NCCN1CCOCC1)n1nc(C)n2c(cc3sccc32)c1=O	nan
	CHEMBL1309746	20596	0	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	6	1	8	1.4	CCC(C(=O)NCCN1CCOCC1)n1nc(C)n2c(cc3sccc32)c1=O	nan
	1831123	20649	8	None	-1	3	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	489	3	1	7	5.2	Cc1nc2c(sc3nc(N4CCOCC4)c4c(c32)CC(C)(C)OC4)c(-c2ccccc2)c1C(=O)O	nan
	CHEMBL1310276	20649	8	None	-1	3	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	489	3	1	7	5.2	Cc1nc2c(sc3nc(N4CCOCC4)c4c(c32)CC(C)(C)OC4)c(-c2ccccc2)c1C(=O)O	nan
	16194788	20836	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	6	1	7	2.2	O=C(CSc1nnc2ccc(-c3ccccc3)nn12)NCC1CCCO1	nan
	CHEMBL1311747	20836	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	6	1	7	2.2	O=C(CSc1nnc2ccc(-c3ccccc3)nn12)NCC1CCCO1	nan
	2820129	20934	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	282	2	2	4	2.2	CSc1sc(C(=O)NNC(C)=O)c2c1C=CCC2	nan
	CHEMBL1312452	20934	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	282	2	2	4	2.2	CSc1sc(C(=O)NNC(C)=O)c2c1C=CCC2	nan
	622563	21007	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	282	2	0	4	3.1	CN1c2ccc(C=O)c3c(C=O)ccc(c23)N(C)C1(C)C	nan
	CHEMBL1312974	21007	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	282	2	0	4	3.1	CN1c2ccc(C=O)c3c(C=O)ccc(c23)N(C)C1(C)C	nan
	4584575	21074	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	3	2	5	3.7	CC(C)N=C(S)n1cc(C(=O)c2cc(Cl)cc(Cl)c2O)cn1	nan
	CHEMBL1313487	21074	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	3	2	5	3.7	CC(C)N=C(S)n1cc(C(=O)c2cc(Cl)cc(Cl)c2O)cn1	nan
	16029652	21303	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	6	1	6	5.0	CCOc1ccc(NC(=O)c2sc3nc(-c4ccc(OC)cc4)cn3c2C)cc1	nan
	CHEMBL1315982	21303	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	6	1	6	5.0	CCOc1ccc(NC(=O)c2sc3nc(-c4ccc(OC)cc4)cn3c2C)cc1	nan
	1116235	21363	15	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	5	1	9	0.7	COc1cc(NC(=O)Cn2cnc3c2c(=O)n(C)c(=O)n3C)c(OC)cc1Cl	nan
	CHEMBL1316844	21363	15	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	5	1	9	0.7	COc1cc(NC(=O)Cn2cnc3c2c(=O)n(C)c(=O)n3C)c(OC)cc1Cl	nan
	16030395	21384	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	8	1	4	4.5	CCCCNC(=O)CSc1nc2ccccc2nc1Cc1ccc(C)cc1	nan
	CHEMBL1317102	21384	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	8	1	4	4.5	CCCCNC(=O)CSc1nc2ccccc2nc1Cc1ccc(C)cc1	nan
	16018828	21389	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	4	1	6	4.1	Cc1ccc(NC(=O)CSc2nncn3c2cc2sccc23)cc1F	nan
	CHEMBL1317182	21389	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	4	1	6	4.1	Cc1ccc(NC(=O)CSc2nncn3c2cc2sccc23)cc1F	nan
	16018832	21419	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	4	1	6	4.3	Cc1ccc(C)c(NC(=O)CSc2nncn3c2cc2sccc23)c1	nan
	CHEMBL1317561	21419	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	4	1	6	4.3	Cc1ccc(C)c(NC(=O)CSc2nncn3c2cc2sccc23)c1	nan
	16025821	21456	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	486	6	1	5	4.9	CN(C)c1ccc(CNC(=O)C2CCN(C(=O)c3ccc(-n4ccc5ccccc54)s3)CC2)cc1	nan
	CHEMBL1318005	21456	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	486	6	1	5	4.9	CN(C)c1ccc(CNC(=O)C2CCN(C(=O)c3ccc(-n4ccc5ccccc54)s3)CC2)cc1	nan
	1482206	21533	16	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	316	3	1	5	2.1	CS(=O)(=O)c1ccc(-c2cn3cc(C(=O)O)ccc3n2)cc1	nan
	CHEMBL1318777	21533	16	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	316	3	1	5	2.1	CS(=O)(=O)c1ccc(-c2cn3cc(C(=O)O)ccc3n2)cc1	nan
	1115262	21554	31	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	4	2	4	5.5	O=C(O)c1ccc(Nc2nc(-c3ccccc3)c3cc(Br)ccc3n2)cc1	nan
	CHEMBL1318956	21554	31	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	4	2	4	5.5	O=C(O)c1ccc(Nc2nc(-c3ccccc3)c3cc(Br)ccc3n2)cc1	nan
	16025794	21556	0	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	457	5	1	4	5.2	Cc1ccc(CNC(=O)C2CCN(C(=O)c3ccc(-n4ccc5ccccc54)s3)CC2)cc1	nan
	CHEMBL1318960	21556	0	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	457	5	1	4	5.2	Cc1ccc(CNC(=O)C2CCN(C(=O)c3ccc(-n4ccc5ccccc54)s3)CC2)cc1	nan
	16021547	21570	0	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	497	6	2	8	1.8	NS(=O)(=O)c1ccc(CCNC(=O)C2CCN(c3ncnc4c3nc3n4CCCCC3)CC2)cc1	nan
	CHEMBL1319081	21570	0	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	497	6	2	8	1.8	NS(=O)(=O)c1ccc(CCNC(=O)C2CCN(c3ncnc4c3nc3n4CCCCC3)CC2)cc1	nan
	6287803	21575	3	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	521	7	1	6	4.6	CC1Cc2cc(C(=O)C3=C(O)C(=O)N(CCCn4ccnc4)C3c3ccc(Br)cc3)ccc2O1	nan
	CHEMBL1319132	21575	3	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	521	7	1	6	4.6	CC1Cc2cc(C(=O)C3=C(O)C(=O)N(CCCn4ccnc4)C3c3ccc(Br)cc3)ccc2O1	nan
	15988299	21598	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	5	1	7	2.9	Cn1c(=O)c2sccc2n2c(CCCC(=O)Nc3ccc(F)cc3F)nnc12	nan
	CHEMBL1319322	21598	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	5	1	7	2.9	Cn1c(=O)c2sccc2n2c(CCCC(=O)Nc3ccc(F)cc3F)nnc12	nan
	3152547	21784	4	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	5	1	5	3.2	O=C(C1=C(O)C(=O)N(CC2CCCO2)C1c1ccccc1F)c1ccco1	nan
	CHEMBL1320921	21784	4	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	5	1	5	3.2	O=C(C1=C(O)C(=O)N(CC2CCCO2)C1c1ccccc1F)c1ccco1	nan
	829953	21896	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	330	5	0	5	2.4	CCN(CC)S(=O)(=O)c1cccc(-c2cn3cccnc3n2)c1	nan
	CHEMBL1321896	21896	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	330	5	0	5	2.4	CCN(CC)S(=O)(=O)c1cccc(-c2cn3cccnc3n2)c1	nan
	3147388	22062	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	316	5	1	4	2.9	Cc1cc(SCC(=O)NCC2CCCO2)nc2ccccc12	nan
	CHEMBL1323473	22062	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	316	5	1	4	2.9	Cc1cc(SCC(=O)NCC2CCCO2)nc2ccccc12	nan
	3154196	22163	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	5	1	8	-0.1	CN(CC(O)Cn1cnc2c1c(=O)n(C)c(=O)n2C)c1ccccc1	nan
	CHEMBL1324245	22163	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	5	1	8	-0.1	CN(CC(O)Cn1cnc2c1c(=O)n(C)c(=O)n2C)c1ccccc1	nan
	16019851	22224	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	467	11	1	9	1.9	CCOCCCNC(=O)CCc1nnc2ccc(N3CCN(c4cccc(OC)c4)CC3)nn12	nan
	CHEMBL1324764	22224	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	467	11	1	9	1.9	CCOCCCNC(=O)CCc1nnc2ccc(N3CCN(c4cccc(OC)c4)CC3)nn12	nan
	16018924	22249	0	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	4	0	5	5.2	CCc1nnc(SCc2cccc(F)c2)c2cc3sc(C)cc3n12	nan
	CHEMBL1324960	22249	0	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	4	0	5	5.2	CCc1nnc(SCc2cccc(F)c2)c2cc3sc(C)cc3n12	nan
	4156222	22308	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	398	4	0	6	2.5	O=C(c1cccc([N+](=O)[O-])c1)N1CCCN(C(=O)c2cccc([N+](=O)[O-])c2)CC1	nan
	CHEMBL1325527	22308	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	398	4	0	6	2.5	O=C(c1cccc([N+](=O)[O-])c1)N1CCCN(C(=O)c2cccc([N+](=O)[O-])c2)CC1	nan
	16012102	22449	0	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	4	1	7	3.2	CCc1cccc(C)c1NC(=O)C1CCN(c2nn3c(=O)cc(C)nc3s2)CC1	nan
	CHEMBL1326931	22449	0	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	4	1	7	3.2	CCc1cccc(C)c1NC(=O)C1CCN(c2nn3c(=O)cc(C)nc3s2)CC1	nan
	342695	22641	3	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	295	3	0	8	0.6	Cn1c([N+](=O)[O-])cnc1N1CCN(c2nncs2)C1=O	nan
	CHEMBL1328402	22641	3	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	295	3	0	8	0.6	Cn1c([N+](=O)[O-])cnc1N1CCN(c2nncs2)C1=O	nan
	5048043	22666	9	None	-2	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	4	0	4	5.0	Cc1nn(C)cc1CN(C)C(=O)c1cc(-c2ccccc2)nc2ccc(Br)cc12	nan
	CHEMBL1328648	22666	9	None	-2	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	4	0	4	5.0	Cc1nn(C)cc1CN(C)C(=O)c1cc(-c2ccccc2)nc2ccc(Br)cc12	nan
	16195662	22758	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	5	0	9	1.6	CCOC(=O)N1CCN(C(=O)CSc2ccc3nnc(-c4ccncc4)n3n2)CC1	nan
	CHEMBL1329498	22758	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	5	0	9	1.6	CCOC(=O)N1CCN(C(=O)CSc2ccc3nnc(-c4ccncc4)n3n2)CC1	nan
	15988282	22795	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	5	1	7	2.0	Cn1c(=O)c2sccc2n2c(CCC(=O)NCc3ccc(F)cc3)nnc12	nan
	CHEMBL1329775	22795	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	5	1	7	2.0	Cn1c(=O)c2sccc2n2c(CCC(=O)NCc3ccc(F)cc3)nnc12	nan
	753118	22977	51	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	347	2	1	3	4.7	Cc1ccc(-c2cc(C(=O)O)c3cc(Br)ccc3n2)s1	nan
	CHEMBL1331202	22977	51	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	347	2	1	3	4.7	Cc1ccc(-c2cc(C(=O)O)c3cc(Br)ccc3n2)s1	nan
	CHEMBL1532594	22977	51	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	347	2	1	3	4.7	Cc1ccc(-c2cc(C(=O)O)c3cc(Br)ccc3n2)s1	nan
	15989826	23103	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	324	3	1	6	3.2	Cc1ccc2nc(NCc3ccccc3Cl)c3nnnn3c2c1	nan
	CHEMBL1332222	23103	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	324	3	1	6	3.2	Cc1ccc2nc(NCc3ccccc3Cl)c3nnnn3c2c1	nan
	7120050	23699	9	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	1	1	4	3.9	O=c1c2oc3ccccc3c2[nH]c(=S)n1-c1ccc(F)cc1	nan
	CHEMBL1336910	23699	9	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	1	1	4	3.9	O=c1c2oc3ccccc3c2[nH]c(=S)n1-c1ccc(F)cc1	nan
	2997990	23737	7	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	5	0	10	-0.2	Cc1cc(C(=O)COC(=O)Cn2cnc3c2c(=O)n(C)c(=O)n3C)c(C)n1C	nan
	CHEMBL1337270	23737	7	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	5	0	10	-0.2	Cc1cc(C(=O)COC(=O)Cn2cnc3c2c(=O)n(C)c(=O)n3C)c(C)n1C	nan
	5827230	23816	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	465	5	1	9	3.4	COc1cccc(C2C(C(=O)c3ccc4c(c3)OCCO4)=C(O)C(=O)N2c2nnc(C)s2)c1	nan
	CHEMBL1338023	23816	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	465	5	1	9	3.4	COc1cccc(C2C(C(=O)c3ccc4c(c3)OCCO4)=C(O)C(=O)N2c2nnc(C)s2)c1	nan
	4385163	23997	11	None	-2	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	6	2	4	4.5	COc1ccc(C(CC(=O)O)NC(=O)c2sc3ccccc3c2Cl)cc1	nan
	CHEMBL1339561	23997	11	None	-2	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	6	2	4	4.5	COc1ccc(C(CC(=O)O)NC(=O)c2sc3ccccc3c2Cl)cc1	nan
	8030040	24170	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	6	2	5	3.2	O=C(NCCNC(=O)c1ccc(-c2ccc(Cl)c(Cl)c2)o1)c1cnccn1	nan
	CHEMBL1341144	24170	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	6	2	5	3.2	O=C(NCCNC(=O)c1ccc(-c2ccc(Cl)c(Cl)c2)o1)c1cnccn1	nan
	661441	24574	7	None	-2	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	233	3	1	3	2.8	CC(Sc1ccc2ccccc2n1)C(=O)O	nan
	CHEMBL1344527	24574	7	None	-2	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	233	3	1	3	2.8	CC(Sc1ccc2ccccc2n1)C(=O)O	nan
	CHEMBL1530959	24574	7	None	-2	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	233	3	1	3	2.8	CC(Sc1ccc2ccccc2n1)C(=O)O	nan
	865623	24579	2	None	-4	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	271	3	0	5	3.5	CN(C)c1ccc(-c2nnc(-c3cccs3)o2)cc1	nan
	CHEMBL1344555	24579	2	None	-4	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	271	3	0	5	3.5	CN(C)c1ccc(-c2nnc(-c3cccs3)o2)cc1	nan
	2937580	24696	15	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	5	1	5	3.5	Cc1ccc(C(=O)C2=C(O)C(=O)N(CC3CCCO3)C2c2ccccc2F)o1	nan
	CHEMBL1345579	24696	15	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	5	1	5	3.5	Cc1ccc(C(=O)C2=C(O)C(=O)N(CC3CCCO3)C2c2ccccc2F)o1	nan
	1375907	24836	5	None	-1	3	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	3	0	7	1.4	CCOC(=O)Cn1cnc2c(C#N)c3n(c2c1=O)CCCCC3	nan
	CHEMBL1346739	24836	5	None	-1	3	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	3	0	7	1.4	CCOC(=O)Cn1cnc2c(C#N)c3n(c2c1=O)CCCCC3	nan
	5037672	24893	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	471	5	1	8	1.4	O=C(Nc1cc(S(=O)(=O)N2CCOCC2)ccc1N1CCOCC1)c1cn2ccccc2n1	nan
	CHEMBL1347181	24893	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	471	5	1	8	1.4	O=C(Nc1cc(S(=O)(=O)N2CCOCC2)ccc1N1CCOCC1)c1cn2ccccc2n1	nan
	3748480	24959	17	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	5	1	7	4.5	COc1cccc(C2C(C(=O)c3cc4ccccc4o3)=C(O)C(=O)N2c2cc(C)on2)c1	nan
	CHEMBL1347701	24959	17	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	5	1	7	4.5	COc1cccc(C2C(C(=O)c3cc4ccccc4o3)=C(O)C(=O)N2c2cc(C)on2)c1	nan
	6463240	24981	14	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	4	0	9	0.6	CC(C)n1c(CN2CCN(C(=O)c3ccco3)CC2)nc2c1c(=O)n(C)c(=O)n2C	nan
	CHEMBL1347878	24981	14	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	4	0	9	0.6	CC(C)n1c(CN2CCN(C(=O)c3ccco3)CC2)nc2c1c(=O)n(C)c(=O)n2C	nan
	4046369	25118	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	400	4	1	7	1.8	Cc1cc(C)n2nc(C(=O)Nc3cccc(S(=O)(=O)N4CCCC4)c3)nc2n1	nan
	CHEMBL1349141	25118	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	400	4	1	7	1.8	Cc1cc(C)n2nc(C(=O)Nc3cccc(S(=O)(=O)N4CCCC4)c3)nc2n1	nan
	5810234	25153	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	4	1	7	3.7	O=C(C1=C(O)C(=O)N(c2nccs2)C1c1ccccc1)c1ccc2c(c1)OCCO2	nan
	CHEMBL1349428	25153	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	4	1	7	3.7	O=C(C1=C(O)C(=O)N(c2nccs2)C1c1ccccc1)c1ccc2c(c1)OCCO2	nan
	664152	25199	14	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	5	1	6	3.1	Cc1nc(SCC(=O)NCC2CCCO2)c2oc3ccccc3c2n1	nan
	CHEMBL1349799	25199	14	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	5	1	6	3.1	Cc1nc(SCC(=O)NCC2CCCO2)c2oc3ccccc3c2n1	nan
	4648816	25241	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	7	1	8	2.4	COc1ccc(S(=O)(=O)N2CCOCC2)cc1NC(=O)CSc1ncnc2ccccc12	nan
	CHEMBL1350189	25241	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	7	1	8	2.4	COc1ccc(S(=O)(=O)N2CCOCC2)cc1NC(=O)CSc1ncnc2ccccc12	nan
	2081076	25272	18	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	304	2	1	5	3.3	O=c1c2c3c(sc2[nH]c(=S)n1Cc1ccco1)CCC3	nan
	CHEMBL1350435	25272	18	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	304	2	1	5	3.3	O=c1c2c3c(sc2[nH]c(=S)n1Cc1ccco1)CCC3	nan
	6618816	25337	0	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	6	1	7	2.4	Cn1c(=O)c2sccc2n2c(CCCC(=O)NCc3ccc(F)cc3)nnc12	nan
	CHEMBL1351035	25337	0	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	6	1	7	2.4	Cn1c(=O)c2sccc2n2c(CCCC(=O)NCc3ccc(F)cc3)nnc12	nan
	3117452	25342	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	265	4	0	3	1.4	Cc1c2ccccc2cc[n+]1CCCS(=O)(=O)[O-]	nan
	CHEMBL1351071	25342	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	265	4	0	3	1.4	Cc1c2ccccc2cc[n+]1CCCS(=O)(=O)[O-]	nan
	5809890	25466	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	446	5	1	6	3.8	O=C(C1=C(O)C(=O)N(Cc2ccncc2)C1c1ccccc1F)c1ccc2c(c1)OCCO2	nan
	CHEMBL1352143	25466	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	446	5	1	6	3.8	O=C(C1=C(O)C(=O)N(Cc2ccncc2)C1c1ccccc1F)c1ccc2c(c1)OCCO2	nan
	24794131	25478	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	6	0	8	2.7	CSc1ccccc1OCc1cc(C(=O)N2CCN(c3ncccn3)CC2)no1	nan
	CHEMBL1352219	25478	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	6	0	8	2.7	CSc1ccccc1OCc1cc(C(=O)N2CCN(c3ncccn3)CC2)no1	nan
	20903685	25525	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	6	0	8	2.1	CCOC(=O)C1CCN(C(=O)CCc2nnc3ccc(N4CCC(C)CC4)nn23)CC1	nan
	CHEMBL1352523	25525	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	6	0	8	2.1	CCOC(=O)C1CCN(C(=O)CCc2nnc3ccc(N4CCC(C)CC4)nn23)CC1	nan
	2322442	25564	7	None	1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	4	1	5	3.3	Cc1noc(NS(=O)(=O)c2ccc(N3Cc4ccccc4C3=O)cc2)c1C	nan
	CHEMBL1352855	25564	7	None	1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	4	1	5	3.3	Cc1noc(NS(=O)(=O)c2ccc(N3Cc4ccccc4C3=O)cc2)c1C	nan
	135490313	25712	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	4	2	10	-0.6	Cc1cc(O)nc(SCC(=O)c2c(N)n(C)c(=O)n(C)c2=O)n1	nan
	CHEMBL1353870	25712	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	4	2	10	-0.6	Cc1cc(O)nc(SCC(=O)c2c(N)n(C)c(=O)n(C)c2=O)n1	nan
	20923143	25823	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	7	1	6	1.6	CCCNS(=O)(=O)c1cc(CN2C(=O)c3cccnc3C2=O)ccc1OC	nan
	CHEMBL1354972	25823	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	7	1	6	1.6	CCCNS(=O)(=O)c1cc(CN2C(=O)c3cccnc3C2=O)ccc1OC	nan
	1116268	25837	14	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	4	1	9	-0.1	COC(=O)c1ccc(NC(=O)Cn2cnc3c2c(=O)n(C)c(=O)n3C)cc1	nan
	CHEMBL1355136	25837	14	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	4	1	9	-0.1	COC(=O)c1ccc(NC(=O)Cn2cnc3c2c(=O)n(C)c(=O)n3C)cc1	nan
	1003440	25953	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	3	2	5	5.9	Nc1c(C(=O)Nc2ccc(C(F)(F)F)cc2)sc2nc(-c3cccs3)ccc12	nan
	CHEMBL1356669	25953	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	3	2	5	5.9	Nc1c(C(=O)Nc2ccc(C(F)(F)F)cc2)sc2nc(-c3cccs3)ccc12	nan
	16024861	26033	0	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	3	1	4	3.0	CCNC(=O)C1CCN(c2nc3ccccc3nc2C(F)(F)F)CC1	nan
	CHEMBL1357771	26033	0	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	3	1	4	3.0	CCNC(=O)C1CCN(c2nc3ccccc3nc2C(F)(F)F)CC1	nan
	25162722	26104	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	9	1	9	1.4	CCN(CC)c1ccc(S(=O)(=O)N2CCOCC2)cc1NC(=O)CSc1nncn1C	nan
	CHEMBL1358718	26104	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	9	1	9	1.4	CCN(CC)c1ccc(S(=O)(=O)N2CCOCC2)cc1NC(=O)CSc1nncn1C	nan
	4312795	26265	20	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	234	3	1	4	2.2	CC(Sc1cnc2ccccc2n1)C(=O)O	nan
	CHEMBL1360045	26265	20	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	234	3	1	4	2.2	CC(Sc1cnc2ccccc2n1)C(=O)O	nan
	3704657	26277	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	361	4	1	6	3.2	Cc1ccc(C2C(C(=O)c3ccco3)=C(O)C(=O)N2c2ncccn2)cc1	nan
	CHEMBL1360163	26277	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	361	4	1	6	3.2	Cc1ccc(C2C(C(=O)c3ccco3)=C(O)C(=O)N2c2ncccn2)cc1	nan
	24000844	26293	2	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	5	2	7	2.9	Cn1c2ccccc2c2nnc(SCC(=O)Nc3cccc(C(=O)O)c3)nc21	nan
	CHEMBL1360279	26293	2	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	5	2	7	2.9	Cn1c2ccccc2c2nnc(SCC(=O)Nc3cccc(C(=O)O)c3)nc21	nan
	791500	26315	15	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	298	3	1	5	3.4	CCOC(=O)c1c(C)nc(S)c(C#N)c1-c1ccccc1	nan
	CHEMBL1360458	26315	15	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	298	3	1	5	3.4	CCOC(=O)c1c(C)nc(S)c(C#N)c1-c1ccccc1	nan
	3178481	26494	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	6	2	9	1.1	CCn1c(SCC(=O)Nc2ccc(NC(C)=O)cc2)nc2c1c(=O)n(C)c(=O)n2C	nan
	CHEMBL1362095	26494	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	6	2	9	1.1	CCn1c(SCC(=O)Nc2ccc(NC(C)=O)cc2)nc2c1c(=O)n(C)c(=O)n2C	nan
	5309057	26575	2	None	1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	2	0	5	3.7	O=C(c1cc2c(s1)-c1ccccc1OC2)N1CCN(c2ccccn2)CC1	nan
	CHEMBL1362711	26575	2	None	1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	2	0	5	3.7	O=C(c1cc2c(s1)-c1ccccc1OC2)N1CCN(c2ccccn2)CC1	nan
	16022478	26596	3	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	6	2	9	4.3	COc1cccc(NC(=O)c2ccc3c(=O)n4nc(Nc5ccccc5OC)sc4nc3c2)c1	nan
	CHEMBL1362937	26596	3	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	6	2	9	4.3	COc1cccc(NC(=O)c2ccc3c(=O)n4nc(Nc5ccccc5OC)sc4nc3c2)c1	nan
	20917857	26886	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	6	1	6	2.4	Cc1ccc(CNS(=O)(=O)c2cc(F)ccc2CN2C(=O)c3cccnc3C2=O)o1	nan
	CHEMBL1365432	26886	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	6	1	6	2.4	Cc1ccc(CNS(=O)(=O)c2cc(F)ccc2CN2C(=O)c3cccnc3C2=O)o1	nan
	2999882	27064	18	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	7	1	5	2.9	COCCCN1C(=O)C(O)=C(C(=O)c2ccco2)C1c1ccccc1	nan
	CHEMBL1367025	27064	18	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	7	1	5	2.9	COCCCN1C(=O)C(O)=C(C(=O)c2ccco2)C1c1ccccc1	nan
	1914729	27152	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	296	11	1	3	4.7	CC(=O)c1ccc(CCCCCCCCCC(=O)O)s1	nan
	CHEMBL1367732	27152	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	296	11	1	3	4.7	CC(=O)c1ccc(CCCCCCCCCC(=O)O)s1	nan
	3820161	27203	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	4	1	6	3.3	Cc1ccc(C(=O)C2=C(O)C(=O)N(c3ncccn3)C2c2ccccc2F)o1	nan
	CHEMBL1368082	27203	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	4	1	6	3.3	Cc1ccc(C(=O)C2=C(O)C(=O)N(c3ncccn3)C2c2ccccc2F)o1	nan
	135419062	27250	6	None	1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	5	1	7	4.5	N#Cc1c(O)nc(SCC(=O)c2ccc(Br)cc2)nc1-c1cccs1	nan
	CHEMBL1368444	27250	6	None	1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	5	1	7	4.5	N#Cc1c(O)nc(SCC(=O)c2ccc(Br)cc2)nc1-c1cccs1	nan
	3154099	27368	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	7	1	8	4.1	C=CCOc1cccc(C2C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2c2nnc(C)s2)c1	nan
	CHEMBL1369329	27368	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	7	1	8	4.1	C=CCOc1cccc(C2C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2c2nnc(C)s2)c1	nan
	2443232	27603	7	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	519	5	1	5	6.4	O=C(COC(=O)c1cc(-c2ccccc2Cl)nc2ccccc12)Nc1ncc(C(F)(F)F)cc1Cl	nan
	CHEMBL1370986	27603	7	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	519	5	1	5	6.4	O=C(COC(=O)c1cc(-c2ccccc2Cl)nc2ccccc12)Nc1ncc(C(F)(F)F)cc1Cl	nan
	22548207	27635	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	5	1	7	0.8	CCOC(=O)CNC(=O)Cn1cnc2c(oc3ccccc32)c1=O	nan
	CHEMBL1371227	27635	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	5	1	7	0.8	CCOC(=O)CNC(=O)Cn1cnc2c(oc3ccccc32)c1=O	nan
	663879	28060	13	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	9	1	7	4.2	Cc1ccc(C(=O)C2=C(O)C(=O)N(CCCn3ccnc3)C2c2ccc(OC(C)C)cc2)o1	nan
	CHEMBL1374204	28060	13	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	9	1	7	4.2	Cc1ccc(C(=O)C2=C(O)C(=O)N(CCCn3ccnc3)C2c2ccc(OC(C)C)cc2)o1	nan
	20917681	28065	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	6	1	7	2.0	O=C1c2cccnc2C(=O)N1Cc1ccc(S(=O)(=O)NCc2ccco2)s1	nan
	CHEMBL1374225	28065	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	6	1	7	2.0	O=C1c2cccnc2C(=O)N1Cc1ccc(S(=O)(=O)NCc2ccco2)s1	nan
	4855374	28339	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	5	0	10	-0.3	CN(C(=O)COC(=O)Cn1cnc2c1c(=O)n(C)c(=O)n2C)C1(C#N)CCCCC1	nan
	CHEMBL1376372	28339	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	5	0	10	-0.3	CN(C(=O)COC(=O)Cn1cnc2c1c(=O)n(C)c(=O)n2C)C1(C#N)CCCCC1	nan
	20917816	28775	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	4	0	5	2.4	CC1CCN(S(=O)(=O)c2cc(F)ccc2CN2C(=O)c3cccnc3C2=O)CC1	nan
	CHEMBL1380363	28775	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	4	0	5	2.4	CC1CCN(S(=O)(=O)c2cc(F)ccc2CN2C(=O)c3cccnc3C2=O)CC1	nan
	661999	28860	14	None	-5	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	460	6	1	8	4.5	COc1cccc(C2C(C(=O)c3cc4ccccc4o3)=C(O)C(=O)N2c2cc(C)on2)c1OC	nan
	CHEMBL1380975	28860	14	None	-5	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	460	6	1	8	4.5	COc1cccc(C2C(C(=O)c3cc4ccccc4o3)=C(O)C(=O)N2c2cc(C)on2)c1OC	nan
	4342649	28973	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	6	1	6	3.5	O=C(C1=C(O)C(=O)N(CCN2CCOCC2)C1c1cccc(F)c1)c1cc2ccccc2o1	nan
	5027943	28973	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	6	1	6	3.5	O=C(C1=C(O)C(=O)N(CCN2CCOCC2)C1c1cccc(F)c1)c1cc2ccccc2o1	nan
	CHEMBL1381980	28973	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	6	1	6	3.5	O=C(C1=C(O)C(=O)N(CCN2CCOCC2)C1c1cccc(F)c1)c1cc2ccccc2o1	nan
	135431552	29041	10	None	-2	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	4	1	6	4.7	N#Cc1c(O)nc(SCc2ccc(Cl)cc2)nc1-c1cccs1	nan
	CHEMBL1382616	29041	10	None	-2	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	4	1	6	4.7	N#Cc1c(O)nc(SCc2ccc(Cl)cc2)nc1-c1cccs1	nan
	921583	29434	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	316	1	1	3	4.3	Sc1nc(-c2ccccc2)nc2ccc(Br)cc12	nan
	CHEMBL1386089	29434	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	316	1	1	3	4.3	Sc1nc(-c2ccccc2)nc2ccc(Br)cc12	nan
	5428525	29754	23	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	262	2	1	5	1.8	COC(=O)Cc1c(C)c2c(O)cc(C)cc2oc1=O	nan
	CHEMBL1388510	29754	23	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	262	2	1	5	1.8	COC(=O)Cc1c(C)c2c(O)cc(C)cc2oc1=O	nan
	5824610	29802	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	296	7	1	5	3.1	CN(C)CCCNc1oc(/C=C/c2ccccc2)nc1C#N	nan
	CHEMBL1388949	29802	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	296	7	1	5	3.1	CN(C)CCCNc1oc(/C=C/c2ccccc2)nc1C#N	nan
	16194879	30150	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	7	1	9	2.9	COc1ccc(NC(=O)CSc2ccc3nnc(-c4cccnc4)n3n2)c(OC)c1	nan
	CHEMBL1391905	30150	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	7	1	9	2.9	COc1ccc(NC(=O)CSc2ccc3nnc(-c4cccnc4)n3n2)c(OC)c1	nan
	1256976	30211	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	496	5	2	5	3.6	NS(=O)(=O)c1ccc(CNC(=O)c2cc(-c3cccnc3)nc3ccc(Br)cc23)cc1	nan
	CHEMBL1392432	30211	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	496	5	2	5	3.6	NS(=O)(=O)c1ccc(CNC(=O)c2cc(-c3cccnc3)nc3ccc(Br)cc23)cc1	nan
	7222624	30504	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	5	1	6	4.2	Cc1nc(C)c(-c2ccc(SCC(=O)Nc3ccc(F)c(F)c3)nn2)s1	nan
	CHEMBL1395178	30504	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	5	1	6	4.2	Cc1nc(C)c(-c2ccc(SCC(=O)Nc3ccc(F)c(F)c3)nn2)s1	nan
	16018363	30528	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	5	1	6	5.5	COc1ccc(NC(=O)c2ccc3c(c2)sc2nc(-c4ccc(OC)cc4)cn23)cc1	nan
	CHEMBL1395439	30528	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	5	1	6	5.5	COc1ccc(NC(=O)c2ccc3c(c2)sc2nc(-c4ccc(OC)cc4)cn23)cc1	nan
	15990211	30679	1	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	3	1	6	3.1	Fc1ccc(CNc2nc3ccc(Cl)cc3n3nnnc23)cc1	nan
	CHEMBL1397707	30679	1	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	3	1	6	3.1	Fc1ccc(CNc2nc3ccc(Cl)cc3n3nnnc23)cc1	nan
	7151328	30740	2	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	4	1	5	3.1	CCS(=O)(=O)Nc1ccc(-c2cn3c(C)csc3n2)cc1	nan
	CHEMBL1398475	30740	2	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	4	1	5	3.1	CCS(=O)(=O)Nc1ccc(-c2cn3c(C)csc3n2)cc1	nan
	20939725	30842	4	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	479	5	0	7	2.9	COc1ccc(CN2C(=O)c3cccnc3C2=O)cc1S(=O)(=O)N1CC(C)Oc2ccccc21	nan
	CHEMBL1399426	30842	4	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	479	5	0	7	2.9	COc1ccc(CN2C(=O)c3cccnc3C2=O)cc1S(=O)(=O)N1CC(C)Oc2ccccc21	nan
	16452548	31094	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	6	2	8	2.7	Cc1cccc(-n2ccc(=O)c(C(=O)Nc3ccc(S(=O)(=O)Nc4nccc(C)n4)cc3)n2)c1	nan
	CHEMBL1401713	31094	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	6	2	8	2.7	Cc1cccc(-n2ccc(=O)c(C(=O)Nc3ccc(S(=O)(=O)Nc4nccc(C)n4)cc3)n2)c1	nan
	3709623	31204	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	4	1	6	3.3	Cc1ccc(C(=O)C2=C(O)C(=O)N(c3ncccn3)C2c2ccc(F)cc2)o1	nan
	CHEMBL1402642	31204	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	4	1	6	3.3	Cc1ccc(C(=O)C2=C(O)C(=O)N(c3ncccn3)C2c2ccc(F)cc2)o1	nan
	5212778	31232	14	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	9	1	6	4.1	CCN(CC)CCCN1C(=O)C(O)=C(C(=O)c2cc3ccccc3o2)C1c1ccccn1	nan
	661982	31232	14	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	9	1	6	4.1	CCN(CC)CCCN1C(=O)C(O)=C(C(=O)c2cc3ccccc3o2)C1c1ccccn1	nan
	CHEMBL1402874	31232	14	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	9	1	6	4.1	CCN(CC)CCCN1C(=O)C(O)=C(C(=O)c2cc3ccccc3o2)C1c1ccccn1	nan
	3152754	31315	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	6	1	5	4.2	O=C(C1=C(O)C(=O)N(CCc2ccccc2)C1c1cccs1)c1ccco1	nan
	CHEMBL1403767	31315	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	6	1	5	4.2	O=C(C1=C(O)C(=O)N(CCc2ccccc2)C1c1cccs1)c1ccco1	nan
	2816622	31392	7	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	396	4	1	6	4.8	COc1ccc(-n2c(=S)[nH]c3sc(-c4ccccc4)cc3c2=O)c(OC)c1	nan
	CHEMBL1404356	31392	7	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	396	4	1	6	4.8	COc1ccc(-n2c(=S)[nH]c3sc(-c4ccccc4)cc3c2=O)c(OC)c1	nan
	7245568	31518	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	5	1	8	2.2	COc1ccc(NC(=O)CCc2nnc3n(C)c(=O)c4sccc4n23)cc1	nan
	CHEMBL1405733	31518	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	5	1	8	2.2	COc1ccc(NC(=O)CCc2nnc3n(C)c(=O)c4sccc4n23)cc1	nan
	4184357	31536	7	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	554	6	1	9	4.3	O=C(O)c1ccc(Cn2c(SCc3cc(=O)n4cc(Br)ccc4n3)nc3ccsc3c2=O)cc1	nan
	CHEMBL1405932	31536	7	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	554	6	1	9	4.3	O=C(O)c1ccc(Cn2c(SCc3cc(=O)n4cc(Br)ccc4n3)nc3ccsc3c2=O)cc1	nan
	757946	31771	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	2	1	2	4.7	Cc1nc2ccc(Br)cc2c(-c2ccccc2)c1C(=O)O	nan
	CHEMBL1407788	31771	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	2	1	2	4.7	Cc1nc2ccc(Br)cc2c(-c2ccccc2)c1C(=O)O	nan
	3160259	31844	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	5	2	7	2.2	Cc1ccc(-c2nn3c(C)nnc3c3ccccc23)cc1S(=O)(=O)NCC(C)O	nan
	CHEMBL1408356	31844	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	5	2	7	2.2	Cc1ccc(-c2nn3c(C)nnc3c3ccccc23)cc1S(=O)(=O)NCC(C)O	nan
	1071246	31917	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	5	1	8	0.6	CCn1c(SCC(=O)NC2CCCC2)nc2c1c(=O)n(C)c(=O)n2C	nan
	CHEMBL1408937	31917	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	5	1	8	0.6	CCn1c(SCC(=O)NC2CCCC2)nc2c1c(=O)n(C)c(=O)n2C	nan
	744304	31952	15	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	231	1	2	4	2.4	COc1ccc2[nH]c3c(S)ncnc3c2c1	nan
	CHEMBL1409203	31952	15	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	231	1	2	4	2.4	COc1ccc2[nH]c3c(S)ncnc3c2c1	nan
	3240452	31954	4	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	5	1	8	0.4	O=C(Cn1cnc2c(nnn2-c2ccc(F)cc2)c1=O)NCC1CCCO1	nan
	CHEMBL1409223	31954	4	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	5	1	8	0.4	O=C(Cn1cnc2c(nnn2-c2ccc(F)cc2)c1=O)NCC1CCCO1	nan
	15989908	32060	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	302	4	0	7	2.2	CCOC(=O)CSc1nc2ccccc2n2c(C)nnc12	nan
	CHEMBL1410062	32060	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	302	4	0	7	2.2	CCOC(=O)CSc1nc2ccccc2n2c(C)nnc12	nan
	20923121	32100	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	7	1	7	2.0	COc1ccc(CN2C(=O)c3cccnc3C2=O)cc1S(=O)(=O)NCc1ccco1	nan
	CHEMBL1410345	32100	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	7	1	7	2.0	COc1ccc(CN2C(=O)c3cccnc3C2=O)cc1S(=O)(=O)NCc1ccco1	nan
	3998353	32293	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	4	1	8	1.0	Cc1cc(C)n2nc(C(=O)Nc3cccc(S(=O)(=O)N4CCOCC4)c3)nc2n1	nan
	CHEMBL1412011	32293	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	4	1	8	1.0	Cc1cc(C)n2nc(C(=O)Nc3cccc(S(=O)(=O)N4CCOCC4)c3)nc2n1	nan
	16034646	32386	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	5	1	7	3.3	Cn1c(=O)c2sccc2n2c(CCCC(=O)Nc3ccc(Cl)cc3)nnc12	nan
	CHEMBL1412706	32386	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	5	1	7	3.3	Cn1c(=O)c2sccc2n2c(CCCC(=O)Nc3ccc(Cl)cc3)nnc12	nan
	1145396	32481	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	3	1	4	4.4	O=C(O)C1CCN(c2nc(-c3ccccc3)c3cc(Br)ccc3n2)CC1	nan
	5026856	32481	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	3	1	4	4.4	O=C(O)C1CCN(c2nc(-c3ccccc3)c3cc(Br)ccc3n2)CC1	nan
	CHEMBL1413474	32481	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	3	1	4	4.4	O=C(O)C1CCN(c2nc(-c3ccccc3)c3cc(Br)ccc3n2)CC1	nan
	652152	32624	19	None	-1	3	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	241	2	1	3	2.7	COc1ccc2c(Cl)c(C(N)=O)sc2c1	nan
	CHEMBL1414671	32624	19	None	-1	3	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	241	2	1	3	2.7	COc1ccc2c(Cl)c(C(N)=O)sc2c1	nan
	1004109	32742	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	3	2	4	5.4	Cc1ccc(NC(=O)c2sc3nc(-c4ccc(F)cc4)ccc3c2N)cc1F	nan
	CHEMBL1415733	32742	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	3	2	4	5.4	Cc1ccc(NC(=O)c2sc3nc(-c4ccc(F)cc4)ccc3c2N)cc1F	nan
	22334931	32802	27	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	5	1	4	3.5	O=C(O)CSc1nc2ccccc2nc1Cc1ccccc1F	nan
	CHEMBL1416271	32802	27	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	5	1	4	3.5	O=C(O)CSc1nc2ccccc2nc1Cc1ccccc1F	nan
	3953394	32907	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	6	1	8	1.5	O=C(CSc1nnc2ccccn12)Nc1cccc(S(=O)(=O)N2CCOCC2)c1	nan
	CHEMBL1417177	32907	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	6	1	8	1.5	O=C(CSc1nnc2ccccn12)Nc1cccc(S(=O)(=O)N2CCOCC2)c1	nan
	24687828	32922	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	7	0	11	-0.1	COc1ccc(C(=O)COC(=O)Cn2cnc3c2c(=O)n(C)c(=O)n3C)c(OC)c1	nan
	CHEMBL1417257	32922	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	7	0	11	-0.1	COc1ccc(C(=O)COC(=O)Cn2cnc3c2c(=O)n(C)c(=O)n3C)c(OC)c1	nan
	7184635	33175	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	7	1	8	2.3	COc1cccc(CNC(=O)CCCc2nnc3n(C)c(=O)c4sccc4n23)c1	nan
	CHEMBL1419486	33175	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	7	1	8	2.3	COc1cccc(CNC(=O)CCCc2nnc3n(C)c(=O)c4sccc4n23)c1	nan
	4796292	33220	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	5	0	6	1.1	CN(C)S(=O)(=O)c1cccc(COC(=O)c2cnccn2)c1	nan
	CHEMBL1419907	33220	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	5	0	6	1.1	CN(C)S(=O)(=O)c1cccc(COC(=O)c2cnccn2)c1	nan
	744542	33243	34	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	261	4	1	3	3.4	Cc1cc(SCCC(=O)O)nc2c(C)cccc12	nan
	CHEMBL1420044	33243	34	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	261	4	1	3	3.4	Cc1cc(SCCC(=O)O)nc2c(C)cccc12	nan
	3789487	33313	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	4	1	6	3.0	O=C(C1=C(O)C(=O)N(c2ncccn2)C1c1ccc(F)cc1)c1ccco1	nan
	CHEMBL1420588	33313	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	4	1	6	3.0	O=C(C1=C(O)C(=O)N(c2ncccn2)C1c1ccc(F)cc1)c1ccco1	nan
	1473006	33366	13	None	1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	1	0	2	4.1	COc1cc2cc(Br)cc(Br)c2nc1C	nan
	CHEMBL1421084	33366	13	None	1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	1	0	2	4.1	COc1cc2cc(Br)cc(Br)c2nc1C	nan
	22421602	33420	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	479	9	2	8	1.0	COc1ccc(-n2nc(C(=O)NCC(=O)NCCCN3CCOCC3)c3ccccc3c2=O)cc1	nan
	CHEMBL1421499	33420	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	479	9	2	8	1.0	COc1ccc(-n2nc(C(=O)NCC(=O)NCCCN3CCOCC3)c3ccccc3c2=O)cc1	nan
	20957484	33427	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	471	10	1	9	1.3	CCOC(=O)C1CCN(C(=O)CCc2nnc3ccc(NCCCN4CCCC4=O)nn23)CC1	nan
	CHEMBL1421579	33427	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	471	10	1	9	1.3	CCOC(=O)C1CCN(C(=O)CCc2nnc3ccc(NCCCN4CCCC4=O)nn23)CC1	nan
	7190683	33442	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	6	1	8	2.9	COc1cccc(NC(=O)CSc2ccc3nnc(-c4cccnc4)n3n2)c1	nan
	CHEMBL1421703	33442	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	6	1	8	2.9	COc1cccc(NC(=O)CSc2ccc3nnc(-c4cccnc4)n3n2)c1	nan
	7190642	33584	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	5	1	7	3.2	Cc1cccc(NC(=O)CSc2ccc3nnc(-c4cccnc4)n3n2)c1	nan
	CHEMBL1422914	33584	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	5	1	7	3.2	Cc1cccc(NC(=O)CSc2ccc3nnc(-c4cccnc4)n3n2)c1	nan
	741274	33814	11	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	286	2	0	7	0.6	COC(=O)Cn1cnc2c(C#N)c3n(c2c1=O)CCCC3	nan
	CHEMBL1424800	33814	11	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	286	2	0	7	0.6	COC(=O)Cn1cnc2c(C#N)c3n(c2c1=O)CCCC3	nan
	3816425	33900	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	7	1	7	5.3	CCCOc1cccc(C2C(C(=O)c3cc4ccccc4o3)=C(O)C(=O)N2c2cc(C)on2)c1	nan
	CHEMBL1425600	33900	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	7	1	7	5.3	CCCOc1cccc(C2C(C(=O)c3cc4ccccc4o3)=C(O)C(=O)N2c2cc(C)on2)c1	nan
	7299201	33908	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	4	1	6	4.6	Cc1cccc(C)c1Nc1c(-c2ccc(N3CCOCC3)cc2)nc2cnccn12	nan
	CHEMBL1425693	33908	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	4	1	6	4.6	Cc1cccc(C)c1Nc1c(-c2ccc(N3CCOCC3)cc2)nc2cnccn12	nan
	5739077	34083	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	466	7	1	8	2.3	COc1cccc(C2C(C(=O)c3ccc4c(c3)OCO4)=C(O)C(=O)N2CCN2CCOCC2)c1	nan
	CHEMBL1427088	34083	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	466	7	1	8	2.3	COc1cccc(C2C(C(=O)c3ccc4c(c3)OCO4)=C(O)C(=O)N2CCN2CCOCC2)c1	nan
	3830309	34216	18	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	4	1	6	4.7	O=C(C1=C(O)C(=O)N(c2nccs2)C1c1ccccc1)c1cc2ccccc2o1	nan
	CHEMBL1428271	34216	18	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	4	1	6	4.7	O=C(C1=C(O)C(=O)N(c2nccs2)C1c1ccccc1)c1cc2ccccc2o1	nan
	20903609	34467	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	517	9	1	10	3.0	COc1cc(NC(=O)CCc2nnc3ccc(N4CCN(c5cccc(OC)c5)CC4)nn23)cc(OC)c1	nan
	CHEMBL1430241	34467	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	517	9	1	10	3.0	COc1cc(NC(=O)CCc2nnc3ccc(N4CCN(c5cccc(OC)c5)CC4)nn23)cc(OC)c1	nan
	990446	34494	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	3	1	9	2.1	COc1cccc(-n2nc3c(-n4ncc(C#N)c4N)nnc(C)c3c2C)c1	nan
	CHEMBL1430459	34494	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	3	1	9	2.1	COc1cccc(-n2nc3c(-n4ncc(C#N)c4N)nnc(C)c3c2C)c1	nan
	2809114	34642	5	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	5	1	4	4.7	CC(=O)c1sc(-c2ccccc2)cc1NS(=O)(=O)c1ccc(C)cc1	nan
	CHEMBL1431741	34642	5	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	5	1	4	4.7	CC(=O)c1sc(-c2ccccc2)cc1NS(=O)(=O)c1ccc(C)cc1	nan
	4968705	34793	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	6	0	10	-0.5	CN(C)S(=O)(=O)c1ccc(C(=O)OCCn2cnc3c2c(=O)n(C)c(=O)n3C)cc1	nan
	CHEMBL1433054	34793	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	6	0	10	-0.5	CN(C)S(=O)(=O)c1ccc(C(=O)OCCn2cnc3c2c(=O)n(C)c(=O)n3C)cc1	nan
	16019549	34886	0	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	479	3	0	9	2.8	O=S(=O)(c1ccc(Br)cc1)c1nnn2c1nc(N1CCOCC1)c1sccc12	nan
	CHEMBL1433993	34886	0	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	479	3	0	9	2.8	O=S(=O)(c1ccc(Br)cc1)c1nnn2c1nc(N1CCOCC1)c1sccc12	nan
	20885693	34994	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	373	7	1	6	2.0	Cc1nn(CCCC(=O)NCCc2ccc(Cl)cc2)c(=O)c2nccn12	nan
	CHEMBL1435443	34994	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	373	7	1	6	2.0	Cc1nn(CCCC(=O)NCCc2ccc(Cl)cc2)c(=O)c2nccn12	nan
	4380857	35000	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	4	0	4	5.0	Cc1c(CN(C)C(=O)c2cc(-c3ccccc3)nc3ccc(Br)cc23)cnn1C	nan
	CHEMBL1435516	35000	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	4	0	4	5.0	Cc1c(CN(C)C(=O)c2cc(-c3ccccc3)nc3ccc(Br)cc23)cnn1C	nan
	5066674	35012	3	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	510	5	1	7	2.7	COC(=O)c1cc(NS(=O)(=O)c2cc(Br)cc3c2N(C(C)=O)CC3)cc(C(=O)OC)c1	nan
	CHEMBL1435676	35012	3	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	510	5	1	7	2.7	COC(=O)c1cc(NS(=O)(=O)c2cc(Br)cc3c2N(C(C)=O)CC3)cc(C(=O)OC)c1	nan
	3993922	35078	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	5	1	7	1.2	O=C(CNC(=O)c1ccccc1)OCc1cc(=O)n2ccsc2n1	nan
	CHEMBL1436555	35078	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	5	1	7	1.2	O=C(CNC(=O)c1ccccc1)OCc1cc(=O)n2ccsc2n1	nan
	16018682	35095	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	366	5	1	6	4.1	CCc1ccccc1NC(=O)CSc1nncn2c1cc1oc(C)cc12	nan
	CHEMBL1436824	35095	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	366	5	1	6	4.1	CCc1ccccc1NC(=O)CSc1nncn2c1cc1oc(C)cc12	nan
	16026770	35115	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	5	1	7	1.7	Cc1csc2nc(COC(=O)CNC(=O)c3ccc(F)cc3)cc(=O)n12	nan
	CHEMBL1437080	35115	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	5	1	7	1.7	Cc1csc2nc(COC(=O)CNC(=O)c3ccc(F)cc3)cc(=O)n12	nan
	90660425	35239	0	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	446	7	1	5	5.1	CCCOc1ccc(C(=O)C2=C(O)C(=O)N(c3ccccn3)C2c2ccccc2F)cc1C	nan
	CHEMBL1438291	35239	0	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	446	7	1	5	5.1	CCCOc1ccc(C(=O)C2=C(O)C(=O)N(c3ccccn3)C2c2ccccc2F)cc1C	nan
	663438	35408	13	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	344	3	0	6	1.4	O=S(=O)(c1cccc(-c2cn3cccnc3n2)c1)N1CCOCC1	nan
	CHEMBL1439795	35408	13	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	344	3	0	6	1.4	O=S(=O)(c1cccc(-c2cn3cccnc3n2)c1)N1CCOCC1	nan
	135544645	35417	7	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	5	2	7	3.7	N#Cc1c(O)nc(SCC(=O)Nc2cccc(Cl)c2)nc1-c1ccco1	nan
	CHEMBL1439904	35417	7	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	5	2	7	3.7	N#Cc1c(O)nc(SCC(=O)Nc2cccc(Cl)c2)nc1-c1ccco1	nan
	3363660	35557	10	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	515	7	1	7	3.3	CCN1C(=O)C2(C(C(=O)c3cc4ccccc4o3)=C(O)C(=O)N2CCCN2CCOCC2)c2ccccc21	nan
	4976974	35557	10	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	515	7	1	7	3.3	CCN1C(=O)C2(C(C(=O)c3cc4ccccc4o3)=C(O)C(=O)N2CCCN2CCOCC2)c2ccccc21	nan
	CHEMBL1441169	35557	10	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	515	7	1	7	3.3	CCN1C(=O)C2(C(C(=O)c3cc4ccccc4o3)=C(O)C(=O)N2CCCN2CCOCC2)c2ccccc21	nan
	2854626	35565	10	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	7	1	5	5.1	CC(=O)C1=C(C)NC(SCC(=O)c2ccc(Cl)cc2)=C(C#N)C1CC(C)C	nan
	CHEMBL1441242	35565	10	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	7	1	5	5.1	CC(=O)C1=C(C)NC(SCC(=O)c2ccc(Cl)cc2)=C(C#N)C1CC(C)C	nan
	20957185	35719	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	440	6	1	8	1.9	O=C(CCc1nnc2ccc(N3CCC4(CC3)OCCO4)nn12)NCc1ccc(F)cc1	nan
	CHEMBL1442625	35719	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	440	6	1	8	1.9	O=C(CCc1nnc2ccc(N3CCC4(CC3)OCCO4)nn12)NCc1ccc(F)cc1	nan
	812443	35913	45	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	278	2	1	4	3.2	C=CCn1c(=S)[nH]c2sc3c(c2c1=O)CCCC3	nan
	CHEMBL1444467	35913	45	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	278	2	1	4	3.2	C=CCn1c(=S)[nH]c2sc3c(c2c1=O)CCCC3	nan
	20923160	35915	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	467	8	1	7	2.4	COc1ccccc1CNS(=O)(=O)c1cc(CN2C(=O)c3cccnc3C2=O)ccc1OC	nan
	CHEMBL1444486	35915	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	467	8	1	7	2.4	COc1ccccc1CNS(=O)(=O)c1cc(CN2C(=O)c3cccnc3C2=O)ccc1OC	nan
	16745544	36292	0	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	2	1	5	2.5	COc1ccc(C2=CC3=C(Br)C(=O)C(C)(O)C(=O)C3=CO2)cc1	nan
	CHEMBL1447877	36292	0	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	2	1	5	2.5	COc1ccc(C2=CC3=C(Br)C(=O)C(C)(O)C(=O)C3=CO2)cc1	nan
	2376086	36356	19	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	296	3	1	5	2.6	COCCn1c(=S)[nH]c2sc3c(c2c1=O)CCCC3	nan
	CHEMBL1448425	36356	19	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	296	3	1	5	2.6	COCCn1c(=S)[nH]c2sc3c(c2c1=O)CCCC3	nan
	16745680	36506	0	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	503	9	0	7	5.7	CCCCC1=CC2=C(c3ccco3)C(=O)C(C)(OC(=O)c3ccc(OC)cc3)C(=O)C2=CN1CC(C)C	nan
	CHEMBL1449527	36506	0	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	503	9	0	7	5.7	CCCCC1=CC2=C(c3ccco3)C(=O)C(C)(OC(=O)c3ccc(OC)cc3)C(=O)C2=CN1CC(C)C	nan
	16018684	36507	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	4	1	6	4.4	Cc1cc(C)c(NC(=O)CSc2nncn3c2cc2oc(C)cc23)c(C)c1	nan
	CHEMBL1449543	36507	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	4	1	6	4.4	Cc1cc(C)c(NC(=O)CSc2nncn3c2cc2oc(C)cc23)c(C)c1	nan
	1094076	36520	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	297	3	1	6	3.0	CC(=O)c1ccc(Nc2nc(=O)c3cccnc3s2)cc1	nan
	CHEMBL1449615	36520	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	297	3	1	6	3.0	CC(=O)c1ccc(Nc2nc(=O)c3cccnc3s2)cc1	nan
	3514089	36664	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	7	1	7	5.3	CCCOc1ccc(C2C(C(=O)c3cc4ccccc4o3)=C(O)C(=O)N2c2cc(C)on2)cc1	nan
	CHEMBL1450861	36664	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	7	1	7	5.3	CCCOc1ccc(C2C(C(=O)c3cc4ccccc4o3)=C(O)C(=O)N2c2cc(C)on2)cc1	nan
	6619005	36882	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	544	5	1	7	4.4	Cc1c(N2C(=O)C(O)=C(C(=O)c3ccc(Br)cc3)C2c2cccnc2)c(=O)n(-c2ccccc2)n1C	nan
	CHEMBL1452549	36882	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	544	5	1	7	4.4	Cc1c(N2C(=O)C(O)=C(C(=O)c3ccc(Br)cc3)C2c2cccnc2)c(=O)n(-c2ccccc2)n1C	nan
	16194575	37059	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	5	1	10	2.1	Cc1nnc(NC(=O)CSc2ccc3nnc(-c4cccnc4)n3n2)s1	nan
	CHEMBL1453968	37059	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	5	1	10	2.1	Cc1nnc(NC(=O)CSc2ccc3nnc(-c4cccnc4)n3n2)s1	nan
	3178522	37123	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	6	0	9	0.2	CCCCn1c(SCC(=O)N2CCOCC2)nc2c1c(=O)n(C)c(=O)n2C	nan
	CHEMBL1454485	37123	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	6	0	9	0.2	CCCCn1c(SCC(=O)N2CCOCC2)nc2c1c(=O)n(C)c(=O)n2C	nan
	2613266	37194	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	344	4	0	8	2.8	O=[N+]([O-])c1cc2c(c(CSc3nnc4ccccn34)c1)OCOC2	nan
	CHEMBL1455089	37194	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	344	4	0	8	2.8	O=[N+]([O-])c1cc2c(c(CSc3nnc4ccccn34)c1)OCOC2	nan
	1084466	37306	17	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	6	2	6	2.5	COc1ccccc1C(=O)Nc1ccc(S(=O)(=O)Nc2ncccn2)cc1	nan
	CHEMBL1456125	37306	17	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	6	2	6	2.5	COc1ccccc1C(=O)Nc1ccc(S(=O)(=O)Nc2ncccn2)cc1	nan
	20885676	37358	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	6	1	6	1.6	Cc1ccc(CNC(=O)CCCn2nc(C)n3ccnc3c2=O)cc1	nan
	CHEMBL1456629	37358	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	6	1	6	1.6	Cc1ccc(CNC(=O)CCCn2nc(C)n3ccnc3c2=O)cc1	nan
	3715206	37367	20	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	294	2	1	5	3.9	CCn1c(=S)[nH]c2scc(-c3cccs3)c2c1=O	nan
	CHEMBL1456701	37367	20	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	294	2	1	5	3.9	CCn1c(=S)[nH]c2scc(-c3cccs3)c2c1=O	nan
	3252203	37520	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	6	1	6	4.2	O=C(CSc1ncnc2ccccc12)Nc1cc(S(=O)(=O)N2CCCCC2)ccc1Cl	nan
	CHEMBL1457998	37520	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	6	1	6	4.2	O=C(CSc1ncnc2ccccc12)Nc1cc(S(=O)(=O)N2CCCCC2)ccc1Cl	nan
	2939635	37623	33	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	247	3	1	3	3.1	Cc1cc(SC(C)C(=O)O)nc2ccccc12	nan
	CHEMBL1458912	37623	33	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	247	3	1	3	3.1	Cc1cc(SC(C)C(=O)O)nc2ccccc12	nan
	1442575	37863	3	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	6	1	4	3.7	CCCc1nc(SCC(=O)NC2CCCC2)c2ccccc2n1	nan
	CHEMBL1460883	37863	3	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	6	1	4	3.7	CCCc1nc(SCC(=O)NC2CCCC2)c2ccccc2n1	nan
	4412828	37961	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	472	9	1	7	2.4	CCN(CC)S(=O)(=O)c1ccc(N2CCOCC2)c(NC(=O)COc2ccc(C#N)cc2)c1	nan
	CHEMBL1461851	37961	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	472	9	1	7	2.4	CCN(CC)S(=O)(=O)c1ccc(N2CCOCC2)c(NC(=O)COc2ccc(C#N)cc2)c1	nan
	1838049	38026	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	410	6	1	8	0.4	COCCNC(=O)/C(C#N)=C/c1c(N2CCN(C)CC2)nc2c(C)cccn2c1=O	nan
	CHEMBL1462354	38026	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	410	6	1	8	0.4	COCCNC(=O)/C(C#N)=C/c1c(N2CCN(C)CC2)nc2c(C)cccn2c1=O	nan
	15945416	38768	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	472	7	1	7	3.5	COc1ccc(S(=O)(=O)N2CCCCC2)cc1NC(=O)CSc1ncnc2ccccc12	nan
	CHEMBL1468328	38768	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	472	7	1	7	3.5	COc1ccc(S(=O)(=O)N2CCCCC2)cc1NC(=O)CSc1ncnc2ccccc12	nan
	4905842	38787	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	6	1	9	4.4	CSc1ccc(C2C(C(=O)c3ccco3)=C(O)C(=O)N2c2nnc(SC)s2)cc1	nan
	CHEMBL1468444	38787	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	6	1	9	4.4	CSc1ccc(C2C(C(=O)c3ccco3)=C(O)C(=O)N2c2nnc(SC)s2)cc1	nan
	6498441	38896	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	3	1	6	2.7	O=C(Cn1c2ccc(F)cc2c2nc3n(c(=O)c21)CCS3)NC1CCCC1	nan
	CHEMBL1469364	38896	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	3	1	6	2.7	O=C(Cn1c2ccc(F)cc2c2nc3n(c(=O)c21)CCS3)NC1CCCC1	nan
	4356276	38999	18	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	7	1	8	4.1	CCOc1ccc(C2C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2c2cc(C)on2)cc1OC	nan
	CHEMBL1470300	38999	18	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	7	1	8	4.1	CCOc1ccc(C2C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2c2cc(C)on2)cc1OC	nan
	3776625	39054	17	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	4	1	6	4.6	Cc1cc(N2C(=O)C(O)=C(C(=O)c3cccs3)C2c2cccc(Br)c2)no1	nan
	CHEMBL1470725	39054	17	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	4	1	6	4.6	Cc1cc(N2C(=O)C(O)=C(C(=O)c3cccs3)C2c2cccc(Br)c2)no1	nan
	3186626	39075	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	6	2	9	1.1	CCC(=O)Nc1cccc(NC(=O)CSc2nc3c(c(=O)n(C)c(=O)n3C)n2C)c1	nan
	CHEMBL1470851	39075	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	6	2	9	1.1	CCC(=O)Nc1cccc(NC(=O)CSc2nc3c(c(=O)n(C)c(=O)n3C)n2C)c1	nan
	7256722	39398	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	4	1	6	2.4	Cc1ccc2nc(SCC(=O)Nc3ccc(F)cc3F)nc(=O)n2c1	nan
	CHEMBL1474450	39398	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	4	1	6	2.4	Cc1ccc2nc(SCC(=O)Nc3ccc(F)cc3F)nc(=O)n2c1	nan
	15990395	39546	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	3	1	5	2.4	CC(=O)c1cccc(NC(=O)c2nc3ccccc3n(C)c2=O)c1	nan
	CHEMBL1476510	39546	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	3	1	5	2.4	CC(=O)c1cccc(NC(=O)c2nc3ccccc3n(C)c2=O)c1	nan
	1506838	39589	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	331	5	1	4	3.1	Cc1cc(CNC(=O)COc2ccc(C#N)cc2)c2ccccc2n1	nan
	CHEMBL1477044	39589	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	331	5	1	4	3.1	Cc1cc(CNC(=O)COc2ccc(C#N)cc2)c2ccccc2n1	nan
	1471774	39632	22	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	242	2	1	4	3.0	CSc1cc(-c2ccccc2)nc(O)c1C#N	nan
	CHEMBL1477426	39632	22	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	242	2	1	4	3.0	CSc1cc(-c2ccccc2)nc(O)c1C#N	nan
	20970002	39642	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	6	1	6	2.5	COc1ccc(CN2C(=O)c3cccnc3C2=O)cc1S(=O)(=O)NC1CCCCC1	nan
	CHEMBL1477514	39642	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	6	1	6	2.5	COc1ccc(CN2C(=O)c3cccnc3C2=O)cc1S(=O)(=O)NC1CCCCC1	nan
	2931382	39936	13	None	-1	3	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	309	4	2	5	2.1	COC(=O)c1sccc1NC(=O)C1CC=CCC1C(=O)O	nan
	CHEMBL1480089	39936	13	None	-1	3	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	309	4	2	5	2.1	COC(=O)c1sccc1NC(=O)C1CC=CCC1C(=O)O	nan
	7120051	39943	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	324	2	1	5	3.8	COc1ccc(-n2c(=S)[nH]c3c(oc4ccccc43)c2=O)cc1	nan
	CHEMBL1480178	39943	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	324	2	1	5	3.8	COc1ccc(-n2c(=S)[nH]c3c(oc4ccccc43)c2=O)cc1	nan
	16018856	39963	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	5	0	8	5.5	COc1ccc(-c2nc(CSc3nnc(C)n4c3cc3sccc34)c(C)o2)cc1	nan
	CHEMBL1480328	39963	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	5	0	8	5.5	COc1ccc(-c2nc(CSc3nnc(C)n4c3cc3sccc34)c(C)o2)cc1	nan
	3451317	39976	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	6	1	7	0.8	CN(C)S(=O)(=O)c1cccc(NC(=O)CSc2nncn2C)c1	nan
	CHEMBL1480436	39976	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	6	1	7	0.8	CN(C)S(=O)(=O)c1cccc(NC(=O)CSc2nncn2C)c1	nan
	3535142	40097	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	9	1	9	3.4	O=C(O)CCCCCn1c(SCc2cc(=O)n3ccccc3n2)nc2ccsc2c1=O	nan
	CHEMBL1481365	40097	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	9	1	9	3.4	O=C(O)CCCCCn1c(SCc2cc(=O)n3ccccc3n2)nc2ccsc2c1=O	nan
	3574141	40148	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	8	0	6	2.1	CCN(CC)S(=O)(=O)c1ccc(N2CCCC2)c(C(=O)OCC(=O)N2CCCC2)c1	nan
	CHEMBL1481920	40148	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	8	0	6	2.1	CCN(CC)S(=O)(=O)c1ccc(N2CCCC2)c(C(=O)OCC(=O)N2CCCC2)c1	nan
	5736472	40440	10	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	6	1	7	2.5	O=c1c2ccccc2nc(/C=C/c2ccc([N+](=O)[O-])o2)n1CCCO	nan
	CHEMBL1484332	40440	10	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	6	1	7	2.5	O=c1c2ccccc2nc(/C=C/c2ccc([N+](=O)[O-])o2)n1CCCO	nan
	5304429	40469	14	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	252	2	1	4	2.4	CC(=O)Nc1cccc(-c2cn3cccnc3n2)c1	nan
	CHEMBL1484671	40469	14	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	252	2	1	4	2.4	CC(=O)Nc1cccc(-c2cn3cccnc3n2)c1	nan
	16012070	40505	1	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	3	1	7	2.9	Cc1cc(=O)n2nc(N3CCC(C(=O)Nc4c(C)cccc4C)CC3)sc2n1	nan
	CHEMBL1484919	40505	1	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	3	1	7	2.9	Cc1cc(=O)n2nc(N3CCC(C(=O)Nc4c(C)cccc4C)CC3)sc2n1	nan
	4399091	40507	18	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	5	1	7	3.7	COc1ccccc1C1C(C(=O)c2ccc(C)o2)=C(O)C(=O)N1c1cc(C)on1	nan
	CHEMBL1484932	40507	18	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	5	1	7	3.7	COc1ccccc1C1C(C(=O)c2ccc(C)o2)=C(O)C(=O)N1c1cc(C)on1	nan
	1387364	40562	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	4	1	7	2.2	CNS(=O)(=O)c1ccc(OC)c(-c2nnc3c4ccccc4c(C)nn23)c1	nan
	CHEMBL1485560	40562	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	4	1	7	2.2	CNS(=O)(=O)c1ccc(OC)c(-c2nnc3c4ccccc4c(C)nn23)c1	nan
	CHEMBL1576237	40562	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	4	1	7	2.2	CNS(=O)(=O)c1ccc(OC)c(-c2nnc3c4ccccc4c(C)nn23)c1	nan
	6622721	40833	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	309	2	1	5	3.6	CNc1nc2c(-c3ccc(Cl)cc3)nnn2c2ccccc12	nan
	CHEMBL1487831	40833	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	309	2	1	5	3.6	CNc1nc2c(-c3ccc(Cl)cc3)nnn2c2ccccc12	nan
	1002526	40874	11	None	-2	3	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	2	1	4	4.1	O=C(O)c1cc(-c2ccc3c(c2)OCO3)nc2ccc(Br)cc12	nan
	CHEMBL1488092	40874	11	None	-2	3	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	2	1	4	4.1	O=C(O)c1cc(-c2ccc3c(c2)OCO3)nc2ccc(Br)cc12	nan
	7190684	40932	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	6	1	8	2.9	COc1ccc(NC(=O)CSc2ccc3nnc(-c4cccnc4)n3n2)cc1	nan
	CHEMBL1488468	40932	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	6	1	8	2.9	COc1ccc(NC(=O)CSc2ccc3nnc(-c4cccnc4)n3n2)cc1	nan
	5881431	41031	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	8	1	7	4.2	C=CCOc1cccc(C2C(C(=O)c3ccc4c(c3)OCCO4)=C(O)C(=O)N2Cc2cccnc2)c1	nan
	CHEMBL1489225	41031	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	8	1	7	4.2	C=CCOc1cccc(C2C(C(=O)c3ccc4c(c3)OCCO4)=C(O)C(=O)N2Cc2cccnc2)c1	nan
	2032322	41146	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	8	1	7	3.5	CCN(CC)CCCNc1nc(SC)nc2sc3c(c12)CCN(C)C3	nan
	CHEMBL1490215	41146	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	8	1	7	3.5	CCN(CC)CCCNc1nc(SC)nc2sc3c(c12)CCN(C)C3	nan
	755499	41253	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	300	2	0	7	1.0	COC(=O)Cn1cnc2c(C#N)c3n(c2c1=O)CCCCC3	nan
	CHEMBL1490891	41253	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	300	2	0	7	1.0	COC(=O)Cn1cnc2c(C#N)c3n(c2c1=O)CCCCC3	nan
	1283516	41444	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	324	2	1	7	0.9	O=c1[nH]n2cc(-n3cc([N+](=O)[O-])cn3)cnc2c1Br	nan
	CHEMBL1492212	41444	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	324	2	1	7	0.9	O=c1[nH]n2cc(-n3cc([N+](=O)[O-])cn3)cnc2c1Br	nan
	774862	41511	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	253	2	0	4	3.1	Cn1c(-c2ccc([N+](=O)[O-])cc2)nc2ccccc21	nan
	CHEMBL1492732	41511	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	253	2	0	4	3.1	Cn1c(-c2ccc([N+](=O)[O-])cc2)nc2ccccc21	nan
	3279901	41606	7	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	5	2	4	3.0	CC(=O)NC(CSc1cc(C)nc2ccc(Br)cc12)C(=O)O	nan
	CHEMBL1493652	41606	7	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	5	2	4	3.0	CC(=O)NC(CSc1cc(C)nc2ccc(Br)cc12)C(=O)O	nan
	4795978	41609	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	5	0	5	3.8	CN(C)S(=O)(=O)c1cccc(COc2ncnc3c(Cl)cc(Cl)cc23)c1	nan
	CHEMBL1493688	41609	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	5	0	5	3.8	CN(C)S(=O)(=O)c1cccc(COc2ncnc3c(Cl)cc(Cl)cc23)c1	nan
	15988336	41690	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	6	1	8	1.9	COc1cccc(CNC(=O)CCc2nnc3n(C)c(=O)c4sccc4n23)c1	nan
	CHEMBL1494501	41690	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	6	1	8	1.9	COc1cccc(CNC(=O)CCc2nnc3n(C)c(=O)c4sccc4n23)c1	nan
	664285	41707	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	258	3	0	5	3.1	CC(=O)CSc1ncnc2c1oc1ccccc12	nan
	CHEMBL1494683	41707	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	258	3	0	5	3.1	CC(=O)CSc1ncnc2c1oc1ccccc12	nan
	748270	41748	41	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	218	0	0	4	2.2	Cc1nnc2c3ccccc3c(Cl)nn12	nan
	CHEMBL1495086	41748	41	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	218	0	0	4	2.2	Cc1nnc2c3ccccc3c(Cl)nn12	nan
	3186635	41858	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	4	0	9	-0.8	CCN1CCN(C(=O)CSc2nc3c(c(=O)n(C)c(=O)n3C)n2C)CC1	nan
	CHEMBL1496152	41858	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	4	0	9	-0.8	CCN1CCN(C(=O)CSc2nc3c(c(=O)n(C)c(=O)n3C)n2C)CC1	nan
	2561752	42094	17	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	4	1	6	3.2	COCCCn1c(=S)[nH]c2sc3c(c2c1=O)CCCS3	nan
	CHEMBL1498284	42094	17	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	4	1	6	3.2	COCCCn1c(=S)[nH]c2sc3c(c2c1=O)CCCS3	nan
	21552	42138	4	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	299	2	1	7	0.1	Cn1c(=O)c2c(nc(Cc3ccc(N)cc3)n2C)n(C)c1=O	nan
	CHEMBL1498782	42138	4	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	299	2	1	7	0.1	Cn1c(=O)c2c(nc(Cc3ccc(N)cc3)n2C)n(C)c1=O	nan
	7677140	42191	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	3	1	5	2.7	O=C(NCc1nnc2c(C(F)(F)F)cc(Cl)cn12)c1cccnc1	nan
	CHEMBL1499143	42191	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	3	1	5	2.7	O=C(NCc1nnc2c(C(F)(F)F)cc(Cl)cn12)c1cccnc1	nan
	2816379	42355	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	330	5	0	8	2.1	CCOC(=O)c1nnn2c1nc(SCC(C)=O)c1ccccc12	nan
	CHEMBL1500551	42355	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	330	5	0	8	2.1	CCOC(=O)c1nnn2c1nc(SCC(C)=O)c1ccccc12	nan
	18554434	42392	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	7	1	8	1.8	O=C(CSc1ncnc2c1nnn2Cc1ccccc1F)NCC1CCCO1	nan
	CHEMBL1500823	42392	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	7	1	8	1.8	O=C(CSc1ncnc2c1nnn2Cc1ccccc1F)NCC1CCCO1	nan
	5077853	42476	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	478	5	1	8	1.5	COc1ccc(-n2nc(C(=O)NCC(=O)N3CCC4(CC3)OCCO4)c3ccccc3c2=O)cc1	nan
	CHEMBL1501692	42476	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	478	5	1	8	1.5	COc1ccc(-n2nc(C(=O)NCC(=O)N3CCC4(CC3)OCCO4)c3ccccc3c2=O)cc1	nan
	7120056	42481	9	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	308	1	1	4	4.1	Cc1ccc(-n2c(=S)[nH]c3c(oc4ccccc43)c2=O)cc1	nan
	CHEMBL1501734	42481	9	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	308	1	1	4	4.1	Cc1ccc(-n2c(=S)[nH]c3c(oc4ccccc43)c2=O)cc1	nan
	3884053	42636	14	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	7	1	5	4.0	CN(C)CCCN1C(=O)C(O)=C(C(=O)c2cc3ccccc3o2)C1c1ccccc1	nan
	661074	42636	14	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	7	1	5	4.0	CN(C)CCCN1C(=O)C(O)=C(C(=O)c2cc3ccccc3o2)C1c1ccccc1	nan
	CHEMBL1503060	42636	14	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	7	1	5	4.0	CN(C)CCCN1C(=O)C(O)=C(C(=O)c2cc3ccccc3o2)C1c1ccccc1	nan
	20957430	42673	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	8	2	9	3.2	CC(=O)c1cccc(NC(=O)CCc2nnc3ccc(NCc4ccc5c(c4)OCO5)nn23)c1	nan
	CHEMBL1503367	42673	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	8	2	9	3.2	CC(=O)c1cccc(NC(=O)CCc2nnc3ccc(NCc4ccc5c(c4)OCO5)nn23)c1	nan
	16452701	42779	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	6	2	8	2.7	Cc1cc(C)nc(NS(=O)(=O)c2ccc(NC(=O)c3nn(-c4ccccc4)ccc3=O)cc2)n1	nan
	CHEMBL1504372	42779	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	6	2	8	2.7	Cc1cc(C)nc(NS(=O)(=O)c2ccc(NC(=O)c3nn(-c4ccccc4)ccc3=O)cc2)n1	nan
	3457991	42909	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	520	5	1	8	3.2	Cc1ccc(F)cc1NC(=O)c1sc2ncn(CC(=O)N3CCN(c4ccccn4)CC3)c(=O)c2c1C	nan
	CHEMBL1505540	42909	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	520	5	1	8	3.2	Cc1ccc(F)cc1NC(=O)c1sc2ncn(CC(=O)N3CCN(c4ccccn4)CC3)c(=O)c2c1C	nan
	5198374	42923	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	6	1	7	2.4	O=C(CSc1ncnc2ccccc12)Nc1cccc(S(=O)(=O)N2CCOCC2)c1	nan
	CHEMBL1505625	42923	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	6	1	7	2.4	O=C(CSc1ncnc2ccccc12)Nc1cccc(S(=O)(=O)N2CCOCC2)c1	nan
	986582	43025	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	358	4	2	4	3.2	CCc1ccc2oc(C(=O)Nc3ccc(S(N)(=O)=O)cc3)c(C)c2c1	nan
	CHEMBL1506399	43025	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	358	4	2	4	3.2	CCc1ccc2oc(C(=O)Nc3ccc(S(N)(=O)=O)cc3)c(C)c2c1	nan
	1811810	43058	14	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	5	1	2	3.5	C=CCNC(=O)Cc1c(OC)ccc2cc(Br)ccc12	nan
	CHEMBL1506727	43058	14	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	5	1	2	3.5	C=CCNC(=O)Cc1c(OC)ccc2cc(Br)ccc12	nan
	135528107	43580	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	6	2	5	3.2	CCN(CC(=O)NC(C)C)Cc1nc(O)c2cc(Br)cc(Br)c2n1	nan
	CHEMBL1511291	43580	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	6	2	5	3.2	CCN(CC(=O)NC(C)C)Cc1nc(O)c2cc(Br)cc(Br)c2n1	nan
	16496658	43696	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	5	1	5	3.1	CC1CCCN(C(=O)COC(=O)CNC(=O)c2sc3ccccc3c2Cl)C1	nan
	CHEMBL1512634	43696	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	5	1	5	3.1	CC1CCCN(C(=O)COC(=O)CNC(=O)c2sc3ccccc3c2Cl)C1	nan
	15988304	43774	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	4	0	8	1.9	Cn1c(=O)c2sccc2n2c(CCC(=O)N3CCN(c4ccccc4)CC3)nnc12	nan
	CHEMBL1513808	43774	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	4	0	8	1.9	Cn1c(=O)c2sccc2n2c(CCC(=O)N3CCN(c4ccccc4)CC3)nnc12	nan
	16026221	43889	0	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	4	0	7	1.2	CCOC(=O)C1CCN(C(=O)Cn2c(=O)cc(C)c3c(C)nn(C)c32)CC1	nan
	CHEMBL1515615	43889	0	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	4	0	7	1.2	CCOC(=O)C1CCN(C(=O)Cn2c(=O)cc(C)c3c(C)nn(C)c32)CC1	nan
	662069	44042	9	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	2	0	6	1.8	COC(=O)c1cc(Br)c(=O)n(-c2nccs2)c1	nan
	CHEMBL1517409	44042	9	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	2	0	6	1.8	COC(=O)c1cc(Br)c(=O)n(-c2nccs2)c1	nan
	3489758	44100	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	3	2	9	0.9	Cn1c(=O)c2ncn(CC(=O)N=Nc3c(O)[nH]c4ccccc34)c2n(C)c1=O	nan
	CHEMBL1518029	44100	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	3	2	9	0.9	Cn1c(=O)c2ncn(CC(=O)N=Nc3c(O)[nH]c4ccccc34)c2n(C)c1=O	nan
	16018686	44263	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	4	1	6	4.3	Cc1cc2c(cc3c(SCC(=O)Nc4ccc(Cl)cc4F)nncn32)o1	nan
	CHEMBL1519470	44263	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	4	1	6	4.3	Cc1cc2c(cc3c(SCC(=O)Nc4ccc(Cl)cc4F)nncn32)o1	nan
	20957225	44281	4	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	423	5	1	9	1.7	Cc1ccc(NC(=O)CCc2nnc3ccc(N4CCC5(CC4)OCCO5)nn23)nc1	nan
	CHEMBL1519640	44281	4	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	423	5	1	9	1.7	Cc1ccc(NC(=O)CCc2nnc3ccc(N4CCC5(CC4)OCCO5)nn23)nc1	nan
	2991435	44299	14	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	4	1	6	2.8	COC(=O)c1ccc(N2CCN(C)CC2)c(NC(=O)c2ccc(Br)o2)c1	nan
	CHEMBL1519787	44299	14	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	4	1	6	2.8	COC(=O)c1ccc(N2CCN(C)CC2)c(NC(=O)c2ccc(Br)o2)c1	nan
	5959865	44413	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	461	7	1	6	4.0	CC1Cc2cc(C(=O)C3=C(O)C(=O)N(CCCn4ccnc4)C3c3ccc(F)cc3)ccc2O1	nan
	CHEMBL1520789	44413	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	461	7	1	6	4.0	CC1Cc2cc(C(=O)C3=C(O)C(=O)N(CCCn4ccnc4)C3c3ccc(F)cc3)ccc2O1	nan
	4197564	44578	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	512	11	1	8	3.9	COc1cc(C2C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2CCN2CCOCC2)ccc1OCCC(C)C	nan
	CHEMBL1522190	44578	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	512	11	1	8	3.9	COc1cc(C2C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2CCN2CCOCC2)ccc1OCCC(C)C	nan
	5064245	44595	4	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	287	5	1	5	1.3	O=C(COc1ncnc2ccccc12)NCC1CCCO1	nan
	CHEMBL1522316	44595	4	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	287	5	1	5	1.3	O=C(COc1ncnc2ccccc12)NCC1CCCO1	nan
	3317909	44598	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	518	7	1	7	4.6	COc1cccc2cc(C(=O)C3=C(O)C(=O)N(CCN4CCOCC4)C3c3ccc(C(C)(C)C)cc3)oc12	nan
	3536112	44598	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	518	7	1	7	4.6	COc1cccc2cc(C(=O)C3=C(O)C(=O)N(CCN4CCOCC4)C3c3ccc(C(C)(C)C)cc3)oc12	nan
	CHEMBL1522365	44598	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	518	7	1	7	4.6	COc1cccc2cc(C(=O)C3=C(O)C(=O)N(CCN4CCOCC4)C3c3ccc(C(C)(C)C)cc3)oc12	nan
	20957467	44673	4	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	9	1	8	1.8	O=C1CCCN1CCCNc1ccc2nnc(CCC(=O)N3CCN(c4ccccc4)CC3)n2n1	nan
	CHEMBL1523099	44673	4	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	9	1	8	1.8	O=C1CCCN1CCCNc1ccc2nnc(CCC(=O)N3CCN(c4ccccc4)CC3)n2n1	nan
	3242118	44686	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	288	2	1	5	2.6	Cc1nn(C(C)C(=O)O)c(=O)c2c1sc1ccccc12	nan
	CHEMBL1523214	44686	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	288	2	1	5	2.6	Cc1nn(C(C)C(=O)O)c(=O)c2c1sc1ccccc12	nan
	3178468	44744	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	4	0	8	0.6	CCn1c(SCC(=O)N2CCCCC2)nc2c1c(=O)n(C)c(=O)n2C	nan
	CHEMBL1523743	44744	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	4	0	8	0.6	CCn1c(SCC(=O)N2CCCCC2)nc2c1c(=O)n(C)c(=O)n2C	nan
	774385	44966	50	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	192	1	1	4	2.3	Cc1ccccc1-c1nnc(S)o1	nan
	CHEMBL1525902	44966	50	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	192	1	1	4	2.3	Cc1ccccc1-c1nnc(S)o1	nan
	6156848	44979	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	7	1	6	3.9	CC1Cc2cc(C(=O)C3=C(O)C(=O)N(CCCn4ccnc4)C3c3ccccc3)ccc2O1	nan
	CHEMBL1525999	44979	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	7	1	6	3.9	CC1Cc2cc(C(=O)C3=C(O)C(=O)N(CCCn4ccnc4)C3c3ccccc3)ccc2O1	nan
	20923115	45238	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	7	0	6	3.1	CCN(c1ccccc1)S(=O)(=O)c1cc(CN2C(=O)c3cccnc3C2=O)ccc1OC	nan
	CHEMBL1528270	45238	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	7	0	6	3.1	CCN(c1ccccc1)S(=O)(=O)c1cc(CN2C(=O)c3cccnc3C2=O)ccc1OC	nan
	1173803	45348	1	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	6	0	9	0.3	CCCn1c(SCCN2CCOCC2)nc2c1c(=O)n(C)c(=O)n2C	nan
	CHEMBL1529195	45348	1	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	6	0	9	0.3	CCCn1c(SCCN2CCOCC2)nc2c1c(=O)n(C)c(=O)n2C	nan
	1150969	45349	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	7	2	6	3.2	CCOc1ccccc1C(=O)Nc1ccc(S(=O)(=O)Nc2nccc(C)n2)cc1	nan
	CHEMBL1529199	45349	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	7	2	6	3.2	CCOc1ccccc1C(=O)Nc1ccc(S(=O)(=O)Nc2nccc(C)n2)cc1	nan
	20957502	45416	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	11	2	8	1.8	COc1cccc(CNC(=O)CCc2nnc3ccc(NCCCN4CCCC4=O)nn23)c1	nan
	CHEMBL1529803	45416	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	11	2	8	1.8	COc1cccc(CNC(=O)CCc2nnc3ccc(NCCCN4CCCC4=O)nn23)c1	nan
	3146230	45598	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	5	1	6	2.7	Cc1sc2ncnc(SCC(=O)NCC3CCCO3)c2c1C	nan
	CHEMBL1531505	45598	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	5	1	6	2.7	Cc1sc2ncnc(SCC(=O)NCC3CCCO3)c2c1C	nan
	20888842	45862	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	8	1	9	1.6	CCCS(=O)(=O)c1nc(S(=O)(=O)c2ccc(C)cc2)c(N2CCN(CCO)CC2)s1	nan
	CHEMBL1533752	45862	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	8	1	9	1.6	CCCS(=O)(=O)c1nc(S(=O)(=O)c2ccc(C)cc2)c(N2CCN(CCO)CC2)s1	nan
	7677714	45864	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	358	3	1	5	3.2	Cc1ccc(C(=O)NCc2nnc3c(C(F)(F)F)cc(Cl)cn23)o1	nan
	CHEMBL1533761	45864	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	358	3	1	5	3.2	Cc1ccc(C(=O)NCc2nnc3c(C(F)(F)F)cc(Cl)cn23)o1	nan
	16018626	45910	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	6	1	8	3.2	COc1ccc(NC(=O)CSc2nncn3c2cc2occc23)c(OC)c1	nan
	CHEMBL1534283	45910	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	6	1	8	3.2	COc1ccc(NC(=O)CSc2nncn3c2cc2occc23)c(OC)c1	nan
	2415319	45912	24	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	3	1	5	4.0	O=C(O)c1ccccc1Sc1ncnc2sc3c(c12)CCC3	nan
	CHEMBL1534296	45912	24	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	3	1	5	4.0	O=C(O)c1ccccc1Sc1ncnc2sc3c(c12)CCC3	nan
	15988400	45941	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	6	1	7	3.0	CCn1c(=O)c2sccc2n2c(CCC(=O)NCc3ccc(Cl)cc3)nnc12	nan
	CHEMBL1534534	45941	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	6	1	7	3.0	CCn1c(=O)c2sccc2n2c(CCC(=O)NCc3ccc(Cl)cc3)nnc12	nan
	3559456	46044	14	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	478	4	1	6	5.3	Cc1cc(N2C(=O)C(O)=C(C(=O)c3cc4ccccc4o3)C2c2cccc(Br)c2)no1	nan
	CHEMBL1535636	46044	14	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	478	4	1	6	5.3	Cc1cc(N2C(=O)C(O)=C(C(=O)c3cc4ccccc4o3)C2c2cccc(Br)c2)no1	nan
	752859	46067	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	291	2	1	6	2.6	Cn1cc(Cl)c(-c2nnc(S)n2-c2ccccc2)n1	nan
	CHEMBL1535864	46067	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	291	2	1	6	2.6	Cn1cc(Cl)c(-c2nnc(S)n2-c2ccccc2)n1	nan
	1258096	46102	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	3	1	7	3.1	O=c1c2ccccc2cnn1Cc1nnc(S)n1-c1ccc(F)c(Cl)c1	nan
	CHEMBL1536340	46102	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	3	1	7	3.1	O=c1c2ccccc2cnn1Cc1nnc(S)n1-c1ccc(F)c(Cl)c1	nan
	5911396	46126	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	4	1	8	3.5	Cc1nnc(N2C(=O)C(O)=C(C(=O)c3ccc4c(c3)OCCO4)C2c2ccc(F)cc2)s1	nan
	CHEMBL1536589	46126	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	4	1	8	3.5	Cc1nnc(N2C(=O)C(O)=C(C(=O)c3ccc4c(c3)OCCO4)C2c2ccc(F)cc2)s1	nan
	2968508	46227	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	4	3	4	3.4	O=C(COc1ccccc1)NC(=S)Nc1cccc2cc(O)ccc12	nan
	CHEMBL1537461	46227	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	4	3	4	3.4	O=C(COc1ccccc1)NC(=S)Nc1cccc2cc(O)ccc12	nan
	973903	46387	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	3	3	7	1.5	O=C(NNc1nc(=O)c2cccnc2s1)c1ccccc1O	nan
	CHEMBL1538711	46387	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	3	3	7	1.5	O=C(NNc1nc(=O)c2cccnc2s1)c1ccccc1O	nan
	4786350	46440	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	284	4	0	6	2.6	COC(=O)c1ccc(COc2ncnc3ccccc23)o1	nan
	CHEMBL1539182	46440	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	284	4	0	6	2.6	COC(=O)c1ccc(COc2ncnc3ccccc23)o1	nan
	4199276	46447	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	4	2	10	-0.3	Cn1c(=O)c2nc(NNC(=O)c3ccc([N+](=O)[O-])cc3)cnc2n(C)c1=O	nan
	CHEMBL1539261	46447	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	4	2	10	-0.3	Cn1c(=O)c2nc(NNC(=O)c3ccc([N+](=O)[O-])cc3)cnc2n(C)c1=O	nan
	20957177	46472	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	6	1	8	2.4	O=C(CCc1nnc2ccc(N3CCC4(CC3)OCCO4)nn12)NCc1ccccc1Cl	nan
	CHEMBL1539515	46472	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	6	1	8	2.4	O=C(CCc1nnc2ccc(N3CCC4(CC3)OCCO4)nn12)NCc1ccccc1Cl	nan
	775376	46756	16	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	319	3	1	7	-0.1	Cn1c(=O)c2c(ncn2CC(=O)NC2CCCCC2)n(C)c1=O	nan
	CHEMBL1541812	46756	16	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	319	3	1	7	-0.1	Cn1c(=O)c2c(ncn2CC(=O)NC2CCCCC2)n(C)c1=O	nan
	2027988	46846	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	3	1	7	2.5	O=c1c2ccccc2cnn1Cc1nnc(S)n1-c1ccc(F)cc1	nan
	CHEMBL1542663	46846	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	3	1	7	2.5	O=c1c2ccccc2cnn1Cc1nnc(S)n1-c1ccc(F)cc1	nan
	7190638	47017	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	5	1	7	2.9	O=C(CSc1ccc2nnc(-c3cccnc3)n2n1)Nc1ccccc1	nan
	CHEMBL1544038	47017	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	5	1	7	2.9	O=C(CSc1ccc2nnc(-c3cccnc3)n2n1)Nc1ccccc1	nan
	5291252	47074	18	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	4	1	4	4.3	Cc1ccc(C(=O)C2=C(O)C(=O)N(c3ccccn3)C2c2ccc(F)cc2)cc1	nan
	CHEMBL1544399	47074	18	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	4	1	4	4.3	Cc1ccc(C(=O)C2=C(O)C(=O)N(c3ccccn3)C2c2ccc(F)cc2)cc1	nan
	3531704	47134	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	6	1	7	5.5	Cc1cc(N2C(=O)C(O)=C(C(=O)c3ccc(C)o3)C2c2cccc(Oc3ccccc3)c2)no1	nan
	CHEMBL1544885	47134	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	6	1	7	5.5	Cc1cc(N2C(=O)C(O)=C(C(=O)c3ccc(C)o3)C2c2cccc(Oc3ccccc3)c2)no1	nan
	1254436	47171	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	2	1	10	-0.3	Cn1c(=O)c2c(nc(Br)n2Cc2nnc(N)s2)n(C)c1=O	nan
	CHEMBL1545144	47171	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	2	1	10	-0.3	Cn1c(=O)c2c(nc(Br)n2Cc2nnc(N)s2)n(C)c1=O	nan
	20923178	47214	4	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	441	7	1	7	2.3	COc1ccc(CN2C(=O)c3cccnc3C2=O)cc1S(=O)(=O)NCc1ccc(C)o1	nan
	CHEMBL1545457	47214	4	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	441	7	1	7	2.3	COc1ccc(CN2C(=O)c3cccnc3C2=O)cc1S(=O)(=O)NCc1ccc(C)o1	nan
	2827527	47227	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	189	0	0	2	3.2	Cc1ccc2c(ccc(=S)n2C)c1	nan
	CHEMBL1545583	47227	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	189	0	0	2	3.2	Cc1ccc2c(ccc(=S)n2C)c1	nan
	4114707	47279	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	356	5	1	6	2.6	Cc1cc2nnc(SCC(=O)NCC3CCCO3)n2c2ccccc12	nan
	CHEMBL1546017	47279	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	356	5	1	6	2.6	Cc1cc2nnc(SCC(=O)NCC3CCCO3)n2c2ccccc12	nan
	6620293	47357	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	2	0	5	3.8	O=C(C1CCN(c2ncnc3c2sc2cccc(F)c23)CC1)N1CCCC1	nan
	CHEMBL1546743	47357	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	2	0	5	3.8	O=C(C1CCN(c2ncnc3c2sc2cccc(F)c23)CC1)N1CCCC1	nan
	2341870	47367	2	None	-3	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	2	0	5	4.1	Cc1ccc(C)n1-c1ccc(-c2nnc3n2CCCCC3)s1	nan
	CHEMBL1546820	47367	2	None	-3	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	2	0	5	4.1	Cc1ccc(C)n1-c1ccc(-c2nnc3n2CCCCC3)s1	nan
	2150404	47610	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	294	1	1	4	3.8	O=c1c2oc3ccccc3c2[nH]c(=S)n1-c1ccccc1	nan
	CHEMBL1549101	47610	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	294	1	1	4	3.8	O=c1c2oc3ccccc3c2[nH]c(=S)n1-c1ccccc1	nan
	2482804	47713	1	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	318	5	2	8	-0.4	C=CCNC(=O)NC(=O)COC(=O)c1nc2nccc(C)n2n1	nan
	CHEMBL1549963	47713	1	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	318	5	2	8	-0.4	C=CCNC(=O)NC(=O)COC(=O)c1nc2nccc(C)n2n1	nan
	7184632	47842	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	6	1	8	2.6	COc1ccc(NC(=O)CCCc2nnc3n(C)c(=O)c4sccc4n23)cc1	nan
	CHEMBL1550958	47842	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	6	1	8	2.6	COc1ccc(NC(=O)CCCc2nnc3n(C)c(=O)c4sccc4n23)cc1	nan
	16030519	47860	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	8	1	5	4.6	COc1ccc(CNC(=O)CSc2nc3ccccc3nc2Cc2ccccc2)cc1	nan
	CHEMBL1551209	47860	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	8	1	5	4.6	COc1ccc(CNC(=O)CSc2nc3ccccc3nc2Cc2ccccc2)cc1	nan
	1116231	47964	15	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	3	1	7	1.4	Cn1c(=O)c2c(ncn2CC(=O)Nc2cccc(Cl)c2Cl)n(C)c1=O	nan
	CHEMBL1552691	47964	15	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	3	1	7	1.4	Cn1c(=O)c2c(ncn2CC(=O)Nc2cccc(Cl)c2Cl)n(C)c1=O	nan
	16031533	47974	2	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	7	1	6	4.5	CCc1ccccc1NC(=O)CSc1nnc(-c2ccc(OC)cc2)s1	nan
	CHEMBL1552858	47974	2	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	7	1	6	4.5	CCc1ccccc1NC(=O)CSc1nnc(-c2ccc(OC)cc2)s1	nan
	16033232	47984	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	5	1	5	5.4	Cc1c(C(=O)NCc2cccc(Cl)c2)sc2ncnc(N(C)C3CCCCC3)c12	nan
	CHEMBL1552980	47984	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	5	1	5	5.4	Cc1c(C(=O)NCc2cccc(Cl)c2)sc2ncnc(N(C)C3CCCCC3)c12	nan
	2136319	48006	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	502	7	1	7	4.2	CCOc1ccc(NC(=O)Cn2cc(C(=O)c3ccc(F)cc3)c(=O)c3cc4c(cc32)OCCO4)cc1	nan
	CHEMBL1553213	48006	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	502	7	1	7	4.2	CCOc1ccc(NC(=O)Cn2cc(C(=O)c3ccc(F)cc3)c(=O)c3cc4c(cc32)OCCO4)cc1	nan
	16018758	48065	0	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	3	0	5	4.5	Cc1cc2c(cc3c(SCc4cccc(F)c4)nnc(C)n32)o1	nan
	CHEMBL1554096	48065	0	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	3	0	5	4.5	Cc1cc2c(cc3c(SCc4cccc(F)c4)nnc(C)n32)o1	nan
	4808155	48243	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	318	4	0	7	0.7	Cn1c(=O)c2c(ncn2CCOc2ccc(F)cc2)n(C)c1=O	nan
	CHEMBL1556293	48243	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	318	4	0	7	0.7	Cn1c(=O)c2c(ncn2CCOc2ccc(F)cc2)n(C)c1=O	nan
	664905	48382	16	None	1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	5	1	6	3.4	O=C(CSc1ncnc2c1oc1ccccc12)NCc1ccco1	nan
	CHEMBL1557499	48382	16	None	1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	5	1	6	3.4	O=C(CSc1ncnc2c1oc1ccccc12)NCc1ccco1	nan
	846378	48496	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	334	4	0	5	3.8	CN(C)CCn1c2ccccc2c2nc3ccc([N+](=O)[O-])cc3cc21	nan
	CHEMBL1558527	48496	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	334	4	0	5	3.8	CN(C)CCn1c2ccccc2c2nc3ccc([N+](=O)[O-])cc3cc21	nan
	20970070	48632	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	481	9	1	7	2.8	CCOc1ccc(CNS(=O)(=O)c2cc(CN3C(=O)c4cccnc4C3=O)ccc2OC)cc1	nan
	CHEMBL1559703	48632	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	481	9	1	7	2.8	CCOc1ccc(CNS(=O)(=O)c2cc(CN3C(=O)c4cccnc4C3=O)ccc2OC)cc1	nan
	749967	48832	50	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	208	2	1	5	2.0	COc1ccccc1-c1nnc(S)o1	nan
	CHEMBL1561641	48832	50	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	208	2	1	5	2.0	COc1ccccc1-c1nnc(S)o1	nan
	2816163	49003	22	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	272	2	0	7	0.8	CCOC(=O)c1nnn2c3ccccc3c(=O)n(C)c12	nan
	CHEMBL1563125	49003	22	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	272	2	0	7	0.8	CCOC(=O)c1nnn2c3ccccc3c(=O)n(C)c12	nan
	754624	49097	15	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	313	2	0	6	3.0	O=c1c2c(-c3ccc([N+](=O)[O-])cc3)csc2nc2n1CCC2	nan
	CHEMBL1563900	49097	15	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	313	2	0	6	3.0	O=c1c2c(-c3ccc([N+](=O)[O-])cc3)csc2nc2n1CCC2	nan
	20923125	49238	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	7	1	6	2.7	COc1ccc(CN2C(=O)c3cccnc3C2=O)cc1S(=O)(=O)NCc1ccc(C)cc1	nan
	CHEMBL1565225	49238	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	7	1	6	2.7	COc1ccc(CN2C(=O)c3cccnc3C2=O)cc1S(=O)(=O)NCc1ccc(C)cc1	nan
	5818870	49247	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	5	1	5	4.3	CC1Cc2cc(C(=O)C3=C(O)C(=O)N(Cc4cccnc4)C3c3ccccc3F)ccc2O1	nan
	CHEMBL1565288	49247	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	5	1	5	4.3	CC1Cc2cc(C(=O)C3=C(O)C(=O)N(Cc4cccnc4)C3c3ccccc3F)ccc2O1	nan
	702333	49729	15	None	-2	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	272	0	1	3	2.9	Cn1c(=S)[nH]c2c(c1=O)C(C)(C)Cc1ccccc1-2	nan
	CHEMBL1569119	49729	15	None	-2	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	272	0	1	3	2.9	Cn1c(=S)[nH]c2c(c1=O)C(C)(C)Cc1ccccc1-2	nan
	1072636	50066	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	483	6	1	11	1.0	CCn1c(SCC(=O)Nc2c(C)n(C)n(-c3ccccc3)c2=O)nc2c1c(=O)n(C)c(=O)n2C	nan
	CHEMBL1572163	50066	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	483	6	1	11	1.0	CCn1c(SCC(=O)Nc2c(C)n(C)n(-c3ccccc3)c2=O)nc2c1c(=O)n(C)c(=O)n2C	nan
	4912148	50074	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	5	1	8	3.6	CSc1nnc(N2C(=O)C(O)=C(C(=O)c3ccco3)C2c2ccccc2)s1	nan
	CHEMBL1572210	50074	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	5	1	8	3.6	CSc1nnc(N2C(=O)C(O)=C(C(=O)c3ccco3)C2c2ccccc2)s1	nan
	719137	50095	16	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	286	1	1	3	3.4	CCn1c(=S)[nH]c2c(c1=O)C(C)(C)Cc1ccccc1-2	nan
	CHEMBL1572461	50095	16	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	286	1	1	3	3.4	CCn1c(=S)[nH]c2c(c1=O)C(C)(C)Cc1ccccc1-2	nan
	22518619	50300	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	481	9	1	8	3.8	CC(C)OCCCn1c(SCC(=O)Nc2ccccc2C(F)(F)F)nc2nccnc2c1=O	nan
	CHEMBL1574369	50300	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	481	9	1	8	3.8	CC(C)OCCCn1c(SCC(=O)Nc2ccccc2C(F)(F)F)nc2nccnc2c1=O	nan
	3516975	50388	14	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	319	2	0	4	4.1	Cc1cc(-c2sccc2Br)nc(-n2cccc2)n1	nan
	CHEMBL1575467	50388	14	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	319	2	0	4	4.1	Cc1cc(-c2sccc2Br)nc(-n2cccc2)n1	nan
	2109682	50414	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	5	1	11	0.2	Cc1ccc(C)c(-n2nnnc2SCC(=O)c2c(N)n(C)c(=O)n(C)c2=O)c1	nan
	CHEMBL1575697	50414	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	5	1	11	0.2	Cc1ccc(C)c(-n2nnnc2SCC(=O)c2c(N)n(C)c(=O)n(C)c2=O)c1	nan
	16189479	50533	4	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	5	0	8	-0.2	Cn1c(=O)c(=O)n(C)c2cc(S(=O)(=O)N3CC(=O)N(CCc4ccccc4)C(=O)C3)ccc21	nan
	CHEMBL1576683	50533	4	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	5	0	8	-0.2	Cn1c(=O)c(=O)n(C)c2cc(S(=O)(=O)N3CC(=O)N(CCc4ccccc4)C(=O)C3)ccc21	nan
	1173783	50567	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	7	2	9	1.5	CCC(=O)Nc1ccc(NC(=O)CSc2nc3c(c(=O)n(C)c(=O)n3C)n2CC)cc1	nan
	CHEMBL1577034	50567	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	7	2	9	1.5	CCC(=O)Nc1ccc(NC(=O)CSc2nc3c(c(=O)n(C)c(=O)n3C)n2CC)cc1	nan
	2960985	50778	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	4	2	5	3.4	N=C(NOC(=O)COc1ccc2ccccc2c1Br)c1cccnc1	nan
	5740252	50778	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	4	2	5	3.4	N=C(NOC(=O)COc1ccc2ccccc2c1Br)c1cccnc1	nan
	9587839	50778	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	4	2	5	3.4	N=C(NOC(=O)COc1ccc2ccccc2c1Br)c1cccnc1	nan
	CHEMBL1578738	50778	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	4	2	5	3.4	N=C(NOC(=O)COc1ccc2ccccc2c1Br)c1cccnc1	nan
	3221467	50790	3	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	8	1	6	3.0	CCOC(=O)CNC(=O)CSc1nc(Cc2ccccc2)nc2ccccc12	nan
	CHEMBL1578803	50790	3	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	8	1	6	3.0	CCOC(=O)CNC(=O)CSc1nc(Cc2ccccc2)nc2ccccc12	nan
	6409200	50925	1	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	336	4	2	5	3.4	O=C(O)c1ccccc1CSc1n[nH]c2c3ccccc3nc-2n1	nan
	CHEMBL1580121	50925	1	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	336	4	2	5	3.4	O=C(O)c1ccccc1CSc1n[nH]c2c3ccccc3nc-2n1	nan
	20957463	50941	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	10	2	7	2.5	O=C(CCc1nnc2ccc(NCCCN3CCCC3=O)nn12)NCc1ccccc1Cl	nan
	CHEMBL1580225	50941	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	10	2	7	2.5	O=C(CCc1nnc2ccc(NCCCN3CCCC3=O)nn12)NCc1ccccc1Cl	nan
	929935	51024	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	331	1	2	6	4.2	CC(C)c1nc2sc3c(O)nc(S)nc3c2c2c1CCCC2	nan
	CHEMBL1580962	51024	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	331	1	2	6	4.2	CC(C)c1nc2sc3c(O)nc(S)nc3c2c2c1CCCC2	nan
	3220371	51032	3	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	6	1	6	2.9	CC(C)C(OC(=O)c1nsc(Cl)c1Cl)C(=O)NCC1CCCO1	nan
	CHEMBL1581023	51032	3	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	6	1	6	2.9	CC(C)C(OC(=O)c1nsc(Cl)c1Cl)C(=O)NCC1CCCO1	nan
	2916260	51109	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	478	8	1	10	0.1	CCN(CC)S(=O)(=O)c1ccc(OC)c(NC(=O)Cn2cnc3c2c(=O)n(C)c(=O)n3C)c1	nan
	CHEMBL1581657	51109	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	478	8	1	10	0.1	CCN(CC)S(=O)(=O)c1ccc(OC)c(NC(=O)Cn2cnc3c2c(=O)n(C)c(=O)n3C)c1	nan
	1324776	51205	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	9	2	8	2.9	CCOc1ccccc1C(=O)Nc1ccc(S(=O)(=O)Nc2cc(OC)nc(OC)n2)cc1	nan
	CHEMBL1582422	51205	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	9	2	8	2.9	CCOc1ccccc1C(=O)Nc1ccc(S(=O)(=O)Nc2cc(OC)nc(OC)n2)cc1	nan
	4976300	51377	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	7	1	9	4.0	CCSc1nnc(N2C(=O)C(O)=C(C(=O)c3ccco3)C2c2cccc(OC)c2)s1	nan
	CHEMBL1583844	51377	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	7	1	9	4.0	CCSc1nnc(N2C(=O)C(O)=C(C(=O)c3ccco3)C2c2cccc(OC)c2)s1	nan
	5083492	51515	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	518	13	1	5	5.1	CC[N+](CC)(CCCCS(=O)(=O)[O-])CCNP1(=O)C=C(c2ccccc2)OC(c2ccccc2)=C1	nan
	CHEMBL1585012	51515	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	518	13	1	5	5.1	CC[N+](CC)(CCCCS(=O)(=O)[O-])CCNP1(=O)C=C(c2ccccc2)OC(c2ccccc2)=C1	nan
	6624747	51746	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	5	1	7	2.6	Cn1c(=O)c2sccc2n2c(CCCC(=O)Nc3ccccc3)nnc12	nan
	CHEMBL1586923	51746	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	5	1	7	2.6	Cn1c(=O)c2sccc2n2c(CCCC(=O)Nc3ccccc3)nnc12	nan
	2384712	52053	21	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	295	1	0	3	4.8	Brc1ccc(-c2nc3ccccc3s2)s1	nan
	CHEMBL1589567	52053	21	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	295	1	0	3	4.8	Brc1ccc(-c2nc3ccccc3s2)s1	nan
	16030403	52128	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	8	1	4	4.8	Cc1ccc(Cc2nc3ccccc3nc2SCC(=O)NCCC(C)C)cc1	nan
	CHEMBL1590296	52128	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	8	1	4	4.8	Cc1ccc(Cc2nc3ccccc3nc2SCC(=O)NCCC(C)C)cc1	nan
	16022890	52179	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	491	8	2	6	5.2	COc1cc2cc(CNc3ccccc3)c(=O)n(CC(=O)Nc3cccc(Cl)c3C)c2cc1OC	nan
	CHEMBL1590948	52179	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	491	8	2	6	5.2	COc1cc2cc(CNc3ccccc3)c(=O)n(CC(=O)Nc3cccc(Cl)c3C)c2cc1OC	nan
	16029271	52264	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	324	4	0	8	1.5	CCOC(=O)c1noc2ncn(Cc3cccc(C#N)c3)c(=O)c12	nan
	CHEMBL1592100	52264	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	324	4	0	8	1.5	CCOC(=O)c1noc2ncn(Cc3cccc(C#N)c3)c(=O)c12	nan
	3431356	52285	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	9	2	4	5.8	CCc1ccc(Nc2cc(C(=O)NCCCN(C)c3ccccc3)c3ccccc3n2)cc1	nan
	CHEMBL1592367	52285	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	9	2	4	5.8	CCc1ccc(Nc2cc(C(=O)NCCCN(C)c3ccccc3)c3ccccc3n2)cc1	nan
	16331440	52310	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	5	0	6	1.9	CC(C(=O)OCC(=O)N(C)C1(C#N)CCCCC1)N1C(=O)c2ccccc2C1=O	nan
	CHEMBL1592707	52310	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	5	0	6	1.9	CC(C(=O)OCC(=O)N(C)C1(C#N)CCCCC1)N1C(=O)c2ccccc2C1=O	nan
	22518595	52441	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	7	1	9	3.0	COc1ccccc1NC(=O)CSc1nc2nccnc2c(=O)n1Cc1cccs1	nan
	CHEMBL1594419	52441	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	7	1	9	3.0	COc1ccccc1NC(=O)CSc1nc2nccnc2c(=O)n1Cc1cccs1	nan
	3630300	52453	15	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	410	4	1	5	4.9	Cc1cccc(N2C(=O)C(O)=C(C(=O)c3cccs3)C2c2ccc(Cl)cc2)n1	nan
	CHEMBL1594498	52453	15	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	410	4	1	5	4.9	Cc1cccc(N2C(=O)C(O)=C(C(=O)c3cccs3)C2c2ccc(Cl)cc2)n1	nan
	16018788	52574	2	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	6	1	6	4.6	CCc1cccc(C)c1NC(=O)CSc1nnc(CC)n2c1cc1occc12	nan
	CHEMBL1595485	52574	2	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	6	1	6	4.6	CCc1cccc(C)c1NC(=O)CSc1nnc(CC)n2c1cc1occc12	nan
	135454734	52653	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	6	3	9	1.2	Nc1cc(O)nc(SCC(=O)Nc2cc(S(=O)(=O)N3CCOCC3)ccc2Cl)n1	nan
	CHEMBL1596208	52653	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	6	3	9	1.2	Nc1cc(O)nc(SCC(=O)Nc2cc(S(=O)(=O)N3CCOCC3)ccc2Cl)n1	nan
	3151377	52670	16	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	4	2	7	2.5	N=c1c(C(=O)NCC2CCCO2)cc2c(=O)n3ccccc3nc2n1C1CCCCC1	nan
	CHEMBL1596336	52670	16	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	4	2	7	2.5	N=c1c(C(=O)NCC2CCCO2)cc2c(=O)n3ccccc3nc2n1C1CCCCC1	nan
	2743162	52768	17	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	245	1	2	3	3.1	Sc1n[nH]c(-c2cc(Cl)cc(Cl)c2)n1	nan
	CHEMBL1597261	52768	17	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	245	1	2	3	3.1	Sc1n[nH]c(-c2cc(Cl)cc(Cl)c2)n1	nan
	5175738	52814	50	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	3	2	5	6.0	Nc1c(C(=O)Nc2ccc(F)cc2)sc2nc(-c3cccs3)cc(C(F)(F)F)c12	nan
	CHEMBL1597711	52814	50	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	3	2	5	6.0	Nc1c(C(=O)Nc2ccc(F)cc2)sc2nc(-c3cccs3)cc(C(F)(F)F)c12	nan
	16018618	52827	3	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	4	1	6	3.8	Cc1cc(C)cc(NC(=O)CSc2nncn3c2cc2occc23)c1	nan
	CHEMBL1597835	52827	3	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	4	1	6	3.8	Cc1cc(C)cc(NC(=O)CSc2nncn3c2cc2occc23)c1	nan
	2931308	52930	10	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	4	2	5	2.4	COC(=O)c1cc(C)sc1NC(=O)C1CC=CCC1C(=O)O	nan
	CHEMBL1598795	52930	10	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	4	2	5	2.4	COC(=O)c1cc(C)sc1NC(=O)C1CC=CCC1C(=O)O	nan
	16033260	52946	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	5	1	5	5.0	Cc1ccc(CNC(=O)c2sc3ncnc(N(C)C4CCCCC4)c3c2C)cc1	nan
	CHEMBL1598947	52946	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	5	1	5	5.0	Cc1ccc(CNC(=O)c2sc3ncnc(N(C)C4CCCCC4)c3c2C)cc1	nan
	7202413	53114	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	3	0	8	1.2	Cc1nnc2sc(SCC(=O)N3CCC(C)CC3)nn2c1=O	nan
	CHEMBL1600469	53114	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	3	0	8	1.2	Cc1nnc2sc(SCC(=O)N3CCC(C)CC3)nn2c1=O	nan
	893043	53138	13	None	-1	3	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	244	1	1	3	2.4	O=c1[nH]c(=S)c2c(n1-c1ccccc1)CCC2	nan
	CHEMBL1600661	53138	13	None	-1	3	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	244	1	1	3	2.4	O=c1[nH]c(=S)c2c(n1-c1ccccc1)CCC2	nan
	15988297	53299	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	5	1	7	3.1	Cc1ccc(NC(=O)CCCc2nnc3n(C)c(=O)c4sccc4n23)cc1F	nan
	CHEMBL1602305	53299	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	5	1	7	3.1	Cc1ccc(NC(=O)CCCc2nnc3n(C)c(=O)c4sccc4n23)cc1F	nan
	20923199	53332	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	441	7	0	7	2.3	COc1ccc(CN2C(=O)c3cccnc3C2=O)cc1S(=O)(=O)N(C)Cc1ccco1	nan
	CHEMBL1602602	53332	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	441	7	0	7	2.3	COc1ccc(CN2C(=O)c3cccnc3C2=O)cc1S(=O)(=O)N(C)Cc1ccco1	nan
	2138501	53336	14	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	298	4	0	7	1.0	COc1ccc(C=O)cc1Cn1cnc2c(cnn2C)c1=O	nan
	CHEMBL1602628	53336	14	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	298	4	0	7	1.0	COc1ccc(C=O)cc1Cn1cnc2c(cnn2C)c1=O	nan
	16301839	53338	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	410	6	2	11	1.2	Cn1c(N)c(C(=O)CSc2nnc(NC3CCCCC3)s2)c(=O)n(C)c1=O	nan
	CHEMBL1602634	53338	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	410	6	2	11	1.2	Cn1c(N)c(C(=O)CSc2nnc(NC3CCCCC3)s2)c(=O)n(C)c1=O	nan
	2960993	53548	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	4	2	5	3.4	N=C(NOC(=O)COc1ccc2ccccc2c1Br)c1ccccn1	nan
	5740253	53548	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	4	2	5	3.4	N=C(NOC(=O)COc1ccc2ccccc2c1Br)c1ccccn1	nan
	9587840	53548	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	4	2	5	3.4	N=C(NOC(=O)COc1ccc2ccccc2c1Br)c1ccccn1	nan
	CHEMBL1604402	53548	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	4	2	5	3.4	N=C(NOC(=O)COc1ccc2ccccc2c1Br)c1ccccn1	nan
	5925277	53565	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	8	1	8	1.2	CCN1CCN(c2nc3c(C)cccn3c(=O)c2/C=C(\C#N)C(=O)NCCCOC)CC1	nan
	CHEMBL1604541	53565	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	8	1	8	1.2	CCN1CCN(c2nc3c(C)cccn3c(=O)c2/C=C(\C#N)C(=O)NCCCOC)CC1	nan
	2928283	53613	16	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	4	2	7	2.5	Cc1cccn2c(=O)c3cc(C(=O)NCC4CCCO4)c(=N)n(C4CCCC4)c3nc12	nan
	CHEMBL1605019	53613	16	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	4	2	7	2.5	Cc1cccn2c(=O)c3cc(C(=O)NCC4CCCO4)c(=N)n(C4CCCC4)c3nc12	nan
	6460757	54198	14	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	5	1	6	2.4	Cc1cc2c(SCC(=O)NCC3CCCO3)ncnc2s1	nan
	CHEMBL1609708	54198	14	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	5	1	6	2.4	Cc1cc2c(SCC(=O)NCC3CCCO3)ncnc2s1	nan
	15991073	54329	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	472	4	1	4	6.7	COc1cccc(C(=O)Nc2ccc3oc(-c4cccc5c(Br)cccc45)nc3c2)c1	nan
	CHEMBL1610897	54329	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	472	4	1	4	6.7	COc1cccc(C(=O)Nc2ccc3oc(-c4cccc5c(Br)cccc45)nc3c2)c1	nan
	7889635	54387	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	5	1	7	1.5	Cc1csc2nc(COC(=O)CNC(=O)c3ccccc3)cc(=O)n12	nan
	CHEMBL1611331	54387	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	5	1	7	1.5	Cc1csc2nc(COC(=O)CNC(=O)c3ccccc3)cc(=O)n12	nan
	778300	54562	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	293	2	1	10	-1.1	Cn1c(=O)c2c(ncn2Cc2nnc(N)s2)n(C)c1=O	nan
	CHEMBL1612871	54562	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	293	2	1	10	-1.1	Cn1c(=O)c2c(ncn2Cc2nnc(N)s2)n(C)c1=O	nan
	705485	54958	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	336	5	2	5	3.9	CCOC(=O)c1cnc2ccccc2c1Nc1cccc(C(=O)O)c1	nan
	CHEMBL1321656	54958	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	336	5	2	5	3.9	CCOC(=O)c1cnc2ccccc2c1Nc1cccc(C(=O)O)c1	nan
	CHEMBL1617945	54958	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	336	5	2	5	3.9	CCOC(=O)c1cnc2ccccc2c1Nc1cccc(C(=O)O)c1	nan
	20279	55070	95	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	285	2	3	8	-0.3	Nc1nc(Cl)nc2c1ncn2[C@H]1C[C@H](O)[C@@H](CO)O1	nan
	CHEMBL1619	55070	95	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	285	2	3	8	-0.3	Nc1nc(Cl)nc2c1ncn2[C@H]1C[C@H](O)[C@@H](CO)O1	nan
	1187262	55342	7	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	4	0	6	3.7	CN1CCC(N(C)c2nc(-c3ccc([N+](=O)[O-])cc3)nc3ccccc23)CC1	nan
	CHEMBL1462585	55342	7	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	4	0	6	3.7	CN1CCC(N(C)c2nc(-c3ccc([N+](=O)[O-])cc3)nc3ccccc23)CC1	nan
	CHEMBL1621394	55342	7	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	4	0	6	3.7	CN1CCC(N(C)c2nc(-c3ccc([N+](=O)[O-])cc3)nc3ccccc23)CC1	nan
	44143728	59931	0	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	4	2	11	-0.4	CC1(C)O[C@@H]2[C@@H](COS(=O)(=O)O)O[C@@H](n3cnc4c(N)ncnc43)[C@@H]2O1	nan
	CHEMBL1553539	59931	0	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	4	2	11	-0.4	CC1(C)O[C@@H]2[C@@H](COS(=O)(=O)O)O[C@@H](n3cnc4c(N)ncnc43)[C@@H]2O1	nan
	CHEMBL1741041	59931	0	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	4	2	11	-0.4	CC1(C)O[C@@H]2[C@@H](COS(=O)(=O)O)O[C@@H](n3cnc4c(N)ncnc43)[C@@H]2O1	nan
	135641876	71821	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	5	2	10	-0.7	COc1cc(/C=N/NC(=O)Cn2cnc3c2c(=O)n(C)c(=O)n3C)ccc1O	nan
	CHEMBL1979668	71821	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	5	2	10	-0.7	COc1cc(/C=N/NC(=O)Cn2cnc3c2c(=O)n(C)c(=O)n3C)ccc1O	nan
	135475570	72313	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	6	1	7	2.3	CCN(CC)S(=O)(=O)c1cccc(N/N=C2/C(=O)Oc3ccccc3C2=O)c1	nan
	CHEMBL1995496	72313	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	6	1	7	2.3	CCN(CC)S(=O)(=O)c1cccc(N/N=C2/C(=O)Oc3ccccc3C2=O)c1	nan
	9632269	72576	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	5	1	9	-0.6	Cn1c(=O)c2c(ncn2CCC(=O)N/N=C/c2cccnc2)n(C)c1=O	nan
	CHEMBL2004582	72576	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	5	1	9	-0.6	Cn1c(=O)c2c(ncn2CCC(=O)N/N=C/c2cccnc2)n(C)c1=O	nan
	9553490	107511	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	356	5	1	9	-0.2	Cn1c(=O)c2c(ncn2CC(=O)N/N=C/C=C/c2ccco2)n(C)c1=O	nan
	CHEMBL3194107	107511	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	356	5	1	9	-0.2	Cn1c(=O)c2c(ncn2CC(=O)N/N=C/C=C/c2ccco2)n(C)c1=O	nan
	6905987	107853	4	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	4	1	7	4.5	Sc1nnc(-c2ccccn2)n1/N=C/c1ccc(-c2ccccc2Br)o1	nan
	CHEMBL3198000	107853	4	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	4	1	7	4.5	Sc1nnc(-c2ccccn2)n1/N=C/c1ccc(-c2ccccc2Br)o1	nan
	540540	107934	6	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	1	0	7	1.1	CC(=O)/N=c1\sc2nc3ccccc3nc2n1N(C(C)=O)C(C)=O	nan
	CHEMBL3198706	107934	6	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	1	0	7	1.1	CC(=O)/N=c1\sc2nc3ccccc3nc2n1N(C(C)=O)C(C)=O	nan
	5339637	108023	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	317	7	2	5	1.4	O=C(COc1ccccc1)NCC(=O)N/N=C/c1cccs1	nan
	CHEMBL3199816	108023	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	317	7	2	5	1.4	O=C(COc1ccccc1)NCC(=O)N/N=C/c1cccs1	nan
	9553411	108415	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	5	1	8	-0.0	Cn1c(=O)c2c(ncn2CCC(=O)N/N=C/c2ccccc2)n(C)c1=O	nan
	CHEMBL3210887	108415	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	5	1	8	-0.0	Cn1c(=O)c2c(ncn2CCC(=O)N/N=C/c2ccccc2)n(C)c1=O	nan
	9634938	108425	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	5	1	9	-0.6	Cn1c(=O)c2c(ncn2CCC(=O)N/N=C/c2ccncc2)n(C)c1=O	nan
	CHEMBL3211064	108425	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	5	1	9	-0.6	Cn1c(=O)c2c(ncn2CCC(=O)N/N=C/c2ccncc2)n(C)c1=O	nan
	1116825	183681	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	4	1	6	2.4	Cc1ccnc(NS(=O)(=O)c2ccc(N3C(=O)c4ccccc4C3=O)cc2)n1	nan
	CHEMBL483773	183681	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	4	1	6	2.4	Cc1ccnc(NS(=O)(=O)c2ccc(N3C(=O)c4ccccc4C3=O)cc2)n1	nan
	7190719	199261	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	4	0	6	3.6	Fc1ccc(CSc2ccc3nnc(-c4cccnc4)n3n2)cc1	nan
	CHEMBL601822	199261	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	4	0	6	3.6	Fc1ccc(CSc2ccc3nnc(-c4cccnc4)n3n2)cc1	nan
	3259	23157	46	None	-	1	Human	3.8	pPotency	=	3.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	836	0	2	5	6.1	O=C1OC2(c3ccccc31)c1cc(I)c(O)c(I)c1Oc1c2cc(I)c(O)c1I	nan
	CHEMBL1332616	23157	46	None	-	1	Human	3.8	pPotency	=	3.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	836	0	2	5	6.1	O=C1OC2(c3ccccc31)c1cc(I)c(O)c(I)c1Oc1c2cc(I)c(O)c1I	nan
	3228920	29525	5	None	-31	2	Human	3.8	pPotency	=	3.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	481	5	2	5	5.9	O=C(CSc1nc(-c2ccccc2F)nc2nc[nH]c12)Nc1c(Cl)cc(Cl)cc1Cl	nan
	CHEMBL1386739	29525	5	None	-31	2	Human	3.8	pPotency	=	3.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	481	5	2	5	5.9	O=C(CSc1nc(-c2ccccc2F)nc2nc[nH]c12)Nc1c(Cl)cc(Cl)cc1Cl	nan
	2099	2997	77	None	-234	3	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	278	5	0	7	0.2	CC(=O)CCCCn1c(=O)c2n(C)cnc2n(c1=O)C	nan
	4740	2997	77	None	-234	3	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	278	5	0	7	0.2	CC(=O)CCCCn1c(=O)c2n(C)cnc2n(c1=O)C	nan
	7095	2997	77	None	-234	3	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	278	5	0	7	0.2	CC(=O)CCCCn1c(=O)c2n(C)cnc2n(c1=O)C	nan
	CHEMBL628	2997	77	None	-234	3	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	278	5	0	7	0.2	CC(=O)CCCCn1c(=O)c2n(C)cnc2n(c1=O)C	nan
	DB00806	2997	77	None	-234	3	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	278	5	0	7	0.2	CC(=O)CCCCn1c(=O)c2n(C)cnc2n(c1=O)C	nan
	3220395	19427	3	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	366	6	1	6	2.7	CCC(OC(=O)c1nsc(Cl)c1Cl)C(=O)NCC1CCCO1	nan
	CHEMBL1300380	19427	3	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	366	6	1	6	2.7	CCC(OC(=O)c1nsc(Cl)c1Cl)C(=O)NCC1CCCO1	nan
	16452711	19549	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	465	6	2	8	2.9	Cc1noc(NS(=O)(=O)c2ccc(NC(=O)c3nn(-c4ccccc4)ccc3=O)cc2)c1C	nan
	CHEMBL1301248	19549	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	465	6	2	8	2.9	Cc1noc(NS(=O)(=O)c2ccc(NC(=O)c3nn(-c4ccccc4)ccc3=O)cc2)c1C	nan
	4134237	19827	9	None	-2	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	301	3	0	4	3.0	CC1CCCN(C(=O)CSc2cnc3ccccc3n2)C1	nan
	CHEMBL1303471	19827	9	None	-2	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	301	3	0	4	3.0	CC1CCCN(C(=O)CSc2cnc3ccccc3n2)C1	nan
	2816749	20036	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	293	1	0	6	1.5	CCOC(=O)N1CCc2c(sc3ncn(C)c(=O)c23)C1	nan
	CHEMBL1305245	20036	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	293	1	0	6	1.5	CCOC(=O)N1CCc2c(sc3ncn(C)c(=O)c23)C1	nan
	225068	20139	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	3	2	6	0.5	CC(=O)Nc1ccc(Cc2nc3c(=O)n(C)c(=O)n(C)c3[nH]2)cc1	nan
	CHEMBL1306052	20139	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	3	2	6	0.5	CC(=O)Nc1ccc(Cc2nc3c(=O)n(C)c(=O)n(C)c3[nH]2)cc1	nan
	2377168	20477	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	7	2	6	1.7	NS(=O)(=O)c1ccc(CCNC(=O)CSc2ncnc3ccccc23)cc1	nan
	CHEMBL1308771	20477	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	7	2	6	1.7	NS(=O)(=O)c1ccc(CCNC(=O)CSc2ncnc3ccccc23)cc1	nan
	6311448	20696	4	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	5	2	6	2.6	CNc1ccc(/C=C(\C#N)C(=O)Nc2ccccn2)cc1[N+](=O)[O-]	nan
	CHEMBL1310631	20696	4	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	5	2	6	2.6	CNc1ccc(/C=C(\C#N)C(=O)Nc2ccccn2)cc1[N+](=O)[O-]	nan
	4454085	20902	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	4	1	8	1.1	CCOC(=O)CC1C(=O)NCCN1C(=O)c1cc2c(=O)n3cccc(C)c3nc2s1	nan
	CHEMBL1312229	20902	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	4	1	8	1.1	CCOC(=O)CC1C(=O)NCCN1C(=O)c1cc2c(=O)n3cccc(C)c3nc2s1	nan
	3269960	20964	1	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	8	1	9	3.7	O=C(O)CCCCn1c(SCc2cc(=O)n3cc(Cl)ccc3n2)nc2ccsc2c1=O	nan
	CHEMBL1312645	20964	1	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	8	1	9	3.7	O=C(O)CCCCn1c(SCc2cc(=O)n3cc(Cl)ccc3n2)nc2ccsc2c1=O	nan
	5811072	20997	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	4	1	7	3.8	O=C(C1=C(O)C(=O)N(c2nccs2)C1c1ccccc1F)c1ccc2c(c1)OCCO2	nan
	CHEMBL1312900	20997	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	4	1	7	3.8	O=C(C1=C(O)C(=O)N(c2nccs2)C1c1ccccc1F)c1ccc2c(c1)OCCO2	nan
	3719872	21078	16	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	366	4	1	6	3.8	Cc1cc(N2C(=O)C(O)=C(C(=O)c3cccs3)C2c2ccccc2)no1	nan
	CHEMBL1313510	21078	16	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	366	4	1	6	3.8	Cc1cc(N2C(=O)C(O)=C(C(=O)c3cccs3)C2c2ccccc2)no1	nan
	7151338	21157	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	307	4	1	5	2.8	CCS(=O)(=O)Nc1ccc(-c2cn3ccsc3n2)cc1	nan
	CHEMBL1314161	21157	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	307	4	1	5	2.8	CCS(=O)(=O)Nc1ccc(-c2cn3ccsc3n2)cc1	nan
	16010497	21199	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	6	1	6	2.0	COc1ccc(CCNC(=O)c2cnc3ccc(C)cn3c2=O)cc1OC	nan
	CHEMBL1314605	21199	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	6	1	6	2.0	COc1ccc(CCNC(=O)c2cnc3ccc(C)cn3c2=O)cc1OC	nan
	4119285	21281	11	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	2	0	7	2.2	Cn1/c(=N/C(=O)c2ccc3c(c2)OCCO3)sc2cc(S(C)(=O)=O)ccc21	nan
	CHEMBL1315733	21281	11	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	2	0	7	2.2	Cn1/c(=N/C(=O)c2ccc3c(c2)OCCO3)sc2cc(S(C)(=O)=O)ccc21	nan
	16020283	21319	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	5	1	5	4.1	CCOc1ccc(CNC(=O)c2cc3c(=O)n(C)c4ccccc4c3s2)cc1	nan
	CHEMBL1316147	21319	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	5	1	5	4.1	CCOc1ccc(CNC(=O)c2cc3c(=O)n(C)c4ccccc4c3s2)cc1	nan
	2645859	21352	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	4	0	6	2.6	Cc1cnc(C(=O)OCC(=O)c2ccc(Br)s2)cn1	nan
	CHEMBL1316688	21352	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	4	0	6	2.6	Cc1cnc(C(=O)OCC(=O)c2ccc(Br)s2)cn1	nan
	16019079	21426	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	436	6	1	5	4.2	CCc1ccc(CNC(=O)c2ccc(Cn3c(=O)c4cccn4c4cccnc43)cc2)cc1	nan
	CHEMBL1317634	21426	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	436	6	1	5	4.2	CCc1ccc(CNC(=O)c2ccc(Cn3c(=O)c4cccn4c4cccnc43)cc2)cc1	nan
	16025698	21454	4	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	4	1	5	6.1	CC(NC(=O)c1ccc(N2Cc3ccccc3Oc3ncccc32)s1)c1ccccc1	nan
	CHEMBL1317991	21454	4	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	4	1	5	6.1	CC(NC(=O)c1ccc(N2Cc3ccccc3Oc3ncccc32)s1)c1ccccc1	nan
	16018836	21511	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	436	4	1	6	4.6	O=C(CSc1nncn2c1cc1sccc12)Nc1ccc(Br)cc1F	nan
	CHEMBL1318579	21511	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	436	4	1	6	4.6	O=C(CSc1nncn2c1cc1sccc12)Nc1ccc(Br)cc1F	nan
	658390	21934	21	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	242	2	1	4	2.7	CSc1sc(C(=O)O)c2c1C(=O)CCC2	nan
	CHEMBL132222	21934	21	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	242	2	1	4	2.7	CSc1sc(C(=O)O)c2c1C(=O)CCC2	nan
	4302597	22168	12	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	2	1	6	3.1	Cc1c(Cl)c(-c2nnc(S)n2-c2ccc(F)cc2)nn1C	nan
	CHEMBL1324305	22168	12	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	2	1	6	3.1	Cc1c(Cl)c(-c2nnc(S)n2-c2ccc(F)cc2)nn1C	nan
	16825458	22423	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	7	1	9	2.9	COc1ccc(NC(=O)CSc2ccc3nnc(-c4cccnc4)n3n2)cc1OC	nan
	CHEMBL1326698	22423	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	7	1	9	2.9	COc1ccc(NC(=O)CSc2ccc3nnc(-c4cccnc4)n3n2)cc1OC	nan
	961104	22728	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	289	5	2	5	1.8	CCOC(=O)c1[nH]cnc1C(=O)Nc1ccccc1OC	nan
	CHEMBL1329229	22728	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	289	5	2	5	1.8	CCOC(=O)c1[nH]cnc1C(=O)Nc1ccccc1OC	nan
	753118	22977	51	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	347	2	1	3	4.7	Cc1ccc(-c2cc(C(=O)O)c3cc(Br)ccc3n2)s1	nan
	CHEMBL1331202	22977	51	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	347	2	1	3	4.7	Cc1ccc(-c2cc(C(=O)O)c3cc(Br)ccc3n2)s1	nan
	CHEMBL1532594	22977	51	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	347	2	1	3	4.7	Cc1ccc(-c2cc(C(=O)O)c3cc(Br)ccc3n2)s1	nan
	5302178	23449	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	2	0	5	2.3	CC1CCCN(S(=O)(=O)c2ccc3c(c2)c(=O)nc2ccccn23)C1	nan
	CHEMBL1334923	23449	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	2	0	5	2.3	CC1CCCN(S(=O)(=O)c2ccc3c(c2)c(=O)nc2ccccn23)C1	nan
	4213677	23550	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	487	5	2	9	2.3	Cc1cccn2c(=O)c3cc(C(=O)NCc4ccc5c(c4)OCO5)c(=N)n(CC4CCCO4)c3nc12	nan
	CHEMBL1335629	23550	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	487	5	2	9	2.3	Cc1cccn2c(=O)c3cc(C(=O)NCc4ccc5c(c4)OCO5)c(=N)n(CC4CCCO4)c3nc12	nan
	2410320	23785	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	7	1	6	2.5	Cc1ccc(S(=O)(=O)NCC(=O)OCC(=O)c2ccc(Br)s2)cc1	nan
	CHEMBL1337652	23785	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	7	1	6	2.5	Cc1ccc(S(=O)(=O)NCC(=O)OCC(=O)c2ccc(Br)s2)cc1	nan
	6624813	24103	3	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	4	0	7	2.0	Cn1c(=O)c2sccc2n2c(CCCC(=O)N3CCCCC3)nnc12	nan
	CHEMBL1340556	24103	3	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	4	0	7	2.0	Cn1c(=O)c2sccc2n2c(CCCC(=O)N3CCCCC3)nnc12	nan
	16189291	24255	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	6	0	8	2.6	CCOC(=O)C(CC)Sc1ccc2nnc(-c3cccnc3)n2n1	nan
	CHEMBL1341871	24255	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	6	0	8	2.6	CCOC(=O)C(CC)Sc1ccc2nnc(-c3cccnc3)n2n1	nan
	2835302	24441	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	272	1	2	4	3.4	CCC1(C)Cc2ccccc2-c2nc(S)nc(O)c21	nan
	CHEMBL1343308	24441	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	272	1	2	4	3.4	CCC1(C)Cc2ccccc2-c2nc(S)nc(O)c21	nan
	9115295	24475	23	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	3	1	4	4.1	O=S(=O)(Nc1nc2ccccc2nc1Cl)c1ccccc1C(F)(F)F	nan
	CHEMBL1343609	24475	23	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	3	1	4	4.1	O=S(=O)(Nc1nc2ccccc2nc1Cl)c1ccccc1C(F)(F)F	nan
	874496	24535	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	254	4	2	2	4.0	CC(C)C(=O)Nc1ccc(Nc2ccccc2)cc1	nan
	CHEMBL1344171	24535	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	254	4	2	2	4.0	CC(C)C(=O)Nc1ccc(Nc2ccccc2)cc1	nan
	5040775	24555	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	300	3	1	5	1.5	CC1CCCCC1NC(=O)Cn1nnc2ccccc2c1=O	nan
	CHEMBL1344340	24555	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	300	3	1	5	1.5	CC1CCCCC1NC(=O)Cn1nnc2ccccc2c1=O	nan
	7190697	24624	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	7	1	9	1.0	CCOC(=O)CNC(=O)CSc1ccc2nnc(-c3cccnc3)n2n1	nan
	CHEMBL1344913	24624	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	7	1	9	1.0	CCOC(=O)CNC(=O)CSc1ccc2nnc(-c3cccnc3)n2n1	nan
	1279973	24669	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	4	0	10	0.8	COCc1cc(C)nc(Sc2nc3c(c(=O)n(C)c(=O)n3C)n2C)c1C#N	nan
	CHEMBL1345308	24669	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	4	0	10	0.8	COCc1cc(C)nc(Sc2nc3c(c(=O)n(C)c(=O)n3C)n2C)c1C#N	nan
	16187878	24749	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	467	10	1	8	3.6	CCOC(=O)CC(NC(=O)CCc1c(C)nc2nc(C)nn2c1C)c1ccc(OC(C)C)cc1	nan
	CHEMBL1346041	24749	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	467	10	1	8	3.6	CCOC(=O)CC(NC(=O)CCc1c(C)nc2nc(C)nn2c1C)c1ccc(OC(C)C)cc1	nan
	4911180	24751	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	7	1	8	4.3	C=CCSc1nnc(N2C(=O)C(O)=C(C(=O)c3ccco3)C2c2ccccc2F)s1	nan
	CHEMBL1346060	24751	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	7	1	8	4.3	C=CCSc1nnc(N2C(=O)C(O)=C(C(=O)c3ccco3)C2c2ccccc2F)s1	nan
	6626039	24833	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	396	7	1	8	2.2	CCn1c(=O)c2sccc2n2c(CCCC(=O)NCc3cccnc3)nnc12	nan
	CHEMBL1346717	24833	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	396	7	1	8	2.2	CCn1c(=O)c2sccc2n2c(CCCC(=O)NCc3cccnc3)nnc12	nan
	4884017	24856	2	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	6	0	6	2.9	CCN1c2ccc(S(=O)(=O)N3CCOCC3)cc2N(Cc2ccc(OC)cc2)C1C	nan
	CHEMBL1346905	24856	2	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	6	0	6	2.9	CCN1c2ccc(S(=O)(=O)N3CCOCC3)cc2N(Cc2ccc(OC)cc2)C1C	nan
	5916900	25150	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	6	1	7	3.6	COc1cccc(C2C(C(=O)c3ccc4c(c3)OCCO4)=C(O)C(=O)N2Cc2cccnc2)c1	nan
	CHEMBL1349404	25150	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	6	1	7	3.6	COc1cccc(C2C(C(=O)c3ccc4c(c3)OCCO4)=C(O)C(=O)N2Cc2cccnc2)c1	nan
	2421577	25243	5	None	-4	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	311	5	0	5	3.2	COC(=O)CCc1c(C)c(C(=O)c2ccco2)c2ccccn12	nan
	CHEMBL1350197	25243	5	None	-4	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	311	5	0	5	3.2	COC(=O)CCc1c(C)c(C(=O)c2ccco2)c2ccccn12	nan
	2429966	25299	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	6	0	7	2.8	COc1ccc(CC(=O)OCc2cc(=O)n3cc(Br)ccc3n2)cc1OC	nan
	CHEMBL1350669	25299	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	6	0	7	2.8	COc1ccc(CC(=O)OCc2cc(=O)n3cc(Br)ccc3n2)cc1OC	nan
	5921143	25488	17	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	515	6	1	10	1.5	CCCN1C(=O)/C(=C/c2c(N3CCNC(=O)C3CC(=O)OC)nc3c(C)cccn3c2=O)SC1=S	nan
	CHEMBL1352285	25488	17	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	515	6	1	10	1.5	CCCN1C(=O)/C(=C/c2c(N3CCNC(=O)C3CC(=O)OC)nc3c(C)cccn3c2=O)SC1=S	nan
	2926991	25519	14	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	4	1	5	4.4	Cc1cccc(N2C(=O)C(O)=C(C(=O)c3cccs3)C2c2ccc(F)cc2)n1	nan
	CHEMBL1352465	25519	14	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	4	1	5	4.4	Cc1cccc(N2C(=O)C(O)=C(C(=O)c3cccs3)C2c2ccc(F)cc2)n1	nan
	16015204	25783	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	6	1	7	4.5	COC(=O)c1c(-c2cccs2)csc1NC(=O)c1ccc(OC)c(OC)c1	nan
	CHEMBL1354415	25783	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	6	1	7	4.5	COC(=O)c1c(-c2cccs2)csc1NC(=O)c1ccc(OC)c(OC)c1	nan
	16030461	25835	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	8	1	4	4.2	CCCCNC(=O)CSc1nc2ccccc2nc1Cc1ccccc1	nan
	CHEMBL1355113	25835	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	8	1	4	4.2	CCCCNC(=O)CSc1nc2ccccc2nc1Cc1ccccc1	nan
	23602530	25917	0	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	5	1	5	2.2	Cc1ccc(Cn2c(CCC(=O)O)nc3ncccc3c2=O)cc1	nan
	CHEMBL1356159	25917	0	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	5	1	5	2.2	Cc1ccc(Cn2c(CCC(=O)O)nc3ncccc3c2=O)cc1	nan
	16018072	25970	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	7	1	4	3.8	Cc1ccc(CCNC(=O)CCCn2c(=O)c3cccn3c3ccc(F)cc32)cc1	nan
	CHEMBL1356862	25970	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	7	1	4	3.8	Cc1ccc(CCNC(=O)CCCn2c(=O)c3cccn3c3ccc(F)cc32)cc1	nan
	1077055	26012	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	4	1	8	0.3	CC(=O)c1cccc(NC(=O)Cn2cnc3c2c(=O)n(C)c(=O)n3C)c1	nan
	CHEMBL1357427	26012	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	4	1	8	0.3	CC(=O)c1cccc(NC(=O)Cn2cnc3c2c(=O)n(C)c(=O)n3C)c1	nan
	16021425	26025	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	6	2	4	6.3	Cc1cccc(OCC(=O)Nc2ccc3nc(Nc4cccc(Cl)c4)cc(C)c3c2)c1	nan
	CHEMBL1357639	26025	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	6	2	4	6.3	Cc1cccc(OCC(=O)Nc2ccc3nc(Nc4cccc(Cl)c4)cc(C)c3c2)c1	nan
	16030521	26039	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	8	1	5	4.6	COc1cccc(CNC(=O)CSc2nc3ccccc3nc2Cc2ccccc2)c1	nan
	CHEMBL1357883	26039	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	8	1	5	4.6	COc1cccc(CNC(=O)CSc2nc3ccccc3nc2Cc2ccccc2)c1	nan
	16030369	26064	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	8	1	5	4.9	COc1cccc(Cc2nc3ccccc3nc2SCC(=O)NCc2ccc(C)cc2)c1	nan
	CHEMBL1358199	26064	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	8	1	5	4.9	COc1cccc(Cc2nc3ccccc3nc2SCC(=O)NCc2ccc(C)cc2)c1	nan
	15987639	26090	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	6	1	4	5.5	Cc1ccc(NC(=O)CSc2nc3ccccc3nc2Cc2ccccc2F)cc1F	nan
	CHEMBL1358546	26090	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	6	1	4	5.5	Cc1ccc(NC(=O)CSc2nc3ccccc3nc2Cc2ccccc2F)cc1F	nan
	881482	26618	16	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	318	3	1	3	3.7	O=S(=O)(Nc1ccccn1)c1ccc(Cl)c2ccccc12	nan
	CHEMBL1363117	26618	16	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	318	3	1	3	3.7	O=S(=O)(Nc1ccccn1)c1ccc(Cl)c2ccccc12	nan
	3193431	26665	3	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	497	7	0	8	4.3	COc1ccc(Cn2nnnc2C(c2ccc3ncccc3c2)N2CCN(C3CCCCC3)CC2)cc1	nan
	CHEMBL1363552	26665	3	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	497	7	0	8	4.3	COc1ccc(Cn2nnnc2C(c2ccc3ncccc3c2)N2CCN(C3CCCCC3)CC2)cc1	nan
	1261960	26669	9	None	-7	3	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	5	2	5	3.5	NS(=O)(=O)c1ccc(CNC(=O)c2cc(-c3ccccn3)nc3ccc(Cl)cc23)cc1	nan
	CHEMBL1363571	26669	9	None	-7	3	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	5	2	5	3.5	NS(=O)(=O)c1ccc(CNC(=O)c2cc(-c3ccccn3)nc3ccc(Cl)cc23)cc1	nan
	7190718	26781	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	4	0	6	3.6	Fc1cccc(CSc2ccc3nnc(-c4cccnc4)n3n2)c1	nan
	CHEMBL1364582	26781	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	4	0	6	3.6	Fc1cccc(CSc2ccc3nnc(-c4cccnc4)n3n2)c1	nan
	20884309	26788	1	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	7	1	8	1.1	CCc1nn(CC(=O)NCCCN2CCOCC2)c(=O)c2cc3sccc3n12	nan
	CHEMBL1364643	26788	1	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	7	1	8	1.1	CCc1nn(CC(=O)NCCCN2CCOCC2)c(=O)c2cc3sccc3n12	nan
	4152428	26823	7	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	6	1	6	5.0	CCOc1ccc(NC(=O)CSc2ncnc3c2sc2ccccc23)cc1	nan
	CHEMBL1364957	26823	7	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	6	1	6	5.0	CCOc1ccc(NC(=O)CSc2ncnc3c2sc2ccccc23)cc1	nan
	5109926	26856	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	487	7	2	8	2.6	COc1ccc(CCn2c(=N)c(C(=O)NCC3CCCO3)cc3c(=O)n4cccc(C)c4nc32)cc1	nan
	CHEMBL1365247	26856	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	487	7	2	8	2.6	COc1ccc(CCn2c(=N)c(C(=O)NCC3CCCO3)cc3c(=O)n4cccc(C)c4nc32)cc1	nan
	2959558	26859	15	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	4	0	4	3.3	CCOC(=O)N1CCN(C(=O)COc2ccc3ccccc3c2Br)CC1	nan
	CHEMBL1365264	26859	15	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	4	0	4	3.3	CCOC(=O)N1CCN(C(=O)COc2ccc3ccccc3c2Br)CC1	nan
	15988059	26915	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	396	3	1	10	2.6	COC(=O)c1cccc(Nc2nn3c(=O)c4cc5c(cc4nc3s2)OCO5)c1	nan
	CHEMBL1365674	26915	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	396	3	1	10	2.6	COC(=O)c1cccc(Nc2nn3c(=O)c4cc5c(cc4nc3s2)OCO5)c1	nan
	16015914	26921	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	454	2	0	4	6.1	Cc1c(C(=O)N2CCC(c3nc4ccccc4s3)CC2)oc2cc(Br)ccc12	nan
	CHEMBL1365703	26921	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	454	2	0	4	6.1	Cc1c(C(=O)N2CCC(c3nc4ccccc4s3)CC2)oc2cc(Br)ccc12	nan
	912209	26934	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	252	2	3	5	1.9	NC(S)=Nc1cccc(-c2nnc(S)o2)c1	nan
	CHEMBL1365893	26934	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	252	2	3	5	1.9	NC(S)=Nc1cccc(-c2nnc(S)o2)c1	nan
	3719648	27509	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	4	1	7	4.4	Cc1nnc(N2C(=O)C(O)=C(C(=O)c3ccco3)C2c2cccc3ccccc23)s1	nan
	CHEMBL1370349	27509	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	4	1	7	4.4	Cc1nnc(N2C(=O)C(O)=C(C(=O)c3ccco3)C2c2cccc3ccccc23)s1	nan
	1775727	27787	16	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	373	3	0	5	4.3	COc1ccccc1CN1COc2ccc3c(oc(=O)c4ccccc43)c2C1	nan
	CHEMBL1372393	27787	16	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	373	3	0	5	4.3	COc1ccccc1CN1COc2ccc3c(oc(=O)c4ccccc43)c2C1	nan
	16193912	28226	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	471	10	1	6	4.8	CCCCN(CC)CCCNC(=O)C1CCN(c2ncnc3c2sc2cccc(F)c23)CC1	nan
	CHEMBL1375345	28226	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	471	10	1	6	4.8	CCCCN(CC)CCCNC(=O)C1CCN(c2ncnc3c2sc2cccc(F)c23)CC1	nan
	2818996	28372	5	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	4	1	6	4.9	COc1ccc(-c2c(C#N)c(N)nc(Sc3ccc(Cl)cc3)c2C#N)cc1	nan
	CHEMBL1376612	28372	5	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	4	1	6	4.9	COc1ccc(-c2c(C#N)c(N)nc(Sc3ccc(Cl)cc3)c2C#N)cc1	nan
	20876288	28979	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	7	1	5	3.5	Cc1ccc(CN2CCSc3ccc(C(=O)NCCCN4CCN(C)CC4)cc32)cc1	nan
	CHEMBL1382060	28979	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	7	1	5	3.5	Cc1ccc(CN2CCSc3ccc(C(=O)NCCCN4CCN(C)CC4)cc32)cc1	nan
	4902824	29051	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	5	1	8	3.8	CSc1nnc(N2C(=O)C(O)=C(C(=O)c3ccco3)C2c2ccccc2F)s1	nan
	CHEMBL1382669	29051	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	5	1	8	3.8	CSc1nnc(N2C(=O)C(O)=C(C(=O)c3ccco3)C2c2ccccc2F)s1	nan
	408543	29404	39	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	219	3	1	3	2.4	O=C(O)CSc1ccc2ccccc2n1	nan
	CHEMBL1385852	29404	39	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	219	3	1	3	2.4	O=C(O)CSc1ccc2ccccc2n1	nan
	16452903	29429	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	6	2	8	2.7	Cc1ccc(-n2ccc(=O)c(C(=O)Nc3ccc(S(=O)(=O)Nc4nccc(C)n4)cc3)n2)cc1	nan
	CHEMBL1386060	29429	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	6	2	8	2.7	Cc1ccc(-n2ccc(=O)c(C(=O)Nc3ccc(S(=O)(=O)Nc4nccc(C)n4)cc3)n2)cc1	nan
	5866058	29454	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	6	1	7	3.2	COc1cccc(C2C(C(=O)c3ccc4c(c3)OCCO4)=C(O)C(=O)N2CC2CCCO2)c1	nan
	CHEMBL1386260	29454	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	6	1	7	3.2	COc1cccc(C2C(C(=O)c3ccc4c(c3)OCCO4)=C(O)C(=O)N2CC2CCCO2)c1	nan
	2219052	29930	10	None	-3	3	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	5	1	6	4.2	CCCCn1nnc(NC(=O)c2sc3cc(Cl)ccc3c2Cl)n1	nan
	CHEMBL1389959	29930	10	None	-3	3	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	5	1	6	4.2	CCCCn1nnc(NC(=O)c2sc3cc(Cl)ccc3c2Cl)n1	nan
	974402	30058	14	None	-4	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	298	3	2	2	3.4	CC(C)NC(=S)NC(=O)c1ccc(-c2ccccc2)cc1	nan
	CHEMBL1391097	30058	14	None	-4	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	298	3	2	2	3.4	CC(C)NC(=S)NC(=O)c1ccc(-c2ccccc2)cc1	nan
	4385170	30202	12	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	7	2	4	4.9	CCOc1ccc(C(CC(=O)O)NC(=O)c2sc3ccccc3c2Cl)cc1	nan
	CHEMBL1392345	30202	12	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	7	2	4	4.9	CCOc1ccc(C(CC(=O)O)NC(=O)c2sc3ccccc3c2Cl)cc1	nan
	2492440	30235	22	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	3	1	4	3.4	Cc1ccccc1S(=O)(=O)Nc1nc2ccccc2nc1Cl	nan
	CHEMBL1392606	30235	22	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	3	1	4	3.4	Cc1ccccc1S(=O)(=O)Nc1nc2ccccc2nc1Cl	nan
	7207181	30282	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	6	1	7	2.9	O=C(CSc1ccc(-c2ccco2)nn1)NCc1ccc2c(c1)OCO2	nan
	CHEMBL1393087	30282	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	6	1	7	2.9	O=C(CSc1ccc(-c2ccco2)nn1)NCc1ccc2c(c1)OCO2	nan
	16025764	30493	0	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	324	2	0	3	4.6	Cc1cc2ccccc2n1-c1ccc(C(=O)N2CCCCC2)s1	nan
	CHEMBL1395096	30493	0	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	324	2	0	3	4.6	Cc1cc2ccccc2n1-c1ccc(C(=O)N2CCCCC2)s1	nan
	5839687	30636	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	6	1	7	1.7	COCCNC(=O)/C(C#N)=C/c1c(N2CCCCCC2)nc2ccccn2c1=O	nan
	CHEMBL1397071	30636	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	6	1	7	1.7	COCCNC(=O)/C(C#N)=C/c1c(N2CCCCCC2)nc2ccccn2c1=O	nan
	5789902	30698	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	5	1	5	4.0	COc1ccc(C(=O)C2=C(O)C(=O)N(c3ccccn3)C2c2ccc(F)cc2)cc1	nan
	CHEMBL1397920	30698	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	5	1	5	4.0	COc1ccc(C(=O)C2=C(O)C(=O)N(c3ccccn3)C2c2ccc(F)cc2)cc1	nan
	3288231	30719	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	5	1	4	5.7	Cc1ccc(-c2cc(C(F)(F)F)c(C#N)c(SCC(=O)Nc3ccccc3)n2)cc1	nan
	CHEMBL1398189	30719	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	5	1	4	5.7	Cc1ccc(-c2cc(C(F)(F)F)c(C#N)c(SCC(=O)Nc3ccccc3)n2)cc1	nan
	15991174	30749	1	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	285	3	3	7	1.6	Cc1cc(Nc2ccc(C(=O)O)c(O)c2)n2ncnc2n1	nan
	CHEMBL1398548	30749	1	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	285	3	3	7	1.6	Cc1cc(Nc2ccc(C(=O)O)c(O)c2)n2ncnc2n1	nan
	16025760	30881	3	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	4	0	5	4.1	CCOC(=O)C1CCN(C(=O)c2ccc(-n3ccc4ccccc43)s2)CC1	nan
	CHEMBL1399794	30881	3	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	4	0	5	4.1	CCOC(=O)C1CCN(C(=O)c2ccc(-n3ccc4ccccc43)s2)CC1	nan
	135444909	30942	10	None	-4	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	547	8	3	10	3.7	Cc1cc(C)nc(NS(=O)(=O)c2ccc(NC(=O)CSc3nc(O)c(C#N)c(-c4ccccc4)n3)cc2)n1	nan
	CHEMBL1400344	30942	10	None	-4	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	547	8	3	10	3.7	Cc1cc(C)nc(NS(=O)(=O)c2ccc(NC(=O)CSc3nc(O)c(C#N)c(-c4ccccc4)n3)cc2)n1	nan
	16023027	30969	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	6	1	6	2.8	CN(Cc1ccc(F)cc1)S(=O)(=O)c1nnc(NC(=O)c2ccccc2)s1	nan
	CHEMBL1400601	30969	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	6	1	6	2.8	CN(Cc1ccc(F)cc1)S(=O)(=O)c1nnc(NC(=O)c2ccccc2)s1	nan
	2005962	30975	8	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	7	0	7	3.5	CC(C)OCCCN1CN(S(=O)(=O)c2cccs2)c2nc3ccccc3nc21	nan
	CHEMBL1400661	30975	8	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	7	0	7	3.5	CC(C)OCCCN1CN(S(=O)(=O)c2cccs2)c2nc3ccccc3nc21	nan
	4176332	31012	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	3	1	5	3.6	CN1CCN(NC(=O)c2cc(-c3ccc(Br)s3)nc3ccccc23)CC1	nan
	CHEMBL1401042	31012	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	3	1	5	3.6	CN1CCN(NC(=O)c2cc(-c3ccc(Br)s3)nc3ccccc23)CC1	nan
	7693269	31052	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	1	1	1	4.1	O=C(c1cc2cc(Br)ccc2[nH]1)N1CCc2ccccc21	nan
	CHEMBL1401345	31052	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	1	1	1	4.1	O=C(c1cc2cc(Br)ccc2[nH]1)N1CCc2ccccc21	nan
	1842681	32400	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	4	0	8	1.2	CCOC(=O)/C(C#N)=C/c1c(N2CCN(C)CC2)nc2c(C)cccn2c1=O	nan
	CHEMBL1412841	32400	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	4	0	8	1.2	CCOC(=O)/C(C#N)=C/c1c(N2CCN(C)CC2)nc2c(C)cccn2c1=O	nan
	3159273	32585	19	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	4	0	5	3.0	Cc1c2c(n3c(nc4ccccc43)c1C#N)N(CCCN(C)C)CC2	nan
	CHEMBL1414335	32585	19	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	4	0	5	3.0	Cc1c2c(n3c(nc4ccccc43)c1C#N)N(CCCN(C)C)CC2	nan
	773430	32701	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	276	1	1	4	2.5	O=C(O)c1ccc2nc3c(nc2c1)-c1ccccc1C3=O	nan
	CHEMBL1415344	32701	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	276	1	1	4	2.5	O=C(O)c1ccc2nc3c(nc2c1)-c1ccccc1C3=O	nan
	1172271	32998	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	6	0	9	0.1	CCCn1c(SCC(=O)N2CCN(CC)CC2)nc2c1c(=O)n(C)c(=O)n2C	nan
	CHEMBL1417950	32998	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	6	0	9	0.1	CCCn1c(SCC(=O)N2CCN(CC)CC2)nc2c1c(=O)n(C)c(=O)n2C	nan
	20957513	33167	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	481	12	2	8	2.6	CSc1ccc(CCNC(=O)CCc2nnc3ccc(NCCCN4CCCC4=O)nn23)cc1	nan
	CHEMBL1419386	33167	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	481	12	2	8	2.6	CSc1ccc(CCNC(=O)CCc2nnc3ccc(NCCCN4CCCC4=O)nn23)cc1	nan
	656126	34115	5	None	-1	3	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	7	1	8	4.1	CCOC(=O)c1c(NC(=O)CSc2nc(C)cc(C)c2C#N)sc(C(C)=O)c1C	nan
	CHEMBL1427319	34115	5	None	-1	3	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	7	1	8	4.1	CCOC(=O)c1c(NC(=O)CSc2nc(C)cc(C)c2C#N)sc(C(C)=O)c1C	nan
	24792443	34191	3	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	5	2	5	3.1	CCc1nc(SCC(=O)NNC(=O)c2ccc(C)cc2)c2ccccc2n1	nan
	CHEMBL1428040	34191	3	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	5	2	5	3.1	CCc1nc(SCC(=O)NNC(=O)c2ccc(C)cc2)c2ccccc2n1	nan
	5295519	34889	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	6	1	10	0.1	COC(=O)c1cc(OC)c(OC)c(OC)c1NC(=O)c1cc(=O)n(C)c(=O)n1C	nan
	CHEMBL1434105	34889	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	6	1	10	0.1	COC(=O)c1cc(OC)c(OC)c(OC)c1NC(=O)c1cc(=O)n(C)c(=O)n1C	nan
	16959503	34973	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	534	8	1	9	2.5	CC(C)Oc1ccc(S(=O)(=O)N2CCOCC2)cc1NC(=O)c1cc([N+](=O)[O-])ccc1N1CCOCC1	nan
	CHEMBL1435220	34973	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	534	8	1	9	2.5	CC(C)Oc1ccc(S(=O)(=O)N2CCOCC2)cc1NC(=O)c1cc([N+](=O)[O-])ccc1N1CCOCC1	nan
	2448286	34996	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	5	1	11	1.6	Cn1c(N)c(C(=O)CSc2nn(-c3ccccc3)c(=S)s2)c(=O)n(C)c1=O	nan
	CHEMBL1435449	34996	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	5	1	11	1.6	Cn1c(N)c(C(=O)CSc2nn(-c3ccccc3)c(=S)s2)c(=O)n(C)c1=O	nan
	16018790	35120	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	5	1	6	4.6	CCc1nnc(SCC(=O)Nc2ccc(Cl)cc2F)c2cc3occc3n12	nan
	CHEMBL1437127	35120	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	5	1	6	4.6	CCc1nnc(SCC(=O)Nc2ccc(Cl)cc2F)c2cc3occc3n12	nan
	135401612	35381	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	311	4	3	7	1.5	Nc1cc(O)nc(SCC(=O)Nc2cccnc2Cl)n1	nan
	CHEMBL1439558	35381	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	311	4	3	7	1.5	Nc1cc(O)nc(SCC(=O)Nc2cccnc2Cl)n1	nan
	15990899	35491	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	567	9	1	10	5.2	COc1cc2nc(SCC(=O)Nc3cccc(C)c3)n3nc(CCn4c(C)nc5ccccc54)nc3c2cc1OC	nan
	CHEMBL1440596	35491	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	567	9	1	10	5.2	COc1cc2nc(SCC(=O)Nc3cccc(C)c3)n3nc(CCn4c(C)nc5ccccc54)nc3c2cc1OC	nan
	16034663	35516	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	6	1	7	2.3	Cn1c(=O)c2sccc2n2c(CCCC(=O)NCc3ccccc3)nnc12	nan
	CHEMBL1440811	35516	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	6	1	7	2.3	Cn1c(=O)c2sccc2n2c(CCCC(=O)NCc3ccccc3)nnc12	nan
	5898351	35686	3	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	457	7	1	6	4.2	Cc1ccc(C2C(C(=O)c3ccc4c(c3)CC(C)O4)=C(O)C(=O)N2CCCn2ccnc2)cc1	nan
	CHEMBL1442346	35686	3	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	457	7	1	6	4.2	Cc1ccc(C2C(C(=O)c3ccc4c(c3)CC(C)O4)=C(O)C(=O)N2CCCn2ccnc2)cc1	nan
	986518	35745	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	3	2	4	3.3	Cc1c(C(=O)Nc2ccc(S(N)(=O)=O)cc2)oc2ccc(Cl)cc12	nan
	CHEMBL1442810	35745	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	3	2	4	3.3	Cc1c(C(=O)Nc2ccc(S(N)(=O)=O)cc2)oc2ccc(Cl)cc12	nan
	16009462	35754	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	4	1	6	2.6	CC(=O)Nc1ccccc1OCc1cc(=O)n2c(C)csc2n1	nan
	CHEMBL1442959	35754	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	4	1	6	2.6	CC(=O)Nc1ccccc1OCc1cc(=O)n2c(C)csc2n1	nan
	7245567	35778	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	6	1	8	1.9	COc1ccc(CNC(=O)CCc2nnc3n(C)c(=O)c4sccc4n23)cc1	nan
	CHEMBL1443187	35778	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	6	1	8	1.9	COc1ccc(CNC(=O)CCc2nnc3n(C)c(=O)c4sccc4n23)cc1	nan
	4920871	36166	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	4	1	7	1.9	O=C(Cn1c2ccc(F)cc2c2nc3n(c(=O)c21)CCS3)NCC1CCCO1	nan
	CHEMBL1446831	36166	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	4	1	7	1.9	O=C(Cn1c2ccc(F)cc2c2nc3n(c(=O)c21)CCS3)NCC1CCCO1	nan
	139030	36189	31	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	196	0	1	2	2.9	O=C1C=C(O)c2cccc3cccc1c23	nan
	CHEMBL1446983	36189	31	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	196	0	1	2	2.9	O=C1C=C(O)c2cccc3cccc1c23	nan
	771978	36200	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	234	3	1	6	1.2	O=C(Nc1ncccn1)c1ccc([N+](=O)[O-])o1	nan
	CHEMBL1447058	36200	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	234	3	1	6	1.2	O=C(Nc1ncccn1)c1ccc([N+](=O)[O-])o1	nan
	1511203	36278	14	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	5	2	7	2.6	Cc1ccc(-c2nn3c(C)nnc3c3ccccc23)cc1S(=O)(=O)NC(C)(C)CO	nan
	CHEMBL1447724	36278	14	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	5	2	7	2.6	Cc1ccc(-c2nn3c(C)nnc3c3ccccc23)cc1S(=O)(=O)NC(C)(C)CO	nan
	5310565	36677	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	356	4	0	8	1.1	O=C(CSc1ccc2nnc(-c3cccnc3)n2n1)N1CCOCC1	nan
	CHEMBL1450965	36677	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	356	4	0	8	1.1	O=C(CSc1ccc2nnc(-c3cccnc3)n2n1)N1CCOCC1	nan
	16457956	36794	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	6	4	8	1.1	CCN(CC)S(=O)(=O)c1cccc(C(=O)NNC(=O)c2ccc3nc(O)c(O)nc3c2)c1	nan
	CHEMBL1451892	36794	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	6	4	8	1.1	CCN(CC)S(=O)(=O)c1cccc(C(=O)NNC(=O)c2ccc3nc(O)c(O)nc3c2)c1	nan
	2173828	37384	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	4	0	3	5.6	CCN(CC)c1nc(-c2ccccc2Cl)c2cc(Br)ccc2n1	nan
	CHEMBL1456908	37384	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	4	0	3	5.6	CCN(CC)c1nc(-c2ccccc2Cl)c2cc(Br)ccc2n1	nan
	20904573	37691	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	464	7	1	8	2.7	Cn1c(=O)c2sccc2n2c(CCCC(=O)NC3CCN(Cc4ccccc4)CC3)nnc12	nan
	CHEMBL1459467	37691	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	464	7	1	8	2.7	Cn1c(=O)c2sccc2n2c(CCCC(=O)NC3CCN(Cc4ccccc4)CC3)nnc12	nan
	734076	37720	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	226	4	1	4	2.4	CCCC(=O)Nc1nc(C)c(C(C)=O)s1	nan
	CHEMBL1459745	37720	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	226	4	1	4	2.4	CCCC(=O)Nc1nc(C)c(C(C)=O)s1	nan
	1511643	37721	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	302	4	1	8	1.3	Cc1cc([N+](=O)[O-])nn1CC(=O)Nc1cccc2nonc12	nan
	CHEMBL1459750	37721	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	302	4	1	8	1.3	Cc1cc([N+](=O)[O-])nn1CC(=O)Nc1cccc2nonc12	nan
	1838806	37851	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	6	1	7	3.6	CCOc1cccc(Nc2cc3n(c(=O)n2)CCc2cc(OC)c(OC)cc2-3)c1	nan
	CHEMBL1460751	37851	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	6	1	7	3.6	CCOc1cccc(Nc2cc3n(c(=O)n2)CCc2cc(OC)c(OC)cc2-3)c1	nan
	16188836	38074	3	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	331	2	0	4	4.0	CC1=NOC(=O)/C1=C\c1ccc(-c2ccccc2Br)o1	nan
	CHEMBL1462764	38074	3	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	331	2	0	4	4.0	CC1=NOC(=O)/C1=C\c1ccc(-c2ccccc2Br)o1	nan
	3332154	38413	1	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	3	1	8	3.2	Cc1nc(N)sc1N=Nc1c(C)n(C)n(-c2ccccc2)c1=O	nan
	CHEMBL1465412	38413	1	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	3	1	8	3.2	Cc1nc(N)sc1N=Nc1c(C)n(C)n(-c2ccccc2)c1=O	nan
	20957223	38520	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	436	6	1	8	2.0	Cc1ccc(CNC(=O)CCc2nnc3ccc(N4CCC5(CC4)OCCO5)nn23)cc1	nan
	CHEMBL1466244	38520	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	436	6	1	8	2.0	Cc1ccc(CNC(=O)CCc2nnc3ccc(N4CCC5(CC4)OCCO5)nn23)cc1	nan
	2350819	38526	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	6	1	9	1.3	Cc1cc(Br)ccc1SCC(=O)OCC(=O)c1c(N)n(C)c(=O)n(C)c1=O	nan
	CHEMBL1466307	38526	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	6	1	9	1.3	Cc1cc(Br)ccc1SCC(=O)OCC(=O)c1c(N)n(C)c(=O)n(C)c1=O	nan
	7190691	38866	1	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	6	1	8	3.1	CC(=O)c1ccc(NC(=O)CSc2ccc3nnc(-c4cccnc4)n3n2)cc1	nan
	CHEMBL1469069	38866	1	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	6	1	8	3.1	CC(=O)c1ccc(NC(=O)CSc2ccc3nnc(-c4cccnc4)n3n2)cc1	nan
	1179824	39046	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	5	2	7	3.6	CCOC(=O)c1sc2ncnc(Nc3cccc(C(=O)O)c3)c2c1C	nan
	CHEMBL1470707	39046	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	5	2	7	3.6	CCOC(=O)c1sc2ncnc(Nc3cccc(C(=O)O)c3)c2c1C	nan
	7207497	39061	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	5	1	5	4.2	Cc1c(Cl)cccc1NC(=O)CSc1ccc(-c2cccnc2)nn1	nan
	CHEMBL1470773	39061	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	5	1	5	4.2	Cc1c(Cl)cccc1NC(=O)CSc1ccc(-c2cccnc2)nn1	nan
	16012892	39275	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	6	2	7	2.9	CCNC(=O)c1c(NC(=O)c2nc(S(=O)(=O)CC)ncc2Cl)sc2c1CCCC2	nan
	CHEMBL1472696	39275	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	6	2	7	2.9	CCNC(=O)c1c(NC(=O)c2nc(S(=O)(=O)CC)ncc2Cl)sc2c1CCCC2	nan
	16030433	39417	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	9	1	6	5.0	COc1cccc(CNC(=O)CSc2nc3ccccc3nc2Cc2ccc(C)cc2)c1OC	nan
	CHEMBL1474670	39417	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	9	1	6	5.0	COc1cccc(CNC(=O)CSc2nc3ccccc3nc2Cc2ccc(C)cc2)c1OC	nan
	4547893	39591	17	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	5	1	6	3.3	COc1ccccc1C(=O)Nc1nc2ccc(S(=O)(=O)N3CCCC3)cc2s1	nan
	CHEMBL1477066	39591	17	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	5	1	6	3.3	COc1ccccc1C(=O)Nc1nc2ccc(S(=O)(=O)N3CCCC3)cc2s1	nan
	1313916	39856	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	4	2	2	5.5	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NC(=O)C1CCCCC1	nan
	CHEMBL1479446	39856	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	4	2	2	5.5	O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1NC(=O)C1CCCCC1	nan
	16021977	40223	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	6	1	6	4.5	CCOC(=O)c1ccc(NC(=O)c2c(C)nn(-c3ccc(F)cc3)c2-n2cccc2)cc1	nan
	CHEMBL1482573	40223	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	6	1	6	4.5	CCOC(=O)c1ccc(NC(=O)c2c(C)nn(-c3ccc(F)cc3)c2-n2cccc2)cc1	nan
	16025700	40442	4	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	4	1	5	5.8	Cc1cccc(CNC(=O)c2ccc(N3Cc4ccccc4Oc4ncccc43)s2)c1	nan
	CHEMBL1484349	40442	4	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	4	1	5	5.8	Cc1cccc(CNC(=O)c2ccc(N3Cc4ccccc4Oc4ncccc43)s2)c1	nan
	4969640	40473	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	7	1	8	1.5	COc1ccc(S(=O)(=O)N(C)C)cc1NC(=O)CSc1nncs1	nan
	CHEMBL1484709	40473	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	7	1	8	1.5	COc1ccc(S(=O)(=O)N(C)C)cc1NC(=O)CSc1nncs1	nan
	2267309	40978	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	345	4	2	6	2.8	Cc1cc(N)n(-c2ccc(Oc3ccccc3)c(S(=O)(=O)O)c2)n1	nan
	CHEMBL1488814	40978	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	345	4	2	6	2.8	Cc1cc(N)n(-c2ccc(Oc3ccccc3)c(S(=O)(=O)O)c2)n1	nan
	3157588	41248	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	5	2	3	3.7	CC(=O)C1=C(O)C(=O)N(CCc2c[nH]c3ccccc23)C1c1ccccc1	nan
	CHEMBL1490855	41248	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	5	2	3	3.7	CC(=O)C1=C(O)C(=O)N(CCc2c[nH]c3ccccc23)C1c1ccccc1	nan
	3755909	41829	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	319	2	0	4	4.1	Cc1cc(-c2ccc(Br)s2)nc(-n2cccc2)n1	nan
	CHEMBL1495948	41829	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	319	2	0	4	4.1	Cc1cc(-c2ccc(Br)s2)nc(-n2cccc2)n1	nan
	6501461	42448	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	6	1	9	2.7	CCC(Sc1nnc(-c2ccco2)n1C)C(=O)Nc1nnc(C)s1	nan
	CHEMBL1501425	42448	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	6	1	9	2.7	CCC(Sc1nnc(-c2ccco2)n1C)C(=O)Nc1nnc(C)s1	nan
	20968950	42498	3	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	7	1	6	0.2	CCN(CC)S(=O)(=O)c1ccc2c(c1)N(CC(=O)N1CCC(C(N)=O)CC1)C(=O)CO2	nan
	CHEMBL1501847	42498	3	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	7	1	6	0.2	CCN(CC)S(=O)(=O)c1ccc2c(c1)N(CC(=O)N1CCC(C(N)=O)CC1)C(=O)CO2	nan
	7692847	42638	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	398	3	1	6	3.1	O=C(NCc1nnc2c(C(F)(F)F)cc(Cl)cn12)c1ccc2c(c1)OCO2	nan
	CHEMBL1503072	42638	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	398	3	1	6	3.1	O=C(NCc1nnc2c(C(F)(F)F)cc(Cl)cn12)c1ccc2c(c1)OCO2	nan
	1243282	42756	13	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	356	2	1	5	4.6	Fc1ccc(-n2c(S)nnc2-c2ccc3ccccc3n2)cc1Cl	nan
	CHEMBL1504174	42756	13	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	356	2	1	5	4.6	Fc1ccc(-n2c(S)nnc2-c2ccc3ccccc3n2)cc1Cl	nan
	20888797	42977	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	479	7	1	9	1.5	CCS(=O)(=O)c1nc(S(=O)(=O)c2ccc(Cl)cc2)c(N2CCN(CCO)CC2)s1	nan
	CHEMBL1506053	42977	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	479	7	1	9	1.5	CCS(=O)(=O)c1nc(S(=O)(=O)c2ccc(Cl)cc2)c(N2CCN(CCO)CC2)s1	nan
	3965652	42999	3	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	288	2	2	5	3.6	Oc1nc(S)ncc1Oc1ccc(Cl)cc1Cl	nan
	CHEMBL1506226	42999	3	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	288	2	2	5	3.6	Oc1nc(S)ncc1Oc1ccc(Cl)cc1Cl	nan
	664243	43238	11	None	-2	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	4	1	7	3.7	Cc1cc(N2C(=O)C(O)=C(C(=O)c3ccc(C)o3)C2c2cccs2)no1	nan
	CHEMBL1508235	43238	11	None	-2	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	4	1	7	3.7	Cc1cc(N2C(=O)C(O)=C(C(=O)c3ccc(C)o3)C2c2cccs2)no1	nan
	1564171	43319	14	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	6	1	8	3.9	C=CCn1c(SCC(=O)Nc2sccc2C#N)nc2sc(C)c(C)c2c1=O	nan
	CHEMBL1509018	43319	14	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	6	1	8	3.9	C=CCn1c(SCC(=O)Nc2sccc2C#N)nc2sc(C)c(C)c2c1=O	nan
	660816	43483	49	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	283	3	1	5	3.2	COc1ccccc1-c1nnc(S)n1-c1ccccc1	nan
	CHEMBL1510509	43483	49	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	283	3	1	5	3.2	COc1ccccc1-c1nnc(S)n1-c1ccccc1	nan
	4736989	43641	14	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	287	4	1	7	1.4	O=C(O)CSc1ccc2nnc(-c3cccnc3)n2n1	nan
	CHEMBL1511802	43641	14	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	287	4	1	7	1.4	O=C(O)CSc1ccc2nnc(-c3cccnc3)n2n1	nan
	16407031	43657	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	544	9	1	9	3.2	COc1ccc2c(c1OC)c(=O)n1c3ccc(OC(C)C(=O)NCCCN4CCOCC4)cc3c3ccnc2c31	nan
	CHEMBL1512174	43657	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	544	9	1	9	3.2	COc1ccc2c(c1OC)c(=O)n1c3ccc(OC(C)C(=O)NCCCN4CCOCC4)cc3c3ccnc2c31	nan
	16021393	43664	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	465	6	2	4	6.6	Cc1cccc(OCC(=O)Nc2ccc3nc(Nc4cccc(C(F)(F)F)c4)cc(C)c3c2)c1	nan
	CHEMBL1512269	43664	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	465	6	2	4	6.6	Cc1cccc(OCC(=O)Nc2ccc3nc(Nc4cccc(C(F)(F)F)c4)cc(C)c3c2)c1	nan
	16018932	43809	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	454	5	0	7	6.7	CCc1nnc(SCc2nc(-c3cccc(Cl)c3)oc2C)c2cc3sc(C)cc3n12	nan
	CHEMBL1514500	43809	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	454	5	0	7	6.7	CCc1nnc(SCc2nc(-c3cccc(Cl)c3)oc2C)c2cc3sc(C)cc3n12	nan
	20885685	43876	4	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	7	1	7	1.3	COc1ccccc1CNC(=O)CCCn1nc(C)n2ccnc2c1=O	nan
	CHEMBL1515364	43876	4	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	7	1	7	1.3	COc1ccccc1CNC(=O)CCCn1nc(C)n2ccnc2c1=O	nan
	16018754	43902	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	6	1	8	3.8	COc1cc(NC(=O)CSc2nnc(C)n3c2cc2oc(C)cc23)cc(OC)c1	nan
	CHEMBL1515810	43902	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	6	1	8	3.8	COc1cc(NC(=O)CSc2nnc(C)n3c2cc2oc(C)cc23)cc(OC)c1	nan
	4350514	44956	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	4	1	6	1.9	Cc1nc2ccccc2c(=O)n1NC(=O)Cc1ccc([N+](=O)[O-])cc1	nan
	CHEMBL1525803	44956	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	4	1	6	1.9	Cc1nc2ccccc2c(=O)n1NC(=O)Cc1ccc([N+](=O)[O-])cc1	nan
	135455188	45265	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	5	2	9	3.3	N#Cc1c(O)nc(SCC(=O)Nc2nnc(C(F)(F)F)s2)nc1-c1ccccc1	nan
	CHEMBL1528492	45265	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	5	2	9	3.3	N#Cc1c(O)nc(SCC(=O)Nc2nnc(C(F)(F)F)s2)nc1-c1ccccc1	nan
	3535143	45429	4	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	482	6	1	9	3.6	O=C(O)C1CCC(Cn2c(SCc3cc(=O)n4ccccc4n3)nc3ccsc3c2=O)CC1	nan
	CHEMBL1529863	45429	4	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	482	6	1	9	3.6	O=C(O)C1CCC(Cn2c(SCc3cc(=O)n4ccccc4n3)nc3ccsc3c2=O)CC1	nan
	16030435	45452	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	447	7	1	4	5.6	Cc1ccc(Cc2nc3ccccc3nc2SCC(=O)NCc2ccccc2Cl)cc1	nan
	CHEMBL1530187	45452	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	447	7	1	4	5.6	Cc1ccc(Cc2nc3ccccc3nc2SCC(=O)NCc2ccccc2Cl)cc1	nan
	54677747	45716	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	426	1	2	7	4.6	O=c1oc2ccccc2c(O)c1[C@H]1c2ccc(O)cc2Oc2c1c(=O)oc1ccccc21	nan
	CHEMBL1532491	45716	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	426	1	2	7	4.6	O=c1oc2ccccc2c(O)c1[C@H]1c2ccc(O)cc2Oc2c1c(=O)oc1ccccc21	nan
	6498569	45750	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	7	2	5	1.0	Cc1ccc(OCC(=O)NCCNC(=O)c2cnccn2)cc1C	nan
	CHEMBL1532759	45750	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	7	2	5	1.0	Cc1ccc(OCC(=O)NCCNC(=O)c2cnccn2)cc1C	nan
	6060971	45754	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	8	1	6	3.4	CC(C)Oc1ccc(C(=O)C2=C(O)C(=O)N(CCN3CCOCC3)C2c2ccccc2)cc1	nan
	CHEMBL1532782	45754	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	8	1	6	3.4	CC(C)Oc1ccc(C(=O)C2=C(O)C(=O)N(CCN3CCOCC3)C2c2ccccc2)cc1	nan
	3262927	46073	1	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	5	0	7	1.3	O=C(OCN1C(=O)c2ccccc2C1=O)c1cc(S(=O)(=O)N2CCOCC2)ccc1F	nan
	CHEMBL1535967	46073	1	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	5	0	7	1.3	O=C(OCN1C(=O)c2ccccc2C1=O)c1cc(S(=O)(=O)N2CCOCC2)ccc1F	nan
	6018171	46075	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	6	1	6	3.9	COc1ccc(C(=O)C2=C(O)C(=O)N(c3ccccn3)C2c2ccc(OC)cc2)cc1	nan
	CHEMBL1535987	46075	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	6	1	6	3.9	COc1ccc(C(=O)C2=C(O)C(=O)N(c3ccccn3)C2c2ccc(OC)cc2)cc1	nan
	7120055	46136	9	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	322	1	1	4	4.4	Cc1ccc(-n2c(=S)[nH]c3c(oc4ccccc43)c2=O)cc1C	nan
	CHEMBL1536665	46136	9	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	322	1	1	4	4.4	Cc1ccc(-n2c(=S)[nH]c3c(oc4ccccc43)c2=O)cc1C	nan
	2086676	46205	2	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	6	1	8	1.3	Cn1c(=O)c(C(=O)COc2ccc(C#N)cc2)c(N)n(Cc2ccccc2)c1=O	nan
	CHEMBL1537193	46205	2	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	6	1	8	1.3	Cn1c(=O)c(C(=O)COc2ccc(C#N)cc2)c(N)n(Cc2ccccc2)c1=O	nan
	20888841	46237	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	457	7	0	8	2.6	CCCS(=O)(=O)c1nc(S(=O)(=O)c2ccc(C)cc2)c(N2CCN(CC)CC2)s1	nan
	CHEMBL1537517	46237	12	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	457	7	0	8	2.6	CCCS(=O)(=O)c1nc(S(=O)(=O)c2ccc(C)cc2)c(N2CCN(CC)CC2)s1	nan
	22334156	46456	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	508	6	1	9	1.5	COc1ccc(-n2nc(C(=O)NCC(=O)N3CCC4(CC3)OCCO4)c3ccccc3c2=O)cc1OC	nan
	CHEMBL1539318	46456	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	508	6	1	9	1.5	COc1ccc(-n2nc(C(=O)NCC(=O)N3CCC4(CC3)OCCO4)c3ccccc3c2=O)cc1OC	nan
	3151316	46459	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	5	2	8	1.5	Cc1cccn2c(=O)c3cc(C(=O)NCC4CCCO4)c(=N)n(CC4CCCO4)c3nc12	nan
	CHEMBL1539382	46459	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	5	2	8	1.5	Cc1cccn2c(=O)c3cc(C(=O)NCC4CCCO4)c(=N)n(CC4CCCO4)c3nc12	nan
	17581317	46677	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	3	1	5	3.7	O=C(NCc1nnc2c(C(F)(F)F)cc(Cl)cn12)c1ccc(Br)o1	nan
	CHEMBL1541200	46677	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	3	1	5	3.7	O=C(NCc1nnc2c(C(F)(F)F)cc(Cl)cn12)c1ccc(Br)o1	nan
	6228228	46790	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	4	1	7	4.0	Cc1nnc(N2C(=O)C(O)=C(C(=O)c3ccc4c(c3)CC(C)O4)C2c2ccccc2)s1	nan
	CHEMBL1542130	46790	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	4	1	7	4.0	Cc1nnc(N2C(=O)C(O)=C(C(=O)c3ccc4c(c3)CC(C)O4)C2c2ccccc2)s1	nan
	2359872	46819	15	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	287	4	1	4	2.8	O=C(CSc1cnc2ccccc2n1)NC1CCCC1	nan
	CHEMBL1542457	46819	15	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	287	4	1	4	2.8	O=C(CSc1cnc2ccccc2n1)NC1CCCC1	nan
	2346972	46838	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	6	1	10	-1.0	CN(C)S(=O)(=O)c1cccc(C(=O)OCC(=O)c2c(N)n(C)c(=O)n(C)c2=O)c1	nan
	CHEMBL1542615	46838	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	6	1	10	-1.0	CN(C)S(=O)(=O)c1cccc(C(=O)OCC(=O)c2c(N)n(C)c(=O)n(C)c2=O)c1	nan
	135420430	46843	11	None	-4	3	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	6	2	8	3.5	CCC(Sc1nc(O)c(C#N)c(-c2ccccc2)n1)C(=O)Nc1cc(C)on1	nan
	CHEMBL1542646	46843	11	None	-4	3	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	6	2	8	3.5	CCC(Sc1nc(O)c(C#N)c(-c2ccccc2)n1)C(=O)Nc1cc(C)on1	nan
	1866349	47179	10	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	233	4	1	3	2.8	O=C(O)CCSc1ccc2ccccc2n1	nan
	661670	47179	10	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	233	4	1	3	2.8	O=C(O)CCSc1ccc2ccccc2n1	nan
	CHEMBL1406059	47179	10	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	233	4	1	3	2.8	O=C(O)CCSc1ccc2ccccc2n1	nan
	CHEMBL1545185	47179	10	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	233	4	1	3	2.8	O=C(O)CCSc1ccc2ccccc2n1	nan
	4876432	47204	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	7	2	6	3.2	CCN(CC)S(=O)(=O)c1ccc(OC)c(NC(=O)c2cc(O)nc3ccccc23)c1	nan
	CHEMBL1545378	47204	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	7	2	6	3.2	CCN(CC)S(=O)(=O)c1ccc(OC)c(NC(=O)c2cc(O)nc3ccccc23)c1	nan
	2595072	47205	14	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	6	1	4	3.1	O=C(CSc1ncnc2ccccc12)NCCc1ccccc1	nan
	CHEMBL1545386	47205	14	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	6	1	4	3.1	O=C(CSc1ncnc2ccccc12)NCCc1ccccc1	nan
	2115012	47272	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	6	1	10	0.2	CCCn1c(N)c(C(=O)COC(=O)c2c(C)noc2C)c(=O)n(C)c1=O	nan
	CHEMBL1545973	47272	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	6	1	10	0.2	CCCn1c(N)c(C(=O)COC(=O)c2c(C)noc2C)c(=O)n(C)c1=O	nan
	241512	47575	3	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	210	1	2	2	3.2	c1ccc(-c2ccc3c(c2)NCCN3)cc1	nan
	CHEMBL1548782	47575	3	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	210	1	2	2	3.2	c1ccc(-c2ccc3c(c2)NCCN3)cc1	nan
	16189384	47794	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	573	10	2	9	1.4	CSCCC(NS(=O)(=O)c1ccc2c(c1)c(=O)n(C)c(=O)n2C)C(=O)NC1CCN(Cc2ccccc2)CC1	nan
	CHEMBL1550614	47794	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	573	10	2	9	1.4	CSCCC(NS(=O)(=O)c1ccc2c(c1)c(=O)n(C)c(=O)n2C)C(=O)NC1CCN(Cc2ccccc2)CC1	nan
	16019521	47866	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	442	3	0	9	2.5	Cc1ccc(C)c(S(=O)(=O)c2nnn3c2nc(N2CCN(C)CC2)c2sccc23)c1	nan
	CHEMBL1551283	47866	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	442	3	0	9	2.5	Cc1ccc(C)c(S(=O)(=O)c2nnn3c2nc(N2CCN(C)CC2)c2sccc23)c1	nan
	6414933	47898	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	7	1	8	4.2	CCOC(=O)c1ccc(NC(=O)C(CC)Sc2nnc3c4ccccc4n(C)c3n2)cc1	nan
	CHEMBL1551836	47898	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	7	1	8	4.2	CCOC(=O)c1ccc(NC(=O)C(CC)Sc2nnc3c4ccccc4n(C)c3n2)cc1	nan
	16018808	47910	1	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	8	1	7	2.7	CCc1nnc(SC(CC)C(=O)NCCOC)c2cc3occc3n12	nan
	CHEMBL1551969	47910	1	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	8	1	7	2.7	CCc1nnc(SC(CC)C(=O)NCCOC)c2cc3occc3n12	nan
	5301786	47934	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	3	1	8	1.0	Cc1ccc(-c2c(C)n3c4c(=O)n(C)c(=O)n(C)c4nc3n2CCO)cc1	nan
	CHEMBL1552221	47934	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	3	1	8	1.0	Cc1ccc(-c2c(C)n3c4c(=O)n(C)c(=O)n(C)c4nc3n2CCO)cc1	nan
	1622536	47997	15	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	6	2	6	4.7	CCCCOC(=O)c1ccc(NC(=O)c2sc3nc(C)cc(C)c3c2N)cc1	nan
	CHEMBL1553105	47997	15	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	6	2	6	4.7	CCCCOC(=O)c1ccc(NC(=O)c2sc3nc(C)cc(C)c3c2N)cc1	nan
	16020969	48033	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	400	4	1	5	5.0	Cc1oc(-c2cccc(Br)c2)nc1CSc1nc2cccnc2[nH]1	nan
	CHEMBL1553552	48033	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	400	4	1	5	5.0	Cc1oc(-c2cccc(Br)c2)nc1CSc1nc2cccnc2[nH]1	nan
	4291583	48068	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	588	14	4	8	2.2	CSCCC(NS(=O)(=O)c1ccc2c(c1)Cc1cc(S(=O)(=O)NC(CCSC)C(=O)O)ccc1-2)C(=O)O	nan
	CHEMBL1554139	48068	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	588	14	4	8	2.2	CSCCC(NS(=O)(=O)c1ccc2c(c1)Cc1cc(S(=O)(=O)NC(CCSC)C(=O)O)ccc1-2)C(=O)O	nan
	20877874	48107	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	3	0	4	3.5	CCCN1CCN(C(=O)c2cc3c(s2)-c2ccccc2OC3)CC1	nan
	CHEMBL1554696	48107	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	3	0	4	3.5	CCCN1CCN(C(=O)c2cc3c(s2)-c2ccccc2OC3)CC1	nan
	16011310	48174	2	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	4	0	5	5.5	CCc1nnc(SCc2cccc(Cl)c2)c2cc3sccc3n12	nan
	CHEMBL1555647	48174	2	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	4	0	5	5.5	CCc1nnc(SCc2cccc(Cl)c2)c2cc3sccc3n12	nan
	16030467	48701	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	7	1	4	5.3	O=C(CSc1nc2ccccc2nc1Cc1ccccc1)NCc1ccccc1Cl	nan
	CHEMBL1560326	48701	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	7	1	4	5.3	O=C(CSc1nc2ccccc2nc1Cc1ccccc1)NCc1ccccc1Cl	nan
	2415608	48753	22	None	-5	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	4	2	7	2.8	CC(=O)Nc1ccc(S(=O)(=O)Nc2nc3cc4c(cc3nc2Cl)OCCO4)cc1	nan
	CHEMBL1560923	48753	22	None	-5	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	4	2	7	2.8	CC(=O)Nc1ccc(S(=O)(=O)Nc2nc3cc4c(cc3nc2Cl)OCCO4)cc1	nan
	15988392	48979	2	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	5	1	7	2.8	CCn1c(=O)c2sccc2n2c(CCC(=O)Nc3ccc(F)cc3)nnc12	nan
	CHEMBL1562908	48979	2	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	5	1	7	2.8	CCn1c(=O)c2sccc2n2c(CCC(=O)Nc3ccc(F)cc3)nnc12	nan
	3805026	49092	19	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	4	1	6	5.2	Cc1cc(N2C(=O)C(O)=C(C(=O)c3cc4ccccc4o3)C2c2ccc(Cl)cc2)no1	nan
	CHEMBL1563863	49092	19	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	4	1	6	5.2	Cc1cc(N2C(=O)C(O)=C(C(=O)c3cc4ccccc4o3)C2c2ccc(Cl)cc2)no1	nan
	6228410	49155	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	4	1	7	4.1	Cc1nnc(N2C(=O)C(O)=C(C(=O)c3ccc4c(c3)CC(C)O4)C2c2ccccc2F)s1	nan
	CHEMBL1564525	49155	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	4	1	7	4.1	Cc1nnc(N2C(=O)C(O)=C(C(=O)c3ccc4c(c3)CC(C)O4)C2c2ccccc2F)s1	nan
	4802105	49323	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	6	1	7	2.8	Cn1cnnc1SCC(=O)Nc1cc(S(=O)(=O)N2CCCCCC2)ccc1Cl	nan
	CHEMBL1565823	49323	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	6	1	7	2.8	Cn1cnnc1SCC(=O)Nc1cc(S(=O)(=O)N2CCCCCC2)ccc1Cl	nan
	225436	49566	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	198	0	1	3	1.2	O=C1c2ccccc2C(=O)c2[nH]cnc21	nan
	CHEMBL1567800	49566	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	198	0	1	3	1.2	O=C1c2ccccc2C(=O)c2[nH]cnc21	nan
	2054020	49676	10	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	4	1	7	4.7	O=C(CSc1ncnc2c1oc1ccccc12)Nc1nc2ccccc2s1	nan
	CHEMBL1568611	49676	10	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	4	1	7	4.7	O=C(CSc1ncnc2c1oc1ccccc12)Nc1nc2ccccc2s1	nan
	2883018	49839	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	227	0	1	5	1.6	N#Cc1c2n(c3c(N)ncnc13)CCCCC2	nan
	CHEMBL1570092	49839	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	227	0	1	5	1.6	N#Cc1c2n(c3c(N)ncnc13)CCCCC2	nan
	16018256	49973	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	9	1	6	3.6	CCOc1ccc(CCNC(=O)Cn2c(=O)c3cccn3c3ccc(F)cc32)cc1OCC	nan
	CHEMBL1571269	49973	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	9	1	6	3.6	CCOc1ccc(CCNC(=O)Cn2c(=O)c3cccn3c3ccc(F)cc32)cc1OCC	nan
	25163648	50106	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	6	0	4	4.3	COc1ccc(S(=O)(=O)N2CCCCCC2)cc1C(=O)N(C)Cc1c(F)cccc1Cl	nan
	CHEMBL1572593	50106	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	6	0	4	4.3	COc1ccc(S(=O)(=O)N2CCCCCC2)cc1C(=O)N(C)Cc1c(F)cccc1Cl	nan
	20957176	50184	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	4	0	9	0.2	CN1CCN(C(=O)CCc2nnc3ccc(N4CCC5(CC4)OCCO5)nn23)CC1	nan
	CHEMBL1573164	50184	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	4	0	9	0.2	CN1CCN(C(=O)CCc2nnc3ccc(N4CCC5(CC4)OCCO5)nn23)CC1	nan
	4200979	50509	3	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	5	1	7	1.0	COC(=O)CCNC(=O)Cn1cnc2sc3c(c2c1=O)CCCC3	nan
	CHEMBL1576536	50509	3	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	5	1	7	1.0	COC(=O)CCNC(=O)Cn1cnc2sc3c(c2c1=O)CCCC3	nan
	1132498	50720	11	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	2	1	5	5.1	Cc1ccc2nsnc2c1NC(=O)c1sc2ccccc2c1Cl	nan
	CHEMBL1578314	50720	11	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	2	1	5	5.1	Cc1ccc2nsnc2c1NC(=O)c1sc2ccccc2c1Cl	nan
	3220367	50975	3	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	7	1	6	2.4	COCCNC(=O)C(OC(=O)c1nsc(Cl)c1Cl)C(C)C	nan
	CHEMBL1580567	50975	3	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	7	1	6	2.4	COCCNC(=O)C(OC(=O)c1nsc(Cl)c1Cl)C(C)C	nan
	4343313	51174	14	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	4	1	5	4.2	Cc1cccc(N2C(=O)C(O)=C(C(=O)c3cccs3)C2c2ccccc2)n1	nan
	CHEMBL1582134	51174	14	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	4	1	5	4.2	Cc1cccc(N2C(=O)C(O)=C(C(=O)c3cccs3)C2c2ccccc2)n1	nan
	3338549	51190	14	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	488	8	1	8	5.3	CCCOc1ccc(C2C(C(=O)c3cc4ccccc4o3)=C(O)C(=O)N2c2cc(C)on2)cc1OC	nan
	CHEMBL1582307	51190	14	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	488	8	1	8	5.3	CCCOc1ccc(C2C(C(=O)c3cc4ccccc4o3)=C(O)C(=O)N2c2cc(C)on2)cc1OC	nan
	20917770	51345	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	6	0	7	2.4	CN(Cc1ccco1)S(=O)(=O)c1ccc(CN2C(=O)c3cccnc3C2=O)s1	nan
	CHEMBL1583626	51345	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	6	0	7	2.4	CN(Cc1ccco1)S(=O)(=O)c1ccc(CN2C(=O)c3cccnc3C2=O)s1	nan
	18562929	51493	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	8	1	9	1.1	COc1ccc(C(=O)NCCc2nnc3ccc(SCC(=O)N4CCOCC4)nn23)cc1	nan
	CHEMBL1584882	51493	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	8	1	9	1.1	COc1ccc(C(=O)NCCc2nnc3ccc(SCC(=O)N4CCOCC4)nn23)cc1	nan
	2427540	51914	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	463	6	1	10	1.4	Cn1c(N)c(C(=O)CSc2nc3ccccc3c(=O)n2Cc2ccccc2)c(=O)n(C)c1=O	nan
	CHEMBL1588321	51914	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	463	6	1	10	1.4	Cn1c(N)c(C(=O)CSc2nc3ccccc3c(=O)n2Cc2ccccc2)c(=O)n(C)c1=O	nan
	20923114	51939	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	9	0	6	2.7	CCCN(CCC)S(=O)(=O)c1cc(CN2C(=O)c3cccnc3C2=O)ccc1OC	nan
	CHEMBL1588547	51939	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	9	0	6	2.7	CCCN(CCC)S(=O)(=O)c1cc(CN2C(=O)c3cccnc3C2=O)ccc1OC	nan
	20885679	52143	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	6	1	6	1.9	Cc1nn(CCCC(=O)NCc2ccccc2Cl)c(=O)c2nccn12	nan
	CHEMBL1590561	52143	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	6	1	6	1.9	Cc1nn(CCCC(=O)NCc2ccccc2Cl)c(=O)c2nccn12	nan
	16023172	52167	1	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	7	1	6	3.4	CCCCNC(=O)CSc1nnc(C)c2c(C)n(-c3ccccc3)nc12	nan
	CHEMBL1590852	52167	1	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	7	1	6	3.4	CCCCNC(=O)CSc1nnc(C)c2c(C)n(-c3ccccc3)nc12	nan
	16016417	52208	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	3	1	5	3.4	Cc1cc(O)c(CN2CCN(c3ccccc3)CC2)c2oc(=O)cc(C)c12	nan
	CHEMBL1591358	52208	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	3	1	5	3.4	Cc1cc(O)c(CN2CCN(c3ccccc3)CC2)c2oc(=O)cc(C)c12	nan
	16009611	52365	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	5	1	6	4.6	O=C(Nc1cccc(OCc2cc(=O)n3c4c(sc3n2)CCCC4)c1)c1ccc(F)cc1	nan
	CHEMBL1593455	52365	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	5	1	6	4.6	O=C(Nc1cccc(OCc2cc(=O)n3c4c(sc3n2)CCCC4)c1)c1ccc(F)cc1	nan
	16453157	52823	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	6	2	8	2.7	O=C(Nc1ccc(S(=O)(=O)Nc2nccs2)cc1)c1nn(-c2ccccc2)ccc1=O	nan
	CHEMBL1597782	52823	13	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	6	2	8	2.7	O=C(Nc1ccc(S(=O)(=O)Nc2nccs2)cc1)c1nn(-c2ccccc2)ccc1=O	nan
	15990388	53029	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	3	1	6	2.4	Cc1c(NC(=O)c2nc3ccccc3n(C)c2=O)cccc1[N+](=O)[O-]	nan
	CHEMBL1599627	53029	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	3	1	6	2.4	Cc1c(NC(=O)c2nc3ccccc3n(C)c2=O)cccc1[N+](=O)[O-]	nan
	20917744	53108	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	6	1	7	2.3	Cc1ccc(CNS(=O)(=O)c2ccc(CN3C(=O)c4cccnc4C3=O)s2)o1	nan
	CHEMBL1600418	53108	5	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	6	1	7	2.3	Cc1ccc(CNS(=O)(=O)c2ccc(CN3C(=O)c4cccnc4C3=O)s2)o1	nan
	3252667	53124	18	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	4	1	6	4.8	Cc1ccc(C2C(C(=O)c3cc4ccccc4o3)=C(O)C(=O)N2c2cc(C)on2)cc1	nan
	CHEMBL1600566	53124	18	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	4	1	6	4.8	Cc1ccc(C2C(C(=O)c3cc4ccccc4o3)=C(O)C(=O)N2c2cc(C)on2)cc1	nan
	5389427	53204	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	7	1	7	4.2	CCOc1ccc(C(=O)C2=C(O)C(=O)N(c3cc(C)on3)C2c2ccccc2OC)cc1	nan
	CHEMBL1601252	53204	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	7	1	7	4.2	CCOc1ccc(C(=O)C2=C(O)C(=O)N(c3cc(C)on3)C2c2ccccc2OC)cc1	nan
	723168	53528	39	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	301	4	1	4	4.2	O=C(O)Cc1sc(-c2ccccc2)nc1-c1cccs1	nan
	CHEMBL1604196	53528	39	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	301	4	1	4	4.2	O=C(O)Cc1sc(-c2ccccc2)nc1-c1cccs1	nan
	2235547	53666	30	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	222	3	1	5	2.4	CCOc1ccccc1-c1nnc(S)o1	nan
	CHEMBL1605444	53666	30	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	222	3	1	5	2.4	CCOc1ccccc1-c1nnc(S)o1	nan
	2927721	53815	17	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	423	7	2	7	2.6	CCOCCCn1c(=N)c(C(=O)NC2CCCCC2)cc2c(=O)n3ccccc3nc21	nan
	CHEMBL1606632	53815	17	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	423	7	2	7	2.6	CCOCCCn1c(=N)c(C(=O)NC2CCCCC2)cc2c(=O)n3ccccc3nc21	nan
	3417563	53905	17	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	7	1	7	3.4	COc1cccc(C2C(C(=O)c3cc4ccccc4o3)=C(O)C(=O)N2CCN2CCOCC2)c1	nan
	3983329	53905	17	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	7	1	7	3.4	COc1cccc(C2C(C(=O)c3cc4ccccc4o3)=C(O)C(=O)N2CCN2CCOCC2)c1	nan
	CHEMBL1607267	53905	17	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	7	1	7	3.4	COc1cccc(C2C(C(=O)c3cc4ccccc4o3)=C(O)C(=O)N2CCN2CCOCC2)c1	nan
	3146573	54130	19	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	4	1	7	3.5	Cc1ccc(C2C(C(=O)c3ccco3)=C(O)C(=O)N2c2nnc(C)s2)cc1	nan
	CHEMBL1609156	54130	19	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	4	1	7	3.5	Cc1ccc(C2C(C(=O)c3ccco3)=C(O)C(=O)N2c2nnc(C)s2)cc1	nan
	1941998	54163	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	4	2	5	5.1	COc1cccc(-c2ccc3c(N)c(C(=O)Nc4cc(F)ccc4F)sc3n2)c1	nan
	CHEMBL1609358	54163	10	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	4	2	5	5.1	COc1cccc(-c2ccc3c(N)c(C(=O)Nc4cc(F)ccc4F)sc3n2)c1	nan
	5389862	54295	6	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	410	9	1	6	3.5	COCCCN1C(=O)C(O)=C(C(=O)c2ccc(OC(C)C)cc2)C1c1cccnc1	nan
	CHEMBL1610515	54295	6	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	410	9	1	6	3.5	COCCCN1C(=O)C(O)=C(C(=O)c2ccc(OC(C)C)cc2)C1c1cccnc1	nan
	9550945	54458	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	2	0	5	3.2	CCOC(=O)N1CCN(C(=O)c2cc3c(s2)-c2ccccc2OC3)CC1	nan
	CHEMBL1611989	54458	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	2	0	5	3.2	CCOC(=O)N1CCN(C(=O)c2cc3c(s2)-c2ccccc2OC3)CC1	nan
	2120111	55414	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	317	3	0	3	4.3	COc1ccc(Br)cc1-c1nc(CCl)cs1	nan
	CHEMBL1484562	55414	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	317	3	0	3	4.3	COc1ccc(Br)cc1-c1nc(CCl)cs1	nan
	CHEMBL1622008	55414	6	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	317	3	0	3	4.3	COc1ccc(Br)cc1-c1nc(CCl)cs1	nan
	1724830	55559	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	4	2	8	1.8	NN1C(=O)/C(=C2/Sc3ccccc3N2CCCS(=O)(=O)O)SC1=S	nan
	CHEMBL1520781	55559	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	4	2	8	1.8	NN1C(=O)/C(=C2/Sc3ccccc3N2CCCS(=O)(=O)O)SC1=S	nan
	CHEMBL1623209	55559	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	4	2	8	1.8	NN1C(=O)/C(=C2/Sc3ccccc3N2CCCS(=O)(=O)O)SC1=S	nan
	9619025	71625	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	400	6	1	10	-0.4	COc1cccc(/C=N/NC(=O)Cn2cnc3c2c(=O)n(C)c(=O)n3C)c1OC	nan
	CHEMBL1973418	71625	8	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	400	6	1	10	-0.4	COc1cccc(/C=N/NC(=O)Cn2cnc3c2c(=O)n(C)c(=O)n3C)c1OC	nan
	5065598	72241	11	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	5	0	8	2.9	CCOC(=O)Cn1/c(=N/C(=O)c2cccs2)sc2cc(C(=O)OC)ccc21	nan
	CHEMBL1992834	72241	11	None	-1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	5	0	8	2.9	CCOC(=O)Cn1/c(=N/C(=O)c2cccs2)sc2cc(C(=O)OC)ccc21	nan
	5286961	72492	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	538	3	2	4	5.3	CC1=C/C(=C(\c2cc(C)c(O)c(Br)c2)c2ccccc2S(=O)(=O)O)C=C(Br)C1=O	nan
	9915251	72492	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	538	3	2	4	5.3	CC1=C/C(=C(\c2cc(C)c(O)c(Br)c2)c2ccccc2S(=O)(=O)O)C=C(Br)C1=O	nan
	CHEMBL2001904	72492	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	538	3	2	4	5.3	CC1=C/C(=C(\c2cc(C)c(O)c(Br)c2)c2ccccc2S(=O)(=O)O)C=C(Br)C1=O	nan
	95028	93375	28	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	270	2	0	6	0.5	Cn1c(=O)c2c(ncn2Cc2ccccc2)n(C)c1=O	nan
	CHEMBL24759	93375	28	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	270	2	0	6	0.5	Cn1c(=O)c2c(ncn2Cc2ccccc2)n(C)c1=O	nan
	135723776	107098	2	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	318	3	2	5	2.6	Cc1cc(O)nc(N/N=C/c2c(F)c(F)c(F)c(F)c2F)n1	nan
	CHEMBL3189383	107098	2	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	318	3	2	5	2.6	Cc1cc(O)nc(N/N=C/c2c(F)c(F)c(F)c(F)c2F)n1	nan
	5342833	107108	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	290	3	3	9	-2.3	Cn1c(=O)c2nc(N/N=C(/C#N)C(N)=O)[nH]c2n(C)c1=O	nan
	CHEMBL3189560	107108	9	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	290	3	3	9	-2.3	Cn1c(=O)c2nc(N/N=C(/C#N)C(N)=O)[nH]c2n(C)c1=O	nan
	4564145	107361	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	3	0	5	3.1	CCOC(=O)c1s/c(=N\C(=O)c2ccc(Br)cc2)n(C)c1C	nan
	CHEMBL3192424	107361	11	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	3	0	5	3.1	CCOC(=O)c1s/c(=N\C(=O)c2ccc(Br)cc2)n(C)c1C	nan
	135526880	107781	5	None	1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	4	2	6	3.0	O=C1CC(C(=O)Nc2ccc(Br)cc2)SC(N/N=C/c2ccco2)=N1	nan
	135643494	107781	5	None	1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	4	2	6	3.0	O=C1CC(C(=O)Nc2ccc(Br)cc2)SC(N/N=C/c2ccco2)=N1	nan
	137199718	107781	5	None	1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	4	2	6	3.0	O=C1CC(C(=O)Nc2ccc(Br)cc2)SC(N/N=C/c2ccco2)=N1	nan
	CHEMBL3197292	107781	5	None	1	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	4	2	6	3.0	O=C1CC(C(=O)Nc2ccc(Br)cc2)SC(N/N=C/c2ccco2)=N1	nan
	9660607	107807	5	None	-2	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	2	1	3	3.8	Cc1ccc(N2C(=O)CS/C2=N\C(=S)Nc2ccccc2)cc1	nan
	CHEMBL3197507	107807	5	None	-2	2	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	2	1	3	3.8	Cc1ccc(N2C(=O)CS/C2=N\C(=S)Nc2ccccc2)cc1	nan
	9583775	108407	2	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	5	2	7	2.1	Nc1c(C(=O)N/N=C/c2ccc([N+](=O)[O-])cc2)cnn1-c1ccccc1	nan
	CHEMBL3210811	108407	2	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	5	2	7	2.1	Nc1c(C(=O)N/N=C/c2ccc([N+](=O)[O-])cc2)cnn1-c1ccccc1	nan
	3669734	197044	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	6	1	7	2.6	CCOC(=O)N1CCN(C(=O)CCCCn2c(=S)[nH]c3ccsc3c2=O)CC1	nan
	CHEMBL582737	197044	7	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	6	1	7	2.6	CCOC(=O)N1CCN(C(=O)CCCCn2c(=S)[nH]c3ccsc3c2=O)CC1	nan
	3324	204712	112	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	7	1	9	0.5	CC(=O)OCC(CCn1cnc2cnc(N)nc21)COC(C)=O	nan
	CHEMBL880	204712	112	None	-	1	Human	4.8	pPotency	=	4.8	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	7	1	9	0.5	CC(=O)OCC(CCn1cnc2cnc(N)nc21)COC(C)=O	nan
	1028	287	69	None	-512	16	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	183	3	4	4	0.4	CNC[C@@H](c1ccc(c(c1)O)O)O	nan
	139148732	287	69	None	-512	16	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	183	3	4	4	0.4	CNC[C@@H](c1ccc(c(c1)O)O)O	nan
	479	287	69	None	-512	16	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	183	3	4	4	0.4	CNC[C@@H](c1ccc(c(c1)O)O)O	nan
	5816	287	69	None	-512	16	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	183	3	4	4	0.4	CNC[C@@H](c1ccc(c(c1)O)O)O	nan
	CHEMBL679	287	69	None	-512	16	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	183	3	4	4	0.4	CNC[C@@H](c1ccc(c(c1)O)O)O	nan
	DB00668	287	69	None	-512	16	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	183	3	4	4	0.4	CNC[C@@H](c1ccc(c(c1)O)O)O	nan
	3289443	6987	2	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	3	2	5	5.0	Nc1c(C(=O)Nc2cccc(F)c2)sc2nc(-c3cccs3)ccc12	nan
	CHEMBL1084955	6987	2	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	3	2	5	5.0	Nc1c(C(=O)Nc2cccc(F)c2)sc2nc(-c3cccs3)ccc12	nan
	4112670	10380	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	454	7	3	4	5.5	O=C(NCCc1ccc(Cl)cc1)C1CCC(CNc2nc(=S)[nH]c3ccccc23)CC1	nan
	CHEMBL1165197	10380	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	454	7	3	4	5.5	O=C(NCCc1ccc(Cl)cc1)C1CCC(CNc2nc(=S)[nH]c3ccccc23)CC1	nan
	1003890	18177	15	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	423	5	2	5	5.1	COc1cccc(-c2ccc3c(N)c(C(=O)NCc4ccc(Cl)cc4)sc3n2)c1	nan
	CHEMBL1271075	18177	15	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	423	5	2	5	5.1	COc1cccc(-c2ccc3c(N)c(C(=O)NCc4ccc(Cl)cc4)sc3n2)c1	nan
	790786	19569	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	283	1	0	1	4.5	CCc1c(C)nc2ccc(Br)cc2c1Cl	nan
	CHEMBL1301385	19569	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	283	1	0	1	4.5	CCc1c(C)nc2ccc(Br)cc2c1Cl	nan
	6621843	19658	2	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	241	3	1	5	2.4	CCCNc1nc2ccccc2n2c(C)nnc12	nan
	CHEMBL1302226	19658	2	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	241	3	1	5	2.4	CCCNc1nc2ccccc2n2c(C)nnc12	nan
	926200	19882	13	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	332	2	0	4	4.0	Fc1cnc(N2CCc3ccccc32)nc1N1CCc2ccccc21	nan
	CHEMBL1303908	19882	13	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	332	2	0	4	4.0	Fc1cnc(N2CCc3ccccc32)nc1N1CCc2ccccc21	nan
	20881176	20170	2	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	8	1	7	2.3	CC(C)CCn1c(=O)c2ccccc2n2c(CCC(=O)NCC3CCCO3)nnc12	nan
	CHEMBL1306246	20170	2	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	8	1	7	2.3	CC(C)CCn1c(=O)c2ccccc2n2c(CCC(=O)NCC3CCCO3)nnc12	nan
	2220688	20321	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	477	3	0	6	4.3	Cc1ccc(-c2cc(C(=O)N3CCN(c4ncccn4)CC3)c3cc(Br)ccc3n2)o1	nan
	CHEMBL1307526	20321	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	477	3	0	6	4.3	Cc1ccc(-c2cc(C(=O)N3CCN(c4ncccn4)CC3)c3cc(Br)ccc3n2)o1	nan
	2962628	20412	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	550	9	3	5	5.0	CCOc1cc(C2NC(=O)NC(c3ccccc3)=C2C(=O)c2ccccc2)c(Br)cc1OCC(=O)O	nan
	CHEMBL1308267	20412	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	550	9	3	5	5.0	CCOc1cc(C2NC(=O)NC(c3ccccc3)=C2C(=O)c2ccccc2)c(Br)cc1OCC(=O)O	nan
	3774396	20630	2	None	-2	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	230	1	3	6	1.7	CSc1nc(S)c2[nH]c(S)nc2n1	nan
	CHEMBL1310138	20630	2	None	-2	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	230	1	3	6	1.7	CSc1nc(S)c2[nH]c(S)nc2n1	nan
	6247103	20943	19	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	5	1	5	4.4	COc1cc(/C=C2\CCc3c2nc2ccccc2c3C(=O)O)cc(OC)c1OC	nan
	CHEMBL1312514	20943	19	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	5	1	5	4.4	COc1cc(/C=C2\CCc3c2nc2ccccc2c3C(=O)O)cc(OC)c1OC	nan
	2927414	21300	20	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	8	2	8	1.9	CCOCCCn1c(=N)c(C(=O)NCc2cccnc2)cc2c(=O)n3ccccc3nc21	nan
	CHEMBL1315953	21300	20	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	8	2	8	1.9	CCOCCCn1c(=N)c(C(=O)NCc2cccnc2)cc2c(=O)n3ccccc3nc21	nan
	16187669	21648	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	501	11	2	7	3.0	CCC1CCCCN1CCCNC(=O)CCCNC(=O)Cn1cnc2sc3c(c2c1=O)CCCC3	nan
	CHEMBL1319736	21648	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	501	11	2	7	3.0	CCC1CCCCN1CCCNC(=O)CCCNC(=O)Cn1cnc2sc3c(c2c1=O)CCCC3	nan
	1473386	21756	23	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	265	4	0	7	0.7	CCOC(=O)CSc1nc(=O)n2ccccc2n1	nan
	CHEMBL1320637	21756	23	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	265	4	0	7	0.7	CCOC(=O)CSc1nc(=O)n2ccccc2n1	nan
	2363935	21797	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	345	6	1	8	0.0	Cn1c(N)c(C(=O)COC(=O)CCc2ccccc2)c(=O)n(C)c1=O	nan
	CHEMBL1321001	21797	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	345	6	1	8	0.0	Cn1c(N)c(C(=O)COC(=O)CCc2ccccc2)c(=O)n(C)c1=O	nan
	1485315	21814	20	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	3	2	5	1.6	CS(=O)(=O)NNC(=O)c1cc2cc3ccccc3nc2s1	nan
	CHEMBL1321144	21814	20	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	3	2	5	1.6	CS(=O)(=O)NNC(=O)c1cc2cc3ccccc3nc2s1	nan
	20903731	21833	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	9	1	7	2.2	CC1CCN(c2ccc3nnc(CCC(=O)NCCCOC(C)C)n3n2)CC1	nan
	CHEMBL1321331	21833	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	9	1	7	2.2	CC1CCN(c2ccc3nnc(CCC(=O)NCCCOC(C)C)n3n2)CC1	nan
	16014625	21865	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	4	2	5	2.3	CC(=O)Nc1ccc(NC(=O)C2CCN(c3cnccn3)CC2)cc1	nan
	CHEMBL1321666	21865	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	4	2	5	2.3	CC(=O)Nc1ccc(NC(=O)C2CCN(c3cnccn3)CC2)cc1	nan
	16031994	22040	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	5	1	6	5.3	Cc1nc(C)c(-c2ccc(SCC(=O)Nc3ccc(Cl)c(Cl)c3)nn2)s1	nan
	CHEMBL1323264	22040	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	5	1	6	5.3	Cc1nc(C)c(-c2ccc(SCC(=O)Nc3ccc(Cl)c(Cl)c3)nn2)s1	nan
	857564	22097	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	5	1	5	4.1	CCc1cc2cccc(C)c2nc1SCC(=O)Nc1cc(C)on1	nan
	CHEMBL1323763	22097	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	5	1	5	4.1	CCc1cc2cccc(C)c2nc1SCC(=O)Nc1cc(C)on1	nan
	1955570	22198	11	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	4	2	5	5.1	COc1cccc(-c2ccc3c(N)c(C(=O)Nc4ccccc4C)sc3n2)c1	nan
	CHEMBL1324540	22198	11	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	4	2	5	5.1	COc1cccc(-c2ccc3c(N)c(C(=O)Nc4ccccc4C)sc3n2)c1	nan
	16019112	22222	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	483	5	1	8	3.6	Cc1ccccc1NC(=O)Cn1c(=O)n(Cc2ccc3c(c2)OCO3)c(=O)c2oc3ccccc3c21	nan
	CHEMBL1324746	22222	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	483	5	1	8	3.6	Cc1ccccc1NC(=O)Cn1c(=O)n(Cc2ccc3c(c2)OCO3)c(=O)c2oc3ccccc3c21	nan
	20957487	22300	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	494	9	1	8	2.0	O=C1CCCN1CCCNc1ccc2nnc(CCC(=O)N3CCN(c4ccccc4F)CC3)n2n1	nan
	CHEMBL1325415	22300	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	494	9	1	8	2.0	O=C1CCCN1CCCNc1ccc2nnc(CCC(=O)N3CCN(c4ccccc4F)CC3)n2n1	nan
	654648	22331	13	None	-3	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	7	1	7	4.4	C=CCOc1cccc(C2C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2c2nccs2)c1	nan
	CHEMBL1325819	22331	13	None	-3	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	7	1	7	4.4	C=CCOc1cccc(C2C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2c2nccs2)c1	nan
	16411657	22485	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	300	2	2	4	0.9	CC1=NN(c2ccccc2)C(=O)C1/C=C1/NC(=S)NC1=O	nan
	CHEMBL1327209	22485	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	300	2	2	4	0.9	CC1=NN(c2ccccc2)C(=O)C1/C=C1/NC(=S)NC1=O	nan
	3725176	22707	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	457	6	1	5	5.7	COc1ccc(-c2cc(C(F)(F)F)c(C#N)c(SCC(=O)Nc3cccc(C)c3)n2)cc1	nan
	CHEMBL1329088	22707	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	457	6	1	5	5.7	COc1ccc(-c2cc(C(F)(F)F)c(C#N)c(SCC(=O)Nc3cccc(C)c3)n2)cc1	nan
	2965680	23608	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	4	1	4	4.4	CC(NC(=O)c1cc(-c2cccnc2)nc2ccc(Br)cc12)C1CCCO1	nan
	CHEMBL1336138	23608	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	4	1	4	4.4	CC(NC(=O)c1cc(-c2cccnc2)nc2ccc(Br)cc12)C1CCCO1	nan
	2928436	23637	17	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	5	2	8	1.7	N=c1c(C(=O)NCC2CCCO2)cc2c(=O)n3ccccc3nc2n1Cc1ccco1	nan
	CHEMBL1336360	23637	17	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	5	2	8	1.7	N=c1c(C(=O)NCC2CCCO2)cc2c(=O)n3ccccc3nc2n1Cc1ccco1	nan
	16023198	23862	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	6	1	6	4.0	Cc1nnc(SCC(=O)NCc2cccc(F)c2)c2nn(-c3ccccc3)c(C)c12	nan
	CHEMBL1338308	23862	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	6	1	6	4.0	Cc1nnc(SCC(=O)NCc2cccc(F)c2)c2nn(-c3ccccc3)c(C)c12	nan
	4907461	23980	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	304	6	1	5	3.7	CCCCNc1ncnc2sc3c(c12)CCN(CCC)C3	nan
	CHEMBL1339392	23980	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	304	6	1	5	3.7	CCCCNc1ncnc2sc3c(c12)CCN(CCC)C3	nan
	4173573	24425	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	5	2	8	0.8	Cc1cccn2c(=O)c3cc(C(N)=S)c(=N)n(CCCN4CCOCC4)c3nc12	nan
	CHEMBL1343182	24425	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	5	2	8	0.8	Cc1cccn2c(=O)c3cc(C(N)=S)c(=N)n(CCCN4CCOCC4)c3nc12	nan
	2439152	24438	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	335	2	0	5	2.2	Cc1ccc2nc(Cn3cc(C(F)(F)F)ccc3=O)cc(=O)n2c1	nan
	CHEMBL1343295	24438	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	335	2	0	5	2.2	Cc1ccc2nc(Cn3cc(C(F)(F)F)ccc3=O)cc(=O)n2c1	nan
	4918386	24788	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	5	1	6	2.5	Cc1cc(CNC(=O)C(C)n2cc([N+](=O)[O-])cn2)c2ccccc2n1	nan
	CHEMBL1346435	24788	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	5	1	6	2.5	Cc1cc(CNC(=O)C(C)n2cc([N+](=O)[O-])cn2)c2ccccc2n1	nan
	20904584	24804	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	5	0	9	1.7	Cn1c(=O)c2sccc2n2c(CCCC(=O)N3CCN(c4ccccn4)CC3)nnc12	nan
	CHEMBL1346578	24804	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	5	0	9	1.7	Cn1c(=O)c2sccc2n2c(CCCC(=O)N3CCN(c4ccccn4)CC3)nnc12	nan
	6112144	24819	3	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	504	9	1	7	3.5	C=CCOc1cccc(C2C(C(=O)c3ccc4c(c3)CC(C)O4)=C(O)C(=O)N2CCN2CCOCC2)c1	nan
	CHEMBL1346652	24819	3	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	504	9	1	7	3.5	C=CCOc1cccc(C2C(C(=O)c3ccc4c(c3)CC(C)O4)=C(O)C(=O)N2CCN2CCOCC2)c1	nan
	5181544	25137	17	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	5	1	8	3.5	COC(=O)c1ccc(C2C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2c2cc(C)on2)cc1	nan
	CHEMBL1349309	25137	17	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	5	1	8	3.5	COC(=O)c1ccc(C2C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2c2cc(C)on2)cc1	nan
	663780	25215	13	None	-5	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	8	2	8	2.2	Cc1ccc2nc3c(cc(C(=O)NCC4CCCO4)c(=N)n3CCCOC(C)C)c(=O)n2c1	nan
	CHEMBL1349978	25215	13	None	-5	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	8	2	8	2.2	Cc1ccc2nc3c(cc(C(=O)NCC4CCCO4)c(=N)n3CCCOC(C)C)c(=O)n2c1	nan
	860395	25224	40	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	273	2	1	3	3.8	O=C(O)c1cc(-c2cccs2)nc2ccc(F)cc12	nan
	CHEMBL1350037	25224	40	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	273	2	1	3	3.8	O=C(O)c1cc(-c2cccs2)nc2ccc(F)cc12	nan
	1013700	25415	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	3	0	3	3.6	O=C(COc1ccc2cc(Br)ccc2c1Br)N1CCOCC1	nan
	CHEMBL1351652	25415	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	3	0	3	3.6	O=C(COc1ccc2cc(Br)ccc2c1Br)N1CCOCC1	nan
	4137672	25559	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	4	1	4	4.1	O=C(O)c1ccccc1SCc1cn2cc(Br)ccc2n1	nan
	CHEMBL1352828	25559	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	4	1	4	4.1	O=C(O)c1ccccc1SCc1cn2cc(Br)ccc2n1	nan
	15991076	25855	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	4	1	4	6.6	COc1cc2ccccc2cc1C(=O)Nc1ccc2oc(-c3ccc(Cl)cc3)nc2c1	nan
	CHEMBL1355303	25855	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	4	1	4	6.6	COc1cc2ccccc2cc1C(=O)Nc1ccc2oc(-c3ccc(Cl)cc3)nc2c1	nan
	16019626	25939	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	3	1	8	3.2	Cc1ccc(-n2nnc(-c3nc(-c4cccs4)no3)c2N)c(C)c1	nan
	CHEMBL1356419	25939	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	3	1	8	3.2	Cc1ccc(-n2nnc(-c3nc(-c4cccs4)no3)c2N)c(C)c1	nan
	16033238	25991	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	4	1	5	5.6	Cc1cccc(NC(=O)c2sc3ncnc(N(C)C4CCCCC4)c3c2C)c1C	nan
	CHEMBL1357134	25991	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	4	1	5	5.6	Cc1cccc(NC(=O)c2sc3ncnc(N(C)C4CCCCC4)c3c2C)c1C	nan
	4084525	26308	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	3	0	6	3.9	CCOC(=O)c1sc2nc(C)nc(N3CCCCC3C)c2c1C	nan
	CHEMBL1360386	26308	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	3	0	6	3.9	CCOC(=O)c1sc2nc(C)nc(N3CCCCC3C)c2c1C	nan
	1130278	26338	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	7	1	6	4.0	Cc1ccc(NC(=O)CSc2nnc(COc3ccccc3C)o2)cc1	nan
	CHEMBL1360712	26338	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	7	1	6	4.0	Cc1ccc(NC(=O)CSc2nnc(COc3ccccc3C)o2)cc1	nan
	2112396	26779	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	495	7	2	7	4.0	CNS(=O)(=O)c1cccc(C(=O)OCC(=O)Nc2ccc(-c3nc4ccc(C)cc4s3)cc2)c1	nan
	CHEMBL1364577	26779	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	495	7	2	7	4.0	CNS(=O)(=O)c1cccc(C(=O)OCC(=O)Nc2ccc(-c3nc4ccc(C)cc4s3)cc2)c1	nan
	3244890	27562	13	None	-5	3	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	294	4	1	2	3.7	O=C(O)CCc1ccc(-c2ccc(Br)cc2)o1	nan
	CHEMBL1370669	27562	13	None	-5	3	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	294	4	1	2	3.7	O=C(O)CCc1ccc(-c2ccc(Br)cc2)o1	nan
	135443907	27905	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	463	7	2	9	4.5	CCOc1ccc2nc(NC(=O)CSc3nc(O)c(C#N)c(-c4ccccc4)n3)sc2c1	nan
	CHEMBL1373145	27905	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	463	7	2	9	4.5	CCOc1ccc2nc(NC(=O)CSc3nc(O)c(C#N)c(-c4ccccc4)n3)sc2c1	nan
	16018180	27907	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	477	6	1	6	5.5	COc1ccc(OC)c(NC(=O)c2oc3c(c2C)-c2nn(Cc4ccc(Cl)cc4)cc2CC3)c1	nan
	CHEMBL1373157	27907	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	477	6	1	6	5.5	COc1ccc(OC)c(NC(=O)c2oc3c(c2C)-c2nn(Cc4ccc(Cl)cc4)cc2CC3)c1	nan
	2727621	28008	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	3	2	7	3.3	CSc1c(C#N)c(N)nc2sc(C(=O)c3ccccc3)c(N)c12	nan
	CHEMBL1373780	28008	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	3	2	7	3.3	CSc1c(C#N)c(N)nc2sc(C(=O)c3ccccc3)c(N)c12	nan
	16019289	28249	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	5	1	5	4.9	Cc1ccc(NC(=O)CSc2ccc(-c3cccs3)nn2)cc1Cl	nan
	CHEMBL1375486	28249	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	5	1	5	4.9	Cc1ccc(NC(=O)CSc2ccc(-c3cccs3)nn2)cc1Cl	nan
	2361888	28410	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	7	1	6	1.2	CCN(CC)S(=O)(=O)c1ccc(O)c(C(=O)OCC(=O)N2CCCC2)c1	nan
	CHEMBL1377052	28410	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	7	1	6	1.2	CCN(CC)S(=O)(=O)c1ccc(O)c(C(=O)OCC(=O)N2CCCC2)c1	nan
	887924	28494	9	None	-3	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	345	2	1	4	4.8	Cc1ccc2c(Cl)c(C(=O)Nc3ccc4c(c3)OCO4)sc2c1	nan
	CHEMBL1377850	28494	9	None	-3	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	345	2	1	4	4.8	Cc1ccc2c(Cl)c(C(=O)Nc3ccc4c(c3)OCO4)sc2c1	nan
	135527311	28982	2	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	4	1	8	3.7	COC(=O)CSc1nc(O)c2c(C(F)(F)F)cc(-c3cccs3)nc2n1	nan
	CHEMBL1382080	28982	2	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	4	1	8	3.7	COC(=O)CSc1nc(O)c2c(C(F)(F)F)cc(-c3cccs3)nc2n1	nan
	15987888	29247	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	7	1	4	4.8	CCN(CC)CCNC(=O)c1cc(-c2ccc(Br)s2)nc2ccccc12	nan
	CHEMBL1384448	29247	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	7	1	4	4.8	CCN(CC)CCNC(=O)c1cc(-c2ccc(Br)s2)nc2ccccc12	nan
	54710218	29544	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	297	2	1	4	3.7	Cc1ccc(Sc2c(O)c3ccccc3n(C)c2=O)cc1	nan
	CHEMBL1386873	29544	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	297	2	1	4	3.7	Cc1ccc(Sc2c(O)c3ccccc3n(C)c2=O)cc1	nan
	4047539	29742	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	4	1	8	0.8	CCOC(=O)CC1C(=O)NCCN1C(=O)c1cc2c(=O)n3ccccc3nc2s1	nan
	CHEMBL1388441	29742	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	4	1	8	0.8	CCOC(=O)CC1C(=O)NCCN1C(=O)c1cc2c(=O)n3ccccc3nc2s1	nan
	733870	29858	34	None	-3	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	294	3	1	4	3.6	CC(=O)c1sc(NC(=O)c2ccc(Cl)cc2)nc1C	nan
	CHEMBL1389324	29858	34	None	-3	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	294	3	1	4	3.6	CC(=O)c1sc(NC(=O)c2ccc(Cl)cc2)nc1C	nan
	829950	29972	14	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	302	3	0	5	1.6	CN(C)S(=O)(=O)c1cccc(-c2cn3cccnc3n2)c1	nan
	CHEMBL1390362	29972	14	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	302	3	0	5	1.6	CN(C)S(=O)(=O)c1cccc(-c2cn3cccnc3n2)c1	nan
	5027542	30016	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	4	0	7	1.5	O=C(CN1C(=O)C2CC=CCC2C1=O)OCc1cc(=O)n2cc(Br)ccc2n1	nan
	CHEMBL1390760	30016	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	4	0	7	1.5	O=C(CN1C(=O)C2CC=CCC2C1=O)OCc1cc(=O)n2cc(Br)ccc2n1	nan
	3634961	30130	17	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	446	6	1	6	3.7	Cc1ccc(C2C(C(=O)c3cc4ccccc4o3)=C(O)C(=O)N2CCN2CCOCC2)cc1	nan
	4315628	30130	17	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	446	6	1	6	3.7	Cc1ccc(C2C(C(=O)c3cc4ccccc4o3)=C(O)C(=O)N2CCN2CCOCC2)cc1	nan
	CHEMBL1391748	30130	17	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	446	6	1	6	3.7	Cc1ccc(C2C(C(=O)c3cc4ccccc4o3)=C(O)C(=O)N2CCN2CCOCC2)cc1	nan
	5898126	30162	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	6	1	6	4.1	COc1ccc(C(=O)C2=C(O)C(=O)N(Cc3ccco3)C2c2cccs2)cc1	nan
	CHEMBL1392030	30162	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	6	1	6	4.1	COc1ccc(C(=O)C2=C(O)C(=O)N(Cc3ccco3)C2c2cccs2)cc1	nan
	4531942	30199	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	5	1	11	0.0	CCSc1nnc(NC(=O)Cn2cnc3c2c(=O)n(C)c(=O)n3C)s1	nan
	CHEMBL1392325	30199	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	5	1	11	0.0	CCSc1nnc(NC(=O)Cn2cnc3c2c(=O)n(C)c(=O)n3C)s1	nan
	1102249	30259	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	4	2	4	4.5	O=C(Nc1ccc(Br)cn1)c1cccc(C(=O)Nc2ccc(Br)cn2)c1	nan
	CHEMBL1392808	30259	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	4	2	4	4.5	O=C(Nc1ccc(Br)cn1)c1cccc(C(=O)Nc2ccc(Br)cn2)c1	nan
	16018254	30758	2	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	273	2	1	4	1.1	CNC(=O)Cn1c(=O)c2cccn2c2ccc(F)cc21	nan
	CHEMBL1398599	30758	2	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	273	2	1	4	1.1	CNC(=O)Cn1c(=O)c2cccn2c2ccc(F)cc21	nan
	16873489	30889	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	396	5	1	8	2.5	O=[N+]([O-])c1ccccc1S(=O)(=O)Nc1cccc(-c2ccc3nncn3n2)c1	nan
	CHEMBL1399932	30889	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	396	5	1	8	2.5	O=[N+]([O-])c1ccccc1S(=O)(=O)Nc1cccc(-c2ccc3nncn3n2)c1	nan
	20957244	31045	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	466	7	0	9	2.5	CCOc1ccc(N(C)C(=O)CCc2nnc3ccc(N4CCC5(CC4)OCCO5)nn23)cc1	nan
	CHEMBL1401299	31045	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	466	7	0	9	2.5	CCOc1ccc(N(C)C(=O)CCc2nnc3ccc(N4CCC5(CC4)OCCO5)nn23)cc1	nan
	5053439	31060	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	5	1	6	1.2	COC(CNC(=O)c1ccc2nc3ccccc3c(=O)n2c1)OC	nan
	CHEMBL1401405	31060	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	5	1	6	1.2	COC(CNC(=O)c1ccc2nc3ccccc3c(=O)n2c1)OC	nan
	5734701	31257	13	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	7	1	6	4.2	CC(C)Oc1ccc(C(=O)C2=C(O)C(=O)N(Cc3cccnc3)C2c2ccco2)cc1	nan
	CHEMBL1403145	31257	13	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	7	1	6	4.2	CC(C)Oc1ccc(C(=O)C2=C(O)C(=O)N(Cc3cccnc3)C2c2ccco2)cc1	nan
	5302177	31343	13	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	2	0	5	2.0	O=c1nc2ccccn2c2ccc(S(=O)(=O)N3CCCCC3)cc12	nan
	CHEMBL1404020	31343	13	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	2	0	5	2.0	O=c1nc2ccccn2c2ccc(S(=O)(=O)N3CCCCC3)cc12	nan
	1504305	31545	13	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	277	5	0	7	1.7	Cc1cc(C)n(C(=O)CCCn2cc([N+](=O)[O-])cn2)n1	nan
	CHEMBL1405977	31545	13	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	277	5	0	7	1.7	Cc1cc(C)n(C(=O)CCCn2cc([N+](=O)[O-])cn2)n1	nan
	5221227	31775	13	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	495	7	2	10	-0.2	Cc1cccn2c(=O)c3cc(C(=O)NCCN4CCOCC4)c(=N)n(CCN4CCOCC4)c3nc12	nan
	CHEMBL1407863	31775	13	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	495	7	2	10	-0.2	Cc1cccn2c(=O)c3cc(C(=O)NCCN4CCOCC4)c(=N)n(CCN4CCOCC4)c3nc12	nan
	975666	31912	22	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	315	4	1	7	1.6	Cc1nnc(NC(=O)CCn2cnc3ccccc3c2=O)s1	nan
	CHEMBL1408899	31912	22	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	315	4	1	7	1.6	Cc1nnc(NC(=O)CCn2cnc3ccccc3c2=O)s1	nan
	3152548	31928	14	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	5	1	5	3.7	O=C(C1=C(O)C(=O)N(CC2CCCO2)C1c1ccc(Cl)cc1)c1ccco1	nan
	CHEMBL1409014	31928	14	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	5	1	5	3.7	O=C(C1=C(O)C(=O)N(CC2CCCO2)C1c1ccc(Cl)cc1)c1ccco1	nan
	3147984	32009	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	5	0	6	2.5	CCN(CC)C(=O)CSc1nnc2c3ccccc3n(C)c2n1	nan
	CHEMBL1409671	32009	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	5	0	6	2.5	CCN(CC)C(=O)CSc1nnc2c3ccccc3n(C)c2n1	nan
	2740105	32078	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	255	2	0	4	3.3	N#Cc1c(N2CCCC2)nsc1-c1ccccc1	nan
	CHEMBL1410151	32078	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	255	2	0	4	3.3	N#Cc1c(N2CCCC2)nsc1-c1ccccc1	nan
	2965406	32083	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	6	1	5	4.1	O=C(NCCCn1ccnc1)c1cc(-c2cccnc2)nc2ccc(Br)cc12	nan
	CHEMBL1410223	32083	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	6	1	5	4.1	O=C(NCCCn1ccnc1)c1cc(-c2cccnc2)nc2ccc(Br)cc12	nan
	609181	32267	11	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	2	1	3	4.1	CC1(C(=O)Nc2nc3ccccc3s2)CC1(Br)Br	nan
	CHEMBL1411818	32267	11	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	2	1	3	4.1	CC1(C(=O)Nc2nc3ccccc3s2)CC1(Br)Br	nan
	2328662	32388	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	320	4	0	7	2.6	CCOC(=O)Cc1csc(-n2sc3ccccc3c2=O)n1	nan
	CHEMBL1412731	32388	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	320	4	0	7	2.6	CCOC(=O)Cc1csc(-n2sc3ccccc3c2=O)n1	nan
	716956	32626	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	4	1	6	3.5	COc1cc(-c2oc3ccc(C)cc3c(=O)c2O)cc(OC)c1OC	nan
	CHEMBL1414686	32626	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	4	1	6	3.5	COc1cc(-c2oc3ccc(C)cc3c(=O)c2O)cc(OC)c1OC	nan
	16019291	32969	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	318	4	0	4	5.2	Clc1cccc(CSc2ccc(-c3cccs3)nn2)c1	nan
	CHEMBL1417757	32969	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	318	4	0	4	5.2	Clc1cccc(CSc2ccc(-c3cccs3)nn2)c1	nan
	17581531	32991	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	4	1	7	3.5	COc1ccc2c(c1)c1nc3n(c(=O)c1n2CC(=O)Nc1ccccc1)CCCS3	nan
	CHEMBL1417902	32991	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	4	1	7	3.5	COc1ccc2c(c1)c1nc3n(c(=O)c1n2CC(=O)Nc1ccccc1)CCCS3	nan
	1505908	33192	11	None	-21	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	3	1	6	1.5	Cc1c(F)cccc1NS(=O)(=O)c1ccc2c(c1)c(=O)n(C)c(=O)n2C	nan
	CHEMBL1419634	33192	11	None	-21	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	3	1	6	1.5	Cc1c(F)cccc1NS(=O)(=O)c1ccc2c(c1)c(=O)n(C)c(=O)n2C	nan
	2138543	33476	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	6	2	7	3.6	Cc1cccc(-c2nnn3c2nc(NCCc2ccc(S(N)(=O)=O)cc2)c2ccccc23)c1	nan
	CHEMBL1422079	33476	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	6	2	7	3.6	Cc1cccc(-c2nnn3c2nc(NCCc2ccc(S(N)(=O)=O)cc2)c2ccccc23)c1	nan
	3937026	34038	16	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	4	1	5	3.5	O=C(CSc1ncnc2c1oc1ccccc12)NC1CCCC1	nan
	CHEMBL1426645	34038	16	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	4	1	5	3.5	O=C(CSc1ncnc2c1oc1ccccc12)NC1CCCC1	nan
	5909825	34680	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	522	8	1	9	2.5	COC(=O)c1ccc(C2C(C(=O)c3ccc4c(c3)OCCO4)=C(O)C(=O)N2CCCN2CCOCC2)cc1	nan
	CHEMBL1432124	34680	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	522	8	1	9	2.5	COC(=O)c1ccc(C2C(C(=O)c3ccc4c(c3)OCCO4)=C(O)C(=O)N2CCCN2CCOCC2)cc1	nan
	16011119	34958	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	4	1	6	3.2	Cc1ccc(CNC(=O)C(C)n2nc(C)n3c(cc4sccc43)c2=O)cc1	nan
	CHEMBL1435058	34958	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	4	1	6	3.2	Cc1ccc(CNC(=O)C(C)n2nc(C)n3c(cc4sccc43)c2=O)cc1	nan
	16018536	35084	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	4	1	5	5.2	O=C(NCc1cccs1)c1ccc2c(c1)sc1nc(-c3ccccc3)cn12	nan
	CHEMBL1436706	35084	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	4	1	5	5.2	O=C(NCc1cccs1)c1ccc2c(c1)sc1nc(-c3ccccc3)cn12	nan
	16011654	35090	2	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	4	1	5	5.8	Cc1ccc(CNC(=O)c2ccc(N3Cc4ccccc4Oc4ncccc43)s2)cc1	nan
	CHEMBL1436776	35090	2	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	4	1	5	5.8	Cc1ccc(CNC(=O)c2ccc(N3Cc4ccccc4Oc4ncccc43)s2)cc1	nan
	790330	35313	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	189	0	1	2	3.1	Cc1ccc2nc(C)cc(S)c2c1	nan
	CHEMBL1439016	35313	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	189	0	1	2	3.1	Cc1ccc2nc(C)cc(S)c2c1	nan
	22333977	35334	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	509	10	2	9	1.0	COc1ccc(-n2nc(C(=O)NCC(=O)NCCCN3CCOCC3)c3ccccc3c2=O)c(OC)c1	nan
	CHEMBL1439223	35334	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	509	10	2	9	1.0	COc1ccc(-n2nc(C(=O)NCC(=O)NCCCN3CCOCC3)c3ccccc3c2=O)c(OC)c1	nan
	974773	35499	7	None	-19	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	222	1	2	2	2.9	O=C(O)c1ccc2cccc(Cl)c2c1O	nan
	CHEMBL1440675	35499	7	None	-19	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	222	1	2	2	2.9	O=C(O)c1ccc2cccc(Cl)c2c1O	nan
	1048151	35995	13	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	5	2	4	3.8	COc1ccc(OCC(=O)NC(=S)Nc2ccc3c4c(cccc24)CC3)cc1	nan
	CHEMBL1445229	35995	13	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	5	2	4	3.8	COc1ccc(OCC(=O)NC(=S)Nc2ccc3c4c(cccc24)CC3)cc1	nan
	16407102	36001	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	530	8	1	9	2.8	COc1ccc2c(c1OC)c(=O)n1c3ccc(OC(C)C(=O)NCCN4CCOCC4)cc3c3ccnc2c31	nan
	CHEMBL1445287	36001	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	530	8	1	9	2.8	COc1ccc2c(c1OC)c(=O)n1c3ccc(OC(C)C(=O)NCCN4CCOCC4)cc3c3ccnc2c31	nan
	3244615	36409	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	460	5	1	8	1.2	O=C(Cn1cnc2sc3c(c2c1=O)CCCC3)NCCC(=O)N1CCC2(CC1)OCCO2	nan
	CHEMBL1448799	36409	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	460	5	1	8	1.2	O=C(Cn1cnc2sc3c(c2c1=O)CCCC3)NCCC(=O)N1CCC2(CC1)OCCO2	nan
	5333438	36510	10	None	1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	252	4	3	5	0.9	O=C(O)/C=C\C(=O)Nc1cc(O)ccc1[N+](=O)[O-]	nan
	CHEMBL1449557	36510	10	None	1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	252	4	3	5	0.9	O=C(O)/C=C\C(=O)Nc1cc(O)ccc1[N+](=O)[O-]	nan
	946874	36924	19	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	6	0	8	2.2	COC(=O)CSc1nc2ccccc2nc1SCC(=O)OC	nan
	CHEMBL1452913	36924	19	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	6	0	8	2.2	COC(=O)CSc1nc2ccccc2nc1SCC(=O)OC	nan
	15990397	36990	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	5	1	7	2.2	COc1cc(NC(=O)c2nc3ccccc3n(C)c2=O)cc(OC)c1OC	nan
	CHEMBL1453389	36990	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	5	1	7	2.2	COc1cc(NC(=O)c2nc3ccccc3n(C)c2=O)cc(OC)c1OC	nan
	2072948	37134	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	3	1	4	3.4	Brc1ccc2ncnc(NCc3cccnc3)c2c1	nan
	CHEMBL1454562	37134	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	3	1	4	3.4	Brc1ccc2ncnc(NCc3cccnc3)c2c1	nan
	20957239	37481	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	440	5	1	8	2.5	Cc1ccc(NC(=O)CCc2nnc3ccc(N4CCC5(CC4)OCCO5)nn23)cc1F	nan
	CHEMBL1457707	37481	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	440	5	1	8	2.5	Cc1ccc(NC(=O)CCc2nnc3ccc(N4CCC5(CC4)OCCO5)nn23)cc1F	nan
	8031083	37677	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	7	1	7	2.1	CCOC(=O)CCc1c(C)c2ccc3c(c2oc1=O)CN(CCCO)CO3	nan
	CHEMBL1459326	37677	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	7	1	7	2.1	CCOC(=O)CCc1c(C)c2ccc3c(c2oc1=O)CN(CCCO)CO3	nan
	1947745	38089	15	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	303	7	1	3	4.5	CCCCc1c(C)nc2ccccc2c1SCCC(=O)O	nan
	1947746	38089	15	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	303	7	1	3	4.5	CCCCc1c(C)nc2ccccc2c1SCCC(=O)O	nan
	CHEMBL1462881	38089	15	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	303	7	1	3	4.5	CCCCc1c(C)nc2ccccc2c1SCCC(=O)O	nan
	3593326	38111	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	5	0	8	1.1	CCOC(=O)C1=NN(c2ccc([N+](=O)[O-])cc2)CC1C(=O)OC	nan
	CHEMBL1463045	38111	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	5	0	8	1.1	CCOC(=O)C1=NN(c2ccc([N+](=O)[O-])cc2)CC1C(=O)OC	nan
	3889908	38194	15	None	1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	463	10	1	7	4.1	CCN(CC)CCCN1C(=O)C(O)=C(C(=O)c2cc3cccc(OC)c3o2)C1c1ccncc1	nan
	663903	38194	15	None	1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	463	10	1	7	4.1	CCN(CC)CCCN1C(=O)C(O)=C(C(=O)c2cc3cccc(OC)c3o2)C1c1ccncc1	nan
	CHEMBL1463781	38194	15	None	1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	463	10	1	7	4.1	CCN(CC)CCCN1C(=O)C(O)=C(C(=O)c2cc3cccc(OC)c3o2)C1c1ccncc1	nan
	4834173	38416	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	442	7	1	6	2.7	CCN(CC)S(=O)(=O)c1ccc(N2CCOCC2)c(NC(=O)c2cccc(C#N)c2)c1	nan
	CHEMBL1465419	38416	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	442	7	1	6	2.7	CCN(CC)S(=O)(=O)c1ccc(N2CCOCC2)c(NC(=O)c2cccc(C#N)c2)c1	nan
	2124679	38506	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	361	5	1	5	2.7	O=C(COc1ncnc2ccc(Br)cc12)NCc1ccco1	nan
	CHEMBL1466120	38506	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	361	5	1	5	2.7	O=C(COc1ncnc2ccc(Br)cc12)NCc1ccco1	nan
	5840379	38642	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	485	4	1	9	0.8	Cc1cccn2c(=O)c(/C=C(\C#N)C(=O)NC3CCS(=O)(=O)C3)c(N3CC(C)OC(C)C3)nc12	nan
	CHEMBL1467214	38642	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	485	4	1	9	0.8	Cc1cccn2c(=O)c(/C=C(\C#N)C(=O)NC3CCS(=O)(=O)C3)c(N3CC(C)OC(C)C3)nc12	nan
	2824481	38794	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	2	0	5	3.9	N#Cc1c(N2CCSCC2)nsc1-c1ccccc1Cl	nan
	CHEMBL1468502	38794	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	2	0	5	3.9	N#Cc1c(N2CCSCC2)nsc1-c1ccccc1Cl	nan
	5911323	38917	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	6	1	6	4.0	CCOc1ccc(C(=O)C2=C(O)C(=O)N(c3ncccn3)C2c2ccc(C)cc2)cc1	nan
	CHEMBL1469507	38917	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	6	1	6	4.0	CCOc1ccc(C(=O)C2=C(O)C(=O)N(c3ncccn3)C2c2ccc(C)cc2)cc1	nan
	3186594	39098	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	4	0	8	0.9	CCC1CCCCN1C(=O)CSc1nc2c(c(=O)n(C)c(=O)n2C)n1C	nan
	CHEMBL1471097	39098	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	4	0	8	0.9	CCC1CCCCN1C(=O)CSc1nc2c(c(=O)n(C)c(=O)n2C)n1C	nan
	5302637	39306	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	5	2	4	6.0	CCc1ccc(NC(=O)c2sc3nc(C)cc(C)c3c2NC(=O)c2ccccc2)cc1	nan
	CHEMBL1473111	39306	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	5	2	4	6.0	CCc1ccc(NC(=O)c2sc3nc(C)cc(C)c3c2NC(=O)c2ccccc2)cc1	nan
	16009440	39371	3	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	7	1	7	4.0	Cc1ccc(OCC(=O)Nc2ccc(OCc3cc(=O)n4ccsc4n3)cc2)cc1C	nan
	CHEMBL1474025	39371	3	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	7	1	7	4.0	Cc1ccc(OCC(=O)Nc2ccc(OCc3cc(=O)n4ccsc4n3)cc2)cc1C	nan
	16018838	39374	1	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	331	3	0	5	4.9	Clc1cccc(CSc2nncn3c2cc2sccc23)c1	nan
	CHEMBL1474070	39374	1	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	331	3	0	5	4.9	Clc1cccc(CSc2nncn3c2cc2sccc23)c1	nan
	16033266	39496	2	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	5	1	5	5.3	Cc1c(C(=O)NC(C)c2ccccc2)sc2ncnc(N(C)C3CCCCC3)c12	nan
	CHEMBL1475712	39496	2	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	5	1	5	5.3	Cc1c(C(=O)NC(C)c2ccccc2)sc2ncnc(N(C)C3CCCCC3)c12	nan
	16030277	39500	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	486	6	0	5	5.1	Cc1ccc(Cc2nc3ccccc3nc2SCC(=O)N2CCN(c3ccc(F)cc3)CC2)cc1	nan
	CHEMBL1475778	39500	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	486	6	0	5	5.1	Cc1ccc(Cc2nc3ccccc3nc2SCC(=O)N2CCN(c3ccc(F)cc3)CC2)cc1	nan
	16018142	39523	3	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	324	6	1	2	4.0	Cn1cc(CCCC(=O)NCc2ccc(F)cc2)c2ccccc21	nan
	CHEMBL1476187	39523	3	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	324	6	1	2	4.0	Cn1cc(CCCC(=O)NCc2ccc(F)cc2)c2ccccc21	nan
	16018630	39531	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	4	1	6	4.0	O=C(CSc1nncn2c1cc1occc12)Nc1ccc(F)c(Cl)c1	nan
	CHEMBL1476304	39531	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	4	1	6	4.0	O=C(CSc1nncn2c1cc1occc12)Nc1ccc(F)c(Cl)c1	nan
	16018040	39544	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	423	7	1	6	3.1	COc1ccc(OC)c(CNC(=O)CCn2c(=O)c3cccn3c3ccc(F)cc32)c1	nan
	CHEMBL1476501	39544	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	423	7	1	6	3.1	COc1ccc(OC)c(CNC(=O)CCn2c(=O)c3cccn3c3ccc(F)cc32)c1	nan
	135407487	39557	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	6	3	6	3.9	Cc1ccc(CNC(=O)CSc2nc3[nH]nc(C)c3c(=N)n2-c2ccccc2Cl)cc1	nan
	CHEMBL1476621	39557	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	6	3	6	3.9	Cc1ccc(CNC(=O)CSc2nc3[nH]nc(C)c3c(=N)n2-c2ccccc2Cl)cc1	nan
	676907	39655	46	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	205	1	1	3	2.8	COc1ccc2c(C)cc(S)nc2c1	nan
	CHEMBL1477596	39655	46	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	205	1	1	3	2.8	COc1ccc2c(C)cc(S)nc2c1	nan
	16018964	39893	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	5	1	5	3.2	CCC(C)NC(=O)c1ccc(Cn2c(=O)c3cccn3c3cccnc32)cc1	nan
	CHEMBL1479750	39893	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	5	1	5	3.2	CCC(C)NC(=O)c1ccc(Cn2c(=O)c3cccn3c3cccnc32)cc1	nan
	16018270	40388	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	5	2	5	5.5	CC(=O)Nc1ccc(NC(=O)c2oc3c(c2C)-c2nn(Cc4ccccc4Cl)cc2CC3)cc1	nan
	CHEMBL1484019	40388	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	5	2	5	5.5	CC(=O)Nc1ccc(NC(=O)c2oc3c(c2C)-c2nn(Cc4ccccc4Cl)cc2CC3)cc1	nan
	4613858	40784	17	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	271	1	2	7	0.9	COC(=O)c1sc2[nH]c(=S)n(N)c(=O)c2c1C	nan
	CHEMBL1487438	40784	17	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	271	1	2	7	0.9	COC(=O)c1sc2[nH]c(=S)n(N)c(=O)c2c1C	nan
	1173795	40933	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	8	2	9	1.9	CCCn1c(SCC(=O)Nc2ccc(NC(=O)CC)cc2)nc2c1c(=O)n(C)c(=O)n2C	nan
	CHEMBL1488482	40933	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	8	2	9	1.9	CCCn1c(SCC(=O)Nc2ccc(NC(=O)CC)cc2)nc2c1c(=O)n(C)c(=O)n2C	nan
	3152454	40965	13	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	6	3	8	0.4	N=c1c(C(=O)NCC2CCCO2)cc2c(=O)n3ccccc3nc2n1CCCO	nan
	CHEMBL1488709	40965	13	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	6	3	8	0.4	N=c1c(C(=O)NCC2CCCO2)cc2c(=O)n3ccccc3nc2n1CCCO	nan
	1294912	41404	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	4	2	8	3.8	COc1ccc(NC(=O)c2sc3nc(N4CCOCC4)c4c(c3c2N)CC(C)(C)OC4)cc1	nan
	CHEMBL1491898	41404	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	4	2	8	3.8	COc1ccc(NC(=O)c2sc3nc(N4CCOCC4)c4c(c3c2N)CC(C)(C)OC4)cc1	nan
	3944710	41411	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	498	5	2	8	2.1	O=C(Nc1cc(S(=O)(=O)N2CCOCC2)ccc1N1CCOCC1)c1cc(O)nc2ccccc12	nan
	CHEMBL1491951	41411	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	498	5	2	8	2.1	O=C(Nc1cc(S(=O)(=O)N2CCOCC2)ccc1N1CCOCC1)c1cc(O)nc2ccccc12	nan
	2958357	41734	14	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	363	5	1	6	2.9	Cc1nc(SCC(=O)NCC2CCCO2)c2c3c(sc2n1)CCC3	nan
	CHEMBL1494894	41734	14	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	363	5	1	6	2.9	Cc1nc(SCC(=O)NCC2CCCO2)c2c3c(sc2n1)CCC3	nan
	3601528	41767	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	487	6	2	7	5.3	COc1ccc(C(=O)Nc2nc3n(n2)C(c2ccc(Cl)cc2)C=C(c2ccccc2)N3)cc1OC	nan
	CHEMBL1495241	41767	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	487	6	2	7	5.3	COc1ccc(C(=O)Nc2nc3n(n2)C(c2ccc(Cl)cc2)C=C(c2ccccc2)N3)cc1OC	nan
	3120647	41774	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	466	3	1	4	6.9	O=C(Nc1ccc2oc(-c3cc(Br)ccc3Cl)nc2c1)c1cc2ccccc2o1	nan
	CHEMBL1495306	41774	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	466	3	1	4	6.9	O=C(Nc1ccc2oc(-c3cc(Br)ccc3Cl)nc2c1)c1cc2ccccc2o1	nan
	3296097	41871	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	508	5	1	9	4.1	CCc1ccc(-n2c(SCc3cc(=O)n4cc(Br)ccc4n3)nc3nncc-3c2O)cc1	nan
	CHEMBL1496299	41871	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	508	5	1	9	4.1	CCc1ccc(-n2c(SCc3cc(=O)n4cc(Br)ccc4n3)nc3nncc-3c2O)cc1	nan
	2175955	42357	2	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	398	7	2	7	3.3	Cc1noc(NS(=O)(=O)c2ccc(N/C=C/C(=O)c3cccnc3)cc2)c1C	nan
	CHEMBL1500554	42357	2	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	398	7	2	7	3.3	Cc1noc(NS(=O)(=O)c2ccc(N/C=C/C(=O)c3cccnc3)cc2)c1C	nan
	2868511	42385	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	4	1	4	3.5	COc1ccc(C2C(C(C)=O)=C(O)C(=O)N2c2ccc(C)cc2)cc1	nan
	CHEMBL1500746	42385	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	4	1	4	3.5	COc1ccc(C2C(C(C)=O)=C(O)C(=O)N2c2ccc(C)cc2)cc1	nan
	3146565	42619	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	4	1	7	4.0	Cc1ccc(C2C(C(=O)c3cccs3)=C(O)C(=O)N2c2nnc(C)s2)cc1	nan
	CHEMBL1502935	42619	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	4	1	7	4.0	Cc1ccc(C2C(C(=O)c3cccs3)=C(O)C(=O)N2c2nnc(C)s2)cc1	nan
	2998667	42791	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	5	1	9	-1.9	CC(=O)OCCNC(=O)Cn1cnc2c1c(=O)n(C)c(=O)n2C	nan
	CHEMBL1504458	42791	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	5	1	9	-1.9	CC(=O)OCCNC(=O)Cn1cnc2c1c(=O)n(C)c(=O)n2C	nan
	2497236	42989	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	7	1	6	4.6	CCOc1ccc(-c2nc(-c3cccs3)c(CC(=O)O)s2)cc1OC	nan
	CHEMBL1506154	42989	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	7	1	6	4.6	CCOc1ccc(-c2nc(-c3cccs3)c(CC(=O)O)s2)cc1OC	nan
	1442564	43395	4	None	-1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	324	5	0	5	3.5	COC(=O)CSc1nc(Cc2ccccc2)nc2ccccc12	nan
	CHEMBL1509687	43395	4	None	-1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	324	5	0	5	3.5	COC(=O)CSc1nc(Cc2ccccc2)nc2ccccc12	nan
	6305743	43406	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	283	7	1	5	3.2	COCCCNc1oc(/C=C/c2ccccc2)nc1C#N	nan
	CHEMBL1509795	43406	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	283	7	1	5	3.2	COCCCNc1oc(/C=C/c2ccccc2)nc1C#N	nan
	15988981	43686	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	538	8	2	7	4.1	Cc1cc(C)c(NC(=O)Cn2c(=O)n(CCC(=O)NCc3ccccc3Cl)c(=O)c3sccc32)c(C)c1	nan
	CHEMBL1512541	43686	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	538	8	2	7	4.1	Cc1cc(C)c(NC(=O)Cn2c(=O)n(CCC(=O)NCc3ccccc3Cl)c(=O)c3sccc32)c(C)c1	nan
	1116224	43804	14	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	3	1	7	1.1	Cn1c(=O)c2c(ncn2CC(=O)Nc2cccc(C(F)(F)F)c2)n(C)c1=O	nan
	CHEMBL1514415	43804	14	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	3	1	7	1.1	Cn1c(=O)c2c(ncn2CC(=O)Nc2cccc(C(F)(F)F)c2)n(C)c1=O	nan
	16018038	43878	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	6	1	5	3.8	CSc1ccc(CNC(=O)CCn2c(=O)c3cccn3c3ccc(F)cc32)cc1	nan
	CHEMBL1515402	43878	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	6	1	5	3.8	CSc1ccc(CNC(=O)CCn2c(=O)c3cccn3c3ccc(F)cc32)cc1	nan
	16016056	43907	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	8	1	7	5.0	COc1ccccc1-c1noc(-c2ccc(NCCc3ccccc3)c([N+](=O)[O-])c2)n1	nan
	CHEMBL1515947	43907	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	8	1	7	5.0	COc1ccccc1-c1noc(-c2ccc(NCCc3ccccc3)c([N+](=O)[O-])c2)n1	nan
	5069160	43981	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	6	2	6	3.5	O=C(CCCn1c(=S)[nH]c2cc3c(cc2c1=O)OCO3)NCc1cccc(Cl)c1	nan
	CHEMBL1516839	43981	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	6	2	6	3.5	O=C(CCCn1c(=S)[nH]c2cc3c(cc2c1=O)OCO3)NCc1cccc(Cl)c1	nan
	5389765	44195	9	None	-1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	396	8	1	6	3.1	COCCN1C(=O)C(O)=C(C(=O)c2ccc(OC(C)C)cc2)C1c1cccnc1	nan
	CHEMBL1518887	44195	9	None	-1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	396	8	1	6	3.1	COCCN1C(=O)C(O)=C(C(=O)c2ccc(OC(C)C)cc2)C1c1cccnc1	nan
	1238913	44338	13	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	3	0	9	-1.1	Cn1c(=O)c2c(nc(SCC(=O)N3CCOCC3)n2C)n(C)c1=O	nan
	CHEMBL1520162	44338	13	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	3	0	9	-1.1	Cn1c(=O)c2c(nc(SCC(=O)N3CCOCC3)n2C)n(C)c1=O	nan
	2165182	44463	11	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	5	1	5	2.9	Cc1ccc(-c2cc(C(=O)NCCN3CCOCC3)c3ccccc3n2)o1	nan
	CHEMBL1521212	44463	11	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	5	1	5	2.9	Cc1ccc(-c2cc(C(=O)NCCN3CCOCC3)c3ccccc3n2)o1	nan
	3111808	44514	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	5	1	4	6.3	CCOc1ccc(C(=O)Nc2ccc3oc(-c4ccc5ccccc5c4)nc3c2)cc1	nan
	CHEMBL1521616	44514	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	5	1	4	6.3	CCOc1ccc(C(=O)Nc2ccc3oc(-c4ccc5ccccc5c4)nc3c2)cc1	nan
	20957509	44635	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	11	2	8	1.8	COc1ccc(CNC(=O)CCc2nnc3ccc(NCCCN4CCCC4=O)nn23)cc1	nan
	CHEMBL1522776	44635	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	11	2	8	1.8	COc1ccc(CNC(=O)CCc2nnc3ccc(NCCCN4CCCC4=O)nn23)cc1	nan
	4126696	44650	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	7	1	5	5.9	COc1ccc(-n2cc(-c3ccccc3)nc2SCC(=O)Nc2ccccc2)cc1Cl	nan
	CHEMBL1522905	44650	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	7	1	5	5.9	COc1ccc(-n2cc(-c3ccccc3)nc2SCC(=O)Nc2ccccc2)cc1Cl	nan
	2561590	45008	7	None	-3	3	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	461	6	0	8	4.1	Cc1cc(C(=O)CSc2nc3ccccc3c(=O)n2C)c(C)n1Cc1ccc2c(c1)OCO2	nan
	CHEMBL1526230	45008	7	None	-3	3	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	461	6	0	8	4.1	Cc1cc(C(=O)CSc2nc3ccccc3c(=O)n2C)c(C)n1Cc1ccc2c(c1)OCO2	nan
	15991183	45158	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	4	1	4	6.8	O=C(Nc1cccc(-c2nc3ccccc3o2)c1)c1ccc(-c2ccc(Br)cc2)o1	nan
	CHEMBL1527553	45158	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	4	1	4	6.8	O=C(Nc1cccc(-c2nc3ccccc3o2)c1)c1ccc(-c2ccc(Br)cc2)o1	nan
	16014288	45509	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	478	7	2	8	3.8	Cc1ccnc(NS(=O)(=O)c2ccc(NC(=O)c3nc(SC(C)C)ncc3Cl)cc2)n1	nan
	CHEMBL1530646	45509	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	478	7	2	8	3.8	Cc1ccnc(NS(=O)(=O)c2ccc(NC(=O)c3nc(SC(C)C)ncc3Cl)cc2)n1	nan
	6078364	45518	3	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	6	1	6	4.2	COc1ccc(C2C(C(=O)c3ccc4c(c3)CC(C)O4)=C(O)C(=O)N2Cc2ccncc2)cc1	nan
	CHEMBL1530717	45518	3	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	6	1	6	4.2	COc1ccc(C2C(C(=O)c3ccc4c(c3)CC(C)O4)=C(O)C(=O)N2Cc2ccncc2)cc1	nan
	950608	45901	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	3	1	6	1.5	N#C/C(=C\c1c(N2CCCCCC2)nc2ccccn2c1=O)C(N)=O	nan
	CHEMBL1534139	45901	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	3	1	6	1.5	N#C/C(=C\c1c(N2CCCCCC2)nc2ccccn2c1=O)C(N)=O	nan
	5310696	45914	13	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	10	1	6	4.0	COCCCN1C(=O)C(O)=C(C(=O)c2ccc(OCC(C)C)cc2C)C1c1cccnc1	nan
	CHEMBL1534309	45914	13	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	10	1	6	4.0	COCCCN1C(=O)C(O)=C(C(=O)c2ccc(OCC(C)C)cc2C)C1c1cccnc1	nan
	1856407	46149	19	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	344	3	0	7	1.1	CCOC(=O)N1CCN(c2nc3c(C)cccn3c(=O)c2C=O)CC1	nan
	CHEMBL1536792	46149	19	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	344	3	0	7	1.1	CCOC(=O)N1CCN(c2nc3c(C)cccn3c(=O)c2C=O)CC1	nan
	1442728	46203	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	5	1	4	4.3	CC(C)c1nc(SCC(=O)NC2CCCCC2)c2ccccc2n1	nan
	CHEMBL1537182	46203	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	5	1	4	4.3	CC(C)c1nc(SCC(=O)NC2CCCCC2)c2ccccc2n1	nan
	6165328	46448	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	6	1	6	4.3	CCOc1ccc(C(=O)C2=C(O)C(=O)N(c3ncccn3)C2c2ccc(Cl)cc2)cc1	nan
	CHEMBL1539268	46448	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	6	1	6	4.3	CCOc1ccc(C(=O)C2=C(O)C(=O)N(c3ncccn3)C2c2ccc(Cl)cc2)cc1	nan
	2944889	46644	13	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	465	10	1	7	5.1	CCCOc1ccc(C2C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2Cc2ccco2)cc1OCC	nan
	CHEMBL1540923	46644	13	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	465	10	1	7	5.1	CCCOc1ccc(C2C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2Cc2ccco2)cc1OCC	nan
	1867273	47121	18	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	5	2	7	1.8	Cc1ccc(-c2nn3c(C)nnc3c3ccccc23)cc1S(=O)(=O)NCCO	nan
	CHEMBL1544770	47121	18	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	5	2	7	1.8	Cc1ccc(-c2nn3c(C)nnc3c3ccccc23)cc1S(=O)(=O)NCCO	nan
	3600899	47152	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	558	4	1	9	4.3	O=c1cc(CSc2nc3nncc-3c(O)n2-c2ccc(Br)cc2)nc2ccc(Br)cn12	nan
	CHEMBL1545051	47152	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	558	4	1	9	4.3	O=c1cc(CSc2nc3nncc-3c(O)n2-c2ccc(Br)cc2)nc2ccc(Br)cn12	nan
	135514845	47351	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	4	2	8	2.7	CN(Cc1nc(O)c2ccccc2n1)Cc1nc(O)c2sccc2n1	nan
	CHEMBL1546713	47351	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	4	2	8	2.7	CN(Cc1nc(O)c2ccccc2n1)Cc1nc(O)c2sccc2n1	nan
	1442627	47558	4	None	-1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	410	7	2	6	3.1	CCCc1nc(SCC(=O)NNC(=O)c2ccc(OC)cc2)c2ccccc2n1	nan
	CHEMBL1548632	47558	4	None	-1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	410	7	2	6	3.1	CCCc1nc(SCC(=O)NNC(=O)c2ccc(OC)cc2)c2ccccc2n1	nan
	16016034	47938	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	6	1	7	4.1	COc1ccccc1-c1noc(-c2ccc(NC(C)C)c([N+](=O)[O-])c2)n1	nan
	CHEMBL1552261	47938	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	6	1	7	4.1	COc1ccccc1-c1noc(-c2ccc(NC(C)C)c([N+](=O)[O-])c2)n1	nan
	16017890	47955	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	5	1	6	1.5	COCCCNC(=O)c1sc2nc3n(c(=O)c2c1C)CCC3	nan
	CHEMBL1552564	47955	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	5	1	6	1.5	COCCCNC(=O)c1sc2nc3n(c(=O)c2c1C)CCC3	nan
	16023050	47956	2	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	4	1	6	3.1	CCNC(=O)C1CCCN(c2nnc(C)c3c(C)n(-c4ccc(C)cc4)nc23)C1	nan
	CHEMBL1552569	47956	2	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	4	1	6	3.1	CCNC(=O)C1CCCN(c2nnc(C)c3c(C)n(-c4ccc(C)cc4)nc23)C1	nan
	3260331	48013	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	396	5	1	3	4.6	O=C(Cn1cc(C(=O)C2CC2)c2ccccc21)Nc1ccc(Br)cc1	nan
	CHEMBL1553312	48013	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	396	5	1	3	4.6	O=C(Cn1cc(C(=O)C2CC2)c2ccccc21)Nc1ccc(Br)cc1	nan
	16030436	48088	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	5	1	5	2.9	CC(C)C(=O)Nc1ccccc1OCc1cc(=O)n2ccccc2n1	nan
	CHEMBL1554451	48088	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	5	1	5	2.9	CC(C)C(=O)Nc1ccccc1OCc1cc(=O)n2ccccc2n1	nan
	16016784	48146	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	442	5	1	4	5.4	CCOC(=O)C1CCCN(C(=O)c2[nH]c3ccccc3c2Sc2ccc(Cl)cc2)C1	nan
	CHEMBL1555295	48146	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	442	5	1	4	5.4	CCOC(=O)C1CCCN(C(=O)c2[nH]c3ccccc3c2Sc2ccc(Cl)cc2)C1	nan
	16196698	48169	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	4	0	7	1.9	Cc1cc2nnc(SCC(=O)N(C)C3CCS(=O)(=O)C3)n2c2ccccc12	nan
	CHEMBL1555603	48169	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	4	0	7	1.9	Cc1cc2nnc(SCC(=O)N(C)C3CCS(=O)(=O)C3)n2c2ccccc12	nan
	2869543	48338	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	307	4	1	5	3.9	CCOC(=O)c1ccc(Nc2nnc(C)c3ccccc23)cc1	nan
	CHEMBL1557161	48338	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	307	4	1	5	3.9	CCOC(=O)c1ccc(Nc2nnc(C)c3ccccc23)cc1	nan
	1272771	48378	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	5	2	6	5.4	COc1ccc(-c2ccc3c(N)c(C(=O)Nc4ccc(C)cc4C)sc3n2)cc1OC	nan
	CHEMBL1557478	48378	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	5	2	6	5.4	COc1ccc(-c2ccc3c(N)c(C(=O)Nc4ccc(C)cc4C)sc3n2)cc1OC	nan
	3239737	48515	1	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	344	4	1	7	1.4	Cc1nn(C(C)C(=O)NCC2CCCO2)c(=O)c2cc3occc3n12	nan
	CHEMBL1558668	48515	1	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	344	4	1	7	1.4	Cc1nn(C(C)C(=O)NCC2CCCO2)c(=O)c2cc3occc3n12	nan
	1503106	48705	11	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	351	6	1	5	3.1	Cc1cc(CNC(=O)COc2ccc([N+](=O)[O-])cc2)c2ccccc2n1	nan
	CHEMBL1560348	48705	11	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	351	6	1	5	3.1	Cc1cc(CNC(=O)COc2ccc([N+](=O)[O-])cc2)c2ccccc2n1	nan
	2456723	48990	7	None	-1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	522	8	2	8	3.7	CCOC(=O)c1cc(-c2ccccc2)sc1NC(=O)COC(=O)c1ccc(Cl)c(S(N)(=O)=O)c1	nan
	CHEMBL1562996	48990	7	None	-1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	522	8	2	8	3.7	CCOC(=O)c1cc(-c2ccccc2)sc1NC(=O)COC(=O)c1ccc(Cl)c(S(N)(=O)=O)c1	nan
	3221518	49099	4	None	-1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	8	1	5	3.8	CCCNC(=O)CSc1nc(COc2ccccc2)nc2ccccc12	nan
	CHEMBL1563919	49099	4	None	-1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	8	1	5	3.8	CCCNC(=O)CSc1nc(COc2ccccc2)nc2ccccc12	nan
	2952819	49164	11	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	6	1	7	2.3	O=C(Cn1nc(-c2cccc([N+](=O)[O-])c2)c2ccccc2c1=O)NCC1CCCO1	nan
	CHEMBL1564585	49164	11	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	6	1	7	2.3	O=C(Cn1nc(-c2cccc([N+](=O)[O-])c2)c2ccccc2c1=O)NCC1CCCO1	nan
	2869470	49359	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	281	3	0	5	3.6	Cc1nnc(Oc2ccc([N+](=O)[O-])cc2)c2ccccc12	nan
	CHEMBL1566109	49359	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	281	3	0	5	3.6	Cc1nnc(Oc2ccc([N+](=O)[O-])cc2)c2ccccc12	nan
	16008434	49448	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	4	0	5	4.7	O=C(c1ccc(Cl)cc1)c1cn(Cc2ccccc2)c2cc3c(cc2c1=O)OCCO3	nan
	CHEMBL1566810	49448	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	4	0	5	4.7	O=C(c1ccc(Cl)cc1)c1cn(Cc2ccccc2)c2cc3c(cc2c1=O)OCCO3	nan
	1017457	49555	16	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	5	1	11	0.2	Cn1c(=O)c2c(nc(Sc3ncnn3CC(=O)NC3CCCCC3)n2C)n(C)c1=O	nan
	CHEMBL1567667	49555	16	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	5	1	11	0.2	Cn1c(=O)c2c(nc(Sc3ncnn3CC(=O)NC3CCCCC3)n2C)n(C)c1=O	nan
	2912191	49644	17	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	5	1	5	4.4	Cc1ccc(C(=O)C2=C(O)C(=O)N(Cc3cccnc3)C2c2ccc(Cl)cc2)o1	nan
	CHEMBL1568384	49644	17	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	5	1	5	4.4	Cc1ccc(C(=O)C2=C(O)C(=O)N(Cc3cccnc3)C2c2ccc(Cl)cc2)o1	nan
	665555	49941	8	None	-1	3	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	4	1	5	4.9	Cc1nc(SCC(=O)Nc2ccc(C)c(F)c2)c2oc3ccccc3c2n1	nan
	CHEMBL1570874	49941	8	None	-1	3	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	4	1	5	4.9	Cc1nc(SCC(=O)Nc2ccc(C)c(F)c2)c2oc3ccccc3c2n1	nan
	4333346	50139	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	8	1	4	4.3	COc1ccc(CCNC(=O)CSc2ccc3ccccc3c2)cc1OC	nan
	CHEMBL1572841	50139	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	8	1	4	4.3	COc1ccc(CCNC(=O)CSc2ccc3ccccc3c2)cc1OC	nan
	20957497	50345	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	10	2	7	2.1	Cc1ccc(CNC(=O)CCc2nnc3ccc(NCCCN4CCCC4=O)nn23)cc1	nan
	CHEMBL1574892	50345	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	10	2	7	2.1	Cc1ccc(CNC(=O)CCc2nnc3ccc(NCCCN4CCCC4=O)nn23)cc1	nan
	1938572	50560	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	6	1	6	3.6	O=C(COc1ccccc1)NCc1nnc2c3ccccc3c(-c3ccccc3)nn12	nan
	CHEMBL1576963	50560	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	6	1	6	3.6	O=C(COc1ccccc1)NCc1nnc2c3ccccc3c(-c3ccccc3)nn12	nan
	1632391	50713	16	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	6	3	4	2.0	O=C(O)CCC(=O)NNC(=O)COc1ccc2ccccc2c1Br	nan
	CHEMBL1578274	50713	16	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	6	3	4	2.0	O=C(O)CCC(=O)NNC(=O)COc1ccc2ccccc2c1Br	nan
	3504887	50765	13	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	3	0	7	1.6	CCOC(=O)C1CCN(C(=O)c2cc3c(=O)n4ccccc4nc3n2C)CC1	nan
	CHEMBL1578618	50765	13	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	3	0	7	1.6	CCOC(=O)C1CCN(C(=O)c2cc3c(=O)n4ccccc4nc3n2C)CC1	nan
	20903631	50771	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	464	6	0	9	1.2	COc1cccc(N2CCN(c3ccc4nnc(CCC(=O)N5CCN(C)CC5)n4n3)CC2)c1	nan
	CHEMBL1578662	50771	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	464	6	0	9	1.2	COc1cccc(N2CCN(c3ccc4nnc(CCC(=O)N5CCN(C)CC5)n4n3)CC2)c1	nan
	16475	51410	40	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	272	3	4	4	1.9	Nc1ccc(-c2ccc(N)c(C(=O)O)c2)cc1C(=O)O	nan
	CHEMBL1584156	51410	40	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	272	3	4	4	1.9	Nc1ccc(-c2ccc(N)c(C(=O)O)c2)cc1C(=O)O	nan
	1997175	51457	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	320	2	0	7	0.9	CN1CCN(c2nc3ccccn3c(=O)c2C=C(C#N)C#N)CC1	nan
	CHEMBL1584587	51457	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	320	2	0	7	0.9	CN1CCN(c2nc3ccccn3c(=O)c2C=C(C#N)C#N)CC1	nan
	20881207	51701	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	10	1	8	2.5	CC(C)OCCCn1c(=O)c2ccccc2n2c(CCC(=O)NCc3ccccn3)nnc12	nan
	CHEMBL1586569	51701	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	10	1	8	2.5	CC(C)OCCCn1c(=O)c2ccccc2n2c(CCC(=O)NCc3ccccn3)nnc12	nan
	3186634	51702	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	366	3	0	9	-1.2	CN1CCN(C(=O)CSc2nc3c(c(=O)n(C)c(=O)n3C)n2C)CC1	nan
	CHEMBL1586576	51702	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	366	3	0	9	-1.2	CN1CCN(C(=O)CSc2nc3c(c(=O)n(C)c(=O)n3C)n2C)CC1	nan
	658021	51974	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	318	1	0	5	3.0	CSC1=NP(=S)(SC)N(C)c2nc3n(c21)CCC3	nan
	CHEMBL1588879	51974	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	318	1	0	5	3.0	CSC1=NP(=S)(SC)N(C)c2nc3n(c21)CCC3	nan
	7190667	52084	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	5	1	7	3.1	O=C(CSc1ccc2nnc(-c3cccnc3)n2n1)Nc1cccc(F)c1	nan
	CHEMBL1589799	52084	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	5	1	7	3.1	O=C(CSc1ccc2nnc(-c3cccnc3)n2n1)Nc1cccc(F)c1	nan
	16030609	52127	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	457	8	0	5	5.7	CCN(C(=O)CSc1nc2ccccc2nc1Cc1cccc(OC)c1)c1cccc(C)c1	nan
	CHEMBL1590288	52127	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	457	8	0	5	5.7	CCN(C(=O)CSc1nc2ccccc2nc1Cc1cccc(OC)c1)c1cccc(C)c1	nan
	6221827	52157	16	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	5	2	5	3.0	COc1ccc(CNC(=O)Cc2c(C)c3c(O)cc(C)cc3oc2=O)cc1	nan
	CHEMBL1590750	52157	16	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	5	2	5	3.0	COc1ccc(CNC(=O)Cc2c(C)c3c(O)cc(C)cc3oc2=O)cc1	nan
	16030275	52238	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	8	0	4	4.9	CCCCN(C)C(=O)CSc1nc2ccccc2nc1Cc1ccc(C)cc1	nan
	CHEMBL1591718	52238	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	8	0	4	4.9	CCCCN(C)C(=O)CSc1nc2ccccc2nc1Cc1ccc(C)cc1	nan
	16031876	52290	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	4	0	5	5.0	CCC1CCCCN1Cc1cn2c(-c3ccc(Br)cc3)nnc2s1	nan
	CHEMBL1592401	52290	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	4	0	5	5.0	CCC1CCCCN1Cc1cn2c(-c3ccc(Br)cc3)nnc2s1	nan
	5768121	52502	12	None	-1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	457	8	1	6	4.6	Cc1cc(OCC(C)C)ccc1C(=O)C1=C(O)C(=O)N(Cc2cccnc2)C1c1ccncc1	nan
	CHEMBL1594882	52502	12	None	-1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	457	8	1	6	4.6	Cc1cc(OCC(C)C)ccc1C(=O)C1=C(O)C(=O)N(Cc2cccnc2)C1c1ccncc1	nan
	4968658	52612	7	None	-5	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	525	8	2	6	6.2	COc1cc(C(=O)Nc2nc(-c3ccc(Cl)cc3)c(C)s2)ccc1OCC(=O)Nc1ccc(F)cc1	nan
	CHEMBL1595841	52612	7	None	-5	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	525	8	2	6	6.2	COc1cc(C(=O)Nc2nc(-c3ccc(Cl)cc3)c(C)s2)ccc1OCC(=O)Nc1ccc(F)cc1	nan
	4875333	53236	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	291	2	1	4	3.5	CCn1c2ccccc2c2nc3cc(C(=O)O)ccc3nc21	nan
	CHEMBL1601617	53236	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	291	2	1	4	3.5	CCn1c2ccccc2c2nc3cc(C(=O)O)ccc3nc21	nan
	15988911	53551	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	436	5	0	7	4.2	COc1cc(OC)cc(-n2c(=O)c3sccc3n(Cc3c(C)cc(C)cc3C)c2=O)c1	nan
	CHEMBL1604412	53551	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	436	5	0	7	4.2	COc1cc(OC)cc(-n2c(=O)c3sccc3n(Cc3c(C)cc(C)cc3C)c2=O)c1	nan
	824096	53643	22	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	220	0	2	5	1.2	N=c1c2c3c(sc2ncn1N)CCCC3	nan
	CHEMBL1605294	53643	22	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	220	0	2	5	1.2	N=c1c2c3c(sc2ncn1N)CCCC3	nan
	16020886	53729	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	7	1	5	6.1	Cc1ccc(CSc2nc3cccnc3n2Cc2ccc(C(=O)NC3CCCCC3)cc2)cc1	nan
	CHEMBL1605955	53729	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	7	1	5	6.1	Cc1ccc(CSc2nc3cccnc3n2Cc2ccc(C(=O)NC3CCCCC3)cc2)cc1	nan
	3973561	54102	3	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	7	0	7	4.1	COc1ccc2cc(C(=O)COC(=O)COc3ccc4c(C)cc(=O)oc4c3)ccc2c1	nan
	CHEMBL1608925	54102	3	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	7	0	7	4.1	COc1ccc2cc(C(=O)COC(=O)COc3ccc4c(C)cc(=O)oc4c3)ccc2c1	nan
	4916122	54221	11	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	275	4	1	6	1.7	Cc1cccc(NC(=O)C(C)n2cc([N+](=O)[O-])cn2)n1	nan
	CHEMBL1609905	54221	11	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	275	4	1	6	1.7	Cc1cccc(NC(=O)C(C)n2cc([N+](=O)[O-])cn2)n1	nan
	3151454	54406	13	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	7	2	8	1.4	COCCCn1c(=N)c(C(=O)NCC2CCCO2)cc2c(=O)n3cc(C)ccc3nc21	nan
	CHEMBL1611459	54406	13	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	7	2	8	1.4	COCCCn1c(=N)c(C(=O)NCC2CCCO2)cc2c(=O)n3cc(C)ccc3nc21	nan
	2810155	54597	6	None	-1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	316	2	1	5	3.6	Cc1ccccc1C(=O)Nc1nc2c(C)csc2c(=O)s1	nan
	CHEMBL1613272	54597	6	None	-1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	316	2	1	5	3.6	Cc1ccccc1C(=O)Nc1nc2c(C)csc2c(=O)s1	nan
	6489921	55063	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	278	4	0	2	3.4	CCCn1c(/C=C/c2cc[n+](C)cc2)nc2ccccc21	nan
	CHEMBL1384004	55063	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	278	4	0	2	3.4	CCCn1c(/C=C/c2cc[n+](C)cc2)nc2ccccc21	nan
	CHEMBL1618913	55063	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	278	4	0	2	3.4	CCCn1c(/C=C/c2cc[n+](C)cc2)nc2ccccc21	nan
	135415554	55492	3	None	1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	4	1	7	4.4	Cc1nn(CCc2nc(-c3ccco3)cs2)c2nc(O)cc(C(F)(F)F)c12	nan
	CHEMBL1494334	55492	3	None	1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	4	1	7	4.4	Cc1nn(CCc2nc(-c3ccco3)cs2)c2nc(O)cc(C(F)(F)F)c12	nan
	CHEMBL1622628	55492	3	None	1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	4	1	7	4.4	Cc1nn(CCc2nc(-c3ccco3)cs2)c2nc(O)cc(C(F)(F)F)c12	nan
	24792259	55551	1	None	1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	3	3	6	2.5	Nc1c(S(=O)(=O)O)cc(NC(=O)c2ccccc2)c2c1C(=O)c1ccccc1C2=O	nan
	CHEMBL1517470	55551	1	None	1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	3	3	6	2.5	Nc1c(S(=O)(=O)O)cc(NC(=O)c2ccccc2)c2c1C(=O)c1ccccc1C2=O	nan
	CHEMBL1623157	55551	1	None	1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	3	3	6	2.5	Nc1c(S(=O)(=O)O)cc(NC(=O)c2ccccc2)c2c1C(=O)c1ccccc1C2=O	nan
	4323731	107211	4	None	-1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	485	3	3	4	5.9	Oc1c(Br)cc(/C=N/c2ccc3[nH]c(-c4ccccc4)nc3c2)c(O)c1Br	nan
	CHEMBL3190756	107211	4	None	-1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	485	3	3	4	5.9	Oc1c(Br)cc(/C=N/c2ccc3[nH]c(-c4ccccc4)nc3c2)c(O)c1Br	nan
	4073001	108227	10	None	-2	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	6	0	8	2.6	COC(=O)Cn1/c(=N/C(=O)c2ccc(OC)c(OC)c2)sc2cc(OC)ccc21	nan
	CHEMBL3208346	108227	10	None	-2	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	6	0	8	2.6	COC(=O)Cn1/c(=N/C(=O)c2ccc(OC)c(OC)c2)sc2cc(OC)ccc21	nan
	6870745	108609	10	None	1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	298	3	0	7	2.1	Cc1nc2ccccc2c(=O)n1/N=C/c1ccc([N+](=O)[O-])o1	nan
	CHEMBL3213340	108609	10	None	1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	298	3	0	7	2.1	Cc1nc2ccccc2c(=O)n1/N=C/c1ccc([N+](=O)[O-])o1	nan
	2941245	146316	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	5	1	5	3.8	Cc1ccc(C(=O)C2=C(O)C(=O)N(Cc3ccccc3)C2c2cccnc2)o1	nan
	CHEMBL392515	146316	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	5	1	5	3.8	Cc1ccc(C(=O)C2=C(O)C(=O)N(Cc3ccccc3)C2c2cccnc2)o1	nan
	1016096	191199	21	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	4	1	6	2.7	Cc1cc(C)nc(NS(=O)(=O)c2ccc(N3C(=O)c4ccccc4C3=O)cc2)n1	nan
	CHEMBL519824	191199	21	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	4	1	6	2.7	Cc1cc(C)nc(NS(=O)(=O)c2ccc(N3C(=O)c4ccccc4C3=O)cc2)n1	nan
	726062	195363	44	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	238	0	2	5	2.6	Oc1nc(S)nc2sc3c(c12)CCCC3	nan
	CHEMBL1583656	195363	44	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	238	0	2	5	2.6	Oc1nc(S)nc2sc3c(c12)CCCC3	nan
	CHEMBL567206	195363	44	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	238	0	2	5	2.6	Oc1nc(S)nc2sc3c(c12)CCCC3	nan
	2998030	31303	6	None	-	1	Human	5.7	pPotency	=	5.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	7	3	6	0.5	COCCNC(=O)NC(=O)COC(=O)C12CC3CC(CC(NC(C)=O)(C3)C1)C2	nan
	CHEMBL1403647	31303	6	None	-	1	Human	5.7	pPotency	=	5.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	7	3	6	0.5	COCCNC(=O)NC(=O)COC(=O)C12CC3CC(CC(NC(C)=O)(C3)C1)C2	nan
	975392	42226	9	None	-1	2	Human	5.7	pPotency	=	5.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	1	1	2	4.3	Cc1cc(Br)c2nc3c(c(C(=O)O)c2c1)CCCCC3	nan
	CHEMBL1499411	42226	9	None	-1	2	Human	5.7	pPotency	=	5.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	1	1	2	4.3	Cc1cc(Br)c2nc3c(c(C(=O)O)c2c1)CCCCC3	nan
	16019550	10607	14	None	-131	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	4	1	8	4.3	O=S(=O)(c1ccccc1)c1nnn2c1nc(NC1CCCCCC1)c1sccc12	nan
	CHEMBL1170886	10607	14	None	-131	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	4	1	8	4.3	O=S(=O)(c1ccccc1)c1nnn2c1nc(NC1CCCCCC1)c1sccc12	nan
	4204374	19373	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	307	6	2	6	3.4	COc1cc2nc(S)nc(NCCC(C)C)c2cc1OC	nan
	CHEMBL1299978	19373	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	307	6	2	6	3.4	COc1cc2nc(S)nc(NCCC(C)C)c2cc1OC	nan
	2421557	19522	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	8	0	7	3.6	COC(=O)CCc1c(C)c(C(=O)c2cc(OC)c(OC)c(OC)c2)c2ccccn12	nan
	CHEMBL1301080	19522	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	8	0	7	3.6	COC(=O)CCc1c(C)c(C(=O)c2cc(OC)c(OC)c(OC)c2)c2ccccn12	nan
	22548258	20093	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	4	1	6	1.7	CC(=O)c1ccc(N2CCN(S(=O)(=O)c3ccc4c(c3)NC(=O)CO4)CC2)cc1	nan
	CHEMBL1305765	20093	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	4	1	6	1.7	CC(=O)c1ccc(N2CCN(S(=O)(=O)c3ccc4c(c3)NC(=O)CO4)CC2)cc1	nan
	16194269	20282	3	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	560	7	1	8	2.4	O=C(CSC1=Nc2ccccc2C2=NC(CC(=O)N3CCN(c4ccccc4)CC3)C(=O)N12)NCC1CCCO1	nan
	CHEMBL1307199	20282	3	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	560	7	1	8	2.4	O=C(CSC1=Nc2ccccc2C2=NC(CC(=O)N3CCN(c4ccccc4)CC3)C(=O)N12)NCC1CCCO1	nan
	3740686	20910	14	None	-7	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	4	1	6	4.0	Cc1cc(N2C(=O)C(O)=C(C(=O)c3cccs3)C2c2ccc(F)cc2)no1	nan
	CHEMBL1312274	20910	14	None	-7	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	4	1	6	4.0	Cc1cc(N2C(=O)C(O)=C(C(=O)c3cccs3)C2c2ccc(F)cc2)no1	nan
	4465171	21058	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	6	1	6	3.1	O=C(CSc1ncnc2ccccc12)Nc1cccc(S(=O)(=O)N2CCCC2)c1	nan
	CHEMBL1313361	21058	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	6	1	6	3.1	O=C(CSc1ncnc2ccccc12)Nc1cccc(S(=O)(=O)N2CCCC2)c1	nan
	2197541	21109	10	None	-2	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	5	1	6	4.3	CC(C)c1ccc(-c2c(C#N)c(N)nc(SCC(=O)N3CCCCC3)c2C#N)cc1	nan
	CHEMBL1313695	21109	10	None	-2	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	5	1	6	4.3	CC(C)c1ccc(-c2c(C#N)c(N)nc(SCC(=O)N3CCCCC3)c2C#N)cc1	nan
	2679228	21164	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	4	1	7	4.0	COc1ccc2oc(C(=O)Nc3nc4ccc(S(C)(=O)=O)cc4s3)c(C)c2c1	nan
	CHEMBL1314240	21164	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	4	1	7	4.0	COc1ccc2oc(C(=O)Nc3nc4ccc(S(C)(=O)=O)cc4s3)c(C)c2c1	nan
	16034516	21196	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	6	1	6	4.6	Cc1nnc(SCC(=O)NCc2ccccc2F)c2nn(-c3ccc(Cl)cc3)c(C)c12	nan
	CHEMBL1314574	21196	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	6	1	6	4.6	Cc1nnc(SCC(=O)NCc2ccccc2F)c2nn(-c3ccc(Cl)cc3)c(C)c12	nan
	135419125	21227	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	346	2	1	3	5.7	Oc1ccc(Cl)cc1C1=Nc2ccccc2N=C(c2ccccc2)C1	nan
	CHEMBL1315137	21227	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	346	2	1	3	5.7	Oc1ccc(Cl)cc1C1=Nc2ccccc2N=C(c2ccccc2)C1	nan
	16012610	21234	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	492	4	0	10	4.0	Cc1cccn2c(=O)c3cc(C#N)c(=O)n(-c4nnc(SCc5ccc(Cl)cc5)s4)c3nc12	nan
	CHEMBL1315199	21234	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	492	4	0	10	4.0	Cc1cccn2c(=O)c3cc(C#N)c(=O)n(-c4nnc(SCc5ccc(Cl)cc5)s4)c3nc12	nan
	4119285	21281	11	None	-1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	2	0	7	2.2	Cn1/c(=N/C(=O)c2ccc3c(c2)OCCO3)sc2cc(S(C)(=O)=O)ccc21	nan
	CHEMBL1315733	21281	11	None	-1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	2	0	7	2.2	Cn1/c(=N/C(=O)c2ccc3c(c2)OCCO3)sc2cc(S(C)(=O)=O)ccc21	nan
	24892214	21297	2	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	7	1	8	2.2	COc1ccc(-c2ccc3nnc(SCC(=O)NCC4CCCO4)n3n2)cc1	nan
	CHEMBL1315929	21297	2	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	7	1	8	2.2	COc1ccc(-c2ccc3nnc(SCC(=O)NCC4CCCO4)n3n2)cc1	nan
	7599144	21305	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	4	1	5	3.1	Cc1cc(NC(=O)c2cccn(Cc3cccc(Cl)c3)c2=O)no1	nan
	CHEMBL1315995	21305	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	4	1	5	3.1	Cc1cc(NC(=O)c2cccn(Cc3cccc(Cl)c3)c2=O)no1	nan
	16018244	21469	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	6	1	5	3.5	Cc1c(C(=O)NCCN(C)C)oc2c1-c1nn(Cc3ccccc3Cl)cc1CC2	nan
	CHEMBL1318247	21469	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	6	1	5	3.5	Cc1c(C(=O)NCCN(C)C)oc2c1-c1nn(Cc3ccccc3Cl)cc1CC2	nan
	15944876	21590	11	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	5	1	5	4.1	Cc1ccc(NC(=O)Cn2cc(S(=O)(=O)c3ccc(F)cc3)c(=O)c3cc(F)ccc32)cc1	nan
	CHEMBL1319259	21590	11	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	5	1	5	4.1	Cc1ccc(NC(=O)Cn2cc(S(=O)(=O)c3ccc(F)cc3)c(=O)c3cc(F)ccc32)cc1	nan
	16010992	21674	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	440	8	1	8	2.6	CCc1cc2c(cc3c(=O)n(CC(=O)NCCc4ccc(OC)c(OC)c4)ncn32)s1	nan
	CHEMBL1319991	21674	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	440	8	1	8	2.6	CCc1cc2c(cc3c(=O)n(CC(=O)NCCc4ccc(OC)c(OC)c4)ncn32)s1	nan
	4164390	21761	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	447	4	1	5	6.1	CC(C)OC(=O)c1c(NC(=O)C2c3ccccc3Oc3ccccc32)sc2c1CCCC2	nan
	CHEMBL1320657	21761	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	447	4	1	5	6.1	CC(C)OC(=O)c1c(NC(=O)C2c3ccccc3Oc3ccccc32)sc2c1CCCC2	nan
	25102515	21783	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	4	1	4	4.1	Cc1cc(=O)oc2cc(NC(=O)COc3cccc(C(F)(F)F)c3)ccc12	nan
	CHEMBL1320916	21783	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	4	1	4	4.1	Cc1cc(=O)oc2cc(NC(=O)COc3cccc(C(F)(F)F)c3)ccc12	nan
	794839	21838	34	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	256	1	1	4	2.8	Sc1nnc(-c2cccc(Br)c2)o1	nan
	CHEMBL1321356	21838	34	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	256	1	1	4	2.8	Sc1nnc(-c2cccc(Br)c2)o1	nan
	16018780	21840	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	3	0	5	5.0	Cc1cc2c(cc3c(SCc4cccc(Cl)c4)nnc(C)n32)o1	nan
	CHEMBL1321426	21840	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	3	0	5	5.0	Cc1cc2c(cc3c(SCc4cccc(Cl)c4)nnc(C)n32)o1	nan
	3996443	21890	7	None	-7	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	6	1	10	-0.7	Cn1c(N)c(C(=O)COC(=O)COc2ccccc2C#N)c(=O)n(C)c1=O	nan
	CHEMBL1321877	21890	7	None	-7	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	6	1	10	-0.7	Cn1c(N)c(C(=O)COC(=O)COc2ccccc2C#N)c(=O)n(C)c1=O	nan
	16009867	22132	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	489	6	1	7	4.5	CCOc1ccccc1NC(=O)Cn1c(=O)n(-c2ccc(F)cc2)c(=O)c2sc3ccccc3c21	nan
	CHEMBL1324000	22132	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	489	6	1	7	4.5	CCOc1ccccc1NC(=O)Cn1c(=O)n(-c2ccc(F)cc2)c(=O)c2sc3ccccc3c21	nan
	1442375	22238	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	4	1	4	4.1	CC(C)(C)c1nc(SCC(=O)NC2CCCC2)c2ccccc2n1	nan
	CHEMBL1324849	22238	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	4	1	4	4.1	CC(C)(C)c1nc(SCC(=O)NC2CCCC2)c2ccccc2n1	nan
	22517548	22353	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	4	1	7	1.6	O=C(Nc1nnc(S(=O)(=O)N2CCOCC2)s1)c1ccccc1Br	nan
	CHEMBL1326013	22353	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	4	1	7	1.6	O=C(Nc1nnc(S(=O)(=O)N2CCOCC2)s1)c1ccccc1Br	nan
	20927538	22466	0	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	8	0	7	1.3	CN(Cc1ccco1)C(=O)Cn1cc(S(=O)(=O)N2CCCC2)c(S(=O)(=O)N2CCCC2)c1	nan
	CHEMBL1327078	22466	0	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	8	0	7	1.3	CN(Cc1ccco1)C(=O)Cn1cc(S(=O)(=O)N2CCCC2)c(S(=O)(=O)N2CCCC2)c1	nan
	2645777	22561	15	None	-2	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	300	1	1	3	4.4	N#Cc1c(S)nc(-c2ccccc2Cl)c2c1CCCC2	nan
	CHEMBL1327817	22561	15	None	-2	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	300	1	1	3	4.4	N#Cc1c(S)nc(-c2ccccc2Cl)c2c1CCCC2	nan
	2816375	22788	26	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	274	2	1	7	1.7	CCOC(=O)c1nnn2c1nc(S)c1ccccc12	nan
	CHEMBL1329724	22788	26	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	274	2	1	7	1.7	CCOC(=O)c1nnn2c1nc(S)c1ccccc12	nan
	3151322	22797	14	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	4	2	7	2.0	N=c1c(C(=O)NC2CCCC2)cc2c(=O)n3ccccc3nc2n1CC1CCCO1	nan
	CHEMBL1329807	22797	14	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	4	2	7	2.0	N=c1c(C(=O)NC2CCCC2)cc2c(=O)n3ccccc3nc2n1CC1CCCO1	nan
	16030826	22946	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	4	2	5	2.9	NC(=O)C1CCN(C(=O)c2ccccc2NC(=O)c2nsc3ccccc23)CC1	nan
	CHEMBL1330985	22946	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	4	2	5	2.9	NC(=O)C1CCN(C(=O)c2ccccc2NC(=O)c2nsc3ccccc23)CC1	nan
	2815453	23184	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	204	0	0	5	0.3	Cn1c2c(c(=O)n3ncnc13)CCCC2	nan
	CHEMBL1332830	23184	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	204	0	0	5	0.3	Cn1c2c(c(=O)n3ncnc13)CCCC2	nan
	16019110	23193	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	5	1	8	3.3	O=C(Cn1c(=O)n(Cc2ccc3c(c2)OCO3)c(=O)c2oc3ccccc3c21)Nc1ccccc1	nan
	CHEMBL1332893	23193	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	5	1	8	3.3	O=C(Cn1c(=O)n(Cc2ccc3c(c2)OCO3)c(=O)c2oc3ccccc3c21)Nc1ccccc1	nan
	16018748	23196	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	3	0	5	4.7	Cc1nnc(SCc2ccc(Cl)cc2)c2cc3occc3n12	nan
	CHEMBL1332908	23196	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	3	0	5	4.7	Cc1nnc(SCc2ccc(Cl)cc2)c2cc3occc3n12	nan
	876371	23260	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	2	1	4	2.2	Cc1cc(/C=C2/C(=O)NC(=O)N(C)C2=O)c(C)n1-c1ccccc1	nan
	CHEMBL1333432	23260	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	2	1	4	2.2	Cc1cc(/C=C2/C(=O)NC(=O)N(C)C2=O)c(C)n1-c1ccccc1	nan
	16031513	23665	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	6	1	6	5.0	COc1ccc(-c2nnc(SCC(=O)Nc3cccc(C(F)(F)F)c3)s2)cc1	nan
	CHEMBL1336578	23665	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	6	1	6	5.0	COc1ccc(-c2nnc(SCC(=O)Nc3cccc(C(F)(F)F)c3)s2)cc1	nan
	16011266	23847	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	3	1	3	3.5	Cc1cccc(CNC(=O)c2ccc3c(c2)N(C)CCS3)c1	nan
	CHEMBL1338231	23847	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	3	1	3	3.5	Cc1cccc(CNC(=O)c2ccc3c(c2)N(C)CCS3)c1	nan
	16009346	23921	11	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	6	1	4	5.1	CCc1ccc2c(c1)c(=O)c(C(=O)c1ccc(C)cc1)cn2CC(=O)Nc1ccccc1C	nan
	CHEMBL1338819	23921	11	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	6	1	4	5.1	CCc1ccc2c(c1)c(=O)c(C(=O)c1ccc(C)cc1)cn2CC(=O)Nc1ccccc1C	nan
	1451340	24040	2	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	7	1	7	4.2	Cc1nonc1NC(=O)CSc1nc(CCC2CCCC2)nc2ccccc12	nan
	CHEMBL1339937	24040	2	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	7	1	7	4.2	Cc1nonc1NC(=O)CSc1nc(CCC2CCCC2)nc2ccccc12	nan
	1173483	24250	3	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	4	1	7	4.1	Cc1cc2cc3c(cc2nc1SCC(=O)Nc1nc(C)c(C)s1)OCO3	nan
	CHEMBL1341833	24250	3	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	4	1	7	4.1	Cc1cc2cc3c(cc2nc1SCC(=O)Nc1nc(C)c(C)s1)OCO3	nan
	3208214	24520	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	5	1	5	4.4	CCc1cc2cc(C)cc(C)c2nc1SCC(=O)Nc1cc(C)on1	nan
	CHEMBL1344061	24520	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	5	1	5	4.4	CCc1cc2cc(C)cc(C)c2nc1SCC(=O)Nc1cc(C)on1	nan
	1442646	24708	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	5	0	4	4.3	CCCc1nc(SCC(=O)N2CCc3ccccc3C2)c2ccccc2n1	nan
	CHEMBL1345722	24708	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	5	0	4	4.3	CCCc1nc(SCC(=O)N2CCc3ccccc3C2)c2ccccc2n1	nan
	2322587	24728	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	9	1	6	1.7	CCN(CC)S(=O)(=O)c1ccc(C(=O)OCCNC(=O)c2cccnc2)cc1	nan
	CHEMBL1345885	24728	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	9	1	6	1.7	CCN(CC)S(=O)(=O)c1ccc(C(=O)OCCNC(=O)c2cccnc2)cc1	nan
	3475758	24748	14	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	490	7	1	9	4.5	COc1cc(C2C(C(=O)c3cc4ccccc4o3)=C(O)C(=O)N2c2cc(C)on2)cc(OC)c1OC	nan
	CHEMBL1346015	24748	14	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	490	7	1	9	4.5	COc1cc(C2C(C(=O)c3cc4ccccc4o3)=C(O)C(=O)N2c2cc(C)on2)cc(OC)c1OC	nan
	911360	24791	16	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	183	0	1	4	1.3	Cn1c(O)nc2c(Cl)nccc21	nan
	CHEMBL1346457	24791	16	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	183	0	1	4	1.3	Cn1c(O)nc2c(Cl)nccc21	nan
	745324	24845	8	None	-1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	3	3	5	4.4	Cc1ccc(NC(S)=Nc2cccc(-c3nnc(S)o3)c2)cc1	nan
	CHEMBL1346824	24845	8	None	-1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	3	3	5	4.4	Cc1ccc(NC(S)=Nc2cccc(-c3nnc(S)o3)c2)cc1	nan
	664458	24886	14	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	326	4	0	6	4.4	O=C(CSc1ncnc2c1oc1ccccc12)c1cccs1	nan
	CHEMBL1347130	24886	14	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	326	4	0	6	4.4	O=C(CSc1ncnc2c1oc1ccccc12)c1cccs1	nan
	866600	24922	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	2	0	6	1.7	CCN1CCN(C(=O)c2cc3c(=O)n4ccccc4nc3s2)CC1	nan
	CHEMBL1347433	24922	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	2	0	6	1.7	CCN1CCN(C(=O)c2cc3c(=O)n4ccccc4nc3s2)CC1	nan
	2158422	25087	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	3	0	7	2.6	CCOC(=O)C1CCN(C(=O)c2cc3c(=O)n4cccc(C)c4nc3s2)CC1	nan
	CHEMBL1348934	25087	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	3	0	7	2.6	CCOC(=O)C1CCN(C(=O)c2cc3c(=O)n4cccc(C)c4nc3s2)CC1	nan
	7711373	25123	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	344	3	1	5	2.9	O=C(NCc1nnc2c(C(F)(F)F)cc(Cl)cn12)c1ccco1	nan
	CHEMBL1349179	25123	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	344	3	1	5	2.9	O=C(NCc1nnc2c(C(F)(F)F)cc(Cl)cn12)c1ccco1	nan
	20920345	25470	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	5	1	6	4.6	Cc1ccc(-n2nc3c(N4CCC(C(=O)NCc5ccccc5C)CC4)nnc(C)c3c2C)cc1	nan
	CHEMBL1352171	25470	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	5	1	6	4.6	Cc1ccc(-n2nc3c(N4CCC(C(=O)NCc5ccccc5C)CC4)nnc(C)c3c2C)cc1	nan
	3742858	25681	14	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	478	4	1	6	5.3	Cc1cc(N2C(=O)C(O)=C(C(=O)c3cc4ccccc4o3)C2c2ccc(Br)cc2)no1	nan
	CHEMBL1353643	25681	14	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	478	4	1	6	5.3	Cc1cc(N2C(=O)C(O)=C(C(=O)c3cc4ccccc4o3)C2c2ccc(Br)cc2)no1	nan
	16009768	25809	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	460	9	2	6	5.1	CCOc1ccc(NC(=O)c2oc3ccccc3c2NC(=O)COc2cccc(OC)c2)cc1	nan
	CHEMBL1354836	25809	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	460	9	2	6	5.1	CCOc1ccc(NC(=O)c2oc3ccccc3c2NC(=O)COc2cccc(OC)c2)cc1	nan
	16022445	25816	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	400	3	1	3	4.8	CC1Cn2c(C(=O)NCc3cccc(Br)c3)cc3cccc(c32)S1	nan
	CHEMBL1354873	25816	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	400	3	1	3	4.8	CC1Cn2c(C(=O)NCc3cccc(Br)c3)cc3cccc(c32)S1	nan
	16024821	25890	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	3	1	4	5.2	O=C(Nc1ccc(Cl)cc1)C1CCN(c2nc3ccccc3nc2C(F)(F)F)CC1	nan
	CHEMBL1355809	25890	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	3	1	4	5.2	O=C(Nc1ccc(Cl)cc1)C1CCN(c2nc3ccccc3nc2C(F)(F)F)CC1	nan
	5292880	25900	11	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	6	1	4	6.5	COc1cc(/C=C(\C#N)c2nc3ccccc3[nH]2)cc(Cl)c1OCc1ccccc1Cl	nan
	CHEMBL1355927	25900	11	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	6	1	4	6.5	COc1cc(/C=C(\C#N)c2nc3ccccc3[nH]2)cc(Cl)c1OCc1ccccc1Cl	nan
	7878585	25904	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	5	1	7	1.9	O=C(CNC(=O)c1ccc(Cl)cc1)OCc1cc(=O)n2ccsc2n1	nan
	CHEMBL1356005	25904	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	5	1	7	1.9	O=C(CNC(=O)c1ccc(Cl)cc1)OCc1cc(=O)n2ccsc2n1	nan
	6200344	25976	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	7	1	6	2.7	COc1cccc(/C=C/c2nc(C#N)c(NCCN(C)C)o2)c1	nan
	CHEMBL1356982	25976	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	7	1	6	2.7	COc1cccc(/C=C/c2nc(C#N)c(NCCN(C)C)o2)c1	nan
	1004107	26164	11	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	5	2	5	5.3	CCOc1cccc(NC(=O)c2sc3nc(-c4ccc(F)cc4)ccc3c2N)c1	nan
	CHEMBL1359199	26164	11	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	5	2	5	5.3	CCOc1cccc(NC(=O)c2sc3nc(-c4ccc(F)cc4)ccc3c2N)c1	nan
	16009637	26466	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	5	1	6	4.5	O=C(Nc1ccc(OCc2cc(=O)n3c4c(sc3n2)CCCC4)cc1)c1ccccc1	nan
	CHEMBL1361843	26466	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	5	1	6	4.5	O=C(Nc1ccc(OCc2cc(=O)n3c4c(sc3n2)CCCC4)cc1)c1ccccc1	nan
	4114478	26817	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	6	1	4	5.1	COc1cccc(NC(=O)Cn2cc(C(=O)C3CCCCC3)c3ccccc32)c1	nan
	CHEMBL1364874	26817	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	6	1	4	5.1	COc1cccc(NC(=O)Cn2cc(C(=O)C3CCCCC3)c3ccccc32)c1	nan
	22641	27065	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	3	1	7	0.8	CC(=O)OCCn1c2nc(=O)[nH]c(=O)c-2nc2cc(C)c(C)cc21	nan
	CHEMBL1367036	27065	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	3	1	7	0.8	CC(=O)OCCn1c2nc(=O)[nH]c(=O)c-2nc2cc(C)c(C)cc21	nan
	2378240	27170	24	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	235	2	1	4	2.7	Fc1ccccc1-c1nnc(S)n1C1CC1	nan
	CHEMBL1367871	27170	24	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	235	2	1	4	2.7	Fc1ccccc1-c1nnc(S)n1C1CC1	nan
	12006141	27497	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	298	4	0	4	4.8	Cc1ccc(CSc2ccc(-c3cccs3)nn2)cc1	nan
	CHEMBL1370265	27497	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	298	4	0	4	4.8	Cc1ccc(CSc2ccc(-c3cccs3)nn2)cc1	nan
	16455091	27609	11	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	483	6	2	8	3.0	Cc1noc(NS(=O)(=O)c2ccc(NC(=O)c3nn(-c4ccc(F)cc4)ccc3=O)cc2)c1C	nan
	CHEMBL1371016	27609	11	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	483	6	2	8	3.0	Cc1noc(NS(=O)(=O)c2ccc(NC(=O)c3nn(-c4ccc(F)cc4)ccc3=O)cc2)c1C	nan
	135406328	27807	16	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	334	3	1	7	1.3	Cc1cc(C)c2c(O)nc(SCC(=O)N3CCOCC3)nc2n1	nan
	CHEMBL1372508	27807	16	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	334	3	1	7	1.3	Cc1cc(C)c2c(O)nc(SCC(=O)N3CCOCC3)nc2n1	nan
	2138011	28186	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	6	1	6	4.1	COc1ccc(S(=O)(=O)c2cn(CC(=O)Nc3cc(C)ccc3C)c3ccccc3c2=O)cc1	nan
	CHEMBL1375055	28186	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	6	1	6	4.1	COc1ccc(S(=O)(=O)c2cn(CC(=O)Nc3cc(C)ccc3C)c3ccccc3c2=O)cc1	nan
	3571741	28191	11	None	-2	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	4	1	4	4.6	Cc1ccc(-c2cc(C(=O)NCc3cnn(C)c3)c3cc(Br)ccc3n2)cc1	nan
	CHEMBL1375116	28191	11	None	-2	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	4	1	4	4.6	Cc1ccc(-c2cc(C(=O)NCc3cnn(C)c3)c3cc(Br)ccc3n2)cc1	nan
	16025702	28222	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	457	6	1	6	5.9	CCOc1ccccc1CNC(=O)c1ccc(N2Cc3ccccc3Oc3ncccc32)s1	nan
	CHEMBL1375311	28222	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	457	6	1	6	5.9	CCOc1ccccc1CNC(=O)c1ccc(N2Cc3ccccc3Oc3ncccc32)s1	nan
	2874807	28711	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	4	1	7	4.6	CC1=C(C(=O)OCC2CCCO2)C(c2coc3ccc(C)cc3c2=O)C2=C(O)CCCC2=N1	nan
	CHEMBL1379763	28711	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	4	1	7	4.6	CC1=C(C(=O)OCC2CCCO2)C(c2coc3ccc(C)cc3c2=O)C2=C(O)CCCC2=N1	nan
	1564382	28891	11	None	-2	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	552	7	1	7	5.8	CCCCn1c(NC(=O)c2ccc(Br)o2)c(S(=O)(=O)c2ccccc2)c2nc3ccccc3nc21	nan
	CHEMBL1381243	28891	11	None	-2	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	552	7	1	7	5.8	CCCCn1c(NC(=O)c2ccc(Br)o2)c(S(=O)(=O)c2ccccc2)c2nc3ccccc3nc21	nan
	666048	29095	11	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	334	3	0	9	2.0	c1cncc(-c2nn3c(Cn4nnc5ccccc54)nnc3s2)c1	nan
	CHEMBL1383055	29095	11	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	334	3	0	9	2.0	c1cncc(-c2nn3c(Cn4nnc5ccccc54)nnc3s2)c1	nan
	220464	29097	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	175	0	0	2	2.9	Cn1ccc(=S)c2ccccc21	nan
	CHEMBL1383064	29097	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	175	0	0	2	2.9	Cn1ccc(=S)c2ccccc21	nan
	4805097	29110	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	2	0	7	0.4	CC1Cc2ccccc2N1C(=O)Cn1cnc2c1c(=O)n(C)c(=O)n2C	nan
	CHEMBL1383239	29110	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	2	0	7	0.4	CC1Cc2ccccc2N1C(=O)Cn1cnc2c1c(=O)n(C)c(=O)n2C	nan
	1186390	29331	12	None	-1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	1	0	3	4.7	O=C(Oc1c(Br)cc(Br)c2cccnc12)N1CCCCC1	nan
	CHEMBL1385192	29331	12	None	-1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	1	0	3	4.7	O=C(Oc1c(Br)cc(Br)c2cccnc12)N1CCCCC1	nan
	4877595	29534	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	6	1	5	3.8	O=C(CSc1nnc(-c2ccc(F)cc2)c2ccccc12)NCC1CCCO1	nan
	CHEMBL1386797	29534	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	6	1	5	3.8	O=C(CSc1nnc(-c2ccc(F)cc2)c2ccccc12)NCC1CCCO1	nan
	865072	29790	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	324	5	0	5	4.0	CCOC(=O)CSc1nc(-c2ccccc2)nc2ccccc12	nan
	CHEMBL1388860	29790	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	324	5	0	5	4.0	CCOC(=O)CSc1nc(-c2ccccc2)nc2ccccc12	nan
	2406693	29813	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	423	5	1	8	2.5	COC(=O)c1sc2nc(C)nc(SCC(=O)N3CCC(C(=O)O)CC3)c2c1C	nan
	CHEMBL1389013	29813	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	423	5	1	8	2.5	COC(=O)c1sc2nc(C)nc(SCC(=O)N3CCC(C(=O)O)CC3)c2c1C	nan
	1261479	29960	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	460	6	2	5	3.5	Cc1cc(C)c2nc(-c3ccccn3)cc(C(=O)NCCc3ccc(S(N)(=O)=O)cc3)c2c1	nan
	CHEMBL1390223	29960	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	460	6	2	5	3.5	Cc1cc(C)c2nc(-c3ccccn3)cc(C(=O)NCCc3ccc(S(N)(=O)=O)cc3)c2c1	nan
	16033258	30408	0	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	398	4	1	5	5.2	Cc1c(C(=O)Nc2ccccc2F)sc2ncnc(N(C)C3CCCCC3)c12	nan
	CHEMBL1394084	30408	0	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	398	4	1	5	5.2	Cc1c(C(=O)Nc2ccccc2F)sc2ncnc(N(C)C3CCCCC3)c12	nan
	16019740	30410	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	6	0	8	2.9	CCn1c(=O)c2sccc2n2c(CCCC(=O)N3CCN(c4ccc(F)cc4)CC3)nnc12	nan
	CHEMBL1394098	30410	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	6	0	8	2.9	CCn1c(=O)c2sccc2n2c(CCCC(=O)N3CCN(c4ccc(F)cc4)CC3)nnc12	nan
	16019075	30438	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	466	7	1	6	4.4	CC(C)Oc1ccc(CNC(=O)c2ccc(Cn3c(=O)c4cccn4c4cccnc43)cc2)cc1	nan
	CHEMBL1394443	30438	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	466	7	1	6	4.4	CC(C)Oc1ccc(CNC(=O)c2ccc(Cn3c(=O)c4cccn4c4cccnc43)cc2)cc1	nan
	1179391	30599	16	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	4	1	5	3.6	Cc1ccc(C(=O)Nc2nc3ccc(S(=O)(=O)N4CCCC4)cc3s2)cc1	nan
	CHEMBL1396599	30599	16	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	4	1	5	3.6	Cc1ccc(C(=O)Nc2nc3ccc(S(=O)(=O)N4CCCC4)cc3s2)cc1	nan
	16031181	30665	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	5	1	6	4.3	COc1cc(NC(=O)c2cc3cc4cc(OC)ccc4nc3o2)cc(OC)c1	nan
	CHEMBL1397472	30665	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	5	1	6	4.3	COc1cc(NC(=O)c2cc3cc4cc(OC)ccc4nc3o2)cc(OC)c1	nan
	16028170	30703	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	3	2	3	4.2	O=C1CC(c2ccccc2)Cc2[nH]c(=O)c(C(=O)Nc3cccc(Cl)c3)cc21	nan
	CHEMBL1397995	30703	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	3	2	3	4.2	O=C1CC(c2ccccc2)Cc2[nH]c(=O)c(C(=O)Nc3cccc(Cl)c3)cc21	nan
	729756	30726	15	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	330	3	1	3	3.9	Cc1ccc(/C=C(\C#N)C(=O)Nc2ccc(Br)cc2)o1	nan
	CHEMBL1398350	30726	15	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	330	3	1	3	3.9	Cc1ccc(/C=C(\C#N)C(=O)Nc2ccc(Br)cc2)o1	nan
	16031340	30733	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	373	5	1	3	4.7	CCc1ccc(CNC(=O)c2cnc(N3CCCCC3)c3ccccc23)cc1	nan
	CHEMBL1398430	30733	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	373	5	1	3	4.7	CCc1ccc(CNC(=O)c2cnc(N3CCCCC3)c3ccccc23)cc1	nan
	15989002	30734	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	481	7	1	8	2.8	O=C(CCn1c(=O)c2sccc2n(Cc2cccc(F)c2)c1=O)NCc1ccc2c(c1)OCO2	nan
	CHEMBL1398440	30734	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	481	7	1	8	2.8	O=C(CCn1c(=O)c2sccc2n(Cc2cccc(F)c2)c1=O)NCc1ccc2c(c1)OCO2	nan
	16026774	30737	3	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	5	1	7	2.2	Cc1csc2nc(COC(=O)CNC(=O)c3ccccc3Cl)cc(=O)n12	nan
	CHEMBL1398452	30737	3	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	5	1	7	2.2	Cc1csc2nc(COC(=O)CNC(=O)c3ccccc3Cl)cc(=O)n12	nan
	24790947	31028	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	454	4	0	5	3.9	O=S(=O)(c1ccc2nc(N3CCN(c4ccc(F)cc4)CC3)ccc2c1)N1CCCCC1	nan
	CHEMBL1401193	31028	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	454	4	0	5	3.9	O=S(=O)(c1ccc2nc(N3CCN(c4ccc(F)cc4)CC3)ccc2c1)N1CCCCC1	nan
	16017881	31308	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	6	1	6	2.3	CCOc1ccc(NC(=O)Cn2ccn(-c3ccc(F)c(F)c3)c(=O)c2=O)cc1	nan
	CHEMBL1403689	31308	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	6	1	6	2.3	CCOc1ccc(NC(=O)Cn2ccn(-c3ccc(F)c(F)c3)c(=O)c2=O)cc1	nan
	654955	31573	5	None	-4	3	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	3	1	6	4.7	CS(=O)(=O)c1sc2nc(-c3cccs3)cc(-c3ccccc3)c2c1N	nan
	CHEMBL1406204	31573	5	None	-4	3	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	3	1	6	4.7	CS(=O)(=O)c1sc2nc(-c3cccs3)cc(-c3ccccc3)c2c1N	nan
	135416200	31575	17	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	5	1	6	3.9	CCN(CC)Cc1c(O)ccc2cc(-c3nc4ccccc4n3C)c(=O)oc12	nan
	45369539	31575	17	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	5	1	6	3.9	CCN(CC)Cc1c(O)ccc2cc(-c3nc4ccccc4n3C)c(=O)oc12	nan
	CHEMBL1406220	31575	17	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	5	1	6	3.9	CCN(CC)Cc1c(O)ccc2cc(-c3nc4ccccc4n3C)c(=O)oc12	nan
	16025790	31625	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	5	1	4	4.5	CCC(C)NC(=O)C1CCN(C(=O)c2ccc(-n3ccc4ccccc43)s2)CC1	nan
	CHEMBL1406711	31625	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	5	1	4	4.5	CCC(C)NC(=O)C1CCN(C(=O)c2ccc(-n3ccc4ccccc43)s2)CC1	nan
	1257542	31693	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	275	4	1	6	1.4	Cc1cccnc1NC(=O)Cn1nc([N+](=O)[O-])cc1C	nan
	CHEMBL1407331	31693	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	275	4	1	6	1.4	Cc1cccnc1NC(=O)Cn1nc([N+](=O)[O-])cc1C	nan
	5834534	31749	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	6	1	5	5.2	CCOc1ccc(C(=O)C2=C(O)C(=O)N(c3ccccn3)C2c2ccc(Cl)cc2)c(C)c1	nan
	CHEMBL1407665	31749	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	6	1	5	5.2	CCOc1ccc(C(=O)C2=C(O)C(=O)N(c3ccccn3)C2c2ccc(Cl)cc2)c(C)c1	nan
	1509257	31770	12	None	-2	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	2	1	5	3.5	CCN1CCc2nc3sc(C(=O)N4CCc5ccccc5C4)c(N)c3cc2C1	nan
	CHEMBL1407777	31770	12	None	-2	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	2	1	5	3.5	CCN1CCc2nc3sc(C(=O)N4CCc5ccccc5C4)c(N)c3cc2C1	nan
	981045	31962	16	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	5	0	9	-0.1	CCn1c(SCCN2CCOCC2)nc2c1c(=O)n(C)c(=O)n2C	nan
	CHEMBL1409260	31962	16	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	5	0	9	-0.1	CCn1c(SCCN2CCOCC2)nc2c1c(=O)n(C)c(=O)n2C	nan
	2649456	32071	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	2	0	5	2.7	O=c1ccc(C(F)(F)F)cn1Cc1cc(=O)n2cc(Br)ccc2n1	nan
	CHEMBL1410109	32071	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	2	0	5	2.7	O=c1ccc(C(F)(F)F)cn1Cc1cc(=O)n2cc(Br)ccc2n1	nan
	1191742	32094	11	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	4	1	5	4.3	O=C(O)CSc1ncnc2scc(-c3ccc(Br)cc3)c12	nan
	CHEMBL1410306	32094	11	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	4	1	5	4.3	O=C(O)CSc1ncnc2scc(-c3ccc(Br)cc3)c12	nan
	15990415	32308	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	4	1	5	5.5	COc1ccc(Cl)cc1NC(=O)c1cn(C2CCCC2)c(=O)c2c1c1ccccc1n2C	nan
	CHEMBL1412135	32308	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	4	1	5	5.5	COc1ccc(Cl)cc1NC(=O)c1cn(C2CCCC2)c(=O)c2c1c1ccccc1n2C	nan
	3151320	32342	17	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	4	2	7	2.4	N=c1c(C(=O)NC2CCCCC2)cc2c(=O)n3ccccc3nc2n1CC1CCCO1	nan
	CHEMBL1412407	32342	17	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	4	2	7	2.4	N=c1c(C(=O)NC2CCCCC2)cc2c(=O)n3ccccc3nc2n1CC1CCCO1	nan
	1484210	32347	14	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	252	4	0	5	3.6	CCSc1nnc(-c2ccccc2SC)o1	nan
	CHEMBL1412417	32347	14	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	252	4	0	5	3.6	CCSc1nnc(-c2ccccc2SC)o1	nan
	4433827	32850	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	6	1	8	2.8	CSc1nc(SCC(=O)NCC2CCCO2)c2c3c(sc2n1)CN(C)CC3	nan
	CHEMBL1416667	32850	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	6	1	8	2.8	CSc1nc(SCC(=O)NCC2CCCO2)c2c3c(sc2n1)CN(C)CC3	nan
	3245881	33394	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	5	1	9	2.6	COc1cc2nc(S)n3nc(CCn4nc(C)cc4C)nc3c2cc1OC	nan
	CHEMBL1421316	33394	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	5	1	9	2.6	COc1cc2nc(S)n3nc(CCn4nc(C)cc4C)nc3c2cc1OC	nan
	5102370	33689	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	9	1	5	1.7	CCN(CC)S(=O)(=O)c1cccc(C(=O)NCCCn2ccnc2)c1	nan
	CHEMBL1423739	33689	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	9	1	5	1.7	CCN(CC)S(=O)(=O)c1cccc(C(=O)NCCCn2ccnc2)c1	nan
	4872167	33916	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	9	1	7	5.2	CCCCCOc1ccc(C2C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2c2cc(C)on2)cc1	nan
	CHEMBL1425797	33916	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	9	1	7	5.2	CCCCCOc1ccc(C2C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2c2cc(C)on2)cc1	nan
	2968003	33971	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	5	1	5	3.3	COc1ccc(-c2cc3ccc(OC(C)C(=O)O)cc3oc2=O)cc1	nan
	CHEMBL1426170	33971	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	5	1	5	3.3	COc1ccc(-c2cc3ccc(OC(C)C(=O)O)cc3oc2=O)cc1	nan
	5933014	34581	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	10	2	6	2.7	CCOc1ccc(C(=O)C2=C(O)C(=O)N(CCOCCO)C2c2ccccc2)cc1	nan
	CHEMBL1431128	34581	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	10	2	6	2.7	CCOc1ccc(C(=O)C2=C(O)C(=O)N(CCOCCO)C2c2ccccc2)cc1	nan
	2365417	34602	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	481	5	1	6	5.2	Cc1ccc2nc(-c3ccc(NC(=O)COC(=O)c4cncc(Br)c4)cc3)sc2c1	nan
	CHEMBL1431340	34602	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	481	5	1	6	5.2	Cc1ccc2nc(-c3ccc(NC(=O)COC(=O)c4cncc(Br)c4)cc3)sc2c1	nan
	2317063	34796	8	None	-2	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	7	2	5	5.6	CCCCOc1ccc(-c2c(C#N)c(S)nc(C)c2C(=O)Nc2ccccc2)cc1	nan
	CHEMBL1433074	34796	8	None	-2	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	7	2	5	5.6	CCCCOc1ccc(-c2c(C#N)c(S)nc(C)c2C(=O)Nc2ccccc2)cc1	nan
	16016637	34849	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	6	1	5	5.0	CCOc1ccc(CNC(=O)c2sc3nc(C)cc(C)c3c2-n2cccc2)cc1	nan
	CHEMBL1433449	34849	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	6	1	5	5.0	CCOc1ccc(CNC(=O)c2sc3nc(C)cc(C)c3c2-n2cccc2)cc1	nan
	16012551	34896	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	6	1	5	5.5	CCOc1ccc(-c2cc(NC(=O)c3cccc(Cl)c3)c(C(=O)OC)s2)cc1	nan
	CHEMBL1434218	34896	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	6	1	5	5.5	CCOc1ccc(-c2cc(NC(=O)c3cccc(Cl)c3)c(C(=O)OC)s2)cc1	nan
	16033555	34945	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	290	2	0	4	4.8	Cc1nc(Oc2ccccc2C)c2oc3ccccc3c2n1	nan
	CHEMBL1434916	34945	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	290	2	0	4	4.8	Cc1nc(Oc2ccccc2C)c2oc3ccccc3c2n1	nan
	16025666	35068	13	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	4	1	7	4.3	Cc1ccc(-n2nnc(-c3nsc(NC(=O)c4ccc(C)c(C)c4)n3)c2C)cc1	nan
	CHEMBL1436433	35068	13	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	4	1	7	4.3	Cc1ccc(-n2nnc(-c3nsc(NC(=O)c4ccc(C)c(C)c4)n3)c2C)cc1	nan
	16015798	35089	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	410	5	1	4	5.6	Cc1ccc(-c2nc3cc(Cl)ccc3o2)cc1NC(=O)COc1ccc(F)cc1	nan
	CHEMBL1436774	35089	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	410	5	1	4	5.6	Cc1ccc(-c2nc3cc(Cl)ccc3o2)cc1NC(=O)COc1ccc(F)cc1	nan
	16018841	35137	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	2	1	4	5.0	Cc1c(C(=O)Nc2ccc(F)cc2F)oc2ccc3c(c12)C(=O)CC(C)(C)O3	nan
	CHEMBL1437356	35137	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	2	1	4	5.0	Cc1c(C(=O)Nc2ccc(F)cc2F)oc2ccc3c(c12)C(=O)CC(C)(C)O3	nan
	1004026	35167	18	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	6	2	6	5.2	CCOc1ccccc1NC(=O)c1sc2nc(-c3ccc(OC)cc3)ccc2c1N	nan
	CHEMBL1437726	35167	18	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	6	2	6	5.2	CCOc1ccccc1NC(=O)c1sc2nc(-c3ccc(OC)cc3)ccc2c1N	nan
	16022287	35267	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	308	5	1	4	3.3	CCCCNC(=O)c1cccc(-n2c(C)nc3cccnc32)c1	nan
	CHEMBL1438563	35267	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	308	5	1	4	3.3	CCCCNC(=O)c1cccc(-n2c(C)nc3cccnc32)c1	nan
	5809896	35328	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	472	7	1	7	4.0	CCOc1cccc(C2C(C(=O)c3ccc4c(c3)OCCO4)=C(O)C(=O)N2Cc2ccncc2)c1	nan
	CHEMBL1439160	35328	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	472	7	1	7	4.0	CCOc1cccc(C2C(C(=O)c3ccc4c(c3)OCCO4)=C(O)C(=O)N2Cc2ccncc2)c1	nan
	15988173	35348	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	4	2	4	2.9	Cc1ccc(CNC(=O)c2ccc3c(=O)n(-c4ccccc4)c(=O)[nH]c3c2)cc1	nan
	CHEMBL1439335	35348	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	4	2	4	2.9	Cc1ccc(CNC(=O)c2ccc3c(=O)n(-c4ccccc4)c(=O)[nH]c3c2)cc1	nan
	1454908	35838	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	268	3	1	4	3.5	Sc1nc(COc2ccccc2)nc2ccccc12	nan
	CHEMBL1443793	35838	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	268	3	1	4	3.5	Sc1nc(COc2ccccc2)nc2ccccc12	nan
	1234247	36081	10	None	-1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	256	1	1	5	2.7	Cc1nnc(S)c2nn(-c3ccccc3)c(C)c12	nan
	CHEMBL1446078	36081	10	None	-1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	256	1	1	5	2.7	Cc1nnc(S)c2nn(-c3ccccc3)c(C)c12	nan
	16026772	36138	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	5	1	7	1.8	Cc1ccc(C(=O)NCC(=O)OCc2cc(=O)n3c(C)csc3n2)cc1	nan
	CHEMBL1446594	36138	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	5	1	7	1.8	Cc1ccc(C(=O)NCC(=O)OCc2cc(=O)n3c(C)csc3n2)cc1	nan
	2957415	36505	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	304	2	0	5	2.5	CC(=O)c1nc(N2C(=O)C3CC=C(C)CC3C2=O)sc1C	nan
	CHEMBL1449518	36505	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	304	2	0	5	2.5	CC(=O)c1nc(N2C(=O)C3CC=C(C)CC3C2=O)sc1C	nan
	2334194	36555	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	9	1	8	3.6	CCOC(=O)c1c(NS(=O)(=O)c2ccccc2)n(CCCOC)c2nc3ccccc3nc12	nan
	CHEMBL1449923	36555	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	9	1	8	3.6	CCOC(=O)c1c(NS(=O)(=O)c2ccccc2)n(CCCOC)c2nc3ccccc3nc12	nan
	4977513	36592	14	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	6	1	7	5.3	Cc1cc(N2C(=O)C(O)=C(C(=O)c3cc4ccccc4o3)C2c2ccc(OC(C)C)cc2)no1	nan
	CHEMBL1450219	36592	14	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	6	1	7	5.3	Cc1cc(N2C(=O)C(O)=C(C(=O)c3cc4ccccc4o3)C2c2ccc(OC(C)C)cc2)no1	nan
	2945668	36767	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	5	1	7	1.8	CCc1nnc(NC(=O)CCn2cnc3ccccc3c2=O)s1	nan
	CHEMBL1451692	36767	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	5	1	7	1.8	CCc1nnc(NC(=O)CCn2cnc3ccccc3c2=O)s1	nan
	24792337	36845	2	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	320	4	2	7	1.6	Cc1cc2nnc(SCC(=O)NC3CCCCC3)n2c(N)n1	nan
	CHEMBL1452223	36845	2	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	320	4	2	7	1.6	Cc1cc2nnc(SCC(=O)NC3CCCCC3)n2c(N)n1	nan
	15988498	36885	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	556	11	2	9	2.9	CCCNC(=O)C1CCC(Cn2c(=O)c3sccc3n(CC(=O)NCc3cccc(OC)c3OC)c2=O)CC1	nan
	CHEMBL1452564	36885	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	556	11	2	9	2.9	CCCNC(=O)C1CCC(Cn2c(=O)c3sccc3n(CC(=O)NCc3cccc(OC)c3OC)c2=O)CC1	nan
	2298970	36891	3	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	398	7	2	7	3.3	Cc1noc(NS(=O)(=O)c2ccc(N/C=C/C(=O)c3ccncc3)cc2)c1C	nan
	CHEMBL1452655	36891	3	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	398	7	2	7	3.3	Cc1noc(NS(=O)(=O)c2ccc(N/C=C/C(=O)c3ccncc3)cc2)c1C	nan
	24790128	37181	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	400	5	1	5	3.2	COc1ccc(-c2[nH]ncc2CN2CCN(C(=O)c3cccs3)CC2)c(F)c1	nan
	CHEMBL1454939	37181	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	400	5	1	5	3.2	COc1ccc(-c2[nH]ncc2CN2CCN(C(=O)c3cccs3)CC2)c(F)c1	nan
	16030361	37241	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	9	1	5	4.7	COc1cccc(Cc2nc3ccccc3nc2SCC(=O)NCCc2ccccc2)c1	nan
	CHEMBL1455531	37241	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	9	1	5	4.7	COc1cccc(Cc2nc3ccccc3nc2SCC(=O)NCCc2ccccc2)c1	nan
	16025668	37440	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	454	5	1	8	4.6	COc1ccc(-n2nnc(-c3nsc(NC(=O)c4ccc(C)c(C)c4)n3)c2C)cc1Cl	nan
	CHEMBL1457411	37440	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	454	5	1	8	4.6	COc1ccc(-n2nnc(-c3nsc(NC(=O)c4ccc(C)c(C)c4)n3)c2C)cc1Cl	nan
	1355891	37556	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	500	11	1	7	3.2	COc1ccc(OC)c(N(CC(=O)NCc2ccccc2)S(=O)(=O)c2ccc(OC)c(OC)c2)c1	nan
	CHEMBL1458278	37556	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	500	11	1	7	3.2	COc1ccc(OC)c(N(CC(=O)NCc2ccccc2)S(=O)(=O)c2ccc(OC)c(OC)c2)c1	nan
	2949787	37654	14	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	5	1	7	3.4	COc1ccccc1C1C(C(=O)c2ccco2)=C(O)C(=O)N1c1cc(C)on1	nan
	CHEMBL1459163	37654	14	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	5	1	7	3.4	COc1ccccc1C1C(C(=O)c2ccco2)=C(O)C(=O)N1c1cc(C)on1	nan
	1445336	37658	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	488	6	0	8	3.9	COc1ccccc1N1CCN(C(=O)CSc2ncnc3c2cnn3-c2ccc(C)c(C)c2)CC1	nan
	CHEMBL1459184	37658	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	488	6	0	8	3.9	COc1ccccc1N1CCN(C(=O)CSc2ncnc3c2cnn3-c2ccc(C)c(C)c2)CC1	nan
	6033330	37798	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	536	11	1	8	3.9	CCCCOc1ccc(C2C(C(=O)c3ccc4c(c3)OCCO4)=C(O)C(=O)N2CCCN2CCOCC2)cc1	nan
	CHEMBL1460387	37798	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	536	11	1	8	3.9	CCCCOc1ccc(C2C(C(=O)c3ccc4c(c3)OCCO4)=C(O)C(=O)N2CCCN2CCOCC2)cc1	nan
	5160710	37838	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	308	5	2	2	4.5	CCCOc1ccc(NC(=O)c2cc3cc(C)ccc3[nH]2)cc1	nan
	CHEMBL1460665	37838	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	308	5	2	2	4.5	CCCOc1ccc(NC(=O)c2cc3cc(C)ccc3[nH]2)cc1	nan
	3502512	37923	14	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	2	2	8	1.0	N#Cc1c(N2CCOCC2)nc(N)c2c(N)nc3c(c12)CC(CCl)O3	nan
	CHEMBL1461443	37923	14	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	2	2	8	1.0	N#Cc1c(N2CCOCC2)nc(N)c2c(N)nc3c(c12)CC(CCl)O3	nan
	2810150	38006	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	2	1	5	4.1	Cc1csc2c(=O)sc(NC(=O)c3ccc(F)cc3Cl)nc12	nan
	CHEMBL1462227	38006	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	2	1	5	4.1	Cc1csc2c(=O)sc(NC(=O)c3ccc(F)cc3Cl)nc12	nan
	4524521	38041	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	4	1	7	0.2	Cn1c(C(=O)NCCN2CCOCC2)cc2c(=O)n3ccccc3nc21	nan
	CHEMBL1462442	38041	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	4	1	7	0.2	Cn1c(C(=O)NCCN2CCOCC2)cc2c(=O)n3ccccc3nc21	nan
	1491130	38097	19	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	5	1	5	3.3	O=C(O)COc1ccc(-c2nccc(-c3cccs3)n2)cc1	nan
	CHEMBL1462936	38097	19	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	5	1	5	3.3	O=C(O)COc1ccc(-c2nccc(-c3cccs3)n2)cc1	nan
	135464100	38209	16	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	5	2	6	3.3	N#Cc1c(O)nc(SCC(=O)NC2CCCCC2)nc1-c1ccccc1	nan
	CHEMBL1463888	38209	16	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	5	2	6	3.3	N#Cc1c(O)nc(SCC(=O)NC2CCCCC2)nc1-c1ccccc1	nan
	2808819	38460	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	4	1	5	4.1	Cc1csc2ncnc(NC3CCN(Cc4ccccc4)CC3)c12	nan
	CHEMBL1465720	38460	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	4	1	5	4.1	Cc1csc2ncnc(NC3CCN(Cc4ccccc4)CC3)c12	nan
	1100812	38501	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	4	0	6	4.4	CCOC(=O)c1nn2c(C(F)(F)F)cc(-c3ccc(OC)cc3)nc2c1Br	nan
	CHEMBL1466098	38501	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	4	0	6	4.4	CCOC(=O)c1nn2c(C(F)(F)F)cc(-c3ccc(OC)cc3)nc2c1Br	nan
	665758	38521	8	None	-1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	5	0	7	4.3	COc1cc(OC)cc(-c2nc(-c3cc4cc(C)ccc4nc3OC)no2)c1	nan
	CHEMBL1466279	38521	8	None	-1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	5	0	7	4.3	COc1cc(OC)cc(-c2nc(-c3cc4cc(C)ccc4nc3OC)no2)c1	nan
	20953708	38823	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	423	5	1	7	3.2	COc1ccc(-c2cc3c(=O)n(CC(=O)Nc4cccc(Cl)c4)nc(C)n3n2)cc1	nan
	CHEMBL1468743	38823	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	423	5	1	7	3.2	COc1ccc(-c2cc3c(=O)n(CC(=O)Nc4cccc(Cl)c4)nc(C)n3n2)cc1	nan
	2913184	38919	15	None	-3	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	4	1	7	3.4	Cc1nnc(N2C(=O)C(O)=C(C(=O)c3ccco3)C2c2ccc(F)cc2)s1	nan
	CHEMBL1469528	38919	15	None	-3	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	4	1	7	3.4	Cc1nnc(N2C(=O)C(O)=C(C(=O)c3ccco3)C2c2ccc(F)cc2)s1	nan
	1226649	38943	14	None	-2	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	2	2	4	4.1	CC(=O)NC(=S)Nc1ccc(-c2nc3ccc(C)cc3s2)cc1	nan
	CHEMBL1469733	38943	14	None	-2	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	2	2	4	4.1	CC(=O)NC(=S)Nc1ccc(-c2nc3ccc(C)cc3s2)cc1	nan
	794237	39070	14	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	311	4	1	5	3.5	COc1ccc(C(=O)Nc2nnc(-c3ccccc3)s2)cc1	nan
	CHEMBL1470825	39070	14	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	311	4	1	5	3.5	COc1ccc(C(=O)Nc2nnc(-c3ccccc3)s2)cc1	nan
	1025062	39254	9	None	-2	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	511	7	1	5	5.6	Cc1nc(SCC(=O)Nc2ccc(F)cc2)c(C#N)c(C)c1CC(=O)c1ccc(Br)cc1	nan
	CHEMBL1472426	39254	9	None	-2	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	511	7	1	5	5.6	Cc1nc(SCC(=O)Nc2ccc(F)cc2)c(C#N)c(C)c1CC(=O)c1ccc(Br)cc1	nan
	16025800	39375	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	7	1	5	3.7	COCCCNC(=O)C1CCN(C(=O)c2ccc(-n3ccc4ccccc43)s2)CC1	nan
	CHEMBL1474073	39375	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	7	1	5	3.7	COCCCNC(=O)C1CCN(C(=O)c2ccc(-n3ccc4ccccc43)s2)CC1	nan
	16017955	39392	0	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	3	1	5	3.3	Cc1ccc(NC(=O)c2nc(-c3ccncc3)no2)c(Cl)c1	nan
	CHEMBL1474407	39392	0	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	3	1	5	3.3	Cc1ccc(NC(=O)c2nc(-c3ccncc3)no2)c(Cl)c1	nan
	923699	39573	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	3	1	4	4.8	Cc1cc(C)cc(C(=O)Nc2ccc(-c3nc4ncccc4o3)cc2)c1	nan
	CHEMBL1476840	39573	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	3	1	4	4.8	Cc1cc(C)cc(C(=O)Nc2ccc(-c3nc4ncccc4o3)cc2)c1	nan
	16030273	39613	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	486	6	0	5	5.1	Cc1ccc(Cc2nc3ccccc3nc2SCC(=O)N2CCN(c3ccccc3F)CC2)cc1	nan
	CHEMBL1477298	39613	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	486	6	0	5	5.1	Cc1ccc(Cc2nc3ccccc3nc2SCC(=O)N2CCN(c3ccccc3F)CC2)cc1	nan
	3492613	39861	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	3	1	4	4.6	COc1ccc(-n2cc(-c3ccc(Br)cc3)nc2S)cc1	nan
	CHEMBL1479477	39861	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	3	1	4	4.6	COc1ccc(-n2cc(-c3ccc(Br)cc3)nc2S)cc1	nan
	1077503	39889	17	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	5	2	7	1.9	CCCn1c(=N)c(C(=O)NCc2cccnc2)cc2c(=O)n3ccccc3nc21	nan
	CHEMBL1479731	39889	17	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	5	2	7	1.9	CCCn1c(=N)c(C(=O)NCc2cccnc2)cc2c(=O)n3ccccc3nc21	nan
	2059287	40169	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	5	0	5	3.5	CCCCN(CC)C(=O)c1cc2c(=O)n3cccc(C)c3nc2s1	nan
	CHEMBL1482087	40169	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	5	0	5	3.5	CCCCN(CC)C(=O)c1cc2c(=O)n3cccc(C)c3nc2s1	nan
	2490618	40188	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	7	1	9	0.0	CCc1ccc(OCC(=O)OCC(=O)c2c(N)n(C)c(=O)n(C)c2=O)cc1	nan
	CHEMBL1482290	40188	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	7	1	9	0.0	CCc1ccc(OCC(=O)OCC(=O)c2c(N)n(C)c(=O)n(C)c2=O)cc1	nan
	16020212	40639	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	562	7	2	8	3.8	Cc1ccc(NC(=O)Cn2c(=O)n(-c3ccccc3)c(=O)c3ccc(C(=O)NCc4ccc5c(c4)OCO5)cc32)cc1	nan
	CHEMBL1486218	40639	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	562	7	2	8	3.8	Cc1ccc(NC(=O)Cn2c(=O)n(-c3ccccc3)c(=O)c3ccc(C(=O)NCc4ccc5c(c4)OCO5)cc32)cc1	nan
	5835099	41104	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	8	1	6	5.0	CCCOc1ccc(C(=O)C2=C(O)C(=O)N(c3ccccn3)C2c2ccc(OC)cc2)cc1C	nan
	CHEMBL1489865	41104	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	8	1	6	5.0	CCCOc1ccc(C(=O)C2=C(O)C(=O)N(c3ccccn3)C2c2ccc(OC)cc2)cc1C	nan
	24791694	41201	3	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	4	0	4	4.0	COc1ccc2cc(C(=O)C3CCCN(C(=O)c4cccnc4)C3)ccc2c1	nan
	CHEMBL1490547	41201	3	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	4	0	4	4.0	COc1ccc2cc(C(=O)C3CCCN(C(=O)c4cccnc4)C3)ccc2c1	nan
	135438626	41466	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	6	3	9	0.8	Cc1ccc(S(=O)(=O)N2CCOCC2)cc1NC(=O)CSc1nc(N)cc(O)n1	nan
	CHEMBL1492401	41466	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	6	3	9	0.8	Cc1ccc(S(=O)(=O)N2CCOCC2)cc1NC(=O)CSc1nc(N)cc(O)n1	nan
	16018070	41502	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	7	1	4	3.5	O=C(CCCn1c(=O)c2cccn2c2ccc(F)cc21)NCCc1ccccc1	nan
	CHEMBL1492679	41502	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	7	1	4	3.5	O=C(CCCn1c(=O)c2cccn2c2ccc(F)cc21)NCCc1ccccc1	nan
	1327115	41592	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	366	3	1	5	4.8	COc1cccc(-c2cc3c(=O)n(-c4ccccc4)c(=S)[nH]c3s2)c1	nan
	CHEMBL1493481	41592	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	366	3	1	5	4.8	COc1cccc(-c2cc3c(=O)n(-c4ccccc4)c(=S)[nH]c3s2)c1	nan
	3034554	41700	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	325	4	1	7	1.5	Cn1c(=S)c2nc(SCCN3CCCC3)[nH]c2n(C)c1=O	nan
	CHEMBL1494615	41700	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	325	4	1	7	1.5	Cn1c(=S)c2nc(SCCN3CCCC3)[nH]c2n(C)c1=O	nan
	976285	42096	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	243	1	0	5	2.1	Cc1csc2nc(=O)c(-c3ccccc3)nn12	nan
	CHEMBL1498297	42096	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	243	1	0	5	2.1	Cc1csc2nc(=O)c(-c3ccccc3)nn12	nan
	3127165	42366	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	6	1	8	0.5	CC(C(O)c1ccccc1)N(C)CCn1cnc2c1c(=O)n(C)c(=O)n2C	nan
	CHEMBL1500612	42366	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	6	1	8	0.5	CC(C(O)c1ccccc1)N(C)CCn1cnc2c1c(=O)n(C)c(=O)n2C	nan
	135413586	42446	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	8	2	10	3.0	CCOC(=O)Cc1csc(NC(=O)CSc2nc(O)c(C#N)c(-c3ccccc3)n2)n1	nan
	CHEMBL1501394	42446	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	8	2	10	3.0	CCOC(=O)Cc1csc(NC(=O)CSc2nc(O)c(C#N)c(-c3ccccc3)n2)n1	nan
	5903312	42584	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	396	6	1	8	0.1	COCCNC(=O)/C(C#N)=C/c1c(N2CCN(C)CC2)nc2ccccn2c1=O	nan
	CHEMBL1502541	42584	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	396	6	1	8	0.1	COCCNC(=O)/C(C#N)=C/c1c(N2CCN(C)CC2)nc2ccccn2c1=O	nan
	790333	43018	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	189	0	1	2	3.1	Cc1cc(S)c2cccc(C)c2n1	nan
	CHEMBL1506363	43018	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	189	0	1	2	3.1	Cc1cc(S)c2cccc(C)c2n1	nan
	2146623	43349	17	None	1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	351	6	1	4	5.0	CC(=O)c1ccc(NC(=O)c2ccc(CSc3ccccc3)o2)cc1	nan
	CHEMBL1509267	43349	17	None	1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	351	6	1	4	5.0	CC(=O)c1ccc(NC(=O)c2ccc(CSc3ccccc3)o2)cc1	nan
	4617873	43662	13	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	6	2	3	4.4	NC(=O)c1ccc(NC(=O)c2ccc(COc3ccccc3Br)cc2)cc1	nan
	CHEMBL1512241	43662	13	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	6	2	3	4.4	NC(=O)c1ccc(NC(=O)c2ccc(COc3ccccc3Br)cc2)cc1	nan
	7877577	43762	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	361	5	1	7	1.4	O=C(CNC(=O)c1ccc(F)cc1)OCc1cc(=O)n2ccsc2n1	nan
	CHEMBL1513627	43762	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	361	5	1	7	1.4	O=C(CNC(=O)c1ccc(F)cc1)OCc1cc(=O)n2ccsc2n1	nan
	7598873	43800	11	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	5	1	3	3.9	CCc1ccccc1NC(=O)c1cccn(Cc2ccccc2F)c1=O	nan
	CHEMBL1514321	43800	11	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	5	1	3	3.9	CCc1ccccc1NC(=O)c1cccn(Cc2ccccc2F)c1=O	nan
	16030561	43813	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	506	6	0	5	5.5	O=C(CSc1nc2ccccc2nc1Cc1ccc(Cl)cc1)N1CCN(c2ccccc2F)CC1	nan
	CHEMBL1514538	43813	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	506	6	0	5	5.5	O=C(CSc1nc2ccccc2nc1Cc1ccc(Cl)cc1)N1CCN(c2ccccc2F)CC1	nan
	16009347	43816	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	4	0	5	4.6	Cc1cc(C)cc(OCc2cc(=O)n3c(-c4ccccc4)csc3n2)c1	nan
	CHEMBL1514567	43816	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	4	0	5	4.6	Cc1cc(C)cc(OCc2cc(=O)n3c(-c4ccccc4)csc3n2)c1	nan
	16018206	43826	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	477	6	1	6	5.5	COc1cc(NC(=O)c2oc3c(c2C)-c2nn(Cc4cccc(Cl)c4)cc2CC3)cc(OC)c1	nan
	CHEMBL1514692	43826	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	477	6	1	6	5.5	COc1cc(NC(=O)c2oc3c(c2C)-c2nn(Cc4cccc(Cl)c4)cc2CC3)cc(OC)c1	nan
	3207800	44074	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	4	1	6	3.8	Cc1cc(C)c2nc(SCC(=O)Nc3cc(C)on3)c(C#N)cc2c1	nan
	CHEMBL1517790	44074	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	4	1	6	3.8	Cc1cc(C)c2nc(SCC(=O)Nc3cc(C)on3)c(C#N)cc2c1	nan
	2091511	44126	2	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	4	0	8	2.5	Cc1ccc2nc(CSc3nnc(-c4ccncc4)n3C)cc(=O)n2c1	nan
	CHEMBL1518274	44126	2	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	4	0	8	2.5	Cc1ccc2nc(CSc3nnc(-c4ccncc4)n3C)cc(=O)n2c1	nan
	24818303	44128	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	4	1	3	4.4	CN(C)C(=O)c1ccc(NC(=O)c2sccc2-c2ccccc2)cc1	nan
	CHEMBL1518303	44128	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	4	1	3	4.4	CN(C)C(=O)c1ccc(NC(=O)c2sccc2-c2ccccc2)cc1	nan
	5151092	44131	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	318	1	1	2	3.2	CNC(=O)c1c2c(nc3ccc(Br)cc13)CCCC2	nan
	CHEMBL1518360	44131	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	318	1	1	2	3.2	CNC(=O)c1c2c(nc3ccc(Br)cc13)CCCC2	nan
	16019804	44295	3	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	9	1	8	1.6	CCCn1c(=O)c2sccc2n2c(CCCC(=O)NCCOC)nnc12	nan
	CHEMBL1519737	44295	3	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	9	1	8	1.6	CCCn1c(=O)c2sccc2n2c(CCCC(=O)NCCOC)nnc12	nan
	4917226	44360	11	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	7	2	4	5.8	O=C(O)CC(NC(=O)c1sc2ccccc2c1Cl)c1ccc(OC2CCCC2)cc1	nan
	CHEMBL1520355	44360	11	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	7	2	4	5.8	O=C(O)CC(NC(=O)c1sc2ccccc2c1Cl)c1ccc(OC2CCCC2)cc1	nan
	24677542	44437	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	8	4	5	3.0	CCCCCNC(=O)c1ccc(NS(=O)(=O)c2ccc3[nH]c(O)nc3c2)cc1	nan
	CHEMBL1520946	44437	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	8	4	5	3.0	CCCCCNC(=O)c1ccc(NS(=O)(=O)c2ccc3[nH]c(O)nc3c2)cc1	nan
	902803	44601	13	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	303	5	1	2	4.5	O=C(Nc1ccccc1)c1ccc(COc2ccccc2)cc1	nan
	CHEMBL1522424	44601	13	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	303	5	1	2	4.5	O=C(Nc1ccccc1)c1ccc(COc2ccccc2)cc1	nan
	15988611	44808	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	6	1	8	3.9	CC(=O)c1ccc(NC(=O)Cn2c(=O)n(Cc3ccco3)c(=O)c3sc4ccccc4c32)cc1	nan
	CHEMBL1524392	44808	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	6	1	8	3.9	CC(=O)c1ccc(NC(=O)Cn2c(=O)n(Cc3ccco3)c(=O)c3sc4ccccc4c32)cc1	nan
	3239863	44967	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	356	7	0	8	2.4	CCOC(=O)CC(=O)CSc1ccc2nnc(-c3ccccc3)n2n1	nan
	CHEMBL1525909	44967	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	356	7	0	8	2.4	CCOC(=O)CC(=O)CSc1ccc2nnc(-c3ccccc3)n2n1	nan
	2930800	45047	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	5	2	7	2.5	COC(=O)c1sc(NC(=O)C2CCCCC2C(=O)O)c(C(=O)OC)c1C	nan
	CHEMBL1526492	45047	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	5	2	7	2.5	COC(=O)c1sc(NC(=O)C2CCCCC2C(=O)O)c(C(=O)OC)c1C	nan
	2349018	45228	20	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	280	2	1	4	3.4	CCCn1c(=S)[nH]c2sc3c(c2c1=O)CCCC3	nan
	CHEMBL1528175	45228	20	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	280	2	1	4	3.4	CCCn1c(=S)[nH]c2sc3c(c2c1=O)CCCC3	nan
	1355435	45242	11	None	-22	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	2	0	4	3.3	Cc1cn(S(=O)(=O)c2ccc(Br)c3ccccc23)cn1	nan
	CHEMBL1528299	45242	11	None	-22	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	2	0	4	3.3	Cc1cn(S(=O)(=O)c2ccc(Br)c3ccccc23)cn1	nan
	5073065	45340	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	330	4	1	6	-0.6	O=C(Cn1cnc2ccccc2c1=O)NCC(=O)N1CCOCC1	nan
	CHEMBL1529152	45340	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	330	4	1	6	-0.6	O=C(Cn1cnc2ccccc2c1=O)NCC(=O)N1CCOCC1	nan
	3240741	45433	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	475	9	1	8	4.6	COc1ccc(CC(=O)Nc2ccc(-c3noc(-c4cc(OC)c(OC)c(OC)c4)n3)cc2)cc1	nan
	CHEMBL1529936	45433	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	475	9	1	8	4.6	COc1ccc(CC(=O)Nc2ccc(-c3noc(-c4cc(OC)c(OC)c(OC)c4)n3)cc2)cc1	nan
	3212225	45458	2	None	-1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	5	1	5	3.1	Cc1cc(C)c2nc(SCC(=O)NCC3CCCO3)c(C#N)cc2c1	nan
	CHEMBL1530244	45458	2	None	-1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	5	1	5	3.1	Cc1cc(C)c2nc(SCC(=O)NCC3CCCO3)c(C#N)cc2c1	nan
	16024952	45460	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	5	1	6	4.0	CCOC(=O)c1cccc(NC(=O)c2ccc3c(c2)nnn3C2CCCC2)c1	nan
	CHEMBL1530263	45460	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	5	1	6	4.0	CCOC(=O)c1cccc(NC(=O)c2ccc3c(c2)nnn3C2CCCC2)c1	nan
	16017576	45471	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	6	1	7	2.2	CN(Cc1ccco1)S(=O)(=O)c1nnc(NC(=O)c2ccccc2)s1	nan
	CHEMBL1530393	45471	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	6	1	7	2.2	CN(Cc1ccco1)S(=O)(=O)c1nnc(NC(=O)c2ccccc2)s1	nan
	4907979	45479	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	6	2	6	3.0	OCCCNc1ncnc2sc3c(c12)CCN(Cc1ccccc1)C3	nan
	CHEMBL1530465	45479	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	6	2	6	3.0	OCCCNc1ncnc2sc3c(c12)CCN(Cc1ccccc1)C3	nan
	1161207	45559	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	8	2	7	3.1	COc1ccccc1OCC(=O)Nc1ccc(S(=O)(=O)Nc2onc(C)c2C)cc1	nan
	CHEMBL1531098	45559	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	8	2	7	3.1	COc1ccccc1OCC(=O)Nc1ccc(S(=O)(=O)Nc2onc(C)c2C)cc1	nan
	1355556	45622	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	3	1	3	3.8	O=S(=O)(Nc1cccnc1)c1ccc(Br)c2ccccc12	nan
	CHEMBL1531651	45622	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	3	1	3	3.8	O=S(=O)(Nc1cccnc1)c1ccc(Br)c2ccccc12	nan
	16025786	45842	3	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	475	5	1	4	5.3	Cc1cc2ccccc2n1-c1ccc(C(=O)N2CCC(C(=O)NCc3ccc(F)cc3)CC2)s1	nan
	CHEMBL1533608	45842	3	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	475	5	1	4	5.3	Cc1cc2ccccc2n1-c1ccc(C(=O)N2CCC(C(=O)NCc3ccc(F)cc3)CC2)s1	nan
	3151323	45927	16	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	4	2	7	2.3	Cc1cccn2c(=O)c3cc(C(=O)NC4CCCC4)c(=N)n(CC4CCCO4)c3nc12	nan
	CHEMBL1534442	45927	16	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	4	2	7	2.3	Cc1cccn2c(=O)c3cc(C(=O)NC4CCCC4)c(=N)n(CC4CCCO4)c3nc12	nan
	3238163	46167	6	None	-1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	5	1	8	0.6	Cc1ccc(-n2nnc3c(=O)n(CC(=O)NCC4CCCO4)cnc32)cc1	nan
	CHEMBL1536880	46167	6	None	-1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	5	1	8	0.6	Cc1ccc(-n2nnc3c(=O)n(CC(=O)NCC4CCCO4)cnc32)cc1	nan
	2989967	46249	19	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	4	1	6	3.5	Cc1cc(N2C(=O)C(O)=C(C(=O)c3ccco3)C2c2ccccc2F)no1	nan
	CHEMBL1537625	46249	19	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	4	1	6	3.5	Cc1cc(N2C(=O)C(O)=C(C(=O)c3ccco3)C2c2ccccc2F)no1	nan
	767265	46504	31	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	277	2	1	5	3.5	Sc1nnc(-c2ccco2)n1-c1ccc(Cl)cc1	nan
	CHEMBL1539766	46504	31	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	277	2	1	5	3.5	Sc1nnc(-c2ccco2)n1-c1ccc(Cl)cc1	nan
	891408	46939	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	259	4	0	6	1.7	O=C(OCc1cccc([N+](=O)[O-])c1)c1cnccn1	nan
	CHEMBL1543385	46939	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	259	4	0	6	1.7	O=C(OCc1cccc([N+](=O)[O-])c1)c1cnccn1	nan
	4634206	47031	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	7	2	10	-0.9	CCOc1ccccc1OCC(=O)NNC(=O)Cn1cnc2c1c(=O)n(C)c(=O)n2C	nan
	CHEMBL1544116	47031	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	7	2	10	-0.9	CCOc1ccccc1OCC(=O)NNC(=O)Cn1cnc2c1c(=O)n(C)c(=O)n2C	nan
	1487485	47035	19	None	-2	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	1	0	3	3.1	Cc1ccc(-n2ncc(Br)c(Br)c2=O)cc1	nan
	CHEMBL1544131	47035	19	None	-2	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	1	0	3	3.1	Cc1ccc(-n2ncc(Br)c(Br)c2=O)cc1	nan
	1867273	47121	18	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	5	2	7	1.8	Cc1ccc(-c2nn3c(C)nnc3c3ccccc23)cc1S(=O)(=O)NCCO	nan
	CHEMBL1544770	47121	18	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	5	2	7	1.8	Cc1ccc(-c2nn3c(C)nnc3c3ccccc23)cc1S(=O)(=O)NCCO	nan
	3781367	47173	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	482	5	2	8	4.2	CCOc1ccc(NC(=O)c2sc3nc(N4CCOCC4)c4c(c3c2N)CC(C)(C)OC4)cc1	nan
	CHEMBL1545158	47173	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	482	5	2	8	4.2	CCOc1ccc(NC(=O)c2sc3nc(N4CCOCC4)c4c(c3c2N)CC(C)(C)OC4)cc1	nan
	28358049	47420	20	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	295	4	1	4	3.3	CCN(CC)Cc1c(O)c(Cl)cc2c(C)cc(=O)oc12	nan
	5398465	47420	20	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	295	4	1	4	3.3	CCN(CC)Cc1c(O)c(Cl)cc2c(C)cc(=O)oc12	nan
	CHEMBL1547311	47420	20	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	295	4	1	4	3.3	CCN(CC)Cc1c(O)c(Cl)cc2c(C)cc(=O)oc12	nan
	7080334	47431	2	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	318	3	1	5	3.6	Cc1c(-c2cccc(NC(=O)c3ccco3)c2)nc2ncccn12	nan
	CHEMBL1547414	47431	2	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	318	3	1	5	3.6	Cc1c(-c2cccc(NC(=O)c3ccco3)c2)nc2ncccn12	nan
	1476696	47458	23	None	-2	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	366	4	0	4	4.8	CSc1cc(-c2ccc(Cl)cc2)n(Cc2ccccc2)c(=O)c1C#N	nan
	CHEMBL1547693	47458	23	None	-2	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	366	4	0	4	4.8	CSc1cc(-c2ccc(Cl)cc2)n(Cc2ccccc2)c(=O)c1C#N	nan
	3830390	47552	3	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	252	2	2	8	-1.2	CN(N)N=Nc1nc2c(=O)n(C)c(=O)n(C)c2[nH]1	nan
	CHEMBL1548599	47552	3	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	252	2	2	8	-1.2	CN(N)N=Nc1nc2c(=O)n(C)c(=O)n(C)c2[nH]1	nan
	20885691	47853	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	7	1	6	1.9	CCc1ccc(CNC(=O)CCCn2nc(C)n3ccnc3c2=O)cc1	nan
	CHEMBL1551091	47853	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	7	1	6	1.9	CCc1ccc(CNC(=O)CCCn2nc(C)n3ccnc3c2=O)cc1	nan
	2053967	47872	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	7	0	5	4.3	CCCCN(CCCC)C(=O)c1cc2c(=O)n3cccc(C)c3nc2s1	nan
	CHEMBL1551348	47872	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	7	0	5	4.3	CCCCN(CCCC)C(=O)c1cc2c(=O)n3cccc(C)c3nc2s1	nan
	7151074	47929	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	6	1	6	4.1	O=C(CSc1nccn1Cc1ccc(Cl)cc1)Nc1ccc2c(c1)OCCO2	nan
	CHEMBL1552167	47929	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	6	1	6	4.1	O=C(CSc1nccn1Cc1ccc(Cl)cc1)Nc1ccc2c(c1)OCCO2	nan
	16025798	48121	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	461	5	1	4	5.0	O=C(NCc1ccc(F)cc1)C1CCN(C(=O)c2ccc(-n3ccc4ccccc43)s2)CC1	nan
	CHEMBL1554965	48121	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	461	5	1	4	5.0	O=C(NCc1ccc(F)cc1)C1CCN(C(=O)c2ccc(-n3ccc4ccccc43)s2)CC1	nan
	16019077	48179	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	6	1	5	4.3	O=C(NCCc1ccccc1Cl)c1ccc(Cn2c(=O)c3cccn3c3cccnc32)cc1	nan
	CHEMBL1555692	48179	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	6	1	5	4.3	O=C(NCCc1ccccc1Cl)c1ccc(Cn2c(=O)c3cccn3c3cccnc32)cc1	nan
	2913061	48285	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	6	1	6	3.8	COc1ccc(C2C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2Cc2cccnc2)cc1	nan
	CHEMBL1556761	48285	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	6	1	6	3.8	COc1ccc(C2C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2Cc2cccnc2)cc1	nan
	4158621	48331	1	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	361	5	1	4	2.9	O=C(CCCN1C(=O)c2cccnc2C1=O)Nc1ccc(F)cc1Cl	nan
	CHEMBL1557087	48331	1	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	361	5	1	4	2.9	O=C(CCCN1C(=O)c2cccnc2C1=O)Nc1ccc(F)cc1Cl	nan
	2448835	48717	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	6	2	9	1.4	CCCn1c(N)c(C(=O)CSc2nc3cc(Cl)c[nH]c-3n2)c(=O)n(C)c1=O	nan
	CHEMBL1560544	48717	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	6	2	9	1.4	CCCn1c(N)c(C(=O)CSc2nc3cc(Cl)c[nH]c-3n2)c(=O)n(C)c1=O	nan
	20921616	48764	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	8	1	8	2.6	COc1ccc(CN(C)S(=O)(=O)c2nnc(NC(=O)c3ccccc3)s2)cc1OC	nan
	CHEMBL1561011	48764	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	8	1	8	2.6	COc1ccc(CN(C)S(=O)(=O)c2nnc(NC(=O)c3ccccc3)s2)cc1OC	nan
	7190686	48939	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	7	1	8	3.3	CCOc1ccccc1NC(=O)CSc1ccc2nnc(-c3cccnc3)n2n1	nan
	CHEMBL1562578	48939	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	7	1	8	3.3	CCOc1ccccc1NC(=O)CSc1ccc2nnc(-c3cccnc3)n2n1	nan
	3152540	48949	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	5	1	5	3.0	O=C(C1=C(O)C(=O)N(CC2CCCO2)C1c1ccccc1)c1ccco1	nan
	CHEMBL1562668	48949	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	5	1	5	3.0	O=C(C1=C(O)C(=O)N(CC2CCCO2)C1c1ccccc1)c1ccco1	nan
	4367682	49357	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	293	1	1	3	2.6	Cc1nc2ccc(Br)cc2c2c1CC(CO)O2	nan
	CHEMBL1566103	49357	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	293	1	1	3	2.6	Cc1nc2ccc(Br)cc2c2c1CC(CO)O2	nan
	1569279	49430	16	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	7	1	6	3.3	CCOC(=O)c1cnc2ccc(Br)cc2c1NCCCN1CCOCC1	nan
	CHEMBL1566690	49430	16	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	7	1	6	3.3	CCOC(=O)c1cnc2ccc(Br)cc2c1NCCCN1CCOCC1	nan
	7881996	49438	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	373	6	1	8	1.2	COc1cccc(C(=O)NCC(=O)OCc2cc(=O)n3ccsc3n2)c1	nan
	CHEMBL1566736	49438	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	373	6	1	8	1.2	COc1cccc(C(=O)NCC(=O)OCc2cc(=O)n3ccsc3n2)c1	nan
	3146574	49503	15	None	-4	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	5	1	8	3.2	COc1ccc(C2C(C(=O)c3ccco3)=C(O)C(=O)N2c2nnc(C)s2)cc1	nan
	CHEMBL1567207	49503	15	None	-4	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	5	1	8	3.2	COc1ccc(C2C(C(=O)c3ccco3)=C(O)C(=O)N2c2nnc(C)s2)cc1	nan
	1226038	49673	14	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	3	0	3	5.3	CC(C)c1ccc(-c2cc(C(=O)N3CCOCC3)c3cc(Br)ccc3n2)cc1	nan
	CHEMBL1568600	49673	14	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	3	0	3	5.3	CC(C)c1ccc(-c2cc(C(=O)N3CCOCC3)c3cc(Br)ccc3n2)cc1	nan
	20904702	49764	3	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	8	1	8	2.1	CCCn1c(=O)c2sccc2n2c(CCCC(=O)NCC3CCCO3)nnc12	nan
	CHEMBL1569451	49764	3	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	8	1	8	2.1	CCCn1c(=O)c2sccc2n2c(CCCC(=O)NCC3CCCO3)nnc12	nan
	16017333	49816	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	5	1	7	1.6	COc1cccc(C(=O)Nc2nnc(S(=O)(=O)N3CCCC3)s2)c1	nan
	CHEMBL1569922	49816	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	5	1	7	1.6	COc1cccc(C(=O)Nc2nnc(S(=O)(=O)N3CCCC3)s2)c1	nan
	1840878	49827	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	5	2	7	1.8	N#C/C(=C\c1c(N2CCC(C(N)=O)CC2)nc2ccccn2c1=O)C(=O)NC1CCCCC1	nan
	CHEMBL1570011	49827	8	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	5	2	7	1.8	N#C/C(=C\c1c(N2CCC(C(N)=O)CC2)nc2ccccn2c1=O)C(=O)NC1CCCCC1	nan
	2134950	49944	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	481	8	1	6	4.0	Cc1cccc(Cn2c(=O)n(CCC(=O)NCCc3ccc(Cl)cc3)c(=O)c3sccc32)c1	nan
	CHEMBL1570886	49944	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	481	8	1	6	4.0	Cc1cccc(Cn2c(=O)n(CCC(=O)NCCc3ccc(Cl)cc3)c(=O)c3sccc32)c1	nan
	16017067	50272	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	5	1	5	4.8	CCC(C(=O)NCc1ccccc1Cl)n1nc(C)c2sc3ccccc3c2c1=O	nan
	CHEMBL1574126	50272	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	5	1	5	4.8	CCC(C(=O)NCc1ccccc1Cl)n1nc(C)c2sc3ccccc3c2c1=O	nan
	860331	50379	2	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	300	4	1	3	3.7	Cc1cc2ccccc2nc1SCC(=O)NC1CCCC1	nan
	CHEMBL1575355	50379	2	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	300	4	1	3	3.7	Cc1cc2ccccc2nc1SCC(=O)NC1CCCC1	nan
	3771682	50469	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	5	1	5	5.4	Cc1cccc(N2C(=O)C(O)=C(C(=O)c3cccs3)C2c2ccc(C(C)C)cc2)n1	nan
	CHEMBL1576217	50469	12	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	5	1	5	5.4	Cc1cccc(N2C(=O)C(O)=C(C(=O)c3cccs3)C2c2ccc(C(C)C)cc2)n1	nan
	20957197	50536	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	6	1	9	2.0	COc1ccc(NC(=O)CCc2nnc3ccc(N4CCC5(CC4)OCCO5)nn23)cc1	nan
	CHEMBL1576697	50536	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	6	1	9	2.0	COc1ccc(NC(=O)CCc2nnc3ccc(N4CCC5(CC4)OCCO5)nn23)cc1	nan
	5738492	50724	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	7	1	6	3.0	COCCCN1C(=O)C(O)=C(C(=O)c2ccc3c(c2)CC(C)O3)C1c1cccnc1	nan
	CHEMBL1578334	50724	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	7	1	6	3.0	COCCCN1C(=O)C(O)=C(C(=O)c2ccc3c(c2)CC(C)O3)C1c1cccnc1	nan
	2503775	50777	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	330	6	1	5	2.3	O=C(CSc1nnc2ccccn12)NCCc1ccc(F)cc1	nan
	CHEMBL1578723	50777	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	330	6	1	5	2.3	O=C(CSc1nnc2ccccn12)NCCc1ccc(F)cc1	nan
	4605879	50799	10	None	-3	3	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	304	4	2	7	2.3	C=CCSc1nc(O)c2c(n1)OC(N)=C(C#N)C2C(C)C	nan
	CHEMBL1578918	50799	10	None	-3	3	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	304	4	2	7	2.3	C=CCSc1nc(O)c2c(n1)OC(N)=C(C#N)C2C(C)C	nan
	2366506	50968	15	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	3	1	6	2.9	O=S(=O)(Nc1nc2ccccc2nc1Cl)c1ccc2c(c1)OCCO2	nan
	CHEMBL1580473	50968	15	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	3	1	6	2.9	O=S(=O)(Nc1nc2ccccc2nc1Cl)c1ccc2c(c1)OCCO2	nan
	135433335	51181	16	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	5	2	7	1.7	O=c1oc2c(CN3CCN(CCO)CC3)c(O)ccc2cc1-c1ccccn1	nan
	1426566	51181	16	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	5	2	7	1.7	O=c1oc2c(CN3CCN(CCO)CC3)c(O)ccc2cc1-c1ccccn1	nan
	CHEMBL1582229	51181	16	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	5	2	7	1.7	O=c1oc2c(CN3CCN(CCO)CC3)c(O)ccc2cc1-c1ccccn1	nan
	5310097	51202	1	None	-4	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	4	1	6	2.7	Cc1ccc(-c2nnc3ccc(SC(C)C(=O)O)nn23)cc1	nan
	CHEMBL1582406	51202	1	None	-4	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	4	1	6	2.7	Cc1ccc(-c2nnc3ccc(SC(C)C(=O)O)nn23)cc1	nan
	4099137	51268	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	500	9	2	6	4.4	O=C(CCCCCn1c(=S)[nH]c2ccc(N3CCOCC3)cc2c1=O)NCc1ccccc1Cl	nan
	CHEMBL1583052	51268	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	500	9	2	6	4.4	O=C(CCCCCn1c(=S)[nH]c2ccc(N3CCOCC3)cc2c1=O)NCc1ccccc1Cl	nan
	661828	51843	14	None	-14	3	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	460	6	1	8	4.5	COc1ccc(OC)c(C2C(C(=O)c3cc4ccccc4o3)=C(O)C(=O)N2c2cc(C)on2)c1	nan
	CHEMBL1587683	51843	14	None	-14	3	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	460	6	1	8	4.5	COc1ccc(OC)c(C2C(C(=O)c3cc4ccccc4o3)=C(O)C(=O)N2c2cc(C)on2)c1	nan
	2004544	51978	16	None	-2	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	4	1	5	4.2	O=C(CSc1ncnc2c1oc1ccccc12)Nc1ccccc1F	nan
	CHEMBL1588950	51978	16	None	-2	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	4	1	5	4.2	O=C(CSc1ncnc2c1oc1ccccc12)Nc1ccccc1F	nan
	1003437	52184	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	3	2	5	5.3	Cc1cc(F)ccc1NC(=O)c1sc2nc(-c3cccs3)ccc2c1N	nan
	CHEMBL1591017	52184	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	3	2	5	5.3	Cc1cc(F)ccc1NC(=O)c1sc2nc(-c3cccs3)ccc2c1N	nan
	16019053	52193	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	9	1	6	4.0	CCCSCCCNC(=O)c1ccc(Cn2c(=O)c3cccn3c3cccnc32)cc1	nan
	CHEMBL1591213	52193	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	9	1	6	4.0	CCCSCCCNC(=O)c1ccc(Cn2c(=O)c3cccn3c3cccnc32)cc1	nan
	16015858	52197	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	396	5	1	4	5.3	O=C(COc1ccccc1Cl)Nc1ccc2oc(-c3ccccc3F)nc2c1	nan
	CHEMBL1591250	52197	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	396	5	1	4	5.3	O=C(COc1ccccc1Cl)Nc1ccc2oc(-c3ccccc3F)nc2c1	nan
	16027414	52255	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	446	6	1	8	3.6	O=C(Nc1ccc(C(=O)OCc2cc(=O)n3nc(C4CC4)sc3n2)cc1)c1ccccc1	nan
	CHEMBL1591957	52255	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	446	6	1	8	3.6	O=C(Nc1ccc(C(=O)OCc2cc(=O)n3nc(C4CC4)sc3n2)cc1)c1ccccc1	nan
	16029938	52301	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	3	1	6	2.8	Cc1ccn2c(=O)c(NC(=O)c3cccc([N+](=O)[O-])c3C)c(C)nc2c1	nan
	CHEMBL1592574	52301	10	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	3	1	6	2.8	Cc1ccn2c(=O)c(NC(=O)c3cccc([N+](=O)[O-])c3C)c(C)nc2c1	nan
	15990931	52321	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	7	2	3	6.1	CC(C)c1ccc(Nc2cc(C(=O)NCCc3ccccc3)c3ccccc3n2)cc1	nan
	CHEMBL1592841	52321	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	7	2	3	6.1	CC(C)c1ccc(Nc2cc(C(=O)NCCc3ccccc3)c3ccccc3n2)cc1	nan
	801483	52438	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	324	3	2	4	5.2	Oc1cccc(-c2nc(-c3cccs3)c(-c3cccs3)[nH]2)c1	nan
	CHEMBL1594404	52438	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	324	3	2	4	5.2	Oc1cccc(-c2nc(-c3cccs3)c(-c3cccs3)[nH]2)c1	nan
	7189836	52632	10	None	-2	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	358	4	1	7	3.3	COc1ccc(C(=O)Nc2nc3cc4c(cc3s2)OCO4)c(OC)c1	nan
	CHEMBL1596046	52632	10	None	-2	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	358	4	1	7	3.3	COc1ccc(C(=O)Nc2nc3cc4c(cc3s2)OCO4)c(OC)c1	nan
	4137685	52678	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	4	1	5	5.8	COc1cccc(C(=O)c2sc3nc(-c4ccccc4)cc(C(F)(F)F)c3c2N)c1	nan
	CHEMBL1596431	52678	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	4	1	5	5.8	COc1cccc(C(=O)c2sc3nc(-c4ccccc4)cc(C(F)(F)F)c3c2N)c1	nan
	3916490	52801	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	8	1	7	2.7	CCN(CC)S(=O)(=O)c1cccc(NC(=O)COc2ncnc3sccc23)c1	nan
	CHEMBL1597614	52801	7	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	8	1	7	2.7	CCN(CC)S(=O)(=O)c1cccc(NC(=O)COc2ncnc3sccc23)c1	nan
	16195124	52995	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	436	7	1	6	2.4	COCCCN1C(=O)C(O)=C(C(=O)c2ccc(OC)cc2)C12C(=O)N(C)c1ccccc12	nan
	CHEMBL1599313	52995	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	436	7	1	6	2.4	COCCCN1C(=O)C(O)=C(C(=O)c2ccc(OC)cc2)C12C(=O)N(C)c1ccccc12	nan
	135419123	53136	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	344	2	1	3	5.5	Cc1ccc(C2=Nc3ccccc3N=C(c3ccc(F)cc3)C2)c(O)c1	nan
	CHEMBL1600651	53136	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	344	2	1	3	5.5	Cc1ccc(C2=Nc3ccccc3N=C(c3ccc(F)cc3)C2)c(O)c1	nan
	16018987	53147	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	482	8	1	7	3.7	COc1ccc(CCNC(=O)c2ccc(Cn3c(=O)c4cccn4c4cccnc43)cc2)cc1OC	nan
	CHEMBL1600729	53147	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	482	8	1	7	3.7	COc1ccc(CCNC(=O)c2ccc(Cn3c(=O)c4cccn4c4cccnc43)cc2)cc1OC	nan
	16009272	53395	1	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	6	1	6	3.2	COc1ccc(CNC(=O)CCc2c(C)nc3c4cccnc4nn3c2C)cc1	nan
	CHEMBL1603189	53395	1	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	6	1	6	3.2	COc1ccc(CNC(=O)CCc2c(C)nc3c4cccnc4nn3c2C)cc1	nan
	2816428	53512	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	256	2	0	5	2.8	C=CCn1c2ccccc2c2nn(C)c(=S)nc21	nan
	CHEMBL1604034	53512	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	256	2	0	5	2.8	C=CCn1c2ccccc2c2nn(C)c(=S)nc21	nan
	3765596	53684	11	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	460	6	1	8	4.5	COc1ccc(C2C(C(=O)c3cc4ccccc4o3)=C(O)C(=O)N2c2cc(C)on2)cc1OC	nan
	CHEMBL1605561	53684	11	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	460	6	1	8	4.5	COc1ccc(C2C(C(=O)c3cc4ccccc4o3)=C(O)C(=O)N2c2cc(C)on2)cc1OC	nan
	4524651	54174	11	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	2	1	5	2.5	CC1CCCCC1NC(=O)c1cc2c(=O)n3ccccc3nc2n1C	nan
	CHEMBL1609461	54174	11	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	2	1	5	2.5	CC1CCCCC1NC(=O)c1cc2c(=O)n3ccccc3nc2n1C	nan
	901441	54185	10	None	-1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	212	1	1	3	3.3	Cc1cc2sc(C(=O)O)c(C)c2s1	nan
	CHEMBL1609556	54185	10	None	-1	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	212	1	1	3	3.3	Cc1cc2sc(C(=O)O)c(C)c2s1	nan
	6498451	54266	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	6	1	9	1.8	COc1cc2c3nc4n(c(=O)c3n(CC(=O)NCC3CCCO3)c2cc1OC)CCS4	nan
	CHEMBL1610295	54266	4	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	6	1	9	1.8	COc1cc2c3nc4n(c(=O)c3n(CC(=O)NCC3CCCO3)c2cc1OC)CCS4	nan
	16022543	54324	11	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	8	2	8	4.1	CCN(CC)CCNC(=O)c1ccc2c(=O)n3nc(Nc4cccc(Cl)c4C)sc3nc2c1	nan
	CHEMBL1610849	54324	11	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	8	2	8	4.1	CCN(CC)CCNC(=O)c1ccc2c(=O)n3nc(Nc4cccc(Cl)c4C)sc3nc2c1	nan
	16013346	54447	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	454	4	1	5	4.2	Cc1cc2oc(C(=O)Nc3ccc(S(=O)(=O)N4CCCCCC4)cc3)cc(=O)c2cc1C	nan
	CHEMBL1611855	54447	9	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	454	4	1	5	4.2	Cc1cc2oc(C(=O)Nc3ccc(S(=O)(=O)N4CCCCCC4)cc3)cc(=O)c2cc1C	nan
	2816611	54511	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	1	2	7	2.8	CCOC(=O)N1CCc2c(sc3nc(S)nc(S)c23)C1	nan
	CHEMBL1612443	54511	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	1	2	7	2.8	CCOC(=O)N1CCc2c(sc3nc(S)nc(S)c23)C1	nan
	2967714	54545	11	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	5	2	3	4.5	COc1ccc(C(=O)Nc2ccc(C(=O)Nc3cccc(C)c3)cc2)cc1	nan
	CHEMBL1612735	54545	11	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	5	2	3	4.5	COc1ccc(C(=O)Nc2ccc(C(=O)Nc3cccc(C)c3)cc2)cc1	nan
	16019073	54583	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	466	8	1	6	4.1	CCOc1ccc(CCNC(=O)c2ccc(Cn3c(=O)c4cccn4c4cccnc43)cc2)cc1	nan
	CHEMBL1613149	54583	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	466	8	1	6	4.1	CCOc1ccc(CCNC(=O)c2ccc(Cn3c(=O)c4cccn4c4cccnc43)cc2)cc1	nan
	4723782	54984	14	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	5	1	3	4.4	Brc1ccc(-c2ccc(CNCc3ccccn3)o2)cc1	nan
	CHEMBL1342613	54984	14	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	5	1	3	4.4	Brc1ccc(-c2ccc(CNCc3ccccn3)o2)cc1	nan
	CHEMBL1618192	54984	14	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	5	1	3	4.4	Brc1ccc(-c2ccc(CNCc3ccccn3)o2)cc1	nan
	20279	55070	95	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	285	2	3	8	-0.3	Nc1nc(Cl)nc2c1ncn2[C@H]1C[C@H](O)[C@@H](CO)O1	nan
	CHEMBL1619	55070	95	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	285	2	3	8	-0.3	Nc1nc(Cl)nc2c1ncn2[C@H]1C[C@H](O)[C@@H](CO)O1	nan
	1712157	55294	11	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	315	6	1	6	1.6	O=C(NCCOC(=O)c1ccc([N+](=O)[O-])cc1)c1cccnc1	nan
	CHEMBL1455081	55294	11	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	315	6	1	6	1.6	O=C(NCCOC(=O)c1ccc([N+](=O)[O-])cc1)c1cccnc1	nan
	CHEMBL1620984	55294	11	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	315	6	1	6	1.6	O=C(NCCOC(=O)c1ccc([N+](=O)[O-])cc1)c1cccnc1	nan
	616262	55432	13	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	233	3	1	5	2.8	CC(=O)c1sc(Nc2ccccn2)nc1C	nan
	CHEMBL1505364	55432	13	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	233	3	1	5	2.8	CC(=O)c1sc(Nc2ccccn2)nc1C	nan
	CHEMBL1622190	55432	13	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	233	3	1	5	2.8	CC(=O)c1sc(Nc2ccccn2)nc1C	nan
	1554378	55864	14	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	6	1	5	3.7	CN(C)CCCNc1ncnc2scc(-c3ccccc3)c12	nan
	CHEMBL1577432	55864	14	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	6	1	5	3.7	CN(C)CCCNc1ncnc2scc(-c3ccccc3)c12	nan
	CHEMBL1625977	55864	14	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	6	1	5	3.7	CN(C)CCCNc1ncnc2scc(-c3ccccc3)c12	nan
	3098134	71744	5	None	-2	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	4	1	7	4.6	C=CCN1C(=O)/C(=C2/Sc3ccc(OC)cc3N2C)S/C1=N\c1cccc(O)c1	nan
	CHEMBL1977502	71744	5	None	-2	2	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	4	1	7	4.6	C=CCN1C(=O)/C(=C2/Sc3ccc(OC)cc3N2C)S/C1=N\c1cccc(O)c1	nan
	9687993	107317	3	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	4	1	6	2.7	C/C(=N\NC(=O)c1c(C)nc2ccccn12)c1cccc([N+](=O)[O-])c1	nan
	CHEMBL3191955	107317	3	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	4	1	6	2.7	C/C(=N\NC(=O)c1c(C)nc2ccccn12)c1cccc([N+](=O)[O-])c1	nan
	3095208	107506	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	293	3	2	4	2.6	O=C1C=C(Nc2ccccc2C(=O)O)c2ccccc2C1=O	nan
	CHEMBL3194086	107506	5	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	293	3	2	4	2.6	O=C1C=C(Nc2ccccc2C(=O)O)c2ccccc2C1=O	nan
	9638310	107686	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	285	4	1	6	1.5	C/C(=N\NC(=O)c1cnccn1)c1ccc([N+](=O)[O-])cc1	nan
	CHEMBL3196238	107686	6	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	285	4	1	6	1.5	C/C(=N\NC(=O)c1cnccn1)c1ccc([N+](=O)[O-])cc1	nan
	102175	140741	66	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	281	3	4	9	-1.5	CNc1ncnc2c1ncn2[C@@H]1O[C@H](CO)[C@@H](O)[C@H]1O	nan
	CHEMBL383144	140741	66	None	-	1	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	281	3	4	9	-1.5	CNc1ncnc2c1ncn2[C@@H]1O[C@H](CO)[C@@H](O)[C@H]1O	nan
	6083	203107	90	None	-44	6	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	347	4	5	10	-1.9	Nc1ncnc2c1ncn2[C@@H]1O[C@H](COP(=O)(O)O)[C@@H](O)[C@H]1O	nan
	CHEMBL1315633	203107	90	None	-44	6	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	347	4	5	10	-1.9	Nc1ncnc2c1ncn2[C@@H]1O[C@H](COP(=O)(O)O)[C@@H](O)[C@H]1O	nan
	CHEMBL752	203107	90	None	-44	6	Human	4.7	pPotency	=	4.7	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	347	4	5	10	-1.9	Nc1ncnc2c1ncn2[C@@H]1O[C@H](COP(=O)(O)O)[C@@H](O)[C@H]1O	nan
	4324298	28415	7	None	-	1	Human	5.6	pPotency	=	5.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	7	1	8	0.9	CCN(CC)S(=O)(=O)c1ccc(N2CCOCC2)c(NC(=O)c2ccc(=O)n(C)n2)c1	nan
	CHEMBL1377104	28415	7	None	-	1	Human	5.6	pPotency	=	5.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	7	1	8	0.9	CCN(CC)S(=O)(=O)c1ccc(N2CCOCC2)c(NC(=O)c2ccc(=O)n(C)n2)c1	nan
	15988970	43807	6	None	-	1	Human	5.6	pPotency	=	5.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	5	1	3	6.2	CCc1ccc(CNC(=O)c2cc(-c3ccc(Br)s3)nc3ccccc23)cc1	nan
	CHEMBL1514445	43807	6	None	-	1	Human	5.6	pPotency	=	5.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	5	1	3	6.2	CCc1ccc(CNC(=O)c2cc(-c3ccc(Br)s3)nc3ccccc23)cc1	nan
	15988960	48260	6	None	-	1	Human	5.6	pPotency	=	5.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	5	1	3	5.5	CC(C)CCNC(=O)c1cc(-c2ccc(Br)s2)nc2ccccc12	nan
	CHEMBL1556439	48260	6	None	-	1	Human	5.6	pPotency	=	5.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	5	1	3	5.5	CC(C)CCNC(=O)c1cc(-c2ccc(Br)s2)nc2ccccc12	nan
	3119935	52425	19	None	-	1	Human	5.6	pPotency	=	5.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	7	2	6	3.7	CCOc1ccccc1C(=O)Nc1ccc(S(=O)(=O)Nc2onc(C)c2C)cc1	nan
	CHEMBL1594298	52425	19	None	-	1	Human	5.6	pPotency	=	5.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	7	2	6	3.7	CCOc1ccccc1C(=O)Nc1ccc(S(=O)(=O)Nc2onc(C)c2C)cc1	nan
	735254	10359	77	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	178	1	1	3	2.4	S=c1[nH]nc(-c2ccccc2)o1	nan
	CHEMBL1164316	10359	77	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	178	1	1	3	2.4	S=c1[nH]nc(-c2ccccc2)o1	nan
	5904441	11246	12	None	-6	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	280	3	1	5	3.1	N#C/C(=C\c1ccc([N+](=O)[O-])o1)c1nc2ccccc2[nH]1	nan
	CHEMBL117966	11246	12	None	-6	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	280	3	1	5	3.1	N#C/C(=C\c1ccc([N+](=O)[O-])o1)c1nc2ccccc2[nH]1	nan
	1004068	18178	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	423	5	2	5	5.1	COc1ccc(-c2ccc3c(N)c(C(=O)NCc4ccc(Cl)cc4)sc3n2)cc1	nan
	CHEMBL1271076	18178	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	423	5	2	5	5.1	COc1ccc(-c2ccc3c(N)c(C(=O)NCc4ccc(Cl)cc4)sc3n2)cc1	nan
	3626929	19342	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	6	1	5	3.7	CC(=O)c1ccc(NC(=O)C(=O)c2cn(CC(=O)N3CCCCC3)c3ccccc23)cc1	nan
	CHEMBL1299573	19342	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	6	1	5	3.7	CC(=O)c1ccc(NC(=O)C(=O)c2cn(CC(=O)N3CCCCC3)c3ccccc23)cc1	nan
	5852174	19432	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	6	1	7	4.0	COC(=O)c1ccc(C2C(C(=O)c3ccc4c(c3)CC(C)O4)=C(O)C(=O)N2Cc2cccnc2)cc1	nan
	CHEMBL1300425	19432	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	6	1	7	4.0	COC(=O)c1ccc(C2C(C(=O)c3ccc4c(c3)CC(C)O4)=C(O)C(=O)N2Cc2cccnc2)cc1	nan
	15988009	19511	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	9	1	9	2.3	COc1ccc(OC)c(CCNC(=O)CCCc2nnc3n(C)c(=O)c4sccc4n23)c1	nan
	CHEMBL1300978	19511	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	9	1	9	2.3	COc1ccc(OC)c(CCNC(=O)CCCc2nnc3n(C)c(=O)c4sccc4n23)c1	nan
	3688325	19602	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	3	2	6	2.9	CC(=O)Nc1cccc(C2=CC(c3ccco3)n3ncnc3N2)c1	nan
	CHEMBL1301688	19602	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	3	2	6	2.9	CC(=O)Nc1cccc(C2=CC(c3ccco3)n3ncnc3N2)c1	nan
	20957233	19642	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	7	1	8	2.3	CC(CNC(=O)CCc1nnc2ccc(N3CCC4(CC3)OCCO4)nn12)c1ccccc1	nan
	CHEMBL1302111	19642	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	7	1	8	2.3	CC(CNC(=O)CCc1nnc2ccc(N3CCC4(CC3)OCCO4)nn12)c1ccccc1	nan
	17584169	19755	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	4	1	5	3.3	O=C(COc1cc2oc(=O)c3c(c2cc1Cl)CCC3)Nc1ccccn1	nan
	CHEMBL1302915	19755	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	4	1	5	3.3	O=C(COc1cc2oc(=O)c3c(c2cc1Cl)CCC3)Nc1ccccn1	nan
	852288	19918	25	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	243	1	1	5	0.9	Cn1c(C(=O)O)cc2c(=O)n3ccccc3nc21	nan
	CHEMBL1304220	19918	25	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	243	1	1	5	0.9	Cn1c(C(=O)O)cc2c(=O)n3ccccc3nc21	nan
	4145244	19927	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	6	1	8	0.6	Cn1cnnc1SCC(=O)Nc1cccc(S(=O)(=O)N2CCOCC2)c1	nan
	CHEMBL1304271	19927	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	6	1	8	0.6	Cn1cnnc1SCC(=O)Nc1cccc(S(=O)(=O)N2CCOCC2)c1	nan
	2429052	20027	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	488	6	1	5	5.8	O=C(COC(=O)CSc1cccc2cccc(Cl)c12)Nc1ncc(C(F)(F)F)cc1Cl	nan
	CHEMBL1305188	20027	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	488	6	1	5	5.8	O=C(COC(=O)CSc1cccc2cccc(Cl)c12)Nc1ncc(C(F)(F)F)cc1Cl	nan
	353380	20197	2	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	2	2	2	5.7	O=C(Nc1ccc(Br)c2ccccc12)c1ccc2ccccc2c1O	nan
	CHEMBL1306524	20197	2	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	2	2	2	5.7	O=C(Nc1ccc(Br)c2ccccc12)c1ccc2ccccc2c1O	nan
	4300736	20325	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	3	2	7	2.0	NS(=O)(=O)c1ccc2nc(NC(=O)c3ccc4c(c3)OCCO4)sc2c1	nan
	CHEMBL1307550	20325	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	3	2	7	2.0	NS(=O)(=O)c1ccc2nc(NC(=O)c3ccc4c(c3)OCCO4)sc2c1	nan
	16194293	20357	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	363	6	1	8	3.4	CCc1nnc(NC(=O)CSc2ccc(-c3cccs3)nn2)s1	nan
	CHEMBL1307806	20357	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	363	6	1	8	3.4	CCc1nnc(NC(=O)CSc2ccc(-c3cccs3)nn2)s1	nan
	24819826	20382	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	6	2	3	4.1	O=C(NCCCSc1ccccc1)c1cc(Br)ccc1O	nan
	CHEMBL1307980	20382	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	6	2	3	4.1	O=C(NCCCSc1ccccc1)c1cc(Br)ccc1O	nan
	713805	20438	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	303	4	0	9	0.6	COc1nc(N2CCCC2)nc(-n2nnc(C(C)=O)c2C)n1	nan
	CHEMBL1308437	20438	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	303	4	0	9	0.6	COc1nc(N2CCCC2)nc(-n2nnc(C(C)=O)c2C)n1	nan
	935829	20456	17	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	315	3	0	4	3.3	Cc1nc2ccccc2nc1SCC(=O)N1CCC(C)CC1	nan
	CHEMBL1308605	20456	17	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	315	3	0	4	3.3	Cc1nc2ccccc2nc1SCC(=O)N1CCC(C)CC1	nan
	2815890	20501	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	296	3	5	10	-1.9	CNc1nc2c(N)ncnc2n1[C@H]1O[C@@H](CO)[C@H](O)[C@@H]1O	nan
	CHEMBL1308946	20501	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	296	3	5	10	-1.9	CNc1nc2c(N)ncnc2n1[C@H]1O[C@@H](CO)[C@H](O)[C@@H]1O	nan
	4619601	20508	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	4	0	7	2.2	CCN(C(=O)CSC1=Nc2ccccc2C2CC=NN12)C1CCS(=O)(=O)C1	nan
	CHEMBL1309010	20508	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	4	0	7	2.2	CCN(C(=O)CSC1=Nc2ccccc2C2CC=NN12)C1CCS(=O)(=O)C1	nan
	4038913	20601	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	530	6	0	6	3.9	CCN(C(=O)COC(=O)c1cc(-c2ccccc2)nc2ccc(Br)cc12)C1CCS(=O)(=O)C1	nan
	CHEMBL1309767	20601	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	530	6	0	6	3.9	CCN(C(=O)COC(=O)c1cc(-c2ccccc2)nc2ccc(Br)cc12)C1CCS(=O)(=O)C1	nan
	20923170	20698	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	6	1	6	2.7	COc1ccc(CN2C(=O)c3cccnc3C2=O)cc1S(=O)(=O)NC1CCCCC1C	nan
	CHEMBL1310648	20698	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	6	1	6	2.7	COc1ccc(CN2C(=O)c3cccnc3C2=O)cc1S(=O)(=O)NC1CCCCC1C	nan
	3163618	20735	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	5	1	6	3.6	Cc1ccc(NC(=O)CSc2nnc(-c3ccncc3)s2)cc1	nan
	CHEMBL1310953	20735	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	5	1	6	3.6	Cc1ccc(NC(=O)CSc2nnc(-c3ccncc3)s2)cc1	nan
	1504615	20784	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	325	5	1	6	2.0	Cc1cc(CNC(=O)Cn2cc([N+](=O)[O-])cn2)c2ccccc2n1	nan
	CHEMBL1311384	20784	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	325	5	1	6	2.0	Cc1cc(CNC(=O)Cn2cc([N+](=O)[O-])cn2)c2ccccc2n1	nan
	652682	20843	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	8	1	6	4.3	C=CCOc1cccc(C2C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2Cc2ccncc2)c1	nan
	CHEMBL1311808	20843	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	8	1	6	4.3	C=CCOc1cccc(C2C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2Cc2ccncc2)c1	nan
	24892134	20860	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	5	1	8	2.7	Cn1c(=O)c2c(SCC(=O)Nc3ccccc3F)nc(-c3ccccc3F)nc2n(C)c1=O	nan
	CHEMBL1311956	20860	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	5	1	8	2.7	Cn1c(=O)c2c(SCC(=O)Nc3ccccc3F)nc(-c3ccccc3F)nc2n(C)c1=O	nan
	2769005	21033	15	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	279	4	0	7	1.1	CCOC(=O)CSc1nc(=O)n2cc(C)ccc2n1	nan
	CHEMBL1313156	21033	15	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	279	4	0	7	1.1	CCOC(=O)CSc1nc(=O)n2cc(C)ccc2n1	nan
	20914264	21036	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	6	1	6	1.9	O=C1c2cccnc2C(=O)N1Cc1ccc(S(=O)(=O)NCc2ccco2)cc1	nan
	CHEMBL1313185	21036	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	6	1	6	1.9	O=C1c2cccnc2C(=O)N1Cc1ccc(S(=O)(=O)NCc2ccco2)cc1	nan
	4002385	21059	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	7	1	6	4.2	CC(C)Oc1ccc(C2C(C(=O)c3ccco3)=C(O)C(=O)N2Cc2cccnc2)cc1	nan
	662194	21059	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	7	1	6	4.2	CC(C)Oc1ccc(C2C(C(=O)c3ccco3)=C(O)C(=O)N2Cc2cccnc2)cc1	nan
	CHEMBL1313374	21059	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	7	1	6	4.2	CC(C)Oc1ccc(C2C(C(=O)c3ccco3)=C(O)C(=O)N2Cc2cccnc2)cc1	nan
	16033288	21184	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	5	1	5	5.3	Cc1ccc(C)c(CNC(=O)c2sc3ncnc(N(C)C4CCCCC4)c3c2C)c1	nan
	CHEMBL1314411	21184	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	5	1	5	5.3	Cc1ccc(C)c(CNC(=O)c2sc3ncnc(N(C)C4CCCCC4)c3c2C)c1	nan
	1046209	21252	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	465	2	1	8	2.8	Cn1c(=O)c2c(nc3n(-c4ccc(O)cc4)c(-c4ccc(Br)cc4)cn23)n(C)c1=O	nan
	CHEMBL1315398	21252	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	465	2	1	8	2.8	Cn1c(=O)c2c(nc3n(-c4ccc(O)cc4)c(-c4ccc(Br)cc4)cn23)n(C)c1=O	nan
	16014663	21263	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	6	1	6	3.8	COc1ccc(-c2nsc(NC(=O)COc3ccc(C)c(C)c3)n2)cc1	nan
	CHEMBL1315498	21263	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	6	1	6	3.8	COc1ccc(-c2nsc(NC(=O)COc3ccc(C)c(C)c3)n2)cc1	nan
	16017636	21311	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	489	5	2	8	4.3	COc1ccc(NC(=O)c2sc3nc(-c4cc5ccc(OC)cc5oc4=O)[nH]c(=O)c3c2C)cc1	nan
	CHEMBL1316057	21311	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	489	5	2	8	4.3	COc1ccc(NC(=O)c2sc3nc(-c4cc5ccc(OC)cc5oc4=O)[nH]c(=O)c3c2C)cc1	nan
	16018724	21317	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	5	1	7	4.2	COc1ccc(Cl)cc1NC(=O)CSc1nnc(C)n2c1cc1occc12	nan
	CHEMBL1316127	21317	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	5	1	7	4.2	COc1ccc(Cl)cc1NC(=O)CSc1nnc(C)n2c1cc1occc12	nan
	16009825	21370	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	491	7	1	9	3.7	COc1cc(NC(=O)Cn2c(=O)n(Cc3ccco3)c(=O)c3sc4ccccc4c32)cc(OC)c1	nan
	CHEMBL1316937	21370	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	491	7	1	9	3.7	COc1cc(NC(=O)Cn2c(=O)n(Cc3ccco3)c(=O)c3sc4ccccc4c32)cc(OC)c1	nan
	24980344	21373	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	6	1	5	3.0	Cc1ccc(C(=O)NCC(=O)OCC(=O)c2ccc(Br)s2)cc1	nan
	CHEMBL1316966	21373	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	6	1	5	3.0	Cc1ccc(C(=O)NCC(=O)OCC(=O)c2ccc(Br)s2)cc1	nan
	7159295	21392	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	356	6	1	9	-0.3	CCOC(=O)CNC(=O)Cn1cnc2c(nnn2-c2ccccc2)c1=O	nan
	CHEMBL1317213	21392	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	356	6	1	9	-0.3	CCOC(=O)CNC(=O)Cn1cnc2c(nnn2-c2ccccc2)c1=O	nan
	17757011	21397	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	2	1	4	5.3	O=C1COc2ccc(-c3cc(-c4ccccc4)c4c(n3)-c3ccccc3OC4)cc2N1	nan
	CHEMBL1317304	21397	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	2	1	4	5.3	O=C1COc2ccc(-c3cc(-c4ccccc4)c4c(n3)-c3ccccc3OC4)cc2N1	nan
	1215486	21398	17	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	5	1	5	5.6	N#Cc1c(C(F)(F)F)cc(-c2cccs2)nc1SCC(=O)Nc1ccc(F)cc1	nan
	CHEMBL1317307	21398	17	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	5	1	5	5.6	N#Cc1c(C(F)(F)F)cc(-c2cccs2)nc1SCC(=O)Nc1ccc(F)cc1	nan
	4318326	21551	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	7	1	6	3.1	COc1ccc2nc(C)cc(SCC(NC(C)=O)C(=O)OC(C)C)c2c1	nan
	CHEMBL1318910	21551	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	7	1	6	3.1	COc1ccc2nc(C)cc(SCC(NC(C)=O)C(=O)OC(C)C)c2c1	nan
	621902	21555	10	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	292	5	0	5	3.5	CCSc1cnn(-c2ccccc2)c(=O)c1SCC	nan
	CHEMBL1318957	21555	10	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	292	5	0	5	3.5	CCSc1cnn(-c2ccccc2)c(=O)c1SCC	nan
	3152777	21681	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	446	4	2	7	5.0	Cc1ccc2nc(N3C(=O)C(O)=C(C(=O)c4ccc(C)o4)C3c3cccc(O)c3)sc2c1	nan
	CHEMBL1320029	21681	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	446	4	2	7	5.0	Cc1ccc2nc(N3C(=O)C(O)=C(C(=O)c4ccc(C)o4)C3c3cccc(O)c3)sc2c1	nan
	15990516	21801	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	396	5	1	4	5.1	COc1ccc2nc3sc(C(=O)NCCc4ccc(Cl)cc4)cc3cc2c1	nan
	CHEMBL1321040	21801	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	396	5	1	4	5.1	COc1ccc2nc3sc(C(=O)NCCc4ccc(Cl)cc4)cc3cc2c1	nan
	2158383	22030	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	331	6	1	6	2.1	CCOCCCNC(=O)c1cc2c(=O)n3ccccc3nc2s1	nan
	CHEMBL1323129	22030	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	331	6	1	6	2.1	CCOCCCNC(=O)c1cc2c(=O)n3ccccc3nc2s1	nan
	864393	22090	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	4	1	3	4.1	Cc1cc(SCC(=O)NC2CCCCC2)nc2ccccc12	nan
	CHEMBL1323679	22090	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	4	1	3	4.1	Cc1cc(SCC(=O)NC2CCCCC2)nc2ccccc12	nan
	2138908	22118	18	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	4	1	4	5.0	CCOC(=O)c1ccc(NC(=O)c2sc3ccccc3c2Cl)cc1	nan
	CHEMBL1323878	22118	18	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	4	1	4	5.0	CCOC(=O)c1ccc(NC(=O)c2sc3ccccc3c2Cl)cc1	nan
	716947	22173	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	296	3	1	4	3.9	CCOc1ccc(-c2oc3ccc(C)cc3c(=O)c2O)cc1	nan
	CHEMBL1324368	22173	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	296	3	1	4	3.9	CCOc1ccc(-c2oc3ccc(C)cc3c(=O)c2O)cc1	nan
	2929091	22182	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	4	2	7	2.2	N=c1c(C(=O)NCC2CCCO2)cc2c(=O)n3ccccc3nc2n1C1CCCC1	nan
	CHEMBL1324435	22182	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	4	2	7	2.2	N=c1c(C(=O)NCC2CCCO2)cc2c(=O)n3ccccc3nc2n1C1CCCC1	nan
	16017079	22204	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	479	4	1	5	6.2	CCC(C(=O)Nc1cc(C(F)(F)F)ccc1Cl)n1nc(C)c2sc3ccccc3c2c1=O	nan
	CHEMBL1324580	22204	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	479	4	1	5	6.2	CCC(C(=O)Nc1cc(C(F)(F)F)ccc1Cl)n1nc(C)c2sc3ccccc3c2c1=O	nan
	6619868	22237	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	467	7	2	5	3.4	NS(=O)(=O)c1ccc(CCNC(=O)c2ccc3c(c2)N(Cc2ccccc2)CCS3)cc1	nan
	CHEMBL1324841	22237	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	467	7	2	5	3.4	NS(=O)(=O)c1ccc(CCNC(=O)c2ccc3c(c2)N(Cc2ccccc2)CCS3)cc1	nan
	135415532	22311	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	351	3	1	7	2.6	Cc1cc(O)nc(SCc2nc3ncccn3c2Br)n1	nan
	CHEMBL1325556	22311	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	351	3	1	7	2.6	Cc1cc(O)nc(SCc2nc3ncccn3c2Br)n1	nan
	1086445	22434	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	5	2	6	3.7	COc1ccc(-c2ccc3c(N)c(C(=O)NC(C)C)sc3n2)cc1OC	nan
	CHEMBL1326816	22434	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	5	2	6	3.7	COc1ccc(-c2ccc3c(N)c(C(=O)NC(C)C)sc3n2)cc1OC	nan
	5739163	22492	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	492	5	1	6	4.4	O=C(C1=C(O)C(=O)N(Cc2cccnc2)C1c1cccc(Br)c1)c1ccc2c(c1)OCO2	nan
	CHEMBL1327274	22492	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	492	5	1	6	4.4	O=C(C1=C(O)C(=O)N(Cc2cccnc2)C1c1cccc(Br)c1)c1ccc2c(c1)OCO2	nan
	2128134	22515	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	5	0	5	2.3	CN(C)S(=O)(=O)c1cccc(COC(=O)c2cccnc2Cl)c1	nan
	CHEMBL1327541	22515	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	5	0	5	2.3	CN(C)S(=O)(=O)c1cccc(COC(=O)c2cccnc2Cl)c1	nan
	5899385	22572	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	7	1	7	3.3	CC1Cc2cc(C(=O)C3=C(O)C(=O)N(CCCn4ccnc4)C3c3cccnc3)ccc2O1	nan
	CHEMBL1327895	22572	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	7	1	7	3.3	CC1Cc2cc(C(=O)C3=C(O)C(=O)N(CCCn4ccnc4)C3c3cccnc3)ccc2O1	nan
	3464558	22606	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	491	6	1	5	3.3	COc1ccc(S(=O)(=O)N2CCN(CC(=O)Nc3ccc(Cl)c(C(F)(F)F)c3)CC2)cc1	nan
	CHEMBL1328124	22606	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	491	6	1	5	3.3	COc1ccc(S(=O)(=O)N2CCN(CC(=O)Nc3ccc(Cl)c(C(F)(F)F)c3)CC2)cc1	nan
	1779937	22771	11	None	-3	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	281	1	1	4	4.3	COc1ccc2sc3c(O)nc4ccccc4c3c2c1	nan
	CHEMBL1329604	22771	11	None	-3	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	281	1	1	4	4.3	COc1ccc2sc3c(O)nc4ccccc4c3c2c1	nan
	16013718	22893	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	3	1	5	3.7	CCc1nonc1NC(=O)c1oc2ccc(Br)cc2c1C	nan
	CHEMBL1330644	22893	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	3	1	5	3.7	CCc1nonc1NC(=O)c1oc2ccc(Br)cc2c1C	nan
	2991043	23099	15	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	5	1	8	0.4	Cn1c(=O)c2c(nc(CN3CCc4ccccc4C3)n2CCCO)n(C)c1=O	nan
	CHEMBL1332170	23099	15	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	5	1	8	0.4	Cn1c(=O)c2c(nc(CN3CCc4ccccc4C3)n2CCCO)n(C)c1=O	nan
	1861856	23172	13	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	4	2	6	2.5	COc1cc2[nH]c(=S)n(NC(=O)c3ccccc3)c(=O)c2cc1OC	nan
	CHEMBL1332727	23172	13	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	4	2	6	2.5	COc1cc2[nH]c(=S)n(NC(=O)c3ccccc3)c(=O)c2cc1OC	nan
	5302228	23542	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	4	0	6	3.3	COc1ccc(N(C)S(=O)(=O)c2ccc3c(c2)c(=O)nc2ccc(Cl)cn23)cc1	nan
	CHEMBL1335569	23542	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	4	0	6	3.3	COc1ccc(N(C)S(=O)(=O)c2ccc3c(c2)c(=O)nc2ccc(Cl)cn23)cc1	nan
	16018981	23621	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	442	5	1	5	4.3	O=C(NCc1ccccc1Cl)c1ccc(Cn2c(=O)c3cccn3c3cccnc32)cc1	nan
	CHEMBL1336206	23621	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	442	5	1	5	4.3	O=C(NCc1ccccc1Cl)c1ccc(Cn2c(=O)c3cccn3c3cccnc32)cc1	nan
	2807849	23643	64	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	217	2	1	3	3.2	CC(=O)c1sc(-c2ccccc2)cc1N	nan
	CHEMBL1336437	23643	64	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	217	2	1	3	3.2	CC(=O)c1sc(-c2ccccc2)cc1N	nan
	2222525	23663	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	4	1	7	3.0	CC(=O)c1sc2nc(SCC(=O)N3CCCCC3)nc(O)c2c1C	nan
	CHEMBL1336564	23663	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	4	1	7	3.0	CC(=O)c1sc2nc(SCC(=O)N3CCCCC3)nc(O)c2c1C	nan
	2844395	23722	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	239	4	2	3	1.3	CC(C)NC(=O)CC(=O)NN=C1CCCCC1	nan
	CHEMBL1337153	23722	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	239	4	2	3	1.3	CC(C)NC(=O)CC(=O)NN=C1CCCCC1	nan
	1480701	23834	17	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	344	3	0	7	2.0	COC(=O)c1nc2ccc(N3CCOCC3)cc2c(C)c1C(=O)OC	nan
	CHEMBL1338156	23834	17	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	344	3	0	7	2.0	COC(=O)c1nc2ccc(N3CCOCC3)cc2c(C)c1C(=O)OC	nan
	861738	23872	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	300	4	1	3	3.7	Cc1cc(SCC(=O)NC2CCCC2)nc2ccccc12	nan
	CHEMBL1338383	23872	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	300	4	1	3	3.7	Cc1cc(SCC(=O)NC2CCCC2)nc2ccccc12	nan
	4677074	24238	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	200	0	1	3	2.8	Sc1nc2ccccc2n2cccc12	nan
	CHEMBL1341748	24238	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	200	0	1	3	2.8	Sc1nc2ccccc2n2cccc12	nan
	2334933	24308	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	6	1	4	3.5	O=C(COC(=O)CSc1ccc2ccccc2c1Br)NC1CC1	nan
	CHEMBL1342297	24308	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	6	1	4	3.5	O=C(COC(=O)CSc1ccc2ccccc2c1Br)NC1CC1	nan
	650550	24373	1	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	3	0	6	3.4	COc1ccc(-c2nsc3c(N4CCCC4)ncnc23)cc1	nan
	CHEMBL1342739	24373	1	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	3	0	6	3.4	COc1ccc(-c2nsc3c(N4CCCC4)ncnc23)cc1	nan
	16445815	24534	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	5	1	8	3.8	CSc1nnc(N2C(=O)C(O)=C(C(=O)c3ccco3)C2c2ccc(F)cc2)s1	nan
	CHEMBL1344160	24534	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	5	1	8	3.8	CSc1nnc(N2C(=O)C(O)=C(C(=O)c3ccco3)C2c2ccc(F)cc2)s1	nan
	7190688	24560	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	7	1	8	3.3	CCOc1ccc(NC(=O)CSc2ccc3nnc(-c4cccnc4)n3n2)cc1	nan
	CHEMBL1344377	24560	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	7	1	8	3.3	CCOc1ccc(NC(=O)CSc2ccc3nnc(-c4cccnc4)n3n2)cc1	nan
	3106500	24585	8	None	1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	306	3	1	7	1.5	CC1=NN(C(N)=S)C(=O)C1N=Nc1ccc([N+](=O)[O-])cc1	nan
	CHEMBL1344603	24585	8	None	1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	306	3	1	7	1.5	CC1=NN(C(N)=S)C(=O)C1N=Nc1ccc([N+](=O)[O-])cc1	nan
	20907339	24644	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	6	1	5	2.6	CCOCCCNC(=O)c1cn2c3c(ccc(Cl)c3c1=O)OC(C)C2	nan
	CHEMBL1345074	24644	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	6	1	5	2.6	CCOCCCNC(=O)c1cn2c3c(ccc(Cl)c3c1=O)OC(C)C2	nan
	6103434	24784	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	506	9	1	7	3.7	CCCOc1cccc(C2C(C(=O)c3ccc4c(c3)CC(C)O4)=C(O)C(=O)N2CCN2CCOCC2)c1	nan
	CHEMBL1346374	24784	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	506	9	1	7	3.7	CCCOc1cccc(C2C(C(=O)c3ccc4c(c3)CC(C)O4)=C(O)C(=O)N2CCN2CCOCC2)c1	nan
	2122298	24919	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	290	5	1	5	2.7	CC(=O)c1sc(NC(=O)COc2ccccc2)nc1C	nan
	CHEMBL1347404	24919	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	290	5	1	5	2.7	CC(=O)c1sc(NC(=O)COc2ccccc2)nc1C	nan
	899068	24967	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	298	1	1	6	3.6	CSc1nc(S)c2c3c(sc2n1)COC(C)(C)C3	nan
	CHEMBL1347767	24967	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	298	1	1	6	3.6	CSc1nc(S)c2c3c(sc2n1)COC(C)(C)C3	nan
	1481616	25033	18	None	-15	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	309	5	0	4	4.3	COc1cccc(CSc2nc3ccccc3cc2C=O)c1	nan
	CHEMBL1348389	25033	18	None	-15	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	309	5	0	4	4.3	COc1cccc(CSc2nc3ccccc3cc2C=O)c1	nan
	1378026	25053	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	7	1	5	4.2	COc1ccc(NC(=O)c2ccc(C(=O)c3cc(OC)ccc3OC)cc2)cc1	nan
	CHEMBL1348606	25053	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	7	1	5	4.2	COc1ccc(NC(=O)c2ccc(C(=O)c3cc(OC)ccc3OC)cc2)cc1	nan
	2205361	25056	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	503	4	3	9	2.3	COC(=O)c1sc(N=C(S)NNC(=O)c2c(Br)c(C)nn2C)c(C(=O)OC)c1C	nan
	CHEMBL1348642	25056	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	503	4	3	9	2.3	COC(=O)c1sc(N=C(S)NNC(=O)c2c(Br)c(C)nn2C)c(C(=O)OC)c1C	nan
	2084877	25070	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	8	1	5	3.8	COCCNC(=O)CSc1cc(-c2ccccc2)c2ccc(OC)cc2n1	nan
	CHEMBL1348812	25070	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	8	1	5	3.8	COCCNC(=O)CSc1cc(-c2ccccc2)c2ccc(OC)cc2n1	nan
	1256964	25076	11	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	423	4	1	4	5.1	O=C(NCc1cccs1)c1cc(-c2ccccn2)nc2ccc(Br)cc12	nan
	CHEMBL1348841	25076	11	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	423	4	1	4	5.1	O=C(NCc1cccs1)c1cc(-c2ccccn2)nc2ccc(Br)cc12	nan
	3783556	25156	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	5	2	7	1.0	C=CCN1C(=O)NC(=O)/C(=C\Nc2c(C)n(C)n(-c3ccccc3)c2=O)C1=O	nan
	CHEMBL1349443	25156	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	5	2	7	1.0	C=CCN1C(=O)NC(=O)/C(=C\Nc2c(C)n(C)n(-c3ccccc3)c2=O)C1=O	nan
	24746879	25169	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	6	0	6	3.5	COC(=O)CSc1nc(COc2ccccc2)nc2ccccc12	nan
	CHEMBL1349543	25169	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	6	0	6	3.5	COC(=O)CSc1nc(COc2ccccc2)nc2ccccc12	nan
	4831863	25249	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	6	1	9	0.5	COc1ccc(S(=O)(=O)N2CCOCC2)cc1NC(=O)Cn1nnc2ccccc2c1=O	nan
	CHEMBL1350232	25249	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	6	1	9	0.5	COc1ccc(S(=O)(=O)N2CCOCC2)cc1NC(=O)Cn1nnc2ccccc2c1=O	nan
	663661	25285	16	None	1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	332	3	1	5	4.5	c1ccc2[nH]c(CSc3ncnc4c3oc3ccccc34)nc2c1	nan
	CHEMBL1350581	25285	16	None	1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	332	3	1	5	4.5	c1ccc2[nH]c(CSc3ncnc4c3oc3ccccc34)nc2c1	nan
	2881707	25414	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	348	3	1	5	3.2	Cc1nnc(Nc2ccc(C(=O)N3CCOCC3)cc2)c2ccccc12	nan
	CHEMBL1351647	25414	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	348	3	1	5	3.2	Cc1nnc(Nc2ccc(C(=O)N3CCOCC3)cc2)c2ccccc12	nan
	5308898	25431	54	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	204	1	1	3	2.4	CCc1cc(=O)oc2cc(C)cc(O)c12	nan
	CHEMBL1351746	25431	54	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	204	1	1	3	2.4	CCc1cc(=O)oc2cc(C)cc(O)c12	nan
	2802516	25486	41	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	253	2	1	4	3.2	Sc1nc(-c2ccccc2)n(-c2ccccc2)n1	nan
	CHEMBL1352266	25486	41	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	253	2	1	4	3.2	Sc1nc(-c2ccccc2)n(-c2ccccc2)n1	nan
	1435022	25576	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	5	1	6	4.3	CCc1nc(SCC(=O)Nc2nc3c(s2)CCCC3)c2ccccc2n1	nan
	CHEMBL1352936	25576	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	5	1	6	4.3	CCc1nc(SCC(=O)Nc2nc3c(s2)CCCC3)c2ccccc2n1	nan
	7285290	25610	19	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	291	2	1	2	3.5	Cc1nc(-c2ccc(Br)cc2)ccc1C(=O)O	nan
	CHEMBL1353200	25610	19	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	291	2	1	2	3.5	Cc1nc(-c2ccc(Br)cc2)ccc1C(=O)O	nan
	15989677	25772	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	539	9	1	9	3.5	COc1cc(NC(=O)Cn2c(=O)n(Cc3ccccc3Cl)c(=O)c3cc(OC)c(OC)cc32)cc(OC)c1	nan
	CHEMBL1354335	25772	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	539	9	1	9	3.5	COc1cc(NC(=O)Cn2c(=O)n(Cc3ccccc3Cl)c(=O)c3cc(OC)c(OC)cc32)cc(OC)c1	nan
	16030401	25808	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	8	1	4	5.0	Cc1ccc(Cc2nc3ccccc3nc2SCC(=O)NCCc2ccccc2)cc1	nan
	CHEMBL1354835	25808	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	8	1	4	5.0	Cc1ccc(Cc2nc3ccccc3nc2SCC(=O)NCCc2ccccc2)cc1	nan
	16010860	25811	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	7	1	6	2.8	CCc1ccc(NC(=O)Cn2c(=O)n(CCC(C)C)c(=O)c3cccnc32)cc1	nan
	CHEMBL1354858	25811	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	7	1	6	2.8	CCc1ccc(NC(=O)Cn2c(=O)n(CCC(C)C)c(=O)c3cccnc32)cc1	nan
	15988167	25874	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	6	1	6	2.9	COc1cccc(NC(=O)Cn2c(=O)n(Cc3ccccc3)c(=O)c3ccccc32)c1	nan
	CHEMBL1355668	25874	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	6	1	6	2.9	COc1cccc(NC(=O)Cn2c(=O)n(Cc3ccccc3)c(=O)c3ccccc32)c1	nan
	16024817	25974	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	3	1	4	5.2	O=C(Nc1ccccc1Cl)C1CCN(c2nc3ccccc3nc2C(F)(F)F)CC1	nan
	CHEMBL1356900	25974	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	3	1	4	5.2	O=C(Nc1ccccc1Cl)C1CCN(c2nc3ccccc3nc2C(F)(F)F)CC1	nan
	1165987	26080	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	8	1	6	4.0	COc1ccc(-c2cc(C(F)(F)F)nc(SCC(=O)NCC(C)C)n2)cc1OC	nan
	CHEMBL1358322	26080	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	8	1	6	4.0	COc1ccc(-c2cc(C(F)(F)F)nc(SCC(=O)NCC(C)C)n2)cc1OC	nan
	1003453	26095	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	3	2	5	5.6	Nc1c(C(=O)Nc2ccccc2Br)sc2nc(-c3cccs3)ccc12	nan
	CHEMBL1358598	26095	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	3	2	5	5.6	Nc1c(C(=O)Nc2ccccc2Br)sc2nc(-c3cccs3)ccc12	nan
	663400	26142	13	None	-1	3	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	4	1	5	4.8	O=C(CSc1ncnc2c1oc1ccccc12)Nc1cccc(Cl)c1	nan
	CHEMBL1359009	26142	13	None	-1	3	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	4	1	5	4.8	O=C(CSc1ncnc2c1oc1ccccc12)Nc1cccc(Cl)c1	nan
	5104589	26223	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	398	3	1	3	6.6	O=C(Nc1ccc2oc(-c3ccc(Cl)cc3)nc2c1)c1ccc2ccccc2c1	nan
	CHEMBL1359625	26223	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	398	3	1	3	6.6	O=C(Nc1ccc2oc(-c3ccc(Cl)cc3)nc2c1)c1ccc2ccccc2c1	nan
	4438847	26350	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	7	1	7	1.1	COc1ccc(S(=O)(=O)N2CCOCC2)cc1NC(=O)CSc1cccc[n+]1[O-]	nan
	CHEMBL1360781	26350	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	7	1	7	1.1	COc1ccc(S(=O)(=O)N2CCOCC2)cc1NC(=O)CSc1cccc[n+]1[O-]	nan
	15989315	26352	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	563	10	1	7	4.6	COc1ccc(CCNC(=O)c2ccc(Cn3c(=O)c4ccccc4n(Cc4cccc(C)c4)c3=O)cc2)cc1OC	nan
	CHEMBL1360796	26352	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	563	10	1	7	4.6	COc1ccc(CCNC(=O)c2ccc(Cn3c(=O)c4ccccc4n(Cc4cccc(C)c4)c3=O)cc2)cc1OC	nan
	15991495	26388	1	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	6	3	5	3.9	O=C(O)Cc1sc(Nc2ccc(C(=O)O)cc2)nc1-c1ccccc1	nan
	CHEMBL1361126	26388	1	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	6	3	5	3.9	O=C(O)Cc1sc(Nc2ccc(C(=O)O)cc2)nc1-c1ccccc1	nan
	2816171	26436	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	3	0	8	1.3	CCOC(=O)c1nnn2c1nc(N1CCOCC1)c1ccccc12	nan
	CHEMBL1361598	26436	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	3	0	8	1.3	CCOC(=O)c1nnn2c1nc(N1CCOCC1)c1ccccc12	nan
	6238059	26507	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	10	2	6	2.8	CCOc1ccc(C(=O)C2=C(O)C(=O)N(CCOCCO)C2c2ccc(F)cc2)cc1	nan
	CHEMBL1362160	26507	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	10	2	6	2.8	CCOc1ccc(C(=O)C2=C(O)C(=O)N(CCOCCO)C2c2ccc(F)cc2)cc1	nan
	15988824	26523	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	7	1	7	4.2	COc1ccc(-c2cc(C(=O)Nc3ccn(Cc4ccc(C)cc4)n3)no2)cc1OC	nan
	CHEMBL1362337	26523	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	7	1	7	4.2	COc1ccc(-c2cc(C(=O)Nc3ccn(Cc4ccc(C)cc4)n3)no2)cc1OC	nan
	6625370	26841	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	373	3	1	7	2.2	Cc1cc(=O)n2nc(N3CCCC3C(=O)Nc3cccc(F)c3)sc2n1	nan
	CHEMBL1365096	26841	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	373	3	1	7	2.2	Cc1cc(=O)n2nc(N3CCCC3C(=O)Nc3cccc(F)c3)sc2n1	nan
	1315619	26874	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	7	3	5	4.3	O=C(Nc1ccccc1C(=O)Nc1ccccc1C(=O)NCc1ccco1)c1ccco1	nan
	CHEMBL1365331	26874	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	7	3	5	4.3	O=C(Nc1ccccc1C(=O)Nc1ccccc1C(=O)NCc1ccco1)c1ccco1	nan
	2138525	26893	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	4	1	7	4.6	Cc1ccc(-c2nnn3c2nc(NCc2ccc4c(c2)OCO4)c2ccccc23)cc1	nan
	CHEMBL1365483	26893	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	4	1	7	4.6	Cc1ccc(-c2nnn3c2nc(NCc2ccc4c(c2)OCO4)c2ccccc23)cc1	nan
	5068934	26942	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	8	1	3	3.0	O=C(CCS(=O)(=O)Cc1cccc(Cl)c1)NCCc1ccccc1	nan
	CHEMBL1365953	26942	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	8	1	3	3.0	O=C(CCS(=O)(=O)Cc1cccc(Cl)c1)NCCc1ccccc1	nan
	7190319	26944	1	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	262	3	0	6	3.0	CCSc1ccc2nnc(-c3cccs3)n2n1	nan
	CHEMBL1365969	26944	1	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	262	3	0	6	3.0	CCSc1ccc2nnc(-c3cccs3)n2n1	nan
	16194607	27122	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	477	10	1	7	1.7	CCN(CC)CCCNC(=O)Cn1cnc2ccc(S(=O)(=O)N3CCC(C)CC3)cc2c1=O	nan
	CHEMBL1367480	27122	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	477	10	1	7	1.7	CCN(CC)CCCNC(=O)Cn1cnc2ccc(S(=O)(=O)N3CCC(C)CC3)cc2c1=O	nan
	16033554	27253	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	4	2	4	1.7	CC(=O)Nc1ccc(NC(=O)CN2C(=O)CN(C)C(=O)c3ccccc32)cc1	nan
	CHEMBL1368494	27253	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	4	2	4	1.7	CC(=O)Nc1ccc(NC(=O)CN2C(=O)CN(C)C(=O)c3ccccc32)cc1	nan
	16009410	27344	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	8	1	7	5.2	CCC(CC)c1nn2c(=O)cc(COc3ccc(NC(=O)c4ccccc4C)cc3)nc2s1	nan
	CHEMBL1369161	27344	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	8	1	7	5.2	CCC(CC)c1nn2c(=O)cc(COc3ccc(NC(=O)c4ccccc4C)cc3)nc2s1	nan
	20880788	27503	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	486	8	1	7	3.4	CC1CCCC(C)N1CCNC(=O)CCc1nnc2n(Cc3ccccc3)c(=O)c3ccccc3n12	nan
	CHEMBL1370306	27503	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	486	8	1	7	3.4	CC1CCCC(C)N1CCNC(=O)CCc1nnc2n(Cc3ccccc3)c(=O)c3ccccc3n12	nan
	2622707	27573	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	286	4	0	6	2.9	O=[N+]([O-])c1cccc(CSc2nnc3ccccn23)c1	nan
	CHEMBL1370729	27573	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	286	4	0	6	2.9	O=[N+]([O-])c1cccc(CSc2nnc3ccccn23)c1	nan
	3178485	27626	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	4	0	8	0.9	CCn1c(SCC(=O)N2CCCCC2C)nc2c1c(=O)n(C)c(=O)n2C	nan
	CHEMBL1371157	27626	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	4	0	8	0.9	CCn1c(SCC(=O)N2CCCCC2C)nc2c1c(=O)n(C)c(=O)n2C	nan
	2155682	27816	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	317	4	0	5	3.1	CC1CCN(C(=O)CSc2nnc(-c3ccccc3)o2)CC1	nan
	CHEMBL1372587	27816	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	317	4	0	5	3.1	CC1CCN(C(=O)CSc2nnc(-c3ccccc3)o2)CC1	nan
	2965534	27838	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	478	8	1	5	5.1	CCOc1ccc(-c2cc(C(=O)NCCCn3ccnc3)c3cc(Br)ccc3n2)cc1	nan
	CHEMBL1372738	27838	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	478	8	1	5	5.1	CCOc1ccc(-c2cc(C(=O)NCCCn3ccnc3)c3cc(Br)ccc3n2)cc1	nan
	2562079	28012	25	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	260	3	1	5	2.6	O=C(O)CSc1ncnc2c1oc1ccccc12	nan
	CHEMBL1373813	28012	25	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	260	3	1	5	2.6	O=C(O)CSc1ncnc2c1oc1ccccc12	nan
	2478421	28166	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	4	1	7	0.8	CC1(C)NC(=O)N(CC(=O)OCc2cc(=O)n3cc(Br)ccc3n2)C1=O	nan
	CHEMBL1374872	28166	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	4	1	7	0.8	CC1(C)NC(=O)N(CC(=O)OCc2cc(=O)n3cc(Br)ccc3n2)C1=O	nan
	3122786	28235	18	None	-10	4	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	334	4	0	4	5.1	COc1ccc(C2CC(c3cccs3)=NN2c2ccccc2)cc1	nan
	CHEMBL1375375	28235	18	None	-10	4	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	334	4	0	4	5.1	COc1ccc(C2CC(c3cccs3)=NN2c2ccccc2)cc1	nan
	4077805	28317	28	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	304	3	1	5	3.9	C=CCn1c(=S)[nH]c2scc(-c3ccc(C)o3)c2c1=O	nan
	CHEMBL1376201	28317	28	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	304	3	1	5	3.9	C=CCn1c(=S)[nH]c2scc(-c3ccc(C)o3)c2c1=O	nan
	2815476	28400	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	4	1	4	4.6	O=S(=O)(Nc1ccccc1C(F)(F)F)c1ccc(-c2ccccn2)s1	nan
	CHEMBL1376936	28400	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	4	1	4	4.6	O=S(=O)(Nc1ccccc1C(F)(F)F)c1ccc(-c2ccccn2)s1	nan
	16016416	28436	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	3	1	5	3.6	Cc1cc(O)c(CN2CCN(c3ccc(F)cc3)CC2)c2oc(=O)cc(C)c12	nan
	CHEMBL1377283	28436	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	3	1	5	3.6	Cc1cc(O)c(CN2CCN(c3ccc(F)cc3)CC2)c2oc(=O)cc(C)c12	nan
	2400757	28470	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	5	1	6	2.1	O=C(CNC(=O)c1cccc(F)c1)OCc1cc(=O)n2cc(Br)ccc2n1	nan
	CHEMBL1377678	28470	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	5	1	6	2.1	O=C(CNC(=O)c1cccc(F)c1)OCc1cc(=O)n2cc(Br)ccc2n1	nan
	2864532	28522	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	335	3	1	3	4.2	CC(C)(C)C(=O)C1=C(O)C(=O)N(c2ccccc2)C1c1ccccc1	nan
	CHEMBL1378083	28522	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	335	3	1	3	4.2	CC(C)(C)C(=O)C1=C(O)C(=O)N(c2ccccc2)C1c1ccccc1	nan
	3522811	28578	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	6	1	8	0.8	Cc1nc(SCC(=O)NCCc2ccccc2)c2c(=O)n(C)c(=O)n(C)c2n1	nan
	CHEMBL1378692	28578	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	6	1	8	0.8	Cc1nc(SCC(=O)NCCc2ccccc2)c2c(=O)n(C)c(=O)n(C)c2n1	nan
	4647380	28653	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	12	1	9	0.8	COCCN(CCOC)S(=O)(=O)c1ccc(C(=O)Nc2nnc(COC)o2)cc1	nan
	CHEMBL1379293	28653	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	12	1	9	0.8	COCCN(CCOC)S(=O)(=O)c1ccc(C(=O)Nc2nnc(COC)o2)cc1	nan
	5904589	28755	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	5	2	6	3.9	O=C(C1=C(O)C(=O)N(Cc2ccccc2)C1c1cccc(O)c1)c1ccc2c(c1)OCCO2	nan
	CHEMBL1380259	28755	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	5	2	6	3.9	O=C(C1=C(O)C(=O)N(Cc2ccccc2)C1c1cccc(O)c1)c1ccc2c(c1)OCCO2	nan
	2768996	28804	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	283	2	1	6	2.2	O=c1c2ccccc2nc(-c2ccc([N+](=O)[O-])cc2)n1O	nan
	CHEMBL1380557	28804	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	283	2	1	6	2.2	O=c1c2ccccc2nc(-c2ccc([N+](=O)[O-])cc2)n1O	nan
	2815634	28820	5	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	3	2	4	5.8	O=C(Nc1ccc(F)cc1)Nc1sccc1-c1nc2ccccc2s1	nan
	CHEMBL1380666	28820	5	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	3	2	4	5.8	O=C(Nc1ccc(F)cc1)Nc1sccc1-c1nc2ccccc2s1	nan
	3604840	28830	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	4	1	5	3.7	COc1cccc(-c2cc(C(=O)Nc3cccnc3Cl)no2)c1	nan
	CHEMBL1380782	28830	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	4	1	5	3.7	COc1cccc(-c2cc(C(=O)Nc3cccnc3Cl)no2)c1	nan
	723113	28850	22	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	2	4	4	3.9	Nc1ccc2[nH]c(-c3ccc(-c4nc5cc(N)ccc5[nH]4)cc3)nc2c1	nan
	CHEMBL1380889	28850	22	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	2	4	4	3.9	Nc1ccc2[nH]c(-c3ccc(-c4nc5cc(N)ccc5[nH]4)cc3)nc2c1	nan
	866607	28903	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	1	0	5	2.8	CC1CCN(C(=O)c2cc3c(=O)n4ccccc4nc3s2)CC1	nan
	CHEMBL1381324	28903	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	1	0	5	2.8	CC1CCN(C(=O)c2cc3c(=O)n4ccccc4nc3s2)CC1	nan
	1247739	29083	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	3	1	6	4.6	Cc1onc(-c2c(F)cccc2Cl)c1C(=O)Nc1nnc(C(F)(F)F)s1	nan
	CHEMBL1382928	29083	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	3	1	6	4.6	Cc1onc(-c2c(F)cccc2Cl)c1C(=O)Nc1nnc(C(F)(F)F)s1	nan
	4908738	29105	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	7	1	8	4.6	CCCSc1nnc(N2C(=O)C(O)=C(C(=O)c3ccco3)C2c2ccccc2F)s1	nan
	CHEMBL1383134	29105	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	7	1	8	4.6	CCCSc1nnc(N2C(=O)C(O)=C(C(=O)c3ccco3)C2c2ccccc2F)s1	nan
	4196061	29271	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	10	2	5	3.4	CCCCCNC(=O)c1ccc2c(=O)n(CCCOCC)c(=S)[nH]c2c1	nan
	CHEMBL1384631	29271	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	10	2	5	3.4	CCCCCNC(=O)c1ccc2c(=O)n(CCCOCC)c(=S)[nH]c2c1	nan
	1392125	29358	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	5	2	6	2.0	O=C1NC(=S)N(Cc2ccc(F)cc2)C(=O)/C1=C/NCc1ccc2c(c1)OCO2	nan
	CHEMBL1385415	29358	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	5	2	6	2.0	O=C1NC(=S)N(Cc2ccc(F)cc2)C(=O)/C1=C/NCc1ccc2c(c1)OCO2	nan
	20876328	29455	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	442	7	1	5	3.3	CN1CCN(CCCNC(=O)c2ccc3c(c2)N(Cc2ccc(F)cc2)CCS3)CC1	nan
	CHEMBL1386262	29455	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	442	7	1	5	3.3	CN1CCN(CCCNC(=O)c2ccc3c(c2)N(Cc2ccc(F)cc2)CCS3)CC1	nan
	17584980	29497	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	478	3	1	7	2.2	Cc1cc(O)c2c(C)c(CC(=O)N3CCN(C(=O)C4COc5ccccc5O4)CC3)c(=O)oc2c1	nan
	CHEMBL1386530	29497	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	478	3	1	7	2.2	Cc1cc(O)c2c(C)c(CC(=O)N3CCN(C(=O)C4COc5ccccc5O4)CC3)c(=O)oc2c1	nan
	3254139	29531	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	4	1	7	3.8	CSc1nc(SC(C)C(=O)O)c2c3c(sc2n1)COC(C)(C)C3	nan
	CHEMBL1386773	29531	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	4	1	7	3.8	CSc1nc(SC(C)C(=O)O)c2c3c(sc2n1)COC(C)(C)C3	nan
	3220391	29581	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	7	1	6	2.1	CCC(OC(=O)c1nsc(Cl)c1Cl)C(=O)NCCOC	nan
	CHEMBL1387168	29581	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	7	1	6	2.1	CCC(OC(=O)c1nsc(Cl)c1Cl)C(=O)NCCOC	nan
	16189864	29614	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	5	0	5	4.4	O=C(c1ccc(C(F)(F)F)cc1)C1CCCN(Cc2cccn2-c2ncccn2)C1	nan
	CHEMBL1387467	29614	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	5	0	5	4.4	O=C(c1ccc(C(F)(F)F)cc1)C1CCCN(Cc2cccn2-c2ncccn2)C1	nan
	899135	29657	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	2	1	3	3.2	NC(=O)c1cc(-c2cccnc2)nc2ccc(Br)cc12	nan
	CHEMBL1387789	29657	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	2	1	3	3.2	NC(=O)c1cc(-c2cccnc2)nc2ccc(Br)cc12	nan
	2360761	29658	24	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	245	1	1	5	2.5	COc1ccc2c(C)cc3nnc(S)n3c2c1	nan
	CHEMBL1387791	29658	24	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	245	1	1	5	2.5	COc1ccc2c(C)cc3nnc(S)n3c2c1	nan
	2377721	29701	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	308	2	0	6	3.9	Cc1cc(C)nc(Sc2ncnc3c2oc2ccccc23)n1	nan
	CHEMBL1388175	29701	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	308	2	0	6	3.9	Cc1cc(C)nc(Sc2ncnc3c2oc2ccccc23)n1	nan
	3303130	29865	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	6	1	6	6.0	Cc1cccc(N2C(=O)C(O)=C(C(=O)c3cccs3)C2c2cccc(Oc3ccccc3)c2)n1	nan
	CHEMBL1389429	29865	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	6	1	6	6.0	Cc1cccc(N2C(=O)C(O)=C(C(=O)c3cccs3)C2c2cccc(Oc3ccccc3)c2)n1	nan
	5047557	29911	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	4	2	5	2.7	COC(=O)c1cc(C)sc1NC(=O)C1C2C=CC(CC2)C1C(=O)O	nan
	CHEMBL1389758	29911	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	4	2	5	2.7	COC(=O)c1cc(C)sc1NC(=O)C1C2C=CC(CC2)C1C(=O)O	nan
	671729	29974	15	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	348	3	1	4	3.8	O=C(Nc1ccc2c(c1)C(=O)N(c1ccccc1)C2=O)c1cccs1	nan
	CHEMBL1390374	29974	15	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	348	3	1	4	3.8	O=C(Nc1ccc2c(c1)C(=O)N(c1ccccc1)C2=O)c1cccs1	nan
	576025	29995	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	264	0	0	4	1.6	O=c1c2ccccc2c(=O)n2n1Cc1ccccc1C2	nan
	CHEMBL1390537	29995	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	264	0	0	4	1.6	O=c1c2ccccc2c(=O)n2n1Cc1ccccc1C2	nan
	1245900	30048	11	None	1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	325	4	1	6	3.8	CCSc1nnc(NC(=O)c2cc3c(s2)CCCC3)s1	nan
	CHEMBL1391017	30048	11	None	1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	325	4	1	6	3.8	CCSc1nnc(NC(=O)c2cc3c(s2)CCCC3)s1	nan
	5260648	30072	33	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	254	1	1	3	2.1	Cc1cc(Br)cn2cc(C(=O)O)nc12	nan
	CHEMBL1391195	30072	33	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	254	1	1	3	2.1	Cc1cc(Br)cn2cc(C(=O)O)nc12	nan
	6619983	30158	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	4	0	7	2.4	COC(=O)C(C)Sc1ccc2nnc(-c3ccccc3)n2n1	nan
	CHEMBL1391987	30158	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	4	0	7	2.4	COC(=O)C(C)Sc1ccc2nnc(-c3ccccc3)n2n1	nan
	3236381	30257	3	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	4	0	8	2.5	CCOC(=O)c1sc2ncnc(N3CCN(C(=O)OCC)CC3)c2c1C	nan
	CHEMBL1392800	30257	3	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	4	0	8	2.5	CCOC(=O)c1sc2ncnc(N3CCN(C(=O)OCC)CC3)c2c1C	nan
	135414599	30354	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	320	1	2	4	0.2	O=C1CC2C(=O)NCCN2C(NC(=O)c2ccc(Cl)cc2)=N1	nan
	CHEMBL1393609	30354	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	320	1	2	4	0.2	O=C1CC2C(=O)NCCN2C(NC(=O)c2ccc(Cl)cc2)=N1	nan
	950424	30452	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	348	3	0	7	1.6	CCN1CCN(c2nc3c(C)cccn3c(=O)c2C=C(C#N)C#N)CC1	nan
	CHEMBL1394651	30452	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	348	3	0	7	1.6	CCN1CCN(c2nc3c(C)cccn3c(=O)c2C=C(C#N)C#N)CC1	nan
	1689018	30466	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	5	1	7	3.2	CCOC(=O)c1sc2ncn(CC(=O)Nc3cc(C)cc(C)c3)c(=O)c2c1C	nan
	CHEMBL1394885	30466	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	5	1	7	3.2	CCOC(=O)c1sc2ncn(CC(=O)Nc3cc(C)cc(C)c3)c(=O)c2c1C	nan
	8087252	30529	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	3	0	5	4.3	COc1cccc(N2CCN(C(=O)c3cc4c(s3)-c3ccccc3OC4)CC2)c1	nan
	CHEMBL1395507	30529	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	3	0	5	4.3	COc1cccc(N2CCN(C(=O)c3cc4c(s3)-c3ccccc3OC4)CC2)c1	nan
	16009438	30538	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	7	1	7	3.7	Cc1ccc(OCC(=O)Nc2ccc(OCc3cc(=O)n4ccsc4n3)cc2)cc1	nan
	CHEMBL1395616	30538	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	7	1	7	3.7	Cc1ccc(OCC(=O)Nc2ccc(OCc3cc(=O)n4ccsc4n3)cc2)cc1	nan
	16017578	30573	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	6	1	7	2.5	Cc1ccc(C(=O)Nc2nnc(S(=O)(=O)N(C)Cc3ccco3)s2)cc1	nan
	CHEMBL1396189	30573	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	6	1	7	2.5	Cc1ccc(C(=O)Nc2nnc(S(=O)(=O)N(C)Cc3ccco3)s2)cc1	nan
	24819156	30590	0	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	471	7	0	6	6.1	COc1ccc(-c2oc3ccc(N4CCOCC4)cc3c2/C=C/c2ccc(OC)c(OC)c2)cc1	nan
	CHEMBL1396464	30590	0	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	471	7	0	6	6.1	COc1ccc(-c2oc3ccc(N4CCOCC4)cc3c2/C=C/c2ccc(OC)c(OC)c2)cc1	nan
	16022449	30627	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	5	1	4	4.9	CC(C)Oc1ccc(CNC(=O)c2cc3cccc4c3n2CC(C)S4)cc1	nan
	CHEMBL1396952	30627	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	5	1	4	4.9	CC(C)Oc1ccc(CNC(=O)c2cc3cccc4c3n2CC(C)S4)cc1	nan
	2017205	30647	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	5	2	6	5.8	COc1ccc(-c2ccc3c(N)c(C(=O)Nc4ccc(C(F)(F)F)cc4)sc3n2)cc1OC	nan
	CHEMBL1397215	30647	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	5	2	6	5.8	COc1ccc(-c2ccc3c(N)c(C(=O)Nc4ccc(C(F)(F)F)cc4)sc3n2)cc1OC	nan
	16019456	30716	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	5	1	8	2.5	COc1cc(NS(=O)(=O)c2c(C)nc3sc(C)c(C)n3c2=O)cc(OC)c1	nan
	CHEMBL1398166	30716	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	5	1	8	2.5	COc1cc(NS(=O)(=O)c2c(C)nc3sc(C)c(C)n3c2=O)cc(OC)c1	nan
	2964735	30757	11	None	-3	3	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	490	7	1	9	4.5	COc1cccc(C2C(C(=O)c3cc4cccc(OC)c4o3)=C(O)C(=O)N2c2cc(C)on2)c1OC	nan
	CHEMBL1398596	30757	11	None	-3	3	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	490	7	1	9	4.5	COc1cccc(C2C(C(=O)c3cc4cccc(OC)c4o3)=C(O)C(=O)N2c2cc(C)on2)c1OC	nan
	16012160	30775	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	5	1	7	2.0	Cc1cc(=O)n2nc(N(C)CC(=O)NCc3cccc(Br)c3)sc2n1	nan
	CHEMBL1398785	30775	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	5	1	7	2.0	Cc1cc(=O)n2nc(N(C)CC(=O)NCc3cccc(Br)c3)sc2n1	nan
	20888752	30872	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	7	1	9	1.2	CCS(=O)(=O)c1nc(S(=O)(=O)c2ccc(C)cc2)c(N2CCN(CCO)CC2)s1	nan
	CHEMBL1399722	30872	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	7	1	9	1.2	CCS(=O)(=O)c1nc(S(=O)(=O)c2ccc(C)cc2)c(N2CCN(CCO)CC2)s1	nan
	7997207	30914	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	5	1	5	3.3	Cc1ccc(NC(=O)COC(=O)c2ccc(-n3cccn3)cc2)cc1C	nan
	CHEMBL1400115	30914	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	5	1	5	3.3	Cc1ccc(NC(=O)COC(=O)c2ccc(-n3cccn3)cc2)cc1C	nan
	2874407	30938	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	463	4	1	7	5.0	CC1=C(C(=O)OCC2CCCO2)C(c2coc3ccccc3c2=O)C2=C(O)CC(C)(C)CC2=N1	nan
	CHEMBL1400295	30938	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	463	4	1	7	5.0	CC1=C(C(=O)OCC2CCCO2)C(c2coc3ccccc3c2=O)C2=C(O)CC(C)(C)CC2=N1	nan
	2157035	31023	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	7	1	6	5.0	Cc1ccc(-c2nc(S(=O)(=O)c3ccccc3)c(SCC(=O)NC3CCCCC3)o2)cc1	nan
	CHEMBL1401131	31023	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	7	1	6	5.0	Cc1ccc(-c2nc(S(=O)(=O)c3ccccc3)c(SCC(=O)NC3CCCCC3)o2)cc1	nan
	5389771	31026	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	9	1	6	2.9	C=CCOc1ccc(C(=O)C2=C(O)C(=O)N(CCOC)C2c2cccnc2)cc1	nan
	CHEMBL1401159	31026	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	9	1	6	2.9	C=CCOc1ccc(C(=O)C2=C(O)C(=O)N(CCOC)C2c2cccnc2)cc1	nan
	20876293	31216	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	8	1	5	3.9	CCN1CCN(CCCNC(=O)c2ccc3c(c2)N(Cc2ccc(C)cc2)CCS3)CC1	nan
	CHEMBL1402721	31216	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	8	1	5	3.9	CCN1CCN(CCCNC(=O)c2ccc3c(c2)N(Cc2ccc(C)cc2)CCS3)CC1	nan
	16025411	31219	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	5	0	7	3.3	COC(=O)CSc1ncc2c(n1)-c1ccccc1N(Cc1cccc(F)c1)S2(=O)=O	nan
	CHEMBL1402769	31219	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	5	0	7	3.3	COC(=O)CSc1ncc2c(n1)-c1ccccc1N(Cc1cccc(F)c1)S2(=O)=O	nan
	1091654	31326	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	7	2	5	4.5	COc1ccc(NC(=O)c2ccco2)cc1NC(=O)COc1ccc(Cl)cc1C	nan
	CHEMBL1403849	31326	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	7	2	5	4.5	COc1ccc(NC(=O)c2ccco2)cc1NC(=O)COc1ccc(Cl)cc1C	nan
	2405342	31462	21	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	3	1	6	2.9	O=S(=O)(Nc1nc2cc3c(cc2nc1Cl)OCCO3)c1ccccc1	nan
	CHEMBL1405208	31462	21	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	3	1	6	2.9	O=S(=O)(Nc1nc2cc3c(cc2nc1Cl)OCCO3)c1ccccc1	nan
	16018264	31497	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	489	6	1	6	5.7	CCOC(=O)c1ccc(NC(=O)c2oc3c(c2C)-c2nn(Cc4ccccc4Cl)cc2CC3)cc1	nan
	CHEMBL1405564	31497	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	489	6	1	6	5.7	CCOC(=O)c1ccc(NC(=O)c2oc3c(c2C)-c2nn(Cc4ccccc4Cl)cc2CC3)cc1	nan
	3258366	31605	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	298	1	2	6	3.5	CCC1(C)Cc2c(sc3nc(S)nc(S)c23)CO1	nan
	CHEMBL1406514	31605	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	298	1	2	6	3.5	CCC1(C)Cc2c(sc3nc(S)nc(S)c23)CO1	nan
	5739089	31653	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	5	1	6	3.7	O=C(C1=C(O)C(=O)N(Cc2cccnc2)C1c1cccc(F)c1)c1ccc2c(c1)OCO2	nan
	CHEMBL1407014	31653	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	5	1	6	3.7	O=C(C1=C(O)C(=O)N(Cc2cccnc2)C1c1cccc(F)c1)c1ccc2c(c1)OCO2	nan
	20877853	31866	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	3	0	5	3.7	CCOC(=O)C1CCN(C(=O)c2cc3c(s2)-c2ccccc2OC3)CC1	nan
	CHEMBL1408512	31866	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	3	0	5	3.7	CCOC(=O)C1CCN(C(=O)c2cc3c(s2)-c2ccccc2OC3)CC1	nan
	704023	32019	39	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	244	1	1	4	3.6	Sc1ncnc2sc(-c3ccccc3)cc12	nan
	CHEMBL1409776	32019	39	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	244	1	1	4	3.6	Sc1ncnc2sc(-c3ccccc3)cc12	nan
	4197372	32038	10	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	4	1	6	4.5	O=C(Nc1nc(-c2cccs2)c(C(=O)C(F)(F)F)s1)c1ccco1	nan
	CHEMBL1409901	32038	10	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	4	1	6	4.5	O=C(Nc1nc(-c2cccs2)c(C(=O)C(F)(F)F)s1)c1ccco1	nan
	1348850	32051	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	6	1	5	5.3	COc1ccc(OCC(=O)Nc2cc(-c3nc4ccccc4s3)ccc2C)cc1	nan
	CHEMBL1409994	32051	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	6	1	5	5.3	COc1ccc(OCC(=O)Nc2cc(-c3nc4ccccc4s3)ccc2C)cc1	nan
	6472686	32080	17	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	304	5	1	5	1.5	COc1cccc2cc(C(=O)NCCN3CCOCC3)oc12	nan
	CHEMBL1410184	32080	17	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	304	5	1	5	1.5	COc1cccc2cc(C(=O)NCCN3CCOCC3)oc12	nan
	16019689	32156	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	457	10	1	8	2.9	COCCCn1c(=O)c2sccc2n2c(CCCC(=O)NCc3ccc(F)cc3)nnc12	nan
	CHEMBL1410849	32156	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	457	10	1	8	2.9	COCCCn1c(=O)c2sccc2n2c(CCCC(=O)NCc3ccc(F)cc3)nnc12	nan
	16025704	32243	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	6	1	7	5.5	COc1ccc(OC)c(CNC(=O)c2ccc(N3Cc4ccccc4Oc4ncccc43)s2)c1	nan
	CHEMBL1411590	32243	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	6	1	7	5.5	COc1ccc(OC)c(CNC(=O)c2ccc(N3Cc4ccccc4Oc4ncccc43)s2)c1	nan
	15988174	32344	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	5	2	4	3.0	Cc1ccc(CCNC(=O)c2ccc3c(=O)n(-c4ccccc4)c(=O)[nH]c3c2)cc1	nan
	CHEMBL1412411	32344	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	5	2	4	3.0	Cc1ccc(CCNC(=O)c2ccc3c(=O)n(-c4ccccc4)c(=O)[nH]c3c2)cc1	nan
	972224	32397	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	335	4	2	5	3.8	CCc1c(C)sc(N=C(S)Nc2cccnc2)c1C(=O)OC	nan
	CHEMBL1412818	32397	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	335	4	2	5	3.8	CCc1c(C)sc(N=C(S)Nc2cccnc2)c1C(=O)OC	nan
	16018140	32407	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	6	1	2	4.5	Cn1cc(CCCC(=O)NCc2ccccc2Cl)c2ccccc21	nan
	CHEMBL1412876	32407	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	6	1	2	4.5	Cn1cc(CCCC(=O)NCc2ccccc2Cl)c2ccccc21	nan
	646994	32441	4	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	6	1	7	3.4	Cc1ccc(S(=O)(=O)N(Cc2cc3cc4c(cc3nc2O)OCCO4)CC2CCCO2)cc1	nan
	CHEMBL1413144	32441	4	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	6	1	7	3.4	Cc1ccc(S(=O)(=O)N(Cc2cc3cc4c(cc3nc2O)OCCO4)CC2CCCO2)cc1	nan
	16018722	32478	1	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	366	4	1	6	4.1	Cc1ccc(C)c(NC(=O)CSc2nnc(C)n3c2cc2occc23)c1	nan
	CHEMBL1413449	32478	1	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	366	4	1	6	4.1	Cc1ccc(C)c(NC(=O)CSc2nnc(C)n3c2cc2occc23)c1	nan
	4149556	32514	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	4	1	3	4.3	CC(C)(C)C(=O)C1=C(O)C(=O)N(Cc2ccccc2)C1c1ccccc1F	nan
	CHEMBL1413747	32514	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	4	1	3	4.3	CC(C)(C)C(=O)C1=C(O)C(=O)N(Cc2ccccc2)C1c1ccccc1F	nan
	16018046	32633	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	6	1	4	3.8	O=C(CCn1c(=O)c2cccn2c2ccc(F)cc21)NCCc1ccccc1Cl	nan
	CHEMBL1414743	32633	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	6	1	4	3.8	O=C(CCn1c(=O)c2cccn2c2ccc(F)cc21)NCCc1ccccc1Cl	nan
	16187993	32690	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	8	1	6	1.2	CCN(CC)S(=O)(=O)c1ccc2c(c1)N(CC(=O)NCc1ccccn1)C(=O)CO2	nan
	CHEMBL1415247	32690	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	8	1	6	1.2	CCN(CC)S(=O)(=O)c1ccc2c(c1)N(CC(=O)NCc1ccccn1)C(=O)CO2	nan
	2910208	32855	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	7	1	6	3.3	O=C(C1=C(O)C(=O)N(CCCn2ccnc2)C1c1ccc(F)cc1)c1ccco1	nan
	CHEMBL1416738	32855	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	7	1	6	3.3	O=C(C1=C(O)C(=O)N(CCCn2ccnc2)C1c1ccc(F)cc1)c1ccco1	nan
	5014048	32899	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	6	2	3	5.9	Cc1ccc(CCNC(=O)c2cc(Nc3ccc(C)c(C)c3)nc3ccccc23)cc1	nan
	CHEMBL1417106	32899	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	6	2	3	5.9	Cc1ccc(CCNC(=O)c2cc(Nc3ccc(C)c(C)c3)nc3ccccc23)cc1	nan
	8901980	32930	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	6	1	5	4.1	CCOC(=O)Nc1ccc2c(CN(C)Cc3ccc(F)cc3)cc(=O)oc2c1	nan
	CHEMBL1417351	32930	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	6	1	5	4.1	CCOC(=O)Nc1ccc2c(CN(C)Cc3ccc(F)cc3)cc(=O)oc2c1	nan
	2911345	33043	15	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	5	1	5	4.5	Cc1ccc(C(=O)C2=C(O)C(=O)N(Cc3cccnc3)C2c2ccc(Br)cc2)o1	nan
	3999653	33043	15	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	5	1	5	4.5	Cc1ccc(C(=O)C2=C(O)C(=O)N(Cc3cccnc3)C2c2ccc(Br)cc2)o1	nan
	CHEMBL1418370	33043	15	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	5	1	5	4.5	Cc1ccc(C(=O)C2=C(O)C(=O)N(Cc3cccnc3)C2c2ccc(Br)cc2)o1	nan
	1388232	33115	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	1	1	4	5.2	Cc1cccc(-n2c(=S)[nH]c3sc4c(c3c2=O)CCc2ccccc2-4)c1	nan
	CHEMBL1418971	33115	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	1	1	4	5.2	Cc1cccc(-n2c(=S)[nH]c3sc4c(c3c2=O)CCc2ccccc2-4)c1	nan
	2077572	33161	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	5	1	6	1.9	O=C(CNC(=O)c1ccccc1)OCc1cc(=O)n2cc(Br)ccc2n1	nan
	CHEMBL1419336	33161	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	5	1	6	1.9	O=C(CNC(=O)c1ccccc1)OCc1cc(=O)n2cc(Br)ccc2n1	nan
	2370216	33495	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	426	3	0	3	4.2	O=C(COc1c(Br)cc(Br)c2cccnc12)N1CCCCC1	nan
	CHEMBL1422190	33495	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	426	3	0	3	4.2	O=C(COc1c(Br)cc(Br)c2cccnc12)N1CCCCC1	nan
	2035062	33518	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	317	3	1	5	2.6	CC(=O)NCc1nnc2c3ccccc3c(-c3ccccc3)nn12	nan
	CHEMBL1422374	33518	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	317	3	1	5	2.6	CC(=O)NCc1nnc2c3ccccc3c(-c3ccccc3)nn12	nan
	16187581	33521	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	8	0	7	2.8	C=CCN(Cc1nc(-c2cc(OC)ccc2OC)oc1C)C1CCS(=O)(=O)C1	nan
	CHEMBL1422392	33521	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	8	0	7	2.8	C=CCN(Cc1nc(-c2cc(OC)ccc2OC)oc1C)C1CCS(=O)(=O)C1	nan
	5931057	33577	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	479	7	1	7	4.0	O=C(C1=C(O)C(=O)N(CCCn2ccnc2)C1c1ccc(Cl)cc1)c1ccc2c(c1)OCCO2	nan
	CHEMBL1422871	33577	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	479	7	1	7	4.0	O=C(C1=C(O)C(=O)N(CCCn2ccnc2)C1c1ccc(Cl)cc1)c1ccc2c(c1)OCCO2	nan
	1609403	33676	6	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	485	7	0	5	4.7	CCCCn1cc[n+](-c2nc3ccccc3nc2[N-]S(=O)(=O)c2ccc(Br)cc2)c1	nan
	CHEMBL1423632	33676	6	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	485	7	0	5	4.7	CCCCn1cc[n+](-c2nc3ccccc3nc2[N-]S(=O)(=O)c2ccc(Br)cc2)c1	nan
	2308387	33711	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	10	0	8	2.6	Cc1c(CCOC(=O)c2cc([N+](=O)[O-])ccc2Cl)sc[n+]1CCCCS(=O)(=O)[O-]	nan
	CHEMBL1423887	33711	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	10	0	8	2.6	Cc1c(CCOC(=O)c2cc([N+](=O)[O-])ccc2Cl)sc[n+]1CCCCS(=O)(=O)[O-]	nan
	3546539	33776	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	319	4	2	4	1.2	O=C1NC(=S)N(C2CC2)C(=O)/C1=C/NCc1ccc(F)cc1	nan
	CHEMBL1424530	33776	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	319	4	2	4	1.2	O=C1NC(=S)N(C2CC2)C(=O)/C1=C/NCc1ccc(F)cc1	nan
	16192280	33922	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	345	4	0	4	4.2	CSc1ccc(C(=O)C2CCCN(C(=O)c3ccsc3)C2)cc1	nan
	CHEMBL1425858	33922	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	345	4	0	4	4.2	CSc1ccc(C(=O)C2CCCN(C(=O)c3ccsc3)C2)cc1	nan
	1229909	34197	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	309	2	1	6	2.7	Cn1cc(Cl)c(-c2nnc(S)n2-c2ccc(F)cc2)n1	nan
	CHEMBL1428119	34197	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	309	2	1	6	2.7	Cn1cc(Cl)c(-c2nnc(S)n2-c2ccc(F)cc2)n1	nan
	20903654	34348	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	478	7	0	9	1.6	CCN1CCN(C(=O)CCc2nnc3ccc(N4CCN(c5cccc(OC)c5)CC4)nn23)CC1	nan
	CHEMBL1429390	34348	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	478	7	0	9	1.6	CCN1CCN(C(=O)CCc2nnc3ccc(N4CCN(c5cccc(OC)c5)CC4)nn23)CC1	nan
	3259805	34353	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	6	1	7	1.9	Cc1ccc(S(=O)(=O)N2CCOCC2)cc1NC(=O)COC(=O)c1cccnc1Cl	nan
	CHEMBL1429423	34353	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	6	1	7	1.9	Cc1ccc(S(=O)(=O)N2CCOCC2)cc1NC(=O)COC(=O)c1cccnc1Cl	nan
	18562990	34400	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	7	1	7	2.0	O=C(NCCc1nnc2ccc(SCC(=O)N3CCCC3)nn12)c1ccc(F)cc1	nan
	CHEMBL1429771	34400	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	7	1	7	2.0	O=C(NCCc1nnc2ccc(SCC(=O)N3CCCC3)nn12)c1ccc(F)cc1	nan
	11834440	34419	7	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	5	1	4	4.9	CC(C)(C)c1ccc(/C(O)=C(/C([S-])=NCc2ccco2)[n+]2ccccc2)cc1	nan
	4030418	34419	7	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	5	1	4	4.9	CC(C)(C)c1ccc(/C(O)=C(/C([S-])=NCc2ccco2)[n+]2ccccc2)cc1	nan
	CHEMBL1429883	34419	7	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	5	1	4	4.9	CC(C)(C)c1ccc(/C(O)=C(/C([S-])=NCc2ccco2)[n+]2ccccc2)cc1	nan
	3402414	34440	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	4	2	10	-2.3	Cn1c(N)c(C(=O)COC(=O)C2=NNC(=O)CC2)c(=O)n(C)c1=O	nan
	CHEMBL1430091	34440	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	4	2	10	-2.3	Cn1c(N)c(C(=O)COC(=O)C2=NNC(=O)CC2)c(=O)n(C)c1=O	nan
	2578265	34444	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	346	2	1	6	1.8	CC1CCC2(CC1)NC(=O)N(Cc1cc(=O)n3ccsc3n1)C2=O	nan
	CHEMBL1430109	34444	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	346	2	1	6	1.8	CC1CCC2(CC1)NC(=O)N(Cc1cc(=O)n3ccsc3n1)C2=O	nan
	4987698	34714	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	6	2	7	3.0	O=C(C1=C(O)C(=O)N(CCN2CCOCC2)C1c1cccc(O)c1)c1cc2ccccc2o1	nan
	CHEMBL1432401	34714	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	6	2	7	3.0	O=C(C1=C(O)C(=O)N(CCN2CCOCC2)C1c1cccc(O)c1)c1cc2ccccc2o1	nan
	657881	34725	10	None	-3	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	203	2	1	5	1.9	CCOC(=O)c1c(C)nsc1S	nan
	CHEMBL1432472	34725	10	None	-3	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	203	2	1	5	1.9	CCOC(=O)c1c(C)nsc1S	nan
	5123174	34745	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	306	4	1	5	3.3	COCCCn1c(=S)[nH]c2c(sc3ccccc32)c1=O	nan
	CHEMBL1432655	34745	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	306	4	1	5	3.3	COCCCn1c(=S)[nH]c2c(sc3ccccc32)c1=O	nan
	16019017	34892	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	5	1	5	3.9	Cc1cccc(CNC(=O)c2ccc(Cn3c(=O)c4cccn4c4cccnc43)cc2)c1	nan
	CHEMBL1434147	34892	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	5	1	5	3.9	Cc1cccc(CNC(=O)c2ccc(Cn3c(=O)c4cccn4c4cccnc43)cc2)c1	nan
	3566323	34940	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	509	9	1	9	4.0	CCOC(=O)CC(NC(=O)c1cc2c(=O)n3cccc(C)c3nc2s1)c1ccc(OCC)c(OC)c1	nan
	CHEMBL1434864	34940	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	509	9	1	9	4.0	CCOC(=O)CC(NC(=O)c1cc2c(=O)n3cccc(C)c3nc2s1)c1ccc(OCC)c(OC)c1	nan
	16015297	35045	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	454	7	1	5	5.3	CCn1c(CN2CCC(C)CC2)nc2cc(NC(=O)COc3ccc(Cl)c(C)c3)ccc21	nan
	CHEMBL1436095	35045	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	454	7	1	5	5.3	CCn1c(CN2CCC(C)CC2)nc2cc(NC(=O)COc3ccc(Cl)c(C)c3)ccc21	nan
	7526401	35058	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	3	1	4	2.2	N#Cc1ccccc1NS(=O)(=O)c1cc2c3c(c1)CCN3C(=O)CC2	nan
	CHEMBL1436243	35058	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	3	1	4	2.2	N#Cc1ccccc1NS(=O)(=O)c1cc2c3c(c1)CCN3C(=O)CC2	nan
	16019444	35060	0	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	5	1	6	2.9	Cc1nc2sc(C)c(C)n2c(=O)c1S(=O)(=O)NCCc1ccc(Cl)cc1	nan
	CHEMBL1436274	35060	0	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	5	1	6	2.9	Cc1nc2sc(C)c(C)n2c(=O)c1S(=O)(=O)NCCc1ccc(Cl)cc1	nan
	1743255	35062	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	423	3	1	5	3.4	N#CCNC(=O)c1nn2c(C(F)(F)F)cc(-c3ccccc3)nc2c1Br	nan
	CHEMBL1436298	35062	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	423	3	1	5	3.4	N#CCNC(=O)c1nn2c(C(F)(F)F)cc(-c3ccccc3)nc2c1Br	nan
	1004082	35108	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	5	2	5	4.8	COc1ccc(-c2ccc3c(N)c(C(=O)NCc4ccc(C)cc4)sc3n2)cc1	nan
	CHEMBL1437042	35108	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	5	2	5	4.8	COc1ccc(-c2ccc3c(N)c(C(=O)NCc4ccc(C)cc4)sc3n2)cc1	nan
	16030497	35138	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	7	1	4	5.8	CCc1cccc(C)c1NC(=O)CSc1nc2ccccc2nc1Cc1ccccc1	nan
	CHEMBL1437361	35138	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	7	1	4	5.8	CCc1cccc(C)c1NC(=O)CSc1nc2ccccc2nc1Cc1ccccc1	nan
	5297283	35172	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	335	2	1	5	2.5	COc1ccc(C2CC(=O)Nc3c2c(=O)nc2c(C)cccn32)cc1	nan
	CHEMBL1437774	35172	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	335	2	1	5	2.5	COc1ccc(C2CC(=O)Nc3c2c(=O)nc2c(C)cccn32)cc1	nan
	2980985	35260	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	3	2	3	3.2	CC(C)(C)C(=O)NNC(=O)COc1ccc2ccccc2c1Br	nan
	CHEMBL1438501	35260	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	3	2	3	3.2	CC(C)(C)C(=O)NNC(=O)COc1ccc2ccccc2c1Br	nan
	16027383	35293	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	463	7	1	8	3.7	Cc1ccccc1OCC(=O)Nc1ccc(C(=O)OCc2cc(=O)n3c(C)csc3n2)cc1	nan
	CHEMBL1438820	35293	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	463	7	1	8	3.7	Cc1ccccc1OCC(=O)Nc1ccc(C(=O)OCc2cc(=O)n3c(C)csc3n2)cc1	nan
	16030423	35432	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	7	1	4	5.2	Cc1ccc(CNC(=O)CSc2nc3ccccc3nc2Cc2ccc(C)cc2)cc1	nan
	CHEMBL1440057	35432	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	7	1	4	5.2	Cc1ccc(CNC(=O)CSc2nc3ccccc3nc2Cc2ccc(C)cc2)cc1	nan
	24816825	35442	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	4	1	3	3.4	O=C(c1ccc(S(=O)(=O)Nc2cccc(C(F)(F)F)c2)cc1)N1CCC1	nan
	CHEMBL1440121	35442	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	4	1	3	3.4	O=C(c1ccc(S(=O)(=O)Nc2cccc(C(F)(F)F)c2)cc1)N1CCC1	nan
	22583638	35562	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	6	1	7	3.9	C=CCn1c(SCC(=O)N2CCN(c3ccccc3)CC2)nc2c3ccccc3nc-2c1O	nan
	CHEMBL1441228	35562	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	6	1	7	3.9	C=CCn1c(SCC(=O)N2CCN(c3ccccc3)CC2)nc2c3ccccc3nc-2c1O	nan
	4066521	35574	11	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	318	3	1	6	2.4	CC(=O)c1sc(NC(=O)C2COc3ccccc3O2)nc1C	nan
	CHEMBL1441350	35574	11	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	318	3	1	6	2.4	CC(=O)c1sc(NC(=O)C2COc3ccccc3O2)nc1C	nan
	2965654	35643	11	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	4	1	5	5.1	O=C(Nc1ccc([N+](=O)[O-])cc1)c1cc(-c2ccccn2)nc2c(Cl)cccc12	nan
	CHEMBL1441978	35643	11	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	4	1	5	5.1	O=C(Nc1ccc([N+](=O)[O-])cc1)c1cc(-c2ccccn2)nc2c(Cl)cccc12	nan
	16008702	35768	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	10	1	8	3.3	CCOC(=O)CC(NC(=O)CCc1c(C)nc2ncnn2c1C)c1ccc(OC(C)C)cc1	nan
	CHEMBL1443046	35768	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	10	1	8	3.3	CCOC(=O)CC(NC(=O)CCc1c(C)nc2ncnn2c1C)c1ccc(OC(C)C)cc1	nan
	2854033	35851	15	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	322	3	0	3	5.2	Fc1ccc(N2N=C(c3cccs3)CC2c2ccccc2)cc1	nan
	CHEMBL1443903	35851	15	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	322	3	0	3	5.2	Fc1ccc(N2N=C(c3cccs3)CC2c2ccccc2)cc1	nan
	5904887	35869	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	8	1	7	3.9	COc1ccc(C2C(C(=O)c3ccc4c(c3)CC(C)O4)=C(O)C(=O)N2CCCn2ccnc2)cc1	nan
	CHEMBL1444052	35869	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	8	1	7	3.9	COc1ccc(C2C(C(=O)c3ccc4c(c3)CC(C)O4)=C(O)C(=O)N2CCCn2ccnc2)cc1	nan
	16249191	36030	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	486	8	2	10	0.0	CC(C)[C@H](NS(=O)(=O)c1ccc(Cl)cc1)C(=O)OCC(=O)c1c(N)n(C)c(=O)n(C)c1=O	nan
	CHEMBL1445550	36030	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	486	8	2	10	0.0	CC(C)[C@H](NS(=O)(=O)c1ccc(Cl)cc1)C(=O)OCC(=O)c1c(N)n(C)c(=O)n(C)c1=O	nan
	6236858	36151	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	5	1	5	4.3	CC1Cc2cc(C(=O)C3=C(O)C(=O)N(Cc4ccncc4)C3c3ccccc3F)ccc2O1	nan
	CHEMBL1446709	36151	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	5	1	5	4.3	CC1Cc2cc(C(=O)C3=C(O)C(=O)N(Cc4ccncc4)C3c3ccccc3F)ccc2O1	nan
	2946413	36250	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	6	1	4	4.9	OC(COc1ccc2ccccc2c1Br)Cn1cnc(-c2ccccc2)c1	nan
	CHEMBL1447526	36250	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	6	1	4	4.9	OC(COc1ccc2ccccc2c1Br)Cn1cnc(-c2ccccc2)c1	nan
	5168521	36268	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	361	3	1	5	3.7	Cc1cc(C)c(NC(=O)Cn2cnc3c(oc4ccccc43)c2=O)c(C)c1	nan
	CHEMBL1447670	36268	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	361	3	1	5	3.7	Cc1cc(C)c(NC(=O)Cn2cnc3c(oc4ccccc43)c2=O)c(C)c1	nan
	975514	36418	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	335	4	1	2	3.7	COc1ccc2cc(Br)ccc2c1CC(=O)NC(C)C	nan
	CHEMBL1448872	36418	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	335	4	1	2	3.7	COc1ccc2cc(Br)ccc2c1CC(=O)NC(C)C	nan
	5003875	36746	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	3	1	4	4.3	O=C(Nc1cccnc1Cl)c1cc(-c2ccc(Cl)cc2)on1	nan
	CHEMBL1451527	36746	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	3	1	4	4.3	O=C(Nc1cccnc1Cl)c1cc(-c2ccc(Cl)cc2)on1	nan
	16009656	36809	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	5	1	6	4.8	Cc1cccc(C(=O)Nc2ccc(OCc3cc(=O)n4c5c(sc4n3)CCCC5)cc2)c1	nan
	CHEMBL1451944	36809	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	5	1	6	4.8	Cc1cccc(C(=O)Nc2ccc(OCc3cc(=O)n4c5c(sc4n3)CCCC5)cc2)c1	nan
	8087990	36825	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	3	0	8	1.3	Cc1nc2scc(C)n2c(=O)c1S(=O)(=O)N1CCN(c2ccccn2)CC1	nan
	CHEMBL1452085	36825	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	3	0	8	1.3	Cc1nc2scc(C)n2c(=O)c1S(=O)(=O)N1CCN(c2ccccn2)CC1	nan
	2172625	36834	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	288	1	2	6	2.6	Cc1cc(C2C(C#N)=C(N)SC(N)=C2C#N)c(C)s1	nan
	CHEMBL1452137	36834	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	288	1	2	6	2.6	Cc1cc(C2C(C#N)=C(N)SC(N)=C2C#N)c(C)s1	nan
	2874437	36893	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	4	0	10	-0.3	Cn1c(=O)c2c(ncn2CC(=O)N2CCN(c3ccc([N+](=O)[O-])cc3)CC2)n(C)c1=O	nan
	CHEMBL1452667	36893	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	4	0	10	-0.3	Cn1c(=O)c2c(ncn2CC(=O)N2CCN(c3ccc([N+](=O)[O-])cc3)CC2)n(C)c1=O	nan
	3242606	36992	7	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	6	1	9	2.0	Cn1c(=O)c2sccc2n2c(CCCC(=O)NCc3ccc4c(c3)OCO4)nnc12	nan
	CHEMBL1453430	36992	7	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	6	1	9	2.0	Cn1c(=O)c2sccc2n2c(CCCC(=O)NCc3ccc4c(c3)OCO4)nnc12	nan
	5924128	37039	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	6	1	6	4.2	COc1ccc(C2C(C(=O)c3ccc4c(c3)CC(C)O4)=C(O)C(=O)N2Cc2cccnc2)cc1	nan
	CHEMBL1453845	37039	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	6	1	6	4.2	COc1ccc(C2C(C(=O)c3ccc4c(c3)CC(C)O4)=C(O)C(=O)N2Cc2cccnc2)cc1	nan
	16025308	37049	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	4	1	5	3.1	O=C(Cn1c2ncccc2c(=O)n1-c1ccccc1)Nc1ccc(F)c(F)c1	nan
	CHEMBL1453921	37049	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	4	1	5	3.1	O=C(Cn1c2ncccc2c(=O)n1-c1ccccc1)Nc1ccc(F)c(F)c1	nan
	16009318	37092	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	300	3	0	5	3.3	Cc1cc(C)cc(OCc2cc(=O)n3cc(C)sc3n2)c1	nan
	CHEMBL1454181	37092	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	300	3	0	5	3.3	Cc1cc(C)cc(OCc2cc(=O)n3cc(C)sc3n2)c1	nan
	16015117	37112	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	6	1	6	4.0	COc1ccccc1OCC(=O)Nc1nc(-c2ccc(Br)cc2)ns1	nan
	CHEMBL1454422	37112	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	6	1	6	4.0	COc1ccccc1OCC(=O)Nc1nc(-c2ccc(Br)cc2)ns1	nan
	20920416	37180	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	6	1	7	4.0	COc1ccc(-n2nc3c(N4CCC(C(=O)NCc5ccccc5)CC4)nnc(C)c3c2C)cc1	nan
	CHEMBL1454925	37180	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	6	1	7	4.0	COc1ccc(-n2nc3c(N4CCC(C(=O)NCc5ccccc5)CC4)nnc(C)c3c2C)cc1	nan
	35802	37182	98	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	313	3	2	4	3.1	COC(=O)Nc1nc2cc(C(=O)c3ccc(F)cc3)ccc2[nH]1	nan
	CHEMBL1454946	37182	98	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	313	3	2	4	3.1	COC(=O)Nc1nc2cc(C(=O)c3ccc(F)cc3)ccc2[nH]1	nan
	5739327	37236	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	6	1	7	3.0	O=C(C1=C(O)C(=O)N(CCN2CCOCC2)C1c1cccc(Cl)c1)c1ccc2c(c1)OCO2	nan
	CHEMBL1455509	37236	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	6	1	7	3.0	O=C(C1=C(O)C(=O)N(CCN2CCOCC2)C1c1cccc(Cl)c1)c1ccc2c(c1)OCO2	nan
	20923165	37333	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	7	1	6	2.4	CCC(C)(C)NS(=O)(=O)c1cc(CN2C(=O)c3cccnc3C2=O)ccc1OC	nan
	CHEMBL1456385	37333	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	7	1	6	2.4	CCC(C)(C)NS(=O)(=O)c1cc(CN2C(=O)c3cccnc3C2=O)ccc1OC	nan
	3356561	37411	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	2	1	6	3.9	CCC1(C)Cc2c(sc3nc(SC)nc(S)c23)CO1	nan
	CHEMBL1457175	37411	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	2	1	6	3.9	CCC1(C)Cc2c(sc3nc(SC)nc(S)c23)CO1	nan
	16018620	37422	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	4	1	6	4.2	O=C(CSc1nncn2c1cc1occc12)Nc1ccccc1C(F)(F)F	nan
	CHEMBL1457242	37422	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	4	1	6	4.2	O=C(CSc1nncn2c1cc1occc12)Nc1ccccc1C(F)(F)F	nan
	24686163	37513	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	6	1	3	5.1	CCN(CC)C(=O)c1ccc(NC(=O)c2sccc2-c2ccccc2)cc1	nan
	CHEMBL1457962	37513	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	6	1	3	5.1	CCN(CC)C(=O)c1ccc(NC(=O)c2sccc2-c2ccccc2)cc1	nan
	3927980	37550	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	8	1	6	3.1	CCCN1C(=O)C2(C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2CCCOC)c2ccccc21	nan
	CHEMBL1458233	37550	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	8	1	6	3.1	CCCN1C(=O)C2(C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2CCCOC)c2ccccc21	nan
	4962629	37584	19	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	351	3	1	4	3.5	Cc1cc(F)ccc1S(=O)(=O)Nc1nc2ccccc2nc1Cl	nan
	CHEMBL1458588	37584	19	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	351	3	1	4	3.5	Cc1cc(F)ccc1S(=O)(=O)Nc1nc2ccccc2nc1Cl	nan
	6460246	37585	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	258	2	0	5	3.1	Cc1nnc2c(SC(C)C)nc3ccccc3n12	nan
	CHEMBL1458589	37585	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	258	2	0	5	3.1	Cc1nnc2c(SC(C)C)nc3ccccc3n12	nan
	7475827	37664	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	5	0	9	0.2	CC(C)Cc1nc(SCC(=O)N2CCOCC2)c2c(=O)n(C)c(=O)n(C)c2n1	nan
	CHEMBL1459222	37664	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	5	0	9	0.2	CC(C)Cc1nc(SCC(=O)N2CCOCC2)c2c(=O)n(C)c(=O)n(C)c2n1	nan
	3239559	37773	4	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	219	2	0	3	3.4	CCn1c(=S)ccc2ccc(OC)cc21	nan
	CHEMBL1460186	37773	4	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	219	2	0	3	3.4	CCn1c(=S)ccc2ccc(OC)cc21	nan
	4091063	37879	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	6	1	7	2.1	COC(=O)c1ccc(NC(=O)C(=O)c2cn(CC(=O)N3CCOCC3)c3ccccc23)cc1	nan
	CHEMBL1461057	37879	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	6	1	7	2.1	COC(=O)c1ccc(NC(=O)C(=O)c2cn(CC(=O)N3CCOCC3)c3ccccc23)cc1	nan
	135413805	37987	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	297	3	3	9	1.2	N#Cc1cc(Nc2c(N)ncnc2O)c([N+](=O)[O-])cc1C#N	nan
	CHEMBL1462053	37987	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	297	3	3	9	1.2	N#Cc1cc(Nc2c(N)ncnc2O)c([N+](=O)[O-])cc1C#N	nan
	4636986	38069	15	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	509	8	2	10	0.2	Cc1cccn2c(=O)c3cc(C(=O)NCCN4CCOCC4)c(=N)n(CCCN4CCOCC4)c3nc12	nan
	CHEMBL1462720	38069	15	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	509	8	2	10	0.2	Cc1cccn2c(=O)c3cc(C(=O)NCCN4CCOCC4)c(=N)n(CCCN4CCOCC4)c3nc12	nan
	993137	38106	17	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	5	1	5	3.4	CC(=O)c1sc(NC(=O)COc2ccc(Br)cc2)nc1C	nan
	CHEMBL1463012	38106	17	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	5	1	5	3.4	CC(=O)c1sc(NC(=O)COc2ccc(Br)cc2)nc1C	nan
	2225463	38160	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	336	5	1	3	3.3	O=C(NCCCN1CCCC1=O)c1sc2ccccc2c1Cl	nan
	CHEMBL1463545	38160	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	336	5	1	3	3.3	O=C(NCCCN1CCCC1=O)c1sc2ccccc2c1Cl	nan
	6184422	38231	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	522	10	1	8	3.5	CCCCOc1cccc(C2C(C(=O)c3ccc4c(c3)OCCO4)=C(O)C(=O)N2CCN2CCOCC2)c1	nan
	CHEMBL1464067	38231	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	522	10	1	8	3.5	CCCCOc1cccc(C2C(C(=O)c3ccc4c(c3)OCCO4)=C(O)C(=O)N2CCN2CCOCC2)c1	nan
	135449395	38238	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	5	2	8	3.1	CCN(Cc1nc(O)c2ccccc2n1)Cc1nc(O)c2sccc2n1	nan
	CHEMBL1464106	38238	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	5	2	8	3.1	CCN(Cc1nc(O)c2ccccc2n1)Cc1nc(O)c2sccc2n1	nan
	5778449	38326	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	7	1	8	0.8	CCN1CCN(c2nc3c(C)cccn3c(=O)c2/C=C(\C#N)C(=O)NCCOC)CC1	nan
	CHEMBL1464778	38326	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	7	1	8	0.8	CCN1CCN(c2nc3c(C)cccn3c(=O)c2/C=C(\C#N)C(=O)NCCOC)CC1	nan
	2457314	38337	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	7	1	10	0.1	COc1ccc(OC)c(/C=C/C(=O)OCC(=O)c2c(N)n(C)c(=O)n(C)c2=O)c1	nan
	CHEMBL1464838	38337	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	7	1	10	0.1	COc1ccc(OC)c(/C=C/C(=O)OCC(=O)c2c(N)n(C)c(=O)n(C)c2=O)c1	nan
	3791918	38348	20	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	245	1	2	3	3.1	Sc1n[nH]c(-c2cc(Cl)ccc2Cl)n1	nan
	CHEMBL1464872	38348	20	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	245	1	2	3	3.1	Sc1n[nH]c(-c2cc(Cl)ccc2Cl)n1	nan
	985269	38393	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	3	0	5	4.7	c1ccc(-c2cc3c(N4CCN(c5ccccc5)CC4)ncnc3s2)cc1	nan
	CHEMBL1465210	38393	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	3	0	5	4.7	c1ccc(-c2cc3c(N4CCN(c5ccccc5)CC4)ncnc3s2)cc1	nan
	1435001	38469	4	None	-3	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	396	6	2	6	2.8	CCc1nc(SCC(=O)NNC(=O)c2ccc(OC)cc2)c2ccccc2n1	nan
	CHEMBL1465814	38469	4	None	-3	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	396	6	2	6	2.8	CCc1nc(SCC(=O)NNC(=O)c2ccc(OC)cc2)c2ccccc2n1	nan
	1479844	38507	15	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	318	3	0	4	5.2	CSc1nc(Sc2ccccc2Cl)c2ccccc2n1	nan
	CHEMBL1466134	38507	15	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	318	3	0	4	5.2	CSc1nc(Sc2ccccc2Cl)c2ccccc2n1	nan
	1836205	38510	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	7	1	8	0.8	COCCCNC(=O)/C(C#N)=C/c1c(N2CCN(C)CC2)nc2c(C)cccn2c1=O	nan
	CHEMBL1466152	38510	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	7	1	8	0.8	COCCCNC(=O)/C(C#N)=C/c1c(N2CCN(C)CC2)nc2c(C)cccn2c1=O	nan
	2982726	38545	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	6	2	7	1.1	CCOC(=O)C1=C(CN2CCOCC2)NC(=O)NC1c1cccc([N+](=O)[O-])c1	nan
	CHEMBL1466461	38545	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	6	2	7	1.1	CCOC(=O)C1=C(CN2CCOCC2)NC(=O)NC1c1cccc([N+](=O)[O-])c1	nan
	5831389	38610	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	442	5	1	6	3.9	Cc1ccc(C2C(C(=O)c3ccc4c(c3)OCCO4)=C(O)C(=O)N2Cc2cccnc2)cc1	nan
	CHEMBL1466919	38610	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	442	5	1	6	3.9	Cc1ccc(C2C(C(=O)c3ccc4c(c3)OCCO4)=C(O)C(=O)N2Cc2cccnc2)cc1	nan
	2161641	38666	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	7	2	7	3.0	CCOc1ncccc1C(=O)Nc1ccc(S(=O)(=O)Nc2nccs2)cc1	nan
	CHEMBL1467371	38666	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	7	2	7	3.0	CCOc1ncccc1C(=O)Nc1ccc(S(=O)(=O)Nc2nccs2)cc1	nan
	2146410	38668	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	4	1	2	3.3	CCNC(=O)Cc1c(OC)ccc2cc(Br)ccc12	nan
	CHEMBL1467397	38668	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	4	1	2	3.3	CCNC(=O)Cc1c(OC)ccc2cc(Br)ccc12	nan
	5028075	38704	5	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	7	1	6	3.9	COc1ccc(NC(=O)COC(=O)c2cc(SC)ccc2Cl)c(OC)c1	nan
	CHEMBL1467702	38704	5	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	7	1	6	3.9	COc1ccc(NC(=O)COC(=O)c2cc(SC)ccc2Cl)c(OC)c1	nan
	5786830	38715	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	5	1	6	3.4	COc1ccc(C(=O)C2=C(O)C(=O)N(c3ncccn3)C2c2ccc(F)cc2)cc1	nan
	CHEMBL1467854	38715	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	5	1	6	3.4	COc1ccc(C(=O)C2=C(O)C(=O)N(c3ncccn3)C2c2ccc(F)cc2)cc1	nan
	652110	38803	4	None	-2	3	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	276	4	0	5	3.0	COC(=O)CSc1nc(C(C)C)nc2ccccc12	nan
	CHEMBL1468599	38803	4	None	-2	3	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	276	4	0	5	3.0	COC(=O)CSc1nc(C(C)C)nc2ccccc12	nan
	20904121	38877	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	6	1	8	1.7	CC(=O)c1cccc(NC(=O)CCc2nnc3ccc(N4CCOCC4)nn23)c1	nan
	CHEMBL1469174	38877	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	6	1	8	1.7	CC(=O)c1cccc(NC(=O)CCc2nnc3ccc(N4CCOCC4)nn23)c1	nan
	5726945	38891	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	266	3	0	4	3.5	CC(=O)c1ccc(/C=C/c2nc3ccccc3n2C)o1	nan
	CHEMBL1469326	38891	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	266	3	0	4	3.5	CC(=O)c1ccc(/C=C/c2nc3ccccc3n2C)o1	nan
	3812545	38997	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	6	1	8	3.7	COc1ccc(OC)c(C2C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2c2cc(C)on2)c1	nan
	CHEMBL1470290	38997	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	6	1	8	3.7	COc1ccc(OC)c(C2C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2c2cc(C)on2)c1	nan
	2964736	39013	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	436	5	1	8	4.6	COc1cccc2cc(C(=O)C3=C(O)C(=O)N(c4cc(C)on4)C3c3cccs3)oc12	nan
	CHEMBL1470378	39013	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	436	5	1	8	4.6	COc1cccc2cc(C(=O)C3=C(O)C(=O)N(c4cc(C)on4)C3c3cccs3)oc12	nan
	15988466	39270	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	4	1	7	2.3	COc1ccc(NC(=O)Cn2c(=O)c3cc(Cl)ccc3n3nncc23)cc1	nan
	CHEMBL1472605	39270	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	4	1	7	2.3	COc1ccc(NC(=O)Cn2c(=O)c3cc(Cl)ccc3n3nncc23)cc1	nan
	16011470	39286	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	508	10	1	6	5.8	COc1ccc(CCNC(=O)c2ccc(Cn3c(SCc4ccccc4)nc4cccnc43)cc2)cc1	nan
	CHEMBL1472792	39286	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	508	10	1	6	5.8	COc1ccc(CCNC(=O)c2ccc(Cn3c(SCc4ccccc4)nc4cccnc43)cc2)cc1	nan
	6229347	39366	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	6	2	5	3.0	COc1ccccc1CCNC(=O)Cc1c(C)c2c(O)cc(C)cc2oc1=O	nan
	CHEMBL1473886	39366	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	6	2	5	3.0	COc1ccccc1CCNC(=O)Cc1c(C)c2c(O)cc(C)cc2oc1=O	nan
	20886471	39378	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	7	1	4	4.3	CCCOc1ccc(CNC(=O)c2ccc3c(c2)N(CC)CCS3)cc1	nan
	CHEMBL1474147	39378	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	7	1	4	4.3	CCCOc1ccc(CNC(=O)c2ccc3c(c2)N(CC)CCS3)cc1	nan
	15988056	39439	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	7	2	4	3.5	CCCCCn1c(=O)[nH]c2cc(C(=O)NCc3ccc(Cl)cc3)ccc2c1=O	nan
	CHEMBL1475000	39439	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	7	2	4	3.5	CCCCCn1c(=O)[nH]c2cc(C(=O)NCc3ccc(Cl)cc3)ccc2c1=O	nan
	5297460	39450	18	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	326	5	1	5	4.0	CCOc1ccc(-c2oc3ccccc3c(=O)c2O)cc1OCC	nan
	CHEMBL1475143	39450	18	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	326	5	1	5	4.0	CCOc1ccc(-c2oc3ccccc3c(=O)c2O)cc1OCC	nan
	16018222	39459	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	4	1	5	3.0	COc1cccc(NC(=O)Cn2c(=O)c3cccn3c3ccc(F)cc32)c1	nan
	CHEMBL1475268	39459	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	4	1	5	3.0	COc1cccc(NC(=O)Cn2c(=O)c3cccn3c3ccc(F)cc32)c1	nan
	135410479	39469	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	4	2	4	5.5	Cc1ccc(NC(=O)c2cnn3c2NC(c2ccccc2)=CC3c2ccccc2)cc1	nan
	CHEMBL1475406	39469	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	4	2	4	5.5	Cc1ccc(NC(=O)c2cnn3c2NC(c2ccccc2)=CC3c2ccccc2)cc1	nan
	16031507	39470	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	6	1	6	4.1	COc1ccc(-c2nnc(SCC(=O)Nc3cccc(F)c3)s2)cc1	nan
	CHEMBL1475415	39470	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	6	1	6	4.1	COc1ccc(-c2nnc(SCC(=O)Nc3cccc(F)c3)s2)cc1	nan
	16015334	39533	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	460	6	1	6	5.7	COc1ccc(Cc2c(C)nn(-c3nc(C)c(C(=O)Nc4ccc(C)cc4C)s3)c2C)cc1	nan
	CHEMBL1476342	39533	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	460	6	1	6	5.7	COc1ccc(Cc2c(C)nn(-c3nc(C)c(C(=O)Nc4ccc(C)cc4C)s3)c2C)cc1	nan
	2033254	39579	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	351	6	1	7	2.8	CSc1nc(NCCCN(C)C)c2c3c(sc2n1)CN(C)CC3	nan
	CHEMBL1476899	39579	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	351	6	1	7	2.8	CSc1nc(NCCCN(C)C)c2c3c(sc2n1)CN(C)CC3	nan
	1138445	39677	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	7	2	9	1.5	CCCn1c(SCC(=O)Nc2ccc(NC(C)=O)cc2)nc2c1c(=O)n(C)c(=O)n2C	nan
	CHEMBL1477799	39677	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	7	2	9	1.5	CCCn1c(SCC(=O)Nc2ccc(NC(C)=O)cc2)nc2c1c(=O)n(C)c(=O)n2C	nan
	1442565	39720	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	6	0	5	3.9	CCOC(=O)CSc1nc(Cc2ccccc2)nc2ccccc12	nan
	CHEMBL1478306	39720	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	6	0	5	3.9	CCOC(=O)CSc1nc(Cc2ccccc2)nc2ccccc12	nan
	1005239	39814	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	2	1	5	5.8	N#Cc1sc2nc(-c3cccs3)cc(-c3ccc(Cl)cc3)c2c1N	nan
	CHEMBL1479144	39814	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	2	1	5	5.8	N#Cc1sc2nc(-c3cccs3)cc(-c3ccc(Cl)cc3)c2c1N	nan
	16018188	39842	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	9	1	5	3.8	CCOc1ccc(CCNC(=O)CCCn2c(=O)c3cccn3c3ccccc32)cc1	nan
	CHEMBL1479369	39842	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	9	1	5	3.8	CCOc1ccc(CCNC(=O)CCCn2c(=O)c3cccn3c3ccccc32)cc1	nan
	5914213	40332	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	5	2	7	3.3	O=C(C1=C(O)C(=O)N(Cc2ccncc2)C1c1cccc(O)c1)c1ccc2c(c1)OCCO2	nan
	CHEMBL1483546	40332	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	5	2	7	3.3	O=C(C1=C(O)C(=O)N(Cc2ccncc2)C1c1cccc(O)c1)c1ccc2c(c1)OCCO2	nan
	796660	40416	4	None	1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	3	0	5	2.9	COc1cc2oc(=O)c(Br)c(C)c2c(OC)c1OC	nan
	CHEMBL1484186	40416	4	None	1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	3	0	5	2.9	COc1cc2oc(=O)c(Br)c(C)c2c(OC)c1OC	nan
	16025365	40490	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	564	7	1	7	5.4	CC(=O)c1cccc(NC(=O)CSc2ncc3c(n2)-c2cc(Cl)ccc2N(Cc2ccccc2)S3(=O)=O)c1	nan
	CHEMBL1484843	40490	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	564	7	1	7	5.4	CC(=O)c1cccc(NC(=O)CSc2ncc3c(n2)-c2cc(Cl)ccc2N(Cc2ccccc2)S3(=O)=O)c1	nan
	2881633	40516	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	3	2	5	2.3	Cc1nnc(Nc2ccc(S(N)(=O)=O)cc2)c2ccccc12	nan
	CHEMBL1485038	40516	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	3	2	5	2.3	Cc1nnc(Nc2ccc(S(N)(=O)=O)cc2)c2ccccc12	nan
	16020293	40548	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	562	8	2	7	4.3	COc1ccc(-n2c(=O)c3ccc(C(=O)NCc4ccc(C)cc4)cc3n(CC(=O)Nc3ccc(C)cc3)c2=O)cc1	nan
	CHEMBL1485379	40548	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	562	8	2	7	4.3	COc1ccc(-n2c(=O)c3ccc(C(=O)NCc4ccc(C)cc4)cc3n(CC(=O)Nc3ccc(C)cc3)c2=O)cc1	nan
	866572	40596	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	1	0	6	1.3	CN1CCN(C(=O)c2cc3c(=O)n4ccccc4nc3s2)CC1	nan
	CHEMBL1485808	40596	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	1	0	6	1.3	CN1CCN(C(=O)c2cc3c(=O)n4ccccc4nc3s2)CC1	nan
	15991110	40615	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	5	1	3	5.2	Cc1ccc2c(c1)c(=O)c1ccccc1n2CCCC(=O)Nc1c(F)cccc1F	nan
	CHEMBL1485996	40615	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	5	1	3	5.2	Cc1ccc2c(c1)c(=O)c1ccccc1n2CCCC(=O)Nc1c(F)cccc1F	nan
	20869704	40619	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	7	1	10	-0.3	CCOC(=O)CNC(=O)Cn1cnc2c(nnn2-c2cccc(OC)c2)c1=O	nan
	CHEMBL1486007	40619	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	7	1	10	-0.3	CCOC(=O)CNC(=O)Cn1cnc2c(nnn2-c2cccc(OC)c2)c1=O	nan
	2951279	40620	13	None	-3	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	6	1	7	4.2	COc1cccc2cc(C(=O)C3=C(O)C(=O)N(Cc4ccco4)C3c3cccnc3)oc12	nan
	CHEMBL1486010	40620	13	None	-3	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	6	1	7	4.2	COc1cccc2cc(C(=O)C3=C(O)C(=O)N(Cc4ccco4)C3c3cccnc3)oc12	nan
	3647805	40707	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	8	2	4	3.1	CCCCC(CC)CNC(=O)CC1N=C2c3ccccc3NC(=S)N2C1=O	nan
	CHEMBL1486794	40707	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	8	2	4	3.1	CCCCC(CC)CNC(=O)CC1N=C2c3ccccc3NC(=S)N2C1=O	nan
	3149629	40758	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	266	3	1	5	2.4	O=C(O)CSc1ncnc2sc3c(c12)CCC3	nan
	CHEMBL1487236	40758	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	266	3	1	5	2.4	O=C(O)CSc1ncnc2sc3c(c12)CCC3	nan
	6296199	40769	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	506	9	1	8	2.9	C=CCOc1cccc(C2C(C(=O)c3ccc4c(c3)OCCO4)=C(O)C(=O)N2CCN2CCOCC2)c1	nan
	CHEMBL1487315	40769	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	506	9	1	8	2.9	C=CCOc1cccc(C2C(C(=O)c3ccc4c(c3)OCCO4)=C(O)C(=O)N2CCN2CCOCC2)c1	nan
	3494131	40962	15	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	4	1	7	4.6	Cc1cc(N2C(=O)C(O)=C(C(=O)c3cc4ccccc4o3)C2c2cccs2)no1	nan
	CHEMBL1488696	40962	15	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	4	1	7	4.6	Cc1cc(N2C(=O)C(O)=C(C(=O)c3cc4ccccc4o3)C2c2cccs2)no1	nan
	16016559	41016	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	311	3	1	4	3.7	Cc1ccc(-c2nonc2NC(=O)c2ccc(F)cc2)cc1C	nan
	CHEMBL1489095	41016	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	311	3	1	4	3.7	Cc1ccc(-c2nonc2NC(=O)c2ccc(F)cc2)cc1C	nan
	4604410	41182	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	5	1	4	3.1	Cc1c(Cl)cccc1NC(=O)CCCN1C(=O)c2cccnc2C1=O	nan
	CHEMBL1490398	41182	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	5	1	4	3.1	Cc1c(Cl)cccc1NC(=O)CCCN1C(=O)c2cccnc2C1=O	nan
	15992220	41191	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	262	1	2	4	0.9	CC(=O)N=C(N)Nc1nc(=O)c2ccccc2s1	nan
	3862718	41191	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	262	1	2	4	0.9	CC(=O)N=C(N)Nc1nc(=O)c2ccccc2s1	nan
	5941821	41191	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	262	1	2	4	0.9	CC(=O)N=C(N)Nc1nc(=O)c2ccccc2s1	nan
	CHEMBL1490493	41191	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	262	1	2	4	0.9	CC(=O)N=C(N)Nc1nc(=O)c2ccccc2s1	nan
	5307465	41324	0	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	300	1	0	6	2.5	Cc1sc2nc3ccc(N4CCCC4)nn3c(=O)c2c1C	nan
	CHEMBL1491386	41324	0	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	300	1	0	6	2.5	Cc1sc2nc3ccc(N4CCCC4)nn3c(=O)c2c1C	nan
	648659	41391	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	5	0	8	1.5	CCCn1c(SCC(=O)N2CCc3ccccc3C2)nc2c1c(=O)n(C)c(=O)n2C	nan
	CHEMBL1491811	41391	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	5	0	8	1.5	CCCn1c(SCC(=O)N2CCc3ccccc3C2)nc2c1c(=O)n(C)c(=O)n2C	nan
	3240716	41406	8	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	11	2	7	3.9	CCOc1cc2[nH]c(=S)n(CCCCC(=O)NCc3ccco3)c(=O)c2cc1OCC	nan
	CHEMBL1491907	41406	8	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	11	2	7	3.9	CCOc1cc2[nH]c(=S)n(CCCCC(=O)NCc3ccco3)c(=O)c2cc1OCC	nan
	20917809	41430	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	6	1	6	2.1	O=C1c2cccnc2C(=O)N1Cc1ccc(F)cc1S(=O)(=O)NCc1ccco1	nan
	CHEMBL1492082	41430	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	6	1	6	2.1	O=C1c2cccnc2C(=O)N1Cc1ccc(F)cc1S(=O)(=O)NCc1ccco1	nan
	6533452	41443	16	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	361	4	1	4	4.4	COc1ccc(/C=C2\CCc3c2nc2ccccc2c3C(=O)O)cc1OC	nan
	CHEMBL1492209	41443	16	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	361	4	1	4	4.4	COc1ccc(/C=C2\CCc3c2nc2ccccc2c3C(=O)O)cc1OC	nan
	135414697	41456	12	None	-3	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	4	1	6	3.7	N#Cc1c(O)nc(SCc2ccc(F)cc2)nc1-c1ccco1	nan
	CHEMBL1492324	41456	12	None	-3	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	4	1	6	3.7	N#Cc1c(O)nc(SCc2ccc(F)cc2)nc1-c1ccco1	nan
	3151464	41493	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	6	2	7	2.1	COCCCn1c(=N)c(C(=O)NC2CCCC2)cc2c(=O)n3cccc(C)c3nc21	nan
	CHEMBL1492596	41493	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	6	2	7	2.1	COCCCn1c(=N)c(C(=O)NC2CCCC2)cc2c(=O)n3cccc(C)c3nc21	nan
	3241814	41499	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	326	3	1	6	1.1	Cn1c(C(=O)NCC2CCCO2)cc2c(=O)n3ccccc3nc21	nan
	CHEMBL1492641	41499	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	326	3	1	6	1.1	Cn1c(C(=O)NCC2CCCO2)cc2c(=O)n3ccccc3nc21	nan
	4118355	41586	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	3	1	4	4.7	Cc1ccc(C(C)(C)C)cc1S(=O)(=O)Nc1nc2ccccc2nc1Cl	nan
	CHEMBL1493417	41586	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	3	1	4	4.7	Cc1ccc(C(C)(C)C)cc1S(=O)(=O)Nc1nc2ccccc2nc1Cl	nan
	7899292	41593	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	6	1	8	1.5	COc1cccc(C(=O)NCC(=O)OCc2cc(=O)n3c(C)csc3n2)c1	nan
	CHEMBL1493482	41593	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	6	1	8	1.5	COc1cccc(C(=O)NCC(=O)OCc2cc(=O)n3c(C)csc3n2)c1	nan
	16014523	41654	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	3	1	5	4.8	Cc1cc(Nc2ccc(C)c(Cl)c2)n2nc(-c3ccccc3)nc2n1	nan
	CHEMBL1494140	41654	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	3	1	5	4.8	Cc1cc(Nc2ccc(C)c(Cl)c2)n2nc(-c3ccccc3)nc2n1	nan
	4578483	41682	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	510	5	1	6	6.0	COc1ccc(-c2cc(C(F)(F)F)n3nc(C(=O)Nc4cccc(Cl)c4Cl)cc3n2)cc1OC	nan
	CHEMBL1494437	41682	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	510	5	1	6	6.0	COc1ccc(-c2cc(C(F)(F)F)n3nc(C(=O)Nc4cccc(Cl)c4Cl)cc3n2)cc1OC	nan
	2740372	41697	10	None	-3	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	317	3	0	5	3.8	CCOC(=O)c1csc(-c2sccc2Br)n1	nan
	CHEMBL1494595	41697	10	None	-3	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	317	3	0	5	3.8	CCOC(=O)c1csc(-c2sccc2Br)n1	nan
	6245779	41722	12	None	-3	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	491	8	1	6	5.1	Cc1cc(OCc2ccccc2)ccc1C(=O)C1=C(O)C(=O)N(Cc2cccnc2)C1c1ccncc1	nan
	CHEMBL1494772	41722	12	None	-3	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	491	8	1	6	5.1	Cc1cc(OCc2ccccc2)ccc1C(=O)C1=C(O)C(=O)N(Cc2cccnc2)C1c1ccncc1	nan
	2961508	41771	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	4	2	5	3.4	N=C(NOC(=O)COc1ccc2ccccc2c1Br)c1ccncc1	nan
	5740308	41771	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	4	2	5	3.4	N=C(NOC(=O)COc1ccc2ccccc2c1Br)c1ccncc1	nan
	9587859	41771	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	4	2	5	3.4	N=C(NOC(=O)COc1ccc2ccccc2c1Br)c1ccncc1	nan
	CHEMBL1495283	41771	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	4	2	5	3.4	N=C(NOC(=O)COc1ccc2ccccc2c1Br)c1ccncc1	nan
	7743649	41876	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	4	1	4	4.3	Cc1cc(SCC(=O)NC2(C#N)CCCCC2)nc2c(C)cccc12	nan
	CHEMBL1496365	41876	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	4	1	4	4.3	Cc1cc(SCC(=O)NC2(C#N)CCCCC2)nc2c(C)cccc12	nan
	7709279	41933	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	4	1	7	3.1	COc1ccc2c(c1)c1nc3n(c(=O)c1n2CC(=O)Nc1ccccc1)CCS3	nan
	CHEMBL1496847	41933	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	4	1	7	3.1	COc1ccc2c(c1)c1nc3n(c(=O)c1n2CC(=O)Nc1ccccc1)CCS3	nan
	5760983	41934	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	512	4	1	4	5.4	O=C(C1=C(O)C(=O)N(c2ccccn2)C1c1ccc(Br)cc1)c1ccc(Br)cc1	nan
	CHEMBL1496850	41934	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	512	4	1	4	5.4	O=C(C1=C(O)C(=O)N(c2ccccn2)C1c1ccc(Br)cc1)c1ccc(Br)cc1	nan
	16195573	41967	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	9	2	7	3.2	CCOc1cc2[nH]c(=S)n(CCC(=O)NCc3ccco3)c(=O)c2cc1OCC	nan
	CHEMBL1497122	41967	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	9	2	7	3.2	CCOc1cc2[nH]c(=S)n(CCC(=O)NCc3ccco3)c(=O)c2cc1OCC	nan
	265605	42132	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	236	1	0	6	0.1	CC(C)c1nc2c(c(=O)n(C)c(=O)n2C)n1C	nan
	CHEMBL1498670	42132	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	236	1	0	6	0.1	CC(C)c1nc2c(c(=O)n(C)c(=O)n2C)n1C	nan
	20875207	42311	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	4	2	3	4.2	O=C(Nc1ccccc1F)c1oc2ccccc2c1NC(=O)C1CC1	nan
	CHEMBL1500175	42311	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	4	2	3	4.2	O=C(Nc1ccccc1F)c1oc2ccccc2c1NC(=O)C1CC1	nan
	17583267	42382	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	7	1	7	3.8	COc1cc(NC(=O)COc2cc(C)cc3oc(=O)c(C)c(C)c23)cc(OC)c1OC	nan
	CHEMBL1500728	42382	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	7	1	7	3.8	COc1cc(NC(=O)COc2cc(C)cc3oc(=O)c(C)c(C)c23)cc(OC)c1OC	nan
	2768366	42579	54	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	245	3	2	4	2.2	COc1ccc(-c2ccc(C(=O)O)c(O)n2)cc1	nan
	CHEMBL1502516	42579	54	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	245	3	2	4	2.2	COc1ccc(-c2ccc(C(=O)O)c(O)n2)cc1	nan
	859554	42631	13	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	334	4	1	7	3.3	Cc1cc(NC(=O)CSc2ncnc3sc(C)c(C)c23)no1	nan
	CHEMBL1503032	42631	13	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	334	4	1	7	3.3	Cc1cc(NC(=O)CSc2ncnc3sc(C)c(C)c23)no1	nan
	5294012	42711	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	6	2	7	4.0	CC(C)n1c2ccccc2c2nnc(SCC(=O)Nc3ccccc3C(=O)O)nc21	nan
	CHEMBL1503589	42711	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	6	2	7	4.0	CC(C)n1c2ccccc2c2nnc(SCC(=O)Nc3ccccc3C(=O)O)nc21	nan
	20956972	42892	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	5	1	7	1.9	Cc1ccc(NC(=O)CCc2nnc3ccc(N4CCN(C)CC4)nn23)cc1F	nan
	CHEMBL1505377	42892	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	5	1	7	1.9	Cc1ccc(NC(=O)CCc2nnc3ccc(N4CCN(C)CC4)nn23)cc1F	nan
	4157311	42902	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	511	5	0	9	4.0	O=c1c2sccc2nc(SCc2cc(=O)n3cc(Br)ccc3n2)n1Cc1ccccn1	nan
	CHEMBL1505478	42902	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	511	5	0	9	4.0	O=c1c2sccc2nc(SCc2cc(=O)n3cc(Br)ccc3n2)n1Cc1ccccn1	nan
	5936247	42903	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	6	1	7	3.6	COc1ccccc1C1C(C(=O)c2ccc3c(c2)OCCO3)=C(O)C(=O)N1Cc1cccnc1	nan
	CHEMBL1505481	42903	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	6	1	7	3.6	COc1ccccc1C1C(C(=O)c2ccc3c(c2)OCCO3)=C(O)C(=O)N1Cc1cccnc1	nan
	3152549	43132	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	5	1	5	3.7	O=C(C1=C(O)C(=O)N(CC2CCCO2)C1c1ccccc1Cl)c1ccco1	nan
	CHEMBL1507420	43132	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	5	1	5	3.7	O=C(C1=C(O)C(=O)N(CC2CCCO2)C1c1ccccc1Cl)c1ccco1	nan
	2905772	43149	18	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	6	1	11	-0.4	CCOC(=O)Cc1csc(NC(=O)Cn2cnc3c2c(=O)n(C)c(=O)n3C)n1	nan
	CHEMBL1507551	43149	18	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	6	1	11	-0.4	CCOC(=O)Cc1csc(NC(=O)Cn2cnc3c2c(=O)n(C)c(=O)n3C)n1	nan
	20888750	43161	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	5	0	8	1.8	CCS(=O)(=O)c1nc(S(=O)(=O)c2ccc(C)cc2)c(N2CCN(C)CC2)s1	nan
	CHEMBL1507635	43161	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	5	0	8	1.8	CCS(=O)(=O)c1nc(S(=O)(=O)c2ccc(C)cc2)c(N2CCN(C)CC2)s1	nan
	664007	43259	17	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	4	1	5	5.5	Cc1cc(NC(=O)c2ccc3nc(-c4ccccc4)c(-c4ccccc4)nc3c2)no1	nan
	CHEMBL1508441	43259	17	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	4	1	5	5.5	Cc1cc(NC(=O)c2ccc3nc(-c4ccccc4)c(-c4ccccc4)nc3c2)no1	nan
	1862355	43288	9	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	302	3	1	5	3.3	COc1ccc(-c2cc(-c3cccnc3)c(C#N)c(N)n2)cc1	nan
	CHEMBL1508668	43288	9	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	302	3	1	5	3.3	COc1ccc(-c2cc(-c3cccnc3)c(C#N)c(N)n2)cc1	nan
	6224737	43357	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	463	5	1	8	4.0	COc1cccc(C2C(C(=O)c3ccc4c(c3)CC(C)O4)=C(O)C(=O)N2c2nnc(C)s2)c1	nan
	CHEMBL1509331	43357	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	463	5	1	8	4.0	COc1cccc(C2C(C(=O)c3ccc4c(c3)CC(C)O4)=C(O)C(=O)N2c2nnc(C)s2)c1	nan
	22514400	43435	1	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	346	4	0	7	0.6	CCOC(=O)C1CCN(C(=O)Cn2nc(C)n3cccc3c2=O)CC1	nan
	CHEMBL1510088	43435	1	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	346	4	0	7	0.6	CCOC(=O)C1CCN(C(=O)Cn2nc(C)n3cccc3c2=O)CC1	nan
	4547589	43459	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	4	1	3	4.9	CC(C)(C)C(=O)C1=C(O)C(=O)N(Cc2ccccc2)C1c1ccccc1Cl	nan
	CHEMBL1510328	43459	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	4	1	3	4.9	CC(C)(C)C(=O)C1=C(O)C(=O)N(Cc2ccccc2)C1c1ccccc1Cl	nan
	24792485	43480	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	6	1	8	3.2	COc1cc2cc(C#N)c(SCC(=O)Nc3cc(C)on3)nc2cc1OC	nan
	CHEMBL1510493	43480	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	6	1	8	3.2	COc1cc2cc(C#N)c(SCC(=O)Nc3cc(C)on3)nc2cc1OC	nan
	6042599	43603	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	5	1	6	3.5	Cc1ccc(C2C(C(=O)c3ccc4c(c3)OCCO4)=C(O)C(=O)N2CC2CCCO2)cc1	nan
	CHEMBL1511435	43603	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	5	1	6	3.5	Cc1ccc(C2C(C(=O)c3ccc4c(c3)OCCO4)=C(O)C(=O)N2CC2CCCO2)cc1	nan
	16027534	43653	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	7	1	9	3.6	COc1ccc(C(=O)Nc2cccc(C(=O)OCc3cc(=O)n4nc(C5CC5)sc4n3)c2)cc1	nan
	CHEMBL1512013	43653	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	7	1	9	3.6	COc1ccc(C(=O)Nc2cccc(C(=O)OCc3cc(=O)n4nc(C5CC5)sc4n3)c2)cc1	nan
	16024951	43671	1	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	373	6	2	6	4.8	CCOc1ccc(Nc2nc(N)c(C(=O)c3ccccc3Cl)s2)cc1	nan
	CHEMBL1512414	43671	1	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	373	6	2	6	4.8	CCOc1ccc(Nc2nc(N)c(C(=O)c3ccccc3Cl)s2)cc1	nan
	4395410	43783	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	4	0	4	6.1	N#Cc1c(C(F)(F)F)cc(-c2cccs2)nc1SCc1ccc(F)cc1	nan
	CHEMBL1514024	43783	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	4	0	4	6.1	N#Cc1c(C(F)(F)F)cc(-c2cccs2)nc1SCc1ccc(F)cc1	nan
	16018164	43812	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	7	1	5	3.4	COc1ccccc1CNC(=O)CCCn1c(=O)c2cccn2c2ccccc21	nan
	CHEMBL1514529	43812	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	7	1	5	3.4	COc1ccccc1CNC(=O)CCCn1c(=O)c2cccn2c2ccccc21	nan
	4081154	43892	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	4	1	3	5.1	O=C(Nc1c(C(=O)c2ccccc2)oc2ccccc12)c1ccc(F)cc1	nan
	CHEMBL1515694	43892	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	4	1	3	5.1	O=C(Nc1c(C(=O)c2ccccc2)oc2ccccc12)c1ccc(F)cc1	nan
	135546812	43909	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	6	2	5	3.6	CCc1ccc(NC(=O)CSc2nc(-c3ccccc3)c(C#N)c(=O)[nH]2)cc1	nan
	CHEMBL1515954	43909	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	6	2	5	3.6	CCc1ccc(NC(=O)CSc2nc(-c3ccccc3)c(C#N)c(=O)[nH]2)cc1	nan
	16022285	43968	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	6	2	6	2.3	Cc1nc2cccnc2n1-c1cccc(C(=O)NCCc2ccc(S(N)(=O)=O)cc2)c1	nan
	CHEMBL1516713	43968	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	6	2	6	2.3	Cc1nc2cccnc2n1-c1cccc(C(=O)NCCc2ccc(S(N)(=O)=O)cc2)c1	nan
	1466061	43979	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	7	1	5	3.8	CCOc1ccc2nc(O)c(CN(CCc3ccccc3)C(=O)N3CCOCC3)cc2c1	nan
	CHEMBL1516817	43979	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	7	1	5	3.8	CCOc1ccc2nc(O)c(CN(CCc3ccccc3)C(=O)N3CCOCC3)cc2c1	nan
	3433386	44067	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	5	2	6	2.0	NS(=O)(=O)c1cccc(NC(=O)CSc2ncnc3ccccc23)c1	nan
	CHEMBL1517698	44067	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	5	2	6	2.0	NS(=O)(=O)c1cccc(NC(=O)CSc2ncnc3ccccc23)c1	nan
	16018535	44208	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	3	1	4	4.2	CC(=O)N1CCOc2cc(S(=O)(=O)Nc3cc(C(F)(F)F)ccc3Cl)c(C)cc21	nan
	CHEMBL1518991	44208	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	3	1	4	4.2	CC(=O)N1CCOc2cc(S(=O)(=O)Nc3cc(C(F)(F)F)ccc3Cl)c(C)cc21	nan
	2135572	44223	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	500	8	1	8	4.0	CCOc1ccc(C(=O)c2cn(CC(=O)Nc3ccc(OC)cc3)c3cc4c(cc3c2=O)OCO4)cc1	nan
	CHEMBL1519131	44223	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	500	8	1	8	4.0	CCOc1ccc(C(=O)c2cn(CC(=O)Nc3ccc(OC)cc3)c3cc4c(cc3c2=O)OCO4)cc1	nan
	16025796	44278	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	457	5	1	4	5.4	CC(NC(=O)C1CCN(C(=O)c2ccc(-n3ccc4ccccc43)s2)CC1)c1ccccc1	nan
	CHEMBL1519614	44278	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	457	5	1	4	5.4	CC(NC(=O)C1CCN(C(=O)c2ccc(-n3ccc4ccccc43)s2)CC1)c1ccccc1	nan
	16030429	44420	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	7	1	4	5.1	Cc1ccc(Cc2nc3ccccc3nc2SCC(=O)NCc2ccc(F)cc2)cc1	nan
	CHEMBL1520828	44420	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	7	1	4	5.1	Cc1ccc(Cc2nc3ccccc3nc2SCC(=O)NCc2ccc(F)cc2)cc1	nan
	15988916	44431	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	556	8	2	8	4.4	Cc1cc(C)c(NC(=O)Cn2c(=O)n(Cc3ccc(C(=O)NCc4ccco4)cc3)c(=O)c3sccc32)c(C)c1	nan
	CHEMBL1520905	44431	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	556	8	2	8	4.4	Cc1cc(C)c(NC(=O)Cn2c(=O)n(Cc3ccc(C(=O)NCc4ccco4)cc3)c(=O)c3sccc32)c(C)c1	nan
	289464	44479	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	300	1	1	1	4.5	O=C(O)c1cc2ccccc2c2cc(Br)ccc12	nan
	CHEMBL1521339	44479	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	300	1	1	1	4.5	O=C(O)c1cc2ccccc2c2cc(Br)ccc12	nan
	2745168	44538	18	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	238	3	1	6	1.2	COCc1nc(S)c(C#N)cc1C(=O)OC	nan
	CHEMBL1521853	44538	18	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	238	3	1	6	1.2	COCc1nc(S)c(C#N)cc1C(=O)OC	nan
	689389	44584	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	6	1	5	3.4	CCN(CC)CCNc1cc(C)c(C#N)c2nc3ccccc3n12	nan
	CHEMBL1522224	44584	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	6	1	5	3.4	CCN(CC)CCNc1cc(C)c(C#N)c2nc3ccccc3n12	nan
	1167955	44717	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	6	2	5	5.0	O=C(CSc1nc(-c2ccc(F)cc2)nc2ccc(F)cc12)Nc1cccc(C(=O)O)c1	nan
	CHEMBL1523483	44717	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	6	2	5	5.0	O=C(CSc1nc(-c2ccc(F)cc2)nc2ccc(F)cc12)Nc1cccc(C(=O)O)c1	nan
	17201681	44779	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	336	2	0	2	2.4	O=C(C1CC(=O)N(c2ccc(Br)cc2)C1)N1CCCC1	nan
	CHEMBL1524084	44779	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	336	2	0	2	2.4	O=C(C1CC(=O)N(c2ccc(Br)cc2)C1)N1CCCC1	nan
	16018239	44823	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	298	3	1	3	3.5	CCOc1ccc(NC(=O)N2CCOc3ccccc32)cc1	nan
	CHEMBL1524566	44823	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	298	3	1	3	3.5	CCOc1ccc(NC(=O)N2CCOc3ccccc32)cc1	nan
	818605	44848	18	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	295	4	0	4	2.3	COc1ccc(C=O)cc1CN1C(=O)c2ccccc2C1=O	nan
	CHEMBL1524802	44848	18	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	295	4	0	4	2.3	COc1ccc(C=O)cc1CN1C(=O)c2ccccc2C1=O	nan
	16015121	44867	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	6	1	6	4.0	COc1ccc(OCC(=O)Nc2nc(-c3ccc(Br)cc3)ns2)cc1	nan
	CHEMBL1525000	44867	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	6	1	6	4.0	COc1ccc(OCC(=O)Nc2nc(-c3ccc(Br)cc3)ns2)cc1	nan
	4624396	44893	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	6	1	6	4.1	CCOc1ccc(-c2csc(NC(=O)c3cccc(N4C(=O)CCC4=O)c3)n2)cc1	nan
	CHEMBL1525327	44893	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	6	1	6	4.1	CCOc1ccc(-c2csc(NC(=O)c3cccc(N4C(=O)CCC4=O)c3)n2)cc1	nan
	551547	44910	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	410	4	1	3	4.6	O=C(NCC1CCCO1)c1cc(-c2ccccc2)nc2ccc(Br)cc12	nan
	CHEMBL1525441	44910	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	410	4	1	3	4.6	O=C(NCC1CCCO1)c1cc(-c2ccccc2)nc2ccc(Br)cc12	nan
	2904040	44937	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	6	2	3	3.0	NS(=O)(=O)c1ccc(CCNC(=O)c2ccc(-c3ccccc3)cc2)cc1	nan
	CHEMBL1525655	44937	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	6	2	3	3.0	NS(=O)(=O)c1ccc(CCNC(=O)c2ccc(-c3ccccc3)cc2)cc1	nan
	2868184	44958	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	3	1	3	4.6	CC(=O)C1=C(O)C(=O)N(c2ccc(Br)cc2)C1c1ccc(Cl)cc1	nan
	CHEMBL1525829	44958	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	3	1	3	4.6	CC(=O)C1=C(O)C(=O)N(c2ccc(Br)cc2)C1c1ccc(Cl)cc1	nan
	16018537	44995	1	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	6	1	7	1.6	CCOC(=O)C1CCCN(C(=O)CCS(=O)(=O)c2cc3c(cc2Cl)NC(=O)CO3)C1	nan
	CHEMBL1526153	44995	1	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	6	1	7	1.6	CCOC(=O)C1CCCN(C(=O)CCS(=O)(=O)c2cc3c(cc2Cl)NC(=O)CO3)C1	nan
	3151412	45128	18	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	6	2	8	0.7	COCCn1c(=N)c(C(=O)NCC2CCCO2)cc2c(=O)n3ccccc3nc21	nan
	CHEMBL1527265	45128	18	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	6	2	8	0.7	COCCn1c(=N)c(C(=O)NCC2CCCO2)cc2c(=O)n3ccccc3nc21	nan
	3772745	45172	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	454	5	1	4	4.9	COc1cccc(-c2cc(C(=O)NCC3CCCO3)c3cc(Br)cc(C)c3n2)c1	nan
	CHEMBL1527660	45172	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	454	5	1	4	4.9	COc1cccc(-c2cc(C(=O)NCC3CCCO3)c3cc(Br)cc(C)c3n2)c1	nan
	1253448	45186	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	3	0	7	2.3	CCOC(=O)C1CCN(C(=O)c2cc3c(=O)n4ccccc4nc3s2)CC1	nan
	CHEMBL1527795	45186	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	3	0	7	2.3	CCOC(=O)C1CCN(C(=O)c2cc3c(=O)n4ccccc4nc3s2)CC1	nan
	661360	45193	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	4	1	7	1.5	COc1ccc(-n2ncc3c(N4CCC(C(N)=O)CC4)ncnc32)cc1	nan
	CHEMBL1527862	45193	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	4	1	7	1.5	COc1ccc(-n2ncc3c(N4CCC(C(N)=O)CC4)ncnc32)cc1	nan
	1077518	45284	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	4	2	6	2.5	CCCn1c(=N)c(C(=O)NC2CCCC2)cc2c(=O)n3cccc(C)c3nc21	nan
	CHEMBL1528629	45284	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	4	2	6	2.5	CCCn1c(=N)c(C(=O)NC2CCCC2)cc2c(=O)n3cccc(C)c3nc21	nan
	16813521	45328	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	440	8	1	8	1.8	COc1ccc(C(=O)NCCc2nnc3ccc(SCC(=O)N4CCCC4)nn23)cc1	nan
	CHEMBL1529059	45328	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	440	8	1	8	1.8	COc1ccc(C(=O)NCCc2nnc3ccc(SCC(=O)N4CCCC4)nn23)cc1	nan
	54694033	45353	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	326	5	2	5	2.6	CCCn1c(=O)c(C(=O)NCc2ccco2)c(O)c2ccccc21	nan
	CHEMBL1529241	45353	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	326	5	2	5	2.6	CCCn1c(=O)c(C(=O)NCc2ccco2)c(O)c2ccccc21	nan
	625773	45519	50	None	-3	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	289	2	1	3	4.3	O=C(O)c1cc(-c2ccc(Cl)s2)nc2ccccc12	nan
	CHEMBL153072	45519	50	None	-3	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	289	2	1	3	4.3	O=C(O)c1cc(-c2ccc(Cl)s2)nc2ccccc12	nan
	3151486	45537	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	8	2	8	1.8	CCOCCCn1c(=N)c(C(=O)NCC2CCCO2)cc2c(=O)n3cccc(C)c3nc21	nan
	CHEMBL1530888	45537	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	8	2	8	1.8	CCOCCCn1c(=N)c(C(=O)NCC2CCCO2)cc2c(=O)n3cccc(C)c3nc21	nan
	4216259	45575	7	None	-4	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	426	7	1	8	2.0	CCCCn1c(=O)[nH]c(=O)c2c1nc(Cn1ncc(Cl)c(Cl)c1=O)n2CCC	nan
	CHEMBL1531245	45575	7	None	-4	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	426	7	1	8	2.0	CCCCn1c(=O)[nH]c(=O)c2c1nc(Cn1ncc(Cl)c(Cl)c1=O)n2CCC	nan
	2737056	45662	46	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	191	1	0	4	1.4	O=C1CC(=O)c2c1cccc2[N+](=O)[O-]	nan
	CHEMBL1532031	45662	46	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	191	1	0	4	1.4	O=C1CC(=O)c2c1cccc2[N+](=O)[O-]	nan
	2085635	45713	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	2	0	5	2.9	Cc1ccc2nc(Cn3cc(C(F)(F)F)cc(Cl)c3=O)cc(=O)n2c1	nan
	CHEMBL1532467	45713	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	2	0	5	2.9	Cc1ccc2nc(Cn3cc(C(F)(F)F)cc(Cl)c3=O)cc(=O)n2c1	nan
	3721626	45744	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	324	3	0	5	3.9	COc1ccc2c(c1)c1ncnc(N(C)C3CCCCC3)c1n2C	nan
	CHEMBL1532723	45744	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	324	3	0	5	3.9	COc1ccc2c(c1)c1ncnc(N(C)C3CCCCC3)c1n2C	nan
	3312243	45985	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	461	5	2	7	2.5	Cc1cccn2c(=O)c3cc(C(=O)NCC4CCCO4)c(=N)n(Cc4ccc(F)cc4)c3nc12	nan
	CHEMBL1535016	45985	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	461	5	2	7	2.5	Cc1cccn2c(=O)c3cc(C(=O)NCC4CCCO4)c(=N)n(Cc4ccc(F)cc4)c3nc12	nan
	135403580	46085	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	7	2	7	4.6	N#Cc1c(O)nc(SCC(=O)Nc2ccc(OC(F)(F)Cl)cc2)nc1-c1ccccc1	nan
	CHEMBL1536174	46085	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	7	2	7	4.6	N#Cc1c(O)nc(SCC(=O)Nc2ccc(OC(F)(F)Cl)cc2)nc1-c1ccccc1	nan
	5310128	46101	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	6	1	8	1.6	O=C(CSc1ccc2nnc(-c3ccncc3)n2n1)NCC1CCCO1	nan
	CHEMBL1536319	46101	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	6	1	8	1.6	O=C(CSc1ccc2nnc(-c3ccncc3)n2n1)NCC1CCCO1	nan
	20878456	46134	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	3	0	8	2.3	Cc1ccc(S(=O)(=O)c2nnn3c2nc(N2CCOCC2)c2ccccc23)cc1	nan
	CHEMBL1536657	46134	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	3	0	8	2.3	Cc1ccc(S(=O)(=O)c2nnn3c2nc(N2CCOCC2)c2ccccc23)cc1	nan
	5059230	46145	3	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	4	2	5	2.5	N#CC1=C([C-](C#N)C#N)NC(O)(C2CC2)C([n+]2ccccc2)C1c1ccccc1F	nan
	CHEMBL1536738	46145	3	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	4	2	5	2.5	N#CC1=C([C-](C#N)C#N)NC(O)(C2CC2)C([n+]2ccccc2)C1c1ccccc1F	nan
	5235682	46213	18	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	4	1	6	4.0	Cc1cc(N2C(=O)C(O)=C(C(=O)c3ccco3)C2c2cccc(Cl)c2)no1	nan
	CHEMBL1537295	46213	18	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	4	1	6	4.0	Cc1cc(N2C(=O)C(O)=C(C(=O)c3ccco3)C2c2cccc(Cl)c2)no1	nan
	7190492	46384	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	7	1	8	3.3	CCOc1ccc(NC(=O)CSc2ccc3nnc(-c4ccccn4)n3n2)cc1	nan
	CHEMBL1538682	46384	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	7	1	8	3.3	CCOc1ccc(NC(=O)CSc2ccc3nnc(-c4ccccn4)n3n2)cc1	nan
	3220383	46458	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	7	1	6	3.3	CC(C)CC(OC(=O)c1nsc(Cl)c1Cl)C(=O)NCC1CCCO1	nan
	CHEMBL1539378	46458	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	7	1	6	3.3	CC(C)CC(OC(=O)c1nsc(Cl)c1Cl)C(=O)NCC1CCCO1	nan
	6133031	46486	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	6	1	7	2.4	O=C(C1=C(O)C(=O)N(CCN2CCOCC2)C1c1ccccc1)c1ccc2c(c1)OCCO2	nan
	CHEMBL1539594	46486	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	6	1	7	2.4	O=C(C1=C(O)C(=O)N(CCN2CCOCC2)C1c1ccccc1)c1ccc2c(c1)OCCO2	nan
	1567287	46591	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	4	1	6	-1.0	CN1C(=O)C(=CNCCN2CCOCC2)C(=O)N(C)C1=S	nan
	CHEMBL1540479	46591	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	4	1	6	-1.0	CN1C(=O)C(=CNCCN2CCOCC2)C(=O)N(C)C1=S	nan
	2983027	46608	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	5	1	6	1.8	O=C(NCc1cccnc1)c1cc([N+](=O)[O-])ccc1N1CCOCC1	nan
	CHEMBL1540590	46608	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	5	1	6	1.8	O=C(NCc1cccnc1)c1cc([N+](=O)[O-])ccc1N1CCOCC1	nan
	2431987	46633	19	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	310	4	1	5	3.0	COCCCn1c(=S)[nH]c2sc3c(c2c1=O)CCCC3	nan
	CHEMBL1540855	46633	19	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	310	4	1	5	3.0	COCCCn1c(=S)[nH]c2sc3c(c2c1=O)CCCC3	nan
	3833515	46658	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	7	1	7	5.1	C=CCOc1cccc(C2C(C(=O)c3cc4ccccc4o3)=C(O)C(=O)N2c2cc(C)on2)c1	nan
	CHEMBL1541029	46658	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	7	1	7	5.1	C=CCOc1cccc(C2C(C(=O)c3cc4ccccc4o3)=C(O)C(=O)N2c2cc(C)on2)c1	nan
	6273159	46744	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	7	1	6	4.6	CCOc1cccc(C2C(C(=O)c3ccc4c(c3)CC(C)O4)=C(O)C(=O)N2Cc2ccncc2)c1	nan
	CHEMBL1541682	46744	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	7	1	6	4.6	CCOc1cccc(C2C(C(=O)c3ccc4c(c3)CC(C)O4)=C(O)C(=O)N2Cc2ccncc2)c1	nan
	659524	46931	7	None	-3	3	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	1	0	3	4.1	Brc1cc(Br)c2ncnc(N3CCCCC3)c2c1	nan
	CHEMBL1543331	46931	7	None	-3	3	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	1	0	3	4.1	Brc1cc(Br)c2ncnc(N3CCCCC3)c2c1	nan
	16194876	47177	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	7	1	9	2.9	COc1ccc(OC)c(NC(=O)CSc2ccc3nnc(-c4cccnc4)n3n2)c1	nan
	CHEMBL1545182	47177	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	7	1	9	2.9	COc1ccc(OC)c(NC(=O)CSc2ccc3nnc(-c4cccnc4)n3n2)c1	nan
	2997987	47208	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	5	1	6	2.0	Cc1sc2ncnc(OCC(=O)NCC3CCCO3)c2c1C	nan
	CHEMBL1545423	47208	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	5	1	6	2.0	Cc1sc2ncnc(OCC(=O)NCC3CCCO3)c2c1C	nan
	16188698	47298	0	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	4	1	2	4.2	Cc1ccccc1CC1(CO)CCCN(C(=O)c2cc(Cl)ccc2F)C1	nan
	CHEMBL1546168	47298	0	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	4	1	2	4.2	Cc1ccccc1CC1(CO)CCCN(C(=O)c2cc(Cl)ccc2F)C1	nan
	5389436	47419	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	7	1	8	3.8	COc1cccc(C2C(C(=O)c3ccc(OC)c(OC)c3)=C(O)C(=O)N2c2cc(C)on2)c1	nan
	CHEMBL1547272	47419	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	7	1	8	3.8	COc1cccc(C2C(C(=O)c3ccc(OC)c(OC)c3)=C(O)C(=O)N2c2cc(C)on2)c1	nan
	16437942	47747	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	496	8	2	9	2.2	CCCS(=O)(=O)c1ncc(Cl)c(C(=O)Nc2ccc(S(=O)(=O)Nc3ncccn3)cc2)n1	nan
	CHEMBL1550174	47747	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	496	8	2	9	2.2	CCCS(=O)(=O)c1ncc(Cl)c(C(=O)Nc2ccc(S(=O)(=O)Nc3ncccn3)cc2)n1	nan
	3579665	47792	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	4	1	7	2.3	COC(=O)c1c(NC(=O)c2cccc(N3C(=O)CCC3=O)c2)sc2c1CCN(C(C)=O)C2	nan
	CHEMBL1550602	47792	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	4	1	7	2.3	COC(=O)c1c(NC(=O)c2cccc(N3C(=O)CCC3=O)c2)sc2c1CCN(C(C)=O)C2	nan
	5308895	47847	1	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	3	0	5	4.0	N#CC1=C2SCN(Cc3ccccc3)CN2C(=O)CC1c1cccs1	nan
	CHEMBL1551015	47847	1	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	3	0	5	4.0	N#CC1=C2SCN(Cc3ccccc3)CN2C(=O)CC1c1cccs1	nan
	16031535	47887	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	6	1	6	4.6	COc1ccc(-c2nnc(SCC(=O)Nc3ccc(C)c(C)c3)s2)cc1	nan
	CHEMBL1551622	47887	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	6	1	6	4.6	COc1ccc(-c2nnc(SCC(=O)Nc3ccc(C)c(C)c3)s2)cc1	nan
	16015115	47896	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	5	1	5	4.3	Cc1ccc(OCC(=O)Nc2nc(-c3ccc(Br)cc3)ns2)cc1	nan
	CHEMBL1551830	47896	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	5	1	5	4.3	Cc1ccc(OCC(=O)Nc2nc(-c3ccc(Br)cc3)ns2)cc1	nan
	15989679	47952	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	539	9	1	9	3.5	COc1ccc(NC(=O)Cn2c(=O)n(Cc3ccccc3Cl)c(=O)c3cc(OC)c(OC)cc32)cc1OC	nan
	CHEMBL1552471	47952	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	539	9	1	9	3.5	COc1ccc(NC(=O)Cn2c(=O)n(Cc3ccccc3Cl)c(=O)c3cc(OC)c(OC)cc32)cc1OC	nan
	16030838	47971	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	440	7	2	8	2.3	COc1ccc(-c2cc3ccc(O)c(CN4CCN(CCO)CC4)c3oc2=O)cc1OC	nan
	53229832	47971	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	440	7	2	8	2.3	COc1ccc(-c2cc3ccc(O)c(CN4CCN(CCO)CC4)c3oc2=O)cc1OC	nan
	CHEMBL1552774	47971	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	440	7	2	8	2.3	COc1ccc(-c2cc3ccc(O)c(CN4CCN(CCO)CC4)c3oc2=O)cc1OC	nan
	1004132	48005	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	4	2	4	4.9	Cc1ccc(CNC(=O)c2sc3nc(-c4ccc(F)cc4)ccc3c2N)cc1	nan
	CHEMBL1553209	48005	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	4	2	4	4.9	Cc1ccc(CNC(=O)c2sc3nc(-c4ccc(F)cc4)ccc3c2N)cc1	nan
	15988065	48008	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	2	1	8	3.6	O=c1c2cc3c(cc2nc2sc(Nc4ccc(F)c(Cl)c4)nn12)OCO3	nan
	CHEMBL1553232	48008	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	2	1	8	3.6	O=c1c2cc3c(cc2nc2sc(Nc4ccc(F)c(Cl)c4)nn12)OCO3	nan
	16008431	48015	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	4	0	5	4.1	O=C(c1ccc(F)cc1)c1cn(Cc2ccccc2)c2cc3c(cc2c1=O)OCO3	nan
	CHEMBL1553329	48015	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	4	0	5	4.1	O=C(c1ccc(F)cc1)c1cn(Cc2ccccc2)c2cc3c(cc2c1=O)OCO3	nan
	16018243	48018	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	302	1	1	2	4.1	Cc1c(Cl)cccc1NC(=O)N1CCOc2ccccc21	nan
	CHEMBL1553372	48018	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	302	1	1	2	4.1	Cc1c(Cl)cccc1NC(=O)N1CCOc2ccccc21	nan
	1364295	48048	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	410	5	2	5	5.3	O=C(COc1ccc(Cl)cc1)Nc1ccc(O)c(-c2nc3ccccc3s2)c1	nan
	CHEMBL1553843	48048	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	410	5	2	5	5.3	O=C(COc1ccc(Cl)cc1)Nc1ccc(O)c(-c2nc3ccccc3s2)c1	nan
	5302298	48058	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	2	2	5	5.5	Nc1c(C(=O)Nc2ccc(Cl)c(C(F)(F)F)c2)sc2nc3c(cc12)N1CCC3CC1	nan
	CHEMBL1554006	48058	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	2	2	5	5.5	Nc1c(C(=O)Nc2ccc(Cl)c(C(F)(F)F)c2)sc2nc3c(cc12)N1CCC3CC1	nan
	16018784	48072	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	7	1	8	3.8	CCc1nnc(SCC(=O)Nc2ccc(OC)c(OC)c2)c2cc3occc3n12	nan
	CHEMBL1554189	48072	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	7	1	8	3.8	CCc1nnc(SCC(=O)Nc2ccc(OC)c(OC)c2)c2cc3occc3n12	nan
	16018201	48113	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	4	1	3	3.8	Cc1ccc2c(c1)N(C(=O)N1CCC(C(=O)NCCc3ccccc3)CC1)CC(C)O2	nan
	CHEMBL1554848	48113	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	4	1	3	3.8	Cc1ccc2c(c1)N(C(=O)N1CCC(C(=O)NCCc3ccccc3)CC1)CC(C)O2	nan
	3151378	48189	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	4	2	7	2.9	Cc1cccn2c(=O)c3cc(C(=O)NCC4CCCO4)c(=N)n(C4CCCCC4)c3nc12	nan
	CHEMBL1555780	48189	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	4	2	7	2.9	Cc1cccn2c(=O)c3cc(C(=O)NCC4CCCO4)c(=N)n(C4CCCCC4)c3nc12	nan
	16019891	48391	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	478	6	0	9	5.1	CCC(=O)Oc1cc(C(C)(C)C)cc2cc(-c3nc(-c4ccc(OC)cc4OC)no3)c(=O)oc12	nan
	CHEMBL1557596	48391	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	478	6	0	9	5.1	CCC(=O)Oc1cc(C(C)(C)C)cc2cc(-c3nc(-c4ccc(OC)cc4OC)no3)c(=O)oc12	nan
	3239255	48481	1	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	6	1	7	3.8	COc1ccc(-c2nn(C)c3sc(C(=O)NCc4ccco4)cc23)cc1OC	nan
	CHEMBL1558431	48481	1	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	6	1	7	3.8	COc1ccc(-c2nn(C)c3sc(C(=O)NCc4ccco4)cc23)cc1OC	nan
	662047	48644	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	396	5	1	7	3.8	COc1cccc(C2C(C(=O)c3cccs3)=C(O)C(=O)N2c2cc(C)on2)c1	nan
	CHEMBL1559829	48644	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	396	5	1	7	3.8	COc1cccc(C2C(C(=O)c3cccs3)=C(O)C(=O)N2c2cc(C)on2)c1	nan
	2612492	48796	6	None	-1	3	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	4	1	7	3.9	Cc1nc(SCC(=O)Nc2cc(C)on2)c2c3c(sc2n1)CCCC3	nan
	CHEMBL1561287	48796	6	None	-1	3	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	4	1	7	3.9	Cc1nc(SCC(=O)Nc2cc(C)on2)c2c3c(sc2n1)CCCC3	nan
	670483	48806	35	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	271	2	1	4	3.4	Fc1cccc(-c2nnc(S)n2-c2ccccc2)c1	nan
	CHEMBL1561393	48806	35	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	271	2	1	4	3.4	Fc1cccc(-c2nnc(S)n2-c2ccccc2)c1	nan
	16025728	48913	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	457	5	1	6	5.8	COc1cccc2c1Oc1ncccc1N(c1ccc(C(=O)NCc3ccccc3C)s1)C2	nan
	CHEMBL1562331	48913	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	457	5	1	6	5.8	COc1cccc2c1Oc1ncccc1N(c1ccc(C(=O)NCc3ccccc3C)s1)C2	nan
	135788252	48960	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	4	1	8	3.1	COC(=O)c1cc(-c2ccc(OC)cc2F)nc2nc(SC)nc(O)c12	nan
	CHEMBL1562765	48960	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	4	1	8	3.1	COC(=O)c1cc(-c2ccc(OC)cc2F)nc2nc(SC)nc(O)c12	nan
	20956964	48961	0	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	6	0	9	0.6	CCOC(=O)C1CCN(C(=O)CCc2nnc3ccc(N4CCN(C)CC4)nn23)CC1	nan
	CHEMBL1562772	48961	0	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	6	0	9	0.6	CCOC(=O)C1CCN(C(=O)CCc2nnc3ccc(N4CCN(C)CC4)nn23)CC1	nan
	15988783	49006	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	567	7	1	10	2.8	Cc1sc2ncn(CC(=O)Nc3ccc(C(C)C)cc3)c(=O)c2c1S(=O)(=O)N1CCN(c2ncccn2)CC1	nan
	CHEMBL1563146	49006	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	567	7	1	10	2.8	Cc1sc2ncn(CC(=O)Nc3ccc(C(C)C)cc3)c(=O)c2c1S(=O)(=O)N1CCN(c2ncccn2)CC1	nan
	20923169	49063	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	5	0	6	2.6	COc1ccc(CN2C(=O)c3cccnc3C2=O)cc1S(=O)(=O)N1CC(C)CC(C)C1	nan
	CHEMBL1563711	49063	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	5	0	6	2.6	COc1ccc(CN2C(=O)c3cccnc3C2=O)cc1S(=O)(=O)N1CC(C)CC(C)C1	nan
	16009570	49199	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	5	1	6	4.2	Cc1cn2c(=O)cc(COc3cccc(NC(=O)c4ccccc4C)c3)nc2s1	nan
	CHEMBL1564898	49199	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	5	1	6	4.2	Cc1cn2c(=O)cc(COc3cccc(NC(=O)c4ccccc4C)c3)nc2s1	nan
	22517528	49211	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	4	1	6	3.0	CC1CCN(S(=O)(=O)c2nnc(NC(=O)c3ccccc3Br)s2)CC1	nan
	CHEMBL1564984	49211	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	4	1	6	3.0	CC1CCN(S(=O)(=O)c2nnc(NC(=O)c3ccccc3Br)s2)CC1	nan
	16001900	49648	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	8	2	8	3.6	COc1ccc(CCNc2nc(S)nc3cc(OC)c(OC)cc23)cc1OC	nan
	CHEMBL1568426	49648	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	8	2	8	3.6	COc1ccc(CCNc2nc(S)nc3cc(OC)c(OC)cc23)cc1OC	nan
	2952518	49717	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	571	9	3	9	6.0	CCOc1ccccc1NC(=O)CSC1=C(C#N)C(c2ccco2)C(C(=O)Nc2nc3ccccc3s2)=C(C)N1	nan
	CHEMBL1569028	49717	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	571	9	3	9	6.0	CCOc1ccccc1NC(=O)CSC1=C(C#N)C(c2ccco2)C(C(=O)Nc2nc3ccccc3s2)=C(C)N1	nan
	18562928	49731	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	454	8	1	8	2.2	COc1ccc(C(=O)NCCc2nnc3ccc(SCC(=O)N4CCCCC4)nn23)cc1	nan
	CHEMBL1569159	49731	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	454	8	1	8	2.2	COc1ccc(C(=O)NCCc2nnc3ccc(SCC(=O)N4CCCCC4)nn23)cc1	nan
	3152775	49956	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	446	4	2	7	5.0	Cc1ccc2nc(N3C(=O)C(O)=C(C(=O)c4ccc(C)o4)C3c3ccc(O)cc3)sc2c1	nan
	CHEMBL1571071	49956	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	446	4	2	7	5.0	Cc1ccc2nc(N3C(=O)C(O)=C(C(=O)c4ccc(C)o4)C3c3ccc(O)cc3)sc2c1	nan
	3564285	50248	13	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	6	1	5	4.3	CN(C)CCN1C(=O)C(O)=C(C(=O)c2cc3ccccc3o2)C1c1cccc(Br)c1	nan
	5036767	50248	13	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	6	1	5	4.3	CN(C)CCN1C(=O)C(O)=C(C(=O)c2cc3ccccc3o2)C1c1cccc(Br)c1	nan
	CHEMBL1573867	50248	13	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	6	1	5	4.3	CN(C)CCN1C(=O)C(O)=C(C(=O)c2cc3ccccc3o2)C1c1cccc(Br)c1	nan
	1325969	50260	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	7	0	7	5.3	COc1cc(-c2nnc(COc3ccc4cc(Br)ccc4c3)o2)cc(OC)c1OC	nan
	CHEMBL1574014	50260	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	7	0	7	5.3	COc1cc(-c2nnc(COc3ccc4cc(Br)ccc4c3)o2)cc(OC)c1OC	nan
	3613213	50424	11	None	-1000	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	5	2	3	4.6	O=C(O)CC(NC(=O)c1sc2ccccc2c1Cl)c1ccc(F)cc1	nan
	CHEMBL1575774	50424	11	None	-1000	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	5	2	3	4.6	O=C(O)CC(NC(=O)c1sc2ccccc2c1Cl)c1ccc(F)cc1	nan
	2352763	50452	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	309	5	1	4	2.6	NC(=O)COC(=O)CSc1cccc2cccc(Cl)c12	nan
	CHEMBL1576037	50452	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	309	5	1	4	2.6	NC(=O)COC(=O)CSc1cccc2cccc(Cl)c12	nan
	135433192	50743	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	286	3	1	4	3.8	Oc1nc(SCc2ccccc2F)nc2ccccc12	nan
	CHEMBL1578484	50743	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	286	3	1	4	3.8	Oc1nc(SCc2ccccc2F)nc2ccccc12	nan
	18107118	50761	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	5	1	5	2.9	COc1ccc(S(=O)(=O)N2CCCCCC2)cc1C(=O)Nc1ccccn1	nan
	CHEMBL1578588	50761	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	5	1	5	2.9	COc1ccc(S(=O)(=O)N2CCCCCC2)cc1C(=O)Nc1ccccn1	nan
	1838209	50807	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	446	6	2	8	1.2	N#C/C(=C\c1c(N2CCC(C(N)=O)CC2)nc2ccccn2c1=O)C(=O)NCc1ccco1	nan
	CHEMBL1578976	50807	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	446	6	2	8	1.2	N#C/C(=C\c1c(N2CCC(C(N)=O)CC2)nc2ccccn2c1=O)C(=O)NCc1ccco1	nan
	3802907	50874	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	510	6	1	6	4.1	O=C(C1=C(O)C(=O)N(CCN2CCOCC2)C1c1cccc(Br)c1)c1cc2ccccc2o1	nan
	4542697	50874	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	510	6	1	6	4.1	O=C(C1=C(O)C(=O)N(CCN2CCOCC2)C1c1cccc(Br)c1)c1cc2ccccc2o1	nan
	CHEMBL1579576	50874	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	510	6	1	6	4.1	O=C(C1=C(O)C(=O)N(CCN2CCOCC2)C1c1cccc(Br)c1)c1cc2ccccc2o1	nan
	16196197	50886	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	491	6	1	4	6.4	Cc1cc(/C(O)=C(/C([S-])=Nc2ccc(F)cc2)[n+]2ccccc2)c(C)n1Cc1ccccc1Cl	nan
	3610394	50886	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	491	6	1	4	6.4	Cc1cc(/C(O)=C(/C([S-])=Nc2ccc(F)cc2)[n+]2ccccc2)c(C)n1Cc1ccccc1Cl	nan
	CHEMBL1579745	50886	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	491	6	1	4	6.4	Cc1cc(/C(O)=C(/C([S-])=Nc2ccc(F)cc2)[n+]2ccccc2)c(C)n1Cc1ccccc1Cl	nan
	2357568	50904	7	None	-5	3	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	6	1	6	4.7	O=C(CSc1nnc(-c2cccs2)n1-c1ccccc1)Nc1ccccc1	nan
	CHEMBL1579942	50904	7	None	-5	3	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	6	1	6	4.7	O=C(CSc1nnc(-c2cccs2)n1-c1ccccc1)Nc1ccccc1	nan
	4831734	50933	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	508	7	1	6	3.8	CCN(CC)S(=O)(=O)c1ccc(N2CCOCC2)c(NC(=O)c2c3c(nc4ccccc24)CCC3)c1	nan
	CHEMBL1580173	50933	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	508	7	1	6	3.8	CCN(CC)S(=O)(=O)c1ccc(N2CCOCC2)c(NC(=O)c2c3c(nc4ccccc24)CCC3)c1	nan
	1476967	50965	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	262	2	0	6	2.0	c1cn(-c2ccc(-c3ccnc4ncnn34)cc2)cn1	nan
	CHEMBL1580435	50965	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	262	2	0	6	2.0	c1cn(-c2ccc(-c3ccnc4ncnn34)cc2)cn1	nan
	7190795	50978	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	347	5	0	7	3.2	O=C(CSc1ccc2nnc(-c3cccnc3)n2n1)c1ccccc1	nan
	CHEMBL1580576	50978	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	347	5	0	7	3.2	O=C(CSc1ccc2nnc(-c3cccnc3)n2n1)c1ccccc1	nan
	16194926	51052	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	6	1	7	2.5	Cc1ccc(-c2ccc3nnc(SCC(=O)NCC4CCCO4)n3n2)cc1	nan
	CHEMBL1581174	51052	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	6	1	7	2.5	Cc1ccc(-c2ccc3nnc(SCC(=O)NCC4CCCO4)n3n2)cc1	nan
	3357076	51129	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	7	1	5	3.4	CCN(CC)S(=O)(=O)c1ccc(N2CCCCC2)c(NC(=O)c2ccncc2)c1	nan
	CHEMBL1581844	51129	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	7	1	5	3.4	CCN(CC)S(=O)(=O)c1ccc(N2CCCCC2)c(NC(=O)c2ccncc2)c1	nan
	3151315	51282	15	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	5	2	8	1.9	Cc1cccn2c(=O)c3cc(C(=O)NCc4cccnc4)c(=N)n(CC4CCCO4)c3nc12	nan
	CHEMBL1583158	51282	15	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	5	2	8	1.9	Cc1cccn2c(=O)c3cc(C(=O)NCc4cccnc4)c(=N)n(CC4CCCO4)c3nc12	nan
	3721854	51399	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	2	1	7	2.1	Nc1c(C(=O)N2CCOCC2)sc2nc(N3CCOCC3)c3c(c12)CCCC3	nan
	CHEMBL1584034	51399	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	2	1	7	2.1	Nc1c(C(=O)N2CCOCC2)sc2nc(N3CCOCC3)c3c(c12)CCCC3	nan
	3911608	51507	18	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	4	1	5	4.5	Cc1ccc(C2C(C(=O)c3cccs3)=C(O)C(=O)N2c2cccc(C)n2)cc1	nan
	CHEMBL1584955	51507	18	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	4	1	5	4.5	Cc1ccc(C2C(C(=O)c3cccs3)=C(O)C(=O)N2c2cccc(C)n2)cc1	nan
	7207569	51686	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	410	7	1	7	1.8	O=C(NCCc1nnc2ccc(SCC(=O)N3CCCC3)nn12)c1ccccc1	nan
	CHEMBL1586420	51686	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	410	7	1	7	1.8	O=C(NCCc1nnc2ccc(SCC(=O)N3CCCC3)nn12)c1ccccc1	nan
	7190486	51782	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	6	1	8	2.9	COc1ccc(NC(=O)CSc2ccc3nnc(-c4ccccn4)n3n2)cc1	nan
	CHEMBL1587249	51782	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	6	1	8	2.9	COc1ccc(NC(=O)CSc2ccc3nnc(-c4ccccn4)n3n2)cc1	nan
	5225306	51818	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	1	0	5	2.9	CC1CCCCN1C(=O)c1cc2c(=O)n3ccccc3nc2s1	nan
	CHEMBL1587533	51818	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	1	0	5	2.9	CC1CCCCN1C(=O)c1cc2c(=O)n3ccccc3nc2s1	nan
	4975167	51831	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	366	7	1	5	3.1	CCCc1cc(=O)oc2c(C)c(OCC(=O)NCc3ccccn3)ccc12	nan
	CHEMBL1587597	51831	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	366	7	1	5	3.1	CCCc1cc(=O)oc2c(C)c(OCC(=O)NCc3ccccn3)ccc12	nan
	5236958	52012	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	8	1	5	2.7	CCN(CC)S(=O)(=O)c1ccc(Cl)c(NC(=O)CSc2cccc[n+]2[O-])c1	nan
	CHEMBL1589189	52012	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	8	1	5	2.7	CCN(CC)S(=O)(=O)c1ccc(Cl)c(NC(=O)CSc2cccc[n+]2[O-])c1	nan
	16022898	52097	0	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	299	7	1	6	2.7	CCOCCCNc1nc2ccccc2n2c(CC)nnc12	nan
	CHEMBL1589922	52097	0	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	299	7	1	6	2.7	CCOCCCNc1nc2ccccc2n2c(CC)nnc12	nan
	16009827	52108	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	491	7	1	9	3.7	COc1ccc(NC(=O)Cn2c(=O)n(Cc3ccco3)c(=O)c3sc4ccccc4c32)cc1OC	nan
	CHEMBL1590063	52108	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	491	7	1	9	3.7	COc1ccc(NC(=O)Cn2c(=O)n(Cc3ccco3)c(=O)c3sc4ccccc4c32)cc1OC	nan
	1391194	52178	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	5	2	4	3.9	O=C(O)CCNc1nc(-c2ccccc2)c2cc(Br)ccc2n1	nan
	1391195	52178	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	5	2	4	3.9	O=C(O)CCNc1nc(-c2ccccc2)c2cc(Br)ccc2n1	nan
	CHEMBL1590944	52178	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	5	2	4	3.9	O=C(O)CCNc1nc(-c2ccccc2)c2cc(Br)ccc2n1	nan
	18572144	52201	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	440	8	2	6	2.6	Cn1c(SCC(=O)NCCc2ccccc2)ncc(C(=O)Nc2ccc(F)cc2)c1=O	nan
	CHEMBL1591283	52201	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	440	8	2	6	2.6	Cn1c(SCC(=O)NCCc2ccccc2)ncc(C(=O)Nc2ccc(F)cc2)c1=O	nan
	20903635	52224	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	492	8	0	9	1.9	CCCN1CCN(C(=O)CCc2nnc3ccc(N4CCN(c5cccc(OC)c5)CC4)nn23)CC1	nan
	CHEMBL1591509	52224	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	492	8	0	9	1.9	CCCN1CCN(C(=O)CCc2nnc3ccc(N4CCN(c5cccc(OC)c5)CC4)nn23)CC1	nan
	16012276	52247	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	315	3	1	5	2.3	Cc1cc(C)n2nc(CNC(=O)c3ccc(Cl)cc3)nc2n1	nan
	CHEMBL1591819	52247	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	315	3	1	5	2.3	Cc1cc(C)n2nc(CNC(=O)c3ccc(Cl)cc3)nc2n1	nan
	5303336	52281	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	346	4	1	5	4.2	CCOc1ccc(-c2oc3cc(Cl)ccc3c(=O)c2O)cc1OC	nan
	CHEMBL1592283	52281	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	346	4	1	5	4.2	CCOc1ccc(-c2oc3cc(Cl)ccc3c(=O)c2O)cc1OC	nan
	2790635	52391	15	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	7	2	4	4.1	Cc1ccc(OCCCC(=O)Nc2sc3c(c2C(N)=O)CCC(C)C3)cc1	nan
	CHEMBL1593935	52391	15	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	7	2	4	4.1	Cc1ccc(OCCCC(=O)Nc2sc3c(c2C(N)=O)CCC(C)C3)cc1	nan
	3476583	52575	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	5	1	4	5.8	Cc1ccc(-c2cc(C(F)(F)F)c(C#N)c(SCC(=O)Nc3ccccc3F)n2)cc1	nan
	CHEMBL1595488	52575	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	5	1	4	5.8	Cc1ccc(-c2cc(C(F)(F)F)c(C#N)c(SCC(=O)Nc3ccccc3F)n2)cc1	nan
	1958370	52593	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	6	1	7	2.5	COCCNS(=O)(=O)c1cc(-c2nn3c(C)nnc3c3ccccc23)ccc1C	nan
	CHEMBL1595653	52593	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	6	1	7	2.5	COCCNS(=O)(=O)c1cc(-c2nn3c(C)nnc3c3ccccc23)ccc1C	nan
	4601439	52767	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	4	2	7	3.9	COc1cccc(NC(=O)c2sc3nc(N4CCOCC4)c4c(c3c2N)CCCC4)c1	nan
	CHEMBL1597228	52767	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	4	2	7	3.9	COc1cccc(NC(=O)c2sc3nc(N4CCOCC4)c4c(c3c2N)CCCC4)c1	nan
	4151069	52979	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	461	5	1	10	0.6	COC(=O)c1cc(NS(=O)(=O)c2ccc3c(c2)c(=O)n(C)c(=O)n3C)cc(C(=O)OC)c1	nan
	CHEMBL1599214	52979	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	461	5	1	10	0.6	COC(=O)c1cc(NS(=O)(=O)c2ccc3c(c2)c(=O)n(C)c(=O)n3C)cc(C(=O)OC)c1	nan
	2890665	53051	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	325	3	1	3	3.6	CC(=O)C1=C(O)C(=O)N(c2ccc(F)cc2)C1c1ccc(C)cc1	nan
	CHEMBL1599834	53051	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	325	3	1	3	3.6	CC(=O)C1=C(O)C(=O)N(c2ccc(F)cc2)C1c1ccc(C)cc1	nan
	16020305	53368	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	554	12	1	6	4.3	CCCN(CCC)C(=O)Cn1c(=O)n(-c2ccc(CC)cc2)c(=O)c2ccc(C(=O)NCCc3ccccc3)cc21	nan
	CHEMBL1602912	53368	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	554	12	1	6	4.3	CCCN(CCC)C(=O)Cn1c(=O)n(-c2ccc(CC)cc2)c(=O)c2ccc(C(=O)NCCc3ccccc3)cc21	nan
	910705	53455	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	229	2	0	4	2.4	O=[N+]([O-])c1ccc(-c2cn3c(n2)CCC3)cc1	nan
	CHEMBL1603668	53455	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	229	2	0	4	2.4	O=[N+]([O-])c1ccc(-c2cn3c(n2)CCC3)cc1	nan
	1146176	53603	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	4	0	4	4.7	CC1CCN(C(=O)CSc2nc(-c3ccc(F)cc3)cc(C(F)(F)F)n2)CC1	nan
	CHEMBL1604923	53603	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	4	0	4	4.7	CC1CCN(C(=O)CSc2nc(-c3ccc(F)cc3)cc(C(F)(F)F)n2)CC1	nan
	16019480	53692	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	5	0	9	2.9	CCc1ccc(S(=O)(=O)c2nnn3c2nc(N2CCN(CC)CC2)c2sccc23)cc1	nan
	CHEMBL1605620	53692	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	5	0	9	2.9	CCc1ccc(S(=O)(=O)c2nnn3c2nc(N2CCN(CC)CC2)c2sccc23)cc1	nan
	1410148	53806	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	5	1	5	4.5	CCOc1ccc(C(=O)Nc2ccc3oc(-c4cccnc4)nc3c2)cc1	nan
	CHEMBL1606536	53806	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	5	1	5	4.5	CCOc1ccc(C(=O)Nc2ccc3oc(-c4cccnc4)nc3c2)cc1	nan
	2918495	53838	17	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	8	1	8	2.5	COc1cccc(C2C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2CCN2CCOCC2)c1OC	nan
	CHEMBL1606762	53838	17	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	8	1	8	2.5	COc1cccc(C2C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2CCN2CCOCC2)c1OC	nan
	5730347	53888	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	280	4	0	4	3.9	CCC(=O)c1ccc(/C=C/c2nc3ccccc3n2C)o1	nan
	CHEMBL1607132	53888	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	280	4	0	4	3.9	CCC(=O)c1ccc(/C=C/c2nc3ccccc3n2C)o1	nan
	4426797	53972	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	6	1	10	-0.6	Cn1c(=O)c2c(nc(CN3CCN(C(=O)c4ccco4)CC3)n2CCCO)n(C)c1=O	nan
	CHEMBL1607800	53972	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	6	1	10	-0.6	Cn1c(=O)c2c(nc(CN3CCN(C(=O)c4ccco4)CC3)n2CCCO)n(C)c1=O	nan
	1325691	54005	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	358	1	1	7	3.2	Sc1ncnc2c1sc1nc(N3CCOCC3)c3c(c12)CCCC3	nan
	CHEMBL1608119	54005	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	358	1	1	7	3.2	Sc1ncnc2c1sc1nc(N3CCOCC3)c3c(c12)CCCC3	nan
	2966904	54009	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	7	2	7	3.4	CC(=O)c1sc2nc(SCC(=O)NCCc3ccccc3)nc(O)c2c1C	nan
	CHEMBL1608140	54009	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	7	2	7	3.4	CC(=O)c1sc2nc(SCC(=O)NCCc3ccccc3)nc(O)c2c1C	nan
	16406841	54015	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	3	0	6	3.1	Cc1c(Br)c(=O)oc2cc(OCC(=O)N3C[C@@H]4C[C@H](C3)Cn3c4cccc3=O)ccc12	nan
	CHEMBL1608190	54015	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	3	0	6	3.1	Cc1c(Br)c(=O)oc2cc(OCC(=O)N3C[C@@H]4C[C@H](C3)Cn3c4cccc3=O)ccc12	nan
	54686430	54080	29	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	286	3	2	4	1.8	CCCNC(=O)c1c(O)c2cccc3c2n(c1=O)CCC3	nan
	CHEMBL1608771	54080	29	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	286	3	2	4	1.8	CCCNC(=O)c1c(O)c2cccc3c2n(c1=O)CCC3	nan
	6107794	54138	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	486	7	1	7	4.2	COc1ccc(C2C(C(=O)c3ccc4c(c3)CC(C)O4)=C(O)C(=O)N2Cc2cccnc2)c(OC)c1	nan
	CHEMBL1609202	54138	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	486	7	1	7	4.2	COc1ccc(C2C(C(=O)c3ccc4c(c3)CC(C)O4)=C(O)C(=O)N2Cc2cccnc2)c(OC)c1	nan
	2576098	54170	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	304	5	1	5	2.7	Cc1sc2ncnc(NCCCN3CCCC3=O)c2c1C	nan
	CHEMBL1609414	54170	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	304	5	1	5	2.7	Cc1sc2ncnc(NCCCN3CCCC3=O)c2c1C	nan
	3641030	54226	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	4	1	3	5.1	CC(=O)c1ccc(NC(=O)c2ccc(-c3ccc(Cl)cc3)o2)cc1	nan
	CHEMBL1609950	54226	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	4	1	3	5.1	CC(=O)c1ccc(NC(=O)c2ccc(-c3ccc(Cl)cc3)o2)cc1	nan
	2868074	54244	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	3	1	3	4.7	CC(=O)C1=C(O)C(=O)N(c2cccc(Br)c2)C1c1ccc(Br)cc1	nan
	CHEMBL1610073	54244	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	3	1	3	4.7	CC(=O)C1=C(O)C(=O)N(c2cccc(Br)c2)C1c1ccc(Br)cc1	nan
	2790804	54355	14	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	5	1	6	3.8	O=[N+]([O-])c1ccc(-c2nc(NCC3CCCO3)c3ccccc3n2)cc1	nan
	CHEMBL1611050	54355	14	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	5	1	6	3.8	O=[N+]([O-])c1ccc(-c2nc(NCC3CCCO3)c3ccccc3n2)cc1	nan
	2934073	54606	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	5	1	5	3.7	O=C(C1=C(O)C(=O)N(CC2CCCO2)C1c1cccc(Cl)c1)c1ccco1	nan
	CHEMBL1613356	54606	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	5	1	5	3.7	O=C(C1=C(O)C(=O)N(CC2CCCO2)C1c1cccc(Cl)c1)c1ccco1	nan
	4581262	55040	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	373	4	1	5	4.4	CC1CCN(CCCn2c(=S)[nH]c3c(sc4ccccc43)c2=O)CC1	nan
	CHEMBL1377318	55040	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	373	4	1	5	4.4	CC1CCN(CCCn2c(=S)[nH]c3c(sc4ccccc43)c2=O)CC1	nan
	CHEMBL1618739	55040	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	373	4	1	5	4.4	CC1CCN(CCCn2c(=S)[nH]c3c(sc4ccccc43)c2=O)CC1	nan
	1099157	55066	12	None	-3	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	4	1	4	4.4	O=C(CN1CCCCC1)Nc1c2c(nc3ccccc13)N(c1ccccc1)CC2	nan
	CHEMBL1389219	55066	12	None	-3	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	4	1	4	4.4	O=C(CN1CCCCC1)Nc1c2c(nc3ccccc13)N(c1ccccc1)CC2	nan
	CHEMBL1618947	55066	12	None	-3	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	4	1	4	4.4	O=C(CN1CCCCC1)Nc1c2c(nc3ccccc13)N(c1ccccc1)CC2	nan
	4055296	55192	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	4	0	5	5.8	O=[N+]([O-])c1cccc(-c2cc3sc4ccccc4[n+]3cc2-c2cccc([N+](=O)[O-])c2)c1	nan
	CHEMBL1420869	55192	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	4	0	5	5.8	O=[N+]([O-])c1cccc(-c2cc3sc4ccccc4[n+]3cc2-c2cccc([N+](=O)[O-])c2)c1	nan
	CHEMBL1620041	55192	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	4	0	5	5.8	O=[N+]([O-])c1cccc(-c2cc3sc4ccccc4[n+]3cc2-c2cccc([N+](=O)[O-])c2)c1	nan
	655842	55339	10	None	-12	3	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	6	2	5	3.0	CSCCC(Nc1ncnc2ccc(Br)cc12)C(=O)O	nan
	CHEMBL1466356	55339	10	None	-12	3	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	6	2	5	3.0	CSCCC(Nc1ncnc2ccc(Br)cc12)C(=O)O	nan
	CHEMBL1621365	55339	10	None	-12	3	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	6	2	5	3.0	CSCCC(Nc1ncnc2ccc(Br)cc12)C(=O)O	nan
	3848238	55713	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	5	1	5	5.5	N#Cc1c(SC(C(=O)O)c2ccccc2)nc2c(c1-c1cccs1)CCCC2	nan
	CHEMBL1548688	55713	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	5	1	5	5.5	N#Cc1c(SC(C(=O)O)c2ccccc2)nc2c(c1-c1cccs1)CCCC2	nan
	CHEMBL1624498	55713	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	5	1	5	5.5	N#Cc1c(SC(C(=O)O)c2ccccc2)nc2c(c1-c1cccs1)CCCC2	nan
	3589783	55726	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	2	2	6	5.1	CC1(C)CC2=NC3=C(C(=O)c4ccccc43)C(c3cc([N+](=O)[O-])ccc3O)C2=C(O)C1	nan
	CHEMBL1566042	55726	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	2	2	6	5.1	CC1(C)CC2=NC3=C(C(=O)c4ccccc43)C(c3cc([N+](=O)[O-])ccc3O)C2=C(O)C1	nan
	CHEMBL1624662	55726	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	2	2	6	5.1	CC1(C)CC2=NC3=C(C(=O)c4ccccc43)C(c3cc([N+](=O)[O-])ccc3O)C2=C(O)C1	nan
	9560158	71854	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	5	1	9	-0.4	COc1cccc(/C=N/NC(=O)Cn2cnc3c2c(=O)n(C)c(=O)n3C)c1	nan
	CHEMBL1980603	71854	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	5	1	9	-0.4	COc1cccc(/C=N/NC(=O)Cn2cnc3c2c(=O)n(C)c(=O)n3C)c1	nan
	9624156	71928	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	6	1	5	4.4	N#CCC(=O)N/N=C/c1ccc(N2N=C(c3ccccc3)CC2c2ccccc2)cc1	nan
	CHEMBL1982521	71928	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	6	1	5	4.4	N#CCC(=O)N/N=C/c1ccc(N2N=C(c3ccccc3)CC2c2ccccc2)cc1	nan
	1995859	72458	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	4	0	7	1.3	COCCCn1/c(=N/C(C)=O)c(C#N)cc2c(=O)n3cccc(C)c3nc21	nan
	CHEMBL2000901	72458	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	4	0	7	1.3	COCCCn1/c(=N/C(C)=O)c(C#N)cc2c(=O)n3cccc(C)c3nc21	nan
	65599	104943	38	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	278	5	0	7	0.2	CC(=O)CCCCn1cnc2c1c(=O)n(C)c(=O)n2C	nan
	CHEMBL311948	104943	38	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	278	5	0	7	0.2	CC(=O)CCCCn1cnc2c1c(=O)n(C)c(=O)n2C	nan
	2864416	106403	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	7	1	7	1.6	Cc1[nH]n(-c2ccc([N+](=O)[O-])cc2)c(=O)c1/C=N/CCN1CCN(C(=O)C(C)C)CC1	nan
	CHEMBL3145301	106403	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	7	1	7	1.6	Cc1[nH]n(-c2ccc([N+](=O)[O-])cc2)c(=O)c1/C=N/CCN1CCN(C(=O)C(C)C)CC1	nan
	5935610	107121	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	306	1	1	3	3.9	CCn1c2c(c3cc(Br)ccc31)CCC/C2=N\O	nan
	CHEMBL3189713	107121	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	306	1	1	3	3.9	CCn1c2c(c3cc(Br)ccc31)CCC/C2=N\O	nan
	6279969	107398	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	272	3	0	6	2.1	CN(C)/C=N/c1nc2nccc(-c3cccs3)n2n1	nan
	CHEMBL3192852	107398	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	272	3	0	6	2.1	CN(C)/C=N/c1nc2nccc(-c3cccs3)n2n1	nan
	6860035	107630	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	7	1	8	3.0	COc1ccc(OC)c(/C=N/n2c(S)nnc2COc2ccccc2)c1	nan
	CHEMBL3195667	107630	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	7	1	8	3.0	COc1ccc(OC)c(/C=N/n2c(S)nnc2COc2ccccc2)c1	nan
	135467322	108210	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	8	1	6	4.3	COC(=O)/C(Nc1ccccc1)=C(\C(=O)C(=O)N(C)c1ccccc1)C(=O)c1ccc(Cl)cc1	nan
	CHEMBL3208147	108210	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	8	1	6	4.3	COC(=O)/C(Nc1ccccc1)=C(\C(=O)C(=O)N(C)c1ccccc1)C(=O)c1ccc(Cl)cc1	nan
	2805193	108323	4	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	280	5	1	7	2.6	CCO/C(O)=C(C#N)/C=N/c1ccsc1C(=O)OC	nan
	CHEMBL3209558	108323	4	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	280	5	1	7	2.6	CCO/C(O)=C(C#N)/C=N/c1ccsc1C(=O)OC	nan
	5867179	108531	3	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	5	1	6	4.1	C/C(N)=C(/C#N)C(=O)COC(=O)c1cc(-c2ccccc2)nc2ccc(Br)cc12	nan
	CHEMBL3212349	108531	3	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	5	1	6	4.1	C/C(N)=C(/C#N)C(=O)COC(=O)c1cc(-c2ccccc2)nc2ccc(Br)cc12	nan
	3221537	112122	5	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	331	5	0	5	3.2	CCOc1ccc2nc3c(cc2c1)CN(CCOC)/C(=N\C)S3	nan
	CHEMBL3209727	112122	5	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	331	5	0	5	3.2	CCOc1ccc2nc3c(cc2c1)CN(CCOC)/C(=N\C)S3	nan
	CHEMBL3302425	112122	5	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	331	5	0	5	3.2	CCOc1ccc2nc3c(cc2c1)CN(CCOC)/C(=N\C)S3	nan
	264006	177988	14	None	1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	307	5	4	9	-1.0	C=CCNc1ncnc2c1ncn2C1OC(CO)C(O)C1O	nan
	CHEMBL46703	177988	14	None	1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	307	5	4	9	-1.0	C=CCNc1ncnc2c1ncn2C1OC(CO)C(O)C1O	nan
	833435	195993	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	3	3	4	2.9	Cc1sc(NC(=S)NC(=O)C2CCCCC2)c(C(N)=O)c1C	nan
	CHEMBL571065	195993	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	3	3	4	2.9	Cc1sc(NC(=S)NC(=O)C2CCCCC2)c(C(N)=O)c1C	nan
	22334103	199225	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	513	9	2	8	1.6	COc1ccc(-n2nc(C(=O)NCC(=O)NCCCN3CCOCC3)c3ccccc3c2=O)cc1Cl	nan
	CHEMBL601585	199225	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	513	9	2	8	1.6	COc1ccc(-n2nc(C(=O)NCC(=O)NCCCN3CCOCC3)c3ccccc3c2=O)cc1Cl	nan
	4167655	28039	11	None	-	1	Human	5.6	pPotency	=	5.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	4	1	5	4.3	Brc1ccc(-c2nnc3sc(CNC4CCCC4)cn23)cc1	nan
	CHEMBL1374064	28039	11	None	-	1	Human	5.6	pPotency	=	5.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	4	1	5	4.3	Brc1ccc(-c2nnc3sc(CNC4CCCC4)cn23)cc1	nan
	16018920	28273	5	None	-	1	Human	5.6	pPotency	=	5.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	5	1	6	4.8	CCc1nnc(SCC(=O)Nc2ccc(F)cc2F)c2cc3sc(C)cc3n12	nan
	CHEMBL1375688	28273	5	None	-	1	Human	5.6	pPotency	=	5.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	5	1	6	4.8	CCc1nnc(SCC(=O)Nc2ccc(F)cc2F)c2cc3sc(C)cc3n12	nan
	3348974	38955	9	None	-	1	Human	5.6	pPotency	=	5.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	5	1	11	0.5	CCc1nnc(NC(=O)CSc2nc(C)nc3c2c(=O)n(C)c(=O)n3C)s1	nan
	CHEMBL1469832	38955	9	None	-	1	Human	5.6	pPotency	=	5.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	5	1	11	0.5	CCc1nnc(NC(=O)CSc2nc(C)nc3c2c(=O)n(C)c(=O)n3C)s1	nan
	4351083	46903	7	None	-	1	Human	5.6	pPotency	=	5.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	423	5	2	8	3.0	O=C(NN1C(=O)c2ccccc2NC1c1ccc([N+](=O)[O-])o1)c1ccc([N+](=O)[O-])cc1	nan
	CHEMBL1543122	46903	7	None	-	1	Human	5.6	pPotency	=	5.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	423	5	2	8	3.0	O=C(NN1C(=O)c2ccccc2NC1c1ccc([N+](=O)[O-])o1)c1ccc([N+](=O)[O-])cc1	nan
	3241486	49654	5	None	1	2	Human	5.6	pPotency	=	5.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	442	6	1	6	4.2	COc1ccc(C(=O)Nc2ccc(N3CCN(c4ccc(OC)cc4)CC3)c(C#N)c2)cc1	nan
	CHEMBL1568468	49654	5	None	1	2	Human	5.6	pPotency	=	5.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	442	6	1	6	4.2	COc1ccc(C(=O)Nc2ccc(N3CCN(c4ccc(OC)cc4)CC3)c(C#N)c2)cc1	nan
	1261644	49810	10	None	1	2	Human	5.6	pPotency	=	5.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	3	1	4	4.7	O=C(Nc1ccncc1)c1cc(-c2ccccn2)nc2ccc(Br)cc12	nan
	CHEMBL1569872	49810	10	None	1	2	Human	5.6	pPotency	=	5.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	3	1	4	4.7	O=C(Nc1ccncc1)c1cc(-c2ccccn2)nc2ccc(Br)cc12	nan
	759120	52283	31	None	-	1	Human	5.6	pPotency	=	5.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	2	1	3	4.4	O=C(O)c1cc(-c2ccc(Br)s2)nc2ccccc12	nan
	CHEMBL1592299	52283	31	None	-	1	Human	5.6	pPotency	=	5.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	2	1	3	4.4	O=C(O)c1cc(-c2ccc(Br)s2)nc2ccccc12	nan
	16010305	7592	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	7	1	8	3.2	COCCCNc1nc2c(S(=O)(=O)c3ccccc3)nnn2c2ccc(Cl)cc12	nan
	CHEMBL1088575	7592	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	7	1	8	3.2	COCCCNc1nc2c(S(=O)(=O)c3ccccc3)nnn2c2ccc(Cl)cc12	nan
	16019548	10781	9	None	-23	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	5	1	8	4.4	O=S(=O)(c1ccccc1)c1nnn2c1nc(NCc1ccc(Cl)cc1)c1sccc12	nan
	CHEMBL1172597	10781	9	None	-23	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	5	1	8	4.4	O=S(=O)(c1ccccc1)c1nnn2c1nc(NCc1ccc(Cl)cc1)c1sccc12	nan
	16019364	10855	5	None	-53	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	467	5	1	8	4.5	Cc1ccc(S(=O)(=O)c2nnn3c2nc(NCc2ccc(F)cc2)c2sccc23)cc1C	nan
	CHEMBL1173283	10855	5	None	-53	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	467	5	1	8	4.5	Cc1ccc(S(=O)(=O)c2nnn3c2nc(NCc2ccc(F)cc2)c2sccc23)cc1C	nan
	5721990	14657	23	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	274	3	0	2	4.5	CN(C)c1ccc(/C=C/c2ccc3ccccc3n2)cc1	nan
	CHEMBL120734	14657	23	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	274	3	0	2	4.5	CN(C)c1ccc(/C=C/c2ccc3ccccc3n2)cc1	nan
	3565	19176	46	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	200	0	2	2	2.2	CC1=NCCc2c1[nH]c1cc(O)ccc21	nan
	CHEMBL129177	19176	46	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	200	0	2	2	2.2	CC1=NCCc2c1[nH]c1cc(O)ccc21	nan
	CHEMBL1473205	19176	46	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	200	0	2	2	2.2	CC1=NCCc2c1[nH]c1cc(O)ccc21	nan
	2803232	19319	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	293	3	2	2	4.3	S=C(Nc1ccccc1)Nc1ccccc1-n1cccc1	nan
	CHEMBL1299459	19319	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	293	3	2	2	4.3	S=C(Nc1ccccc1)Nc1ccccc1-n1cccc1	nan
	1305405	19475	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	3	3	4	4.4	O=C(O)c1ccccc1NC(=S)NC(=O)c1sc2ccccc2c1Cl	nan
	CHEMBL1300720	19475	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	3	3	4	4.4	O=C(O)c1ccccc1NC(=S)NC(=O)c1sc2ccccc2c1Cl	nan
	24790327	19510	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	5	0	5	4.4	COc1ccc2cc(C(=O)C3CCCN(C(=O)c4cnn(C(C)C)c4)C3)ccc2c1	nan
	CHEMBL1300972	19510	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	5	0	5	4.4	COc1ccc2cc(C(=O)C3CCCN(C(=O)c4cnn(C(C)C)c4)C3)ccc2c1	nan
	5826640	19578	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	520	10	1	7	4.1	CCCCOc1cccc(C2C(C(=O)c3ccc4c(c3)CC(C)O4)=C(O)C(=O)N2CCN2CCOCC2)c1	nan
	CHEMBL1301431	19578	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	520	10	1	7	4.1	CCCCOc1cccc(C2C(C(=O)c3ccc4c(c3)CC(C)O4)=C(O)C(=O)N2CCN2CCOCC2)c1	nan
	2410711	19597	17	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	363	5	1	5	3.5	CCOc1ccc(S(=O)(=O)Nc2nc3ccccc3nc2Cl)cc1	nan
	CHEMBL1301615	19597	17	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	363	5	1	5	3.5	CCOc1ccc(S(=O)(=O)Nc2nc3ccccc3nc2Cl)cc1	nan
	5918716	19666	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	4	1	7	0.8	CCN1CCN(c2nc3c(C)cccn3c(=O)c2/C=C(\C#N)C(=O)NC)CC1	nan
	CHEMBL1302267	19666	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	4	1	7	0.8	CCN1CCN(c2nc3c(C)cccn3c(=O)c2/C=C(\C#N)C(=O)NC)CC1	nan
	910973	19793	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	284	1	2	6	1.6	N#CC(C#N)=C1NC(N)=C(C#N)C(c2ccccc2)=C1C#N	nan
	CHEMBL1303255	19793	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	284	1	2	6	1.6	N#CC(C#N)=C1NC(N)=C(C#N)C(c2ccccc2)=C1C#N	nan
	2472728	19967	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	4	1	7	2.7	Cc1sc2ncnc(SCC(=O)NC(=O)c3cccn3C)c2c1C	nan
	CHEMBL1304667	19967	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	4	1	7	2.7	Cc1sc2ncnc(SCC(=O)NC(=O)c3cccn3C)c2c1C	nan
	3544771	19989	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	5	0	9	3.2	O=c1c2sccc2nc(SCc2cc(=O)n3ccccc3n2)n1Cc1ccccn1	nan
	CHEMBL1304859	19989	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	5	0	9	3.2	O=c1c2sccc2nc(SCc2cc(=O)n3ccccc3n2)n1Cc1ccccn1	nan
	7295015	20129	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	325	5	1	5	3.6	CSc1ccccc1-c1nnc(NC(=O)Cc2ccccc2)o1	nan
	CHEMBL1305973	20129	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	325	5	1	5	3.6	CSc1ccccc1-c1nnc(NC(=O)Cc2ccccc2)o1	nan
	654420	20132	4	None	-28	3	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	276	5	0	5	2.8	CCOC(=O)CSc1nc(CC)nc2ccccc12	nan
	CHEMBL1305990	20132	4	None	-28	3	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	276	5	0	5	2.8	CCOC(=O)CSc1nc(CC)nc2ccccc12	nan
	4021231	20142	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	461	5	2	7	2.7	Cc1cccn2c(=O)c3cc(C(=O)NCc4ccc(F)cc4)c(=N)n(CC4CCCO4)c3nc12	nan
	CHEMBL1306067	20142	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	461	5	2	7	2.7	Cc1cccn2c(=O)c3cc(C(=O)NCc4ccc(F)cc4)c(=N)n(CC4CCCO4)c3nc12	nan
	833786	20193	14	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	284	3	1	4	4.2	Sc1nc(SCc2ccccc2)nc2ccccc12	nan
	CHEMBL1306480	20193	14	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	284	3	1	4	4.2	Sc1nc(SCc2ccccc2)nc2ccccc12	nan
	865618	20204	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	283	3	0	4	3.6	CN(C)c1ccc(-c2nnc(-c3ccccc3F)o2)cc1	nan
	CHEMBL1306590	20204	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	283	3	0	4	3.6	CN(C)c1ccc(-c2nnc(-c3ccccc3F)o2)cc1	nan
	6078291	20311	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	7	1	6	4.6	CCOc1cccc(C2C(C(=O)c3ccc4c(c3)CC(C)O4)=C(O)C(=O)N2Cc2cccnc2)c1	nan
	CHEMBL1307444	20311	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	7	1	6	4.6	CCOc1cccc(C2C(C(=O)c3ccc4c(c3)CC(C)O4)=C(O)C(=O)N2Cc2cccnc2)c1	nan
	2820469	20390	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	4	1	5	3.4	CSc1sc(C(=O)NCC2CC2)c2c1S(=O)(=O)N(C)c1ccccc1-2	nan
	CHEMBL1308054	20390	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	4	1	5	3.4	CSc1sc(C(=O)NCC2CC2)c2c1S(=O)(=O)N(C)c1ccccc1-2	nan
	5012705	20400	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	9	2	6	3.7	O=C(CCCCCn1c(=S)[nH]c2cc3c(cc2c1=O)OCO3)NCCc1ccccc1	nan
	CHEMBL1308124	20400	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	9	2	6	3.7	O=C(CCCCCn1c(=S)[nH]c2cc3c(cc2c1=O)OCO3)NCCc1ccccc1	nan
	1201985	20550	9	None	-2	3	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	6	0	6	3.8	O=C(CSc1nc2ccccc2nc1SCC(=O)N1CCCCC1)N1CCCCC1	nan
	CHEMBL1309335	20550	9	None	-2	3	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	6	0	6	3.8	O=C(CSc1nc2ccccc2nc1SCC(=O)N1CCCCC1)N1CCCCC1	nan
	24891893	20558	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	6	1	9	-0.0	CCc1nc(SCC(=O)NCC2CCCO2)c2c(=O)n(C)c(=O)n(C)c2n1	nan
	CHEMBL1309394	20558	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	6	1	9	-0.0	CCc1nc(SCC(=O)NCC2CCCO2)c2c(=O)n(C)c(=O)n(C)c2n1	nan
	1596915	20572	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	3	2	7	4.6	Cc1csc(NC(=O)c2sc3nc(-c4cccs4)ccc3c2N)n1	nan
	CHEMBL1309478	20572	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	3	2	7	4.6	Cc1csc(NC(=O)c2sc3nc(-c4cccs4)ccc3c2N)n1	nan
	3236246	20654	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	7	1	8	2.8	CCC(Sc1ccc2nnc(-c3ccc(OC)c(OC)c3)n2n1)C(=O)O	nan
	CHEMBL1310295	20654	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	7	1	8	2.8	CCC(Sc1ccc2nnc(-c3ccc(OC)c(OC)c3)n2n1)C(=O)O	nan
	4881170	20761	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	294	2	0	6	3.0	Cc1nc(SC2CCOC2=O)c2c(C)c(C)sc2n1	nan
	CHEMBL1311178	20761	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	294	2	0	6	3.0	Cc1nc(SC2CCOC2=O)c2c(C)c(C)sc2n1	nan
	5813760	20807	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	506	5	1	6	4.4	O=C(C1=C(O)C(=O)N(Cc2cccnc2)C1c1ccc(Br)cc1)c1ccc2c(c1)OCCO2	nan
	CHEMBL1311567	20807	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	506	5	1	6	4.4	O=C(C1=C(O)C(=O)N(Cc2cccnc2)C1c1ccc(Br)cc1)c1ccc2c(c1)OCCO2	nan
	3682235	20882	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	5	1	7	3.7	COc1cccc(C2C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2c2cc(C)on2)c1	nan
	CHEMBL1312109	20882	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	5	1	7	3.7	COc1cccc(C2C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2c2cc(C)on2)c1	nan
	3588555	20961	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	580	5	1	8	3.8	Cc1cc(Br)ccc1NC(=O)c1sc2ncn(CC(=O)N3CCN(c4ccccn4)CC3)c(=O)c2c1C	nan
	CHEMBL1312634	20961	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	580	5	1	8	3.8	Cc1cc(Br)ccc1NC(=O)c1sc2ncn(CC(=O)N3CCN(c4ccccn4)CC3)c(=O)c2c1C	nan
	2332949	20972	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	363	3	2	5	4.7	Cc1ccc(-c2c(C#N)c(S)nc(C)c2C(=O)Nc2ccccc2C)o1	nan
	CHEMBL1312698	20972	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	363	3	2	5	4.7	Cc1ccc(-c2c(C#N)c(S)nc(C)c2C(=O)Nc2ccccc2C)o1	nan
	20957089	20981	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	426	8	1	9	2.1	CCOC(=O)C1CCN(C(=O)CCc2nnc3ccc(NCc4ccco4)nn23)CC1	nan
	CHEMBL1312760	20981	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	426	8	1	9	2.1	CCOC(=O)C1CCN(C(=O)CCc2nnc3ccc(NCc4ccco4)nn23)CC1	nan
	7064857	21273	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	5	1	5	5.1	CCc1cccc(C)c1Nc1c(-c2ccc(N(C)C)cc2)nc2cnccn12	nan
	CHEMBL1315626	21273	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	5	1	5	5.1	CCc1cccc(C)c1Nc1c(-c2ccc(N(C)C)cc2)nc2cnccn12	nan
	16299684	21284	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	483	7	1	7	2.8	CCN(CC)S(=O)(=O)c1ccc(N2CCCC2)c(NC(=O)c2nn(C)c(=O)c3ccccc23)c1	nan
	CHEMBL1315774	21284	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	483	7	1	7	2.8	CCN(CC)S(=O)(=O)c1ccc(N2CCCC2)c(NC(=O)c2nn(C)c(=O)c3ccccc23)c1	nan
	16010795	21294	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	8	1	8	2.8	COc1ccc(CCn2c(=O)c3cccnc3n(CC(=O)Nc3cccc(C)c3)c2=O)cc1OC	nan
	CHEMBL1315899	21294	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	8	1	8	2.8	COc1ccc(CCn2c(=O)c3cccnc3n(CC(=O)Nc3cccc(C)c3)c2=O)cc1OC	nan
	16018148	21374	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	3	1	4	4.4	CCn1cc2c(n1)-c1c(oc(C(=O)Nc3cccc(C)c3C)c1C)CC2	nan
	CHEMBL1316992	21374	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	3	1	4	4.4	CCn1cc2c(n1)-c1c(oc(C(=O)Nc3cccc(C)c3C)c1C)CC2	nan
	5921518	21432	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	472	8	1	8	2.1	COCCCNC(=O)/C(C#N)=C/c1c(N2CCN(c3ccccc3)CC2)nc2ccccn2c1=O	nan
	CHEMBL1317700	21432	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	472	8	1	8	2.1	COCCCNC(=O)/C(C#N)=C/c1c(N2CCN(c3ccccc3)CC2)nc2ccccn2c1=O	nan
	4062026	21479	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	504	4	1	6	4.5	Cc1ccc(Cl)cc1NC(=O)c1oc2ccc(S(=O)(=O)N3CCC4(CC3)OCCO4)cc2c1C	nan
	CHEMBL1318364	21479	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	504	4	1	6	4.5	Cc1ccc(Cl)cc1NC(=O)c1oc2ccc(S(=O)(=O)N3CCC4(CC3)OCCO4)cc2c1C	nan
	16027568	21480	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	460	6	1	8	3.9	Cc1cccc(C(=O)Nc2ccccc2C(=O)OCc2cc(=O)n3nc(C4CC4)sc3n2)c1	nan
	CHEMBL1318374	21480	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	460	6	1	8	3.9	Cc1cccc(C(=O)Nc2ccccc2C(=O)OCc2cc(=O)n3nc(C4CC4)sc3n2)c1	nan
	16028281	21494	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	7	1	7	3.4	CCc1cccc(NC(=O)Cn2ccn3nc(-c4ccc(OC)c(OC)c4)cc3c2=O)c1	nan
	CHEMBL1318465	21494	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	7	1	7	3.4	CCc1cccc(NC(=O)Cn2ccn3nc(-c4ccc(OC)c(OC)c4)cc3c2=O)c1	nan
	16017220	21515	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	8	1	6	4.8	Cc1nn(CCCC(=O)NCc2ccc(OC(C)C)cc2)c(=O)c2c1sc1ccccc12	nan
	CHEMBL1318645	21515	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	8	1	6	4.8	Cc1nn(CCCC(=O)NCc2ccc(OC(C)C)cc2)c(=O)c2c1sc1ccccc12	nan
	16027652	21566	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	490	9	1	8	4.3	CC(C)Cc1nn2c(=O)cc(COC(=O)c3ccc(NC(=O)CCc4ccccc4)cc3)nc2s1	nan
	CHEMBL1319006	21566	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	490	9	1	8	4.3	CC(C)Cc1nn2c(=O)cc(COC(=O)c3ccc(NC(=O)CCc4ccccc4)cc3)nc2s1	nan
	2998240	21673	5	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	347	3	1	5	4.2	O=C(NCc1ccc(Cl)cc1)c1cc2c(nc3sccn32)s1	nan
	CHEMBL1319990	21673	5	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	347	3	1	5	4.2	O=C(NCc1ccc(Cl)cc1)c1cc2c(nc3sccn32)s1	nan
	16007411	21691	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	3	2	3	4.4	CC(C)c1ccc(NC(=O)c2cc3c(=O)[nH]c4ccccc4c3n2C)cc1	nan
	CHEMBL1320105	21691	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	3	2	3	4.4	CC(C)c1ccc(NC(=O)c2cc3c(=O)[nH]c4ccccc4c3n2C)cc1	nan
	7692481	21729	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	336	3	1	3	3.4	COc1cc2cc(C(=O)N3CCc4ccccc4C3)[nH]c2cc1OC	nan
	CHEMBL1320436	21729	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	336	3	1	3	3.4	COc1cc2cc(C(=O)N3CCc4ccccc4C3)[nH]c2cc1OC	nan
	16019337	21799	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	3	0	9	2.6	Cc1ccc(S(=O)(=O)c2nnn3c2nc(N2CCOCC2)c2sccc23)cc1C	nan
	CHEMBL1321011	21799	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	3	0	9	2.6	Cc1ccc(S(=O)(=O)c2nnn3c2nc(N2CCOCC2)c2sccc23)cc1C	nan
	16017632	21842	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	463	3	2	6	5.0	Cc1c(C(=O)Nc2ccccc2)sc2nc(-c3cc4cc(Cl)ccc4oc3=O)[nH]c(=O)c12	nan
	CHEMBL1321440	21842	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	463	3	2	6	5.0	Cc1c(C(=O)Nc2ccccc2)sc2nc(-c3cc4cc(Cl)ccc4oc3=O)[nH]c(=O)c12	nan
	15988428	21844	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	1	0	5	3.6	Cn1c(=O)n(-c2cccc(Cl)c2)c(=O)c2sc3ccccc3c21	nan
	CHEMBL1321495	21844	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	1	0	5	3.6	Cn1c(=O)n(-c2cccc(Cl)c2)c(=O)c2sc3ccccc3c21	nan
	2988303	21846	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	345	4	0	6	3.2	Cn1c2ccc(F)cc2c2nnc(SCCN3CCCCC3)nc21	nan
	CHEMBL1321509	21846	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	345	4	0	6	3.2	Cn1c2ccc(F)cc2c2nnc(SCCN3CCCCC3)nc21	nan
	16017566	21877	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	6	1	6	2.9	Cc1ccccc1C(=O)Nc1nnc(S(=O)(=O)N(C)Cc2ccccc2)s1	nan
	CHEMBL1321733	21877	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	6	1	6	2.9	Cc1ccccc1C(=O)Nc1nnc(S(=O)(=O)N(C)Cc2ccccc2)s1	nan
	2158383	22030	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	331	6	1	6	2.1	CCOCCCNC(=O)c1cc2c(=O)n3ccccc3nc2s1	nan
	CHEMBL1323129	22030	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	331	6	1	6	2.1	CCOCCCNC(=O)c1cc2c(=O)n3ccccc3nc2s1	nan
	6076700	22162	6	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	10	2	7	2.1	CCOc1ccc(C(=O)C2=C(O)C(=O)N(CCOCCO)C2c2cccnc2)cc1	nan
	CHEMBL1324242	22162	6	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	10	2	7	2.1	CCOc1ccc(C(=O)C2=C(O)C(=O)N(CCOCCO)C2c2cccnc2)cc1	nan
	16805712	22206	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	8	2	9	1.0	Cn1c(=O)c2sccc2n2c(CCCC(=O)NCCc3ccc(S(N)(=O)=O)cc3)nnc12	nan
	CHEMBL1324587	22206	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	8	2	9	1.0	Cn1c(=O)c2sccc2n2c(CCCC(=O)NCCc3ccc(S(N)(=O)=O)cc3)nnc12	nan
	3152453	22444	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	6	3	8	1.1	Cc1cccn2c(=O)c3cc(C(=O)NCc4cccnc4)c(=N)n(CCCO)c3nc12	nan
	CHEMBL1326883	22444	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	6	3	8	1.1	Cc1cccn2c(=O)c3cc(C(=O)NCc4cccnc4)c(=N)n(CCCO)c3nc12	nan
	5048043	22666	9	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	4	0	4	5.0	Cc1nn(C)cc1CN(C)C(=O)c1cc(-c2ccccc2)nc2ccc(Br)cc12	nan
	CHEMBL1328648	22666	9	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	4	0	4	5.0	Cc1nn(C)cc1CN(C)C(=O)c1cc(-c2ccccc2)nc2ccc(Br)cc12	nan
	135706200	22689	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	454	5	1	6	3.2	CN(Cc1nc(O)c2ccccc2n1)C(=O)c1cccc(S(=O)(=O)N2CCCCCC2)c1	nan
	CHEMBL1328897	22689	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	454	5	1	6	3.2	CN(Cc1nc(O)c2ccccc2n1)C(=O)c1cccc(S(=O)(=O)N2CCCCCC2)c1	nan
	5730619	22714	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	398	7	2	7	3.3	Cc1noc(NS(=O)(=O)c2ccc(N/C=C\C(=O)c3ccncc3)cc2)c1C	nan
	CHEMBL1329130	22714	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	398	7	2	7	3.3	Cc1noc(NS(=O)(=O)c2ccc(N/C=C\C(=O)c3ccncc3)cc2)c1C	nan
	2937900	22749	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	5	1	5	4.3	O=C(C1=C(O)C(=O)N(Cc2ccco2)C1c1ccccc1F)c1cccs1	nan
	CHEMBL1329400	22749	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	5	1	5	4.3	O=C(C1=C(O)C(=O)N(Cc2ccco2)C1c1ccccc1F)c1cccs1	nan
	2765497	22763	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	7	1	5	2.4	Cc1ccc(S(=O)(=O)C(C)C(=O)NCCS(=O)(=O)c2ccc(Cl)cc2)cc1	nan
	CHEMBL1329544	22763	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	7	1	5	2.4	Cc1ccc(S(=O)(=O)C(C)C(=O)NCCS(=O)(=O)c2ccc(Cl)cc2)cc1	nan
	44142302	22766	0	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	3	1	4	2.8	CN(C)c1ccc(C#Cc2ccc3cc(CCO)oc(=O)c3c2)cc1	nan
	CHEMBL1329575	22766	0	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	3	1	4	2.8	CN(C)c1ccc(C#Cc2ccc3cc(CCO)oc(=O)c3c2)cc1	nan
	16011595	22819	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	467	9	1	7	4.7	CCCCOc1ccc(CNC(=O)C2CCCN(c3nnc(-n4c(C)ccc4C)s3)C2)cc1	nan
	CHEMBL1330008	22819	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	467	9	1	7	4.7	CCCCOc1ccc(CNC(=O)C2CCCN(c3nnc(-n4c(C)ccc4C)s3)C2)cc1	nan
	4181210	22843	15	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	348	4	1	5	3.9	Cc1ccc(NC(=O)CSc2nnc3ccc4ccccc4n23)cc1	nan
	CHEMBL1330254	22843	15	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	348	4	1	5	3.9	Cc1ccc(NC(=O)CSc2nnc3ccc4ccccc4n23)cc1	nan
	1548033	22845	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	229	3	3	7	-0.6	CN(C)C(=O)CNc1nnc(S)nc1O	nan
	CHEMBL1330266	22845	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	229	3	3	7	-0.6	CN(C)C(=O)CNc1nnc(S)nc1O	nan
	1960924	22937	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	4	4	6	2.4	COc1ccc(C(=O)NC(=S)Nc2ccc3[nH]c(O)nc3c2)c(OC)c1	nan
	CHEMBL1330933	22937	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	4	4	6	2.4	COc1ccc(C(=O)NC(=S)Nc2ccc3[nH]c(O)nc3c2)c(OC)c1	nan
	16022880	23006	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	9	2	7	4.3	COc1ccccc1NC(=O)Cn1c(=O)c(CNc2ccccc2)cc2cc(OC)c(OC)cc21	nan
	CHEMBL1331405	23006	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	9	2	7	4.3	COc1ccccc1NC(=O)Cn1c(=O)c(CNc2ccccc2)cc2cc(OC)c(OC)cc21	nan
	995088	23045	12	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	4	1	4	4.9	Cc1ccc(-c2cc(C(=O)NCc3cnn(C)c3C)c3cc(Br)ccc3n2)cc1	nan
	CHEMBL1331738	23045	12	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	4	1	4	4.9	Cc1ccc(-c2cc(C(=O)NCc3cnn(C)c3C)c3cc(Br)ccc3n2)cc1	nan
	4975488	23228	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	3	0	8	1.8	Cc1nn2c(-c3ccc(S(=O)(=O)N4CCN(C)CC4)o3)nnc2c2ccccc12	nan
	CHEMBL1333127	23228	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	3	0	8	1.8	Cc1nn2c(-c3ccc(S(=O)(=O)N4CCN(C)CC4)o3)nnc2c2ccccc12	nan
	5219389	23287	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	485	7	1	7	2.9	CCN(CC)S(=O)(=O)c1ccc(N2CCOCC2)c(NC(=O)c2cc3ccccc3oc2=O)c1	nan
	CHEMBL1333624	23287	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	485	7	1	7	2.9	CCN(CC)S(=O)(=O)c1ccc(N2CCOCC2)c(NC(=O)c2cc3ccccc3oc2=O)c1	nan
	1298840	23297	10	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	6	1	7	5.1	CCn1c(SCC(=O)Nc2nc3ccccc3s2)nnc1-c1ccc(Br)cc1	nan
	CHEMBL1333690	23297	10	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	6	1	7	5.1	CCn1c(SCC(=O)Nc2nc3ccccc3s2)nnc1-c1ccc(Br)cc1	nan
	3586634	23318	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	8	1	7	5.2	CCCCn1c(SCC(=O)Nc2cccc(OC)c2)nc2c(sc3ccccc32)c1=O	nan
	CHEMBL1333854	23318	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	8	1	7	5.2	CCCCn1c(SCC(=O)Nc2cccc(OC)c2)nc2c(sc3ccccc32)c1=O	nan
	1088584	23323	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	306	4	1	3	3.8	CC(=O)c1cn(CC(=O)Nc2ccc(C)cc2)c2ccccc12	nan
	CHEMBL1333897	23323	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	306	4	1	3	3.8	CC(=O)c1cn(CC(=O)Nc2ccc(C)cc2)c2ccccc12	nan
	1912959	23432	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	5	4	7	2.5	Cc1cc(C)nc(NC(=N)Nc2ccc(S(=O)(=O)Nc3nccc(C)n3)cc2)n1	nan
	5728937	23432	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	5	4	7	2.5	Cc1cc(C)nc(NC(=N)Nc2ccc(S(=O)(=O)Nc3nccc(C)n3)cc2)n1	nan
	5925428	23432	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	5	4	7	2.5	Cc1cc(C)nc(NC(=N)Nc2ccc(S(=O)(=O)Nc3nccc(C)n3)cc2)n1	nan
	CHEMBL1334749	23432	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	5	4	7	2.5	Cc1cc(C)nc(NC(=N)Nc2ccc(S(=O)(=O)Nc3nccc(C)n3)cc2)n1	nan
	5302178	23449	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	2	0	5	2.3	CC1CCCN(S(=O)(=O)c2ccc3c(c2)c(=O)nc2ccccn23)C1	nan
	CHEMBL1334923	23449	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	2	0	5	2.3	CC1CCCN(S(=O)(=O)c2ccc3c(c2)c(=O)nc2ccccn23)C1	nan
	15988344	23539	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	485	8	1	7	4.6	COc1ccc(CNC(=O)CSc2nc3ccsc3c(=O)n2Cc2ccccc2Cl)cc1	nan
	CHEMBL1335550	23539	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	485	8	1	7	4.6	COc1ccc(CNC(=O)CSc2nc3ccsc3c(=O)n2Cc2ccccc2Cl)cc1	nan
	3236871	23579	7	None	-8	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	203	1	0	2	3.7	CCn1c(C)cc(=S)c2ccccc21	nan
	CHEMBL1335833	23579	7	None	-8	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	203	1	0	2	3.7	CCn1c(C)cc(=S)c2ccccc21	nan
	3323389	23598	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	4	2	7	4.0	CC(=O)c1ccc(NC(=O)c2sc3nc(N4CCOCC4)c4c(c3c2N)CCCC4)cc1	nan
	CHEMBL1336041	23598	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	4	2	7	4.0	CC(=O)c1ccc(NC(=O)c2sc3nc(N4CCOCC4)c4c(c3c2N)CCCC4)cc1	nan
	135413771	23689	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	6	1	7	4.9	COc1cc(C2CC(c3c(C)cc(C)nc3O)=NN2c2ccccc2F)cc(OC)c1OC	nan
	CHEMBL1336821	23689	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	6	1	7	4.9	COc1cc(C2CC(c3c(C)cc(C)nc3O)=NN2c2ccccc2F)cc(OC)c1OC	nan
	2140203	23694	1	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	309	3	0	7	2.9	COc1ccc(-n2nnnc2-c2nc3ccccc3s2)cc1	nan
	CHEMBL1336848	23694	1	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	309	3	0	7	2.9	COc1ccc(-n2nnnc2-c2nc3ccccc3s2)cc1	nan
	2088251	23740	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	6	0	6	3.1	CCOc1ccc(CC(=O)OCc2cc(=O)n3cc(Br)ccc3n2)cc1	nan
	CHEMBL1337298	23740	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	6	0	6	3.1	CCOc1ccc(CC(=O)OCc2cc(=O)n3cc(Br)ccc3n2)cc1	nan
	1301366	23755	14	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	366	5	1	5	4.1	O=C(CCSc1nnc2ccc3ccccc3n12)Nc1ccc(F)cc1	nan
	CHEMBL1337428	23755	14	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	366	5	1	5	4.1	O=C(CCSc1nnc2ccc3ccccc3n12)Nc1ccc(F)cc1	nan
	16015123	23797	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	5	1	5	4.6	Cc1cccc(C)c1OCC(=O)Nc1nc(-c2ccc(Br)cc2)ns1	nan
	CHEMBL1337810	23797	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	5	1	5	4.6	Cc1cccc(C)c1OCC(=O)Nc1nc(-c2ccc(Br)cc2)ns1	nan
	16034823	23822	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	467	6	1	4	4.9	Cc1oc(-c2cccc(Br)c2)nc1CN1CCC(C(=O)NCc2ccccc2)CC1	nan
	CHEMBL1338052	23822	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	467	6	1	4	4.9	Cc1oc(-c2cccc(Br)c2)nc1CN1CCC(C(=O)NCc2ccccc2)CC1	nan
	2137854	23926	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	5	1	6	4.6	COc1ccc(-c2nnn3c2nc(NCc2ccccc2)c2ccccc23)cc1	nan
	CHEMBL1338842	23926	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	5	1	6	4.6	COc1ccc(-c2nnn3c2nc(NCc2ccccc2)c2ccccc23)cc1	nan
	16023227	23940	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	475	6	2	6	4.7	O=C(Cn1c(=O)c(CNc2ccccc2)cc2cc3c(cc21)OCCO3)Nc1ccccc1Cl	nan
	CHEMBL1339042	23940	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	475	6	2	6	4.7	O=C(Cn1c(=O)c(CNc2ccccc2)cc2cc3c(cc21)OCCO3)Nc1ccccc1Cl	nan
	4012037	24010	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	282	3	0	5	4.3	c1coc(CSc2ncnc3c2oc2ccccc23)c1	nan
	CHEMBL1339672	24010	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	282	3	0	5	4.3	c1coc(CSc2ncnc3c2oc2ccccc23)c1	nan
	16406923	24149	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	442	7	3	6	2.3	Cc1coc2c1c(C)cc1oc(=O)c(CC(=O)NCC(=O)N[C@H](C(=O)O)C(C)C)c(C)c12	nan
	CHEMBL1340985	24149	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	442	7	3	6	2.3	Cc1coc2c1c(C)cc1oc(=O)c(CC(=O)NCC(=O)N[C@H](C(=O)O)C(C)C)c(C)c12	nan
	1859832	24196	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	485	6	0	7	4.3	COc1ccc(CCn2c(-c3ccc(F)cc3)nc3c(c(=O)c4ccccc4n3C)c2=O)cc1OC	nan
	CHEMBL1341311	24196	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	485	6	0	7	4.3	COc1ccc(CCn2c(-c3ccc(F)cc3)nc3c(c(=O)c4ccccc4n3C)c2=O)cc1OC	nan
	6402475	24431	10	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	2	1	4	4.2	Nc1nc(-c2ccc(Cl)cc2)nnc1-c1ccc(Br)cc1	nan
	CHEMBL1343242	24431	10	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	2	1	4	4.2	Nc1nc(-c2ccc(Cl)cc2)nnc1-c1ccc(Br)cc1	nan
	1831284	24461	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	344	4	1	5	3.5	Cc1cc(C)n(-c2ccc(Oc3ccccc3)c(S(=O)(=O)O)c2)n1	nan
	4401304	24461	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	344	4	1	5	3.5	Cc1cc(C)n(-c2ccc(Oc3ccccc3)c(S(=O)(=O)O)c2)n1	nan
	CHEMBL1343474	24461	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	344	4	1	5	3.5	Cc1cc(C)n(-c2ccc(Oc3ccccc3)c(S(=O)(=O)O)c2)n1	nan
	3238813	24474	11	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	336	5	1	5	3.8	COc1ccc(-c2cc(C(=O)Nc3cccc(C(C)=O)c3)no2)cc1	nan
	CHEMBL1343596	24474	11	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	336	5	1	5	3.8	COc1ccc(-c2cc(C(=O)Nc3cccc(C(C)=O)c3)no2)cc1	nan
	2821813	24543	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	322	2	1	3	4.9	O=C(Nc1ccc(Cl)cc1Cl)c1ccc2ncsc2c1	nan
	CHEMBL1344238	24543	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	322	2	1	3	4.9	O=C(Nc1ccc(Cl)cc1Cl)c1ccc2ncsc2c1	nan
	3158796	24619	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	311	2	2	5	2.9	Cc1cccc(N2C(S)=C(C#N)C(=O)NC2c2ccco2)c1	nan
	CHEMBL1344888	24619	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	311	2	2	5	2.9	Cc1cccc(N2C(S)=C(C#N)C(=O)NC2c2ccco2)c1	nan
	2558333	24687	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	5	1	9	4.8	CCc1cc2c(SCc3nc(O)c4c(C)c(C(C)=O)sc4n3)ncnc2s1	nan
	CHEMBL1345471	24687	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	5	1	9	4.8	CCc1cc2c(SCc3nc(O)c4c(C)c(C(C)=O)sc4n3)ncnc2s1	nan
	7708092	24744	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	6	1	7	2.8	COc1ccc(C(=O)Nc2nnc(S(=O)(=O)Cc3ccccc3)s2)cc1	nan
	CHEMBL1346001	24744	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	6	1	7	2.8	COc1ccc(C(=O)Nc2nnc(S(=O)(=O)Cc3ccccc3)s2)cc1	nan
	4519571	24895	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	317	2	1	6	2.9	O=c1c2cc(Cl)ccc2nc(-c2ccc([N+](=O)[O-])cc2)n1O	nan
	CHEMBL1347185	24895	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	317	2	1	6	2.9	O=c1c2cc(Cl)ccc2nc(-c2ccc([N+](=O)[O-])cc2)n1O	nan
	24790251	25059	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	5	1	4	4.2	O=C(NCC1CCOCC1)c1ccc2nc(Cc3cccc(Cl)c3)oc2c1	nan
	CHEMBL1348671	25059	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	5	1	4	4.2	O=C(NCC1CCOCC1)c1ccc2nc(Cc3cccc(Cl)c3)oc2c1	nan
	16194270	25165	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	7	1	6	3.6	COc1cccc(CNC(=O)CSc2ccc(-c3cccs3)nn2)c1	nan
	CHEMBL1349515	25165	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	7	1	6	3.6	COc1cccc(CNC(=O)CSc2ccc(-c3cccs3)nn2)c1	nan
	2308471	25240	6	None	-8	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	6	0	5	5.7	N#Cc1c(-c2ccc(F)cc2)cc(C2CC2)nc1SCC(=O)c1cccs1	nan
	CHEMBL1350179	25240	6	None	-8	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	6	0	5	5.7	N#Cc1c(-c2ccc(F)cc2)cc(C2CC2)nc1SCC(=O)c1cccs1	nan
	1246228	25314	12	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	310	2	1	4	4.5	Cc1sc(NC(=O)c2oc3ccccc3c2C)c(C#N)c1C	nan
	CHEMBL1350806	25314	12	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	310	2	1	4	4.5	Cc1sc(NC(=O)c2oc3ccccc3c2C)c(C#N)c1C	nan
	3810755	25492	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	6	1	6	3.5	O=C(C1=C(O)C(=O)N(CCN2CCOCC2)C1c1ccc(F)cc1)c1cc2ccccc2o1	nan
	5224304	25492	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	6	1	6	3.5	O=C(C1=C(O)C(=O)N(CCN2CCOCC2)C1c1ccc(F)cc1)c1cc2ccccc2o1	nan
	CHEMBL1352306	25492	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	6	1	6	3.5	O=C(C1=C(O)C(=O)N(CCN2CCOCC2)C1c1ccc(F)cc1)c1cc2ccccc2o1	nan
	3710699	25604	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	238	3	0	5	3.2	CSc1nnc(-c2ccccc2SC)o1	nan
	CHEMBL1353167	25604	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	238	3	0	5	3.2	CSc1nnc(-c2ccccc2SC)o1	nan
	2408978	25699	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	3	1	4	3.8	O=S(=O)(Nc1nc2ccccc2nc1Cl)c1ccc(Br)cc1	nan
	CHEMBL1353794	25699	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	3	1	4	3.8	O=S(=O)(Nc1nc2ccccc2nc1Cl)c1ccc(Br)cc1	nan
	2137114	25788	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	482	5	1	5	4.4	Cc1ccc(C)c(NC(=O)Cn2cc(S(=O)(=O)c3ccc(F)cc3)c(=O)c3cc(F)ccc32)c1	nan
	CHEMBL1354500	25788	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	482	5	1	5	4.4	Cc1ccc(C)c(NC(=O)Cn2cc(S(=O)(=O)c3ccc(F)cc3)c(=O)c3cc(F)ccc32)c1	nan
	7177775	25817	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	4	0	7	1.8	Cc1ccc2nc(SCC(=O)N3CCN(c4ccccc4)CC3)nc(=O)n2c1	nan
	CHEMBL1354880	25817	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	4	0	7	1.8	Cc1ccc2nc(SCC(=O)N3CCN(c4ccccc4)CC3)nc(=O)n2c1	nan
	16015313	25821	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	466	6	1	6	5.8	COc1cccc(NC(=O)c2sc(-n3nc(C)c(Cc4ccccc4Cl)c3C)nc2C)c1	nan
	CHEMBL1354922	25821	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	466	6	1	6	5.8	COc1cccc(NC(=O)c2sc(-n3nc(C)c(Cc4ccccc4Cl)c3C)nc2C)c1	nan
	16019333	25822	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	5	1	8	4.8	CCc1ccc(Nc2nc3c(S(=O)(=O)c4ccc(C)cc4)nnn3c3ccsc23)cc1	nan
	CHEMBL1354928	25822	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	5	1	8	4.8	CCc1ccc(Nc2nc3c(S(=O)(=O)c4ccc(C)cc4)nnn3c3ccsc23)cc1	nan
	15988332	25852	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	464	5	0	9	2.1	CC(=O)c1ccc(N2CCN(C(=O)CCc3nnc4n(C)c(=O)c5sccc5n34)CC2)cc1	nan
	CHEMBL1355272	25852	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	464	5	0	9	2.1	CC(=O)c1ccc(N2CCN(C(=O)CCc3nnc4n(C)c(=O)c5sccc5n34)CC2)cc1	nan
	15988502	25885	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	4	1	4	4.5	O=C(Cn1c(=O)nc(-c2ccccc2)c2ccccc21)Nc1ccc(Cl)cc1F	nan
	CHEMBL1355773	25885	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	4	1	4	4.5	O=C(Cn1c(=O)nc(-c2ccccc2)c2ccccc21)Nc1ccc(Cl)cc1F	nan
	2893260	25990	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	6	1	9	4.0	CCC(Sc1nnc2c3ccccc3n(C)c2n1)C(=O)Nc1nnc(C(C)C)s1	nan
	CHEMBL1357131	25990	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	6	1	9	4.0	CCC(Sc1nnc2c3ccccc3n(C)c2n1)C(=O)Nc1nnc(C(C)C)s1	nan
	16018894	25998	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	5	0	7	5.8	CCc1nnc(SCc2nc(-c3ccccc3)oc2C)c2cc3sccc3n12	nan
	CHEMBL1357169	25998	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	5	0	7	5.8	CCc1nnc(SCc2nc(-c3ccccc3)oc2C)c2cc3sccc3n12	nan
	16012142	26034	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	7	1	5	5.0	CC(CNC(=O)Cn1ncc2c3ccccc3n(Cc3cccc(Cl)c3)c2c1=O)c1ccccc1	nan
	CHEMBL1357797	26034	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	7	1	5	5.0	CC(CNC(=O)Cn1ncc2c3ccccc3n(Cc3cccc(Cl)c3)c2c1=O)c1ccccc1	nan
	16018042	26052	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	6	1	5	3.2	CN(C)c1ccc(CNC(=O)CCn2c(=O)c3cccn3c3ccc(F)cc32)cc1	nan
	CHEMBL1358052	26052	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	6	1	5	3.2	CN(C)c1ccc(CNC(=O)CCn2c(=O)c3cccn3c3ccc(F)cc32)cc1	nan
	7711889	26112	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	4	1	6	0.2	Cn1c(CNS(=O)(=O)c2ccc(Cl)cc2)cc(=O)n(C)c1=O	nan
	CHEMBL1358800	26112	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	4	1	6	0.2	Cn1c(CNS(=O)(=O)c2ccc(Cl)cc2)cc(=O)n(C)c1=O	nan
	16018591	26175	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	6	1	7	2.7	COc1cc(NS(=O)(=O)c2cc3c(cc2C)N(C)CCO3)cc(OC)c1OC	nan
	CHEMBL1359260	26175	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	6	1	7	2.7	COc1cc(NS(=O)(=O)c2cc3c(cc2C)N(C)CCO3)cc(OC)c1OC	nan
	4302860	26186	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	7	1	6	4.2	CCOc1ccc(C2C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2Cc2cccnc2)cc1	nan
	4302861	26186	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	7	1	6	4.2	CCOc1ccc(C2C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2Cc2cccnc2)cc1	nan
	CHEMBL1359331	26186	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	7	1	6	4.2	CCOc1ccc(C2C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2Cc2cccnc2)cc1	nan
	1270409	26196	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	4	1	11	-0.4	Cn1c(=O)c2c(nc(Sc3ncnn3CC(=O)NC(C)(C)C)n2C)n(C)c1=O	nan
	CHEMBL1359403	26196	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	4	1	11	-0.4	Cn1c(=O)c2c(nc(Sc3ncnn3CC(=O)NC(C)(C)C)n2C)n(C)c1=O	nan
	1472977	26263	15	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	446	2	0	3	5.3	Brc1cc(Br)c2nc(-c3ccc(N4CCOCC4)cc3)ccc2c1	nan
	CHEMBL1360031	26263	15	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	446	2	0	3	5.3	Brc1cc(Br)c2nc(-c3ccc(N4CCOCC4)cc3)ccc2c1	nan
	5910118	26298	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	5	2	7	3.3	O=C(C1=C(O)C(=O)N(Cc2cccnc2)C1c1cccc(O)c1)c1ccc2c(c1)OCCO2	nan
	CHEMBL1360299	26298	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	5	2	7	3.3	O=C(C1=C(O)C(=O)N(Cc2cccnc2)C1c1cccc(O)c1)c1ccc2c(c1)OCCO2	nan
	2519123	26357	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	302	5	1	5	2.2	Cc1cccc(-c2nnc(SCC(=O)NC3CC3)n2C)c1	nan
	CHEMBL1360828	26357	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	302	5	1	5	2.2	Cc1cccc(-c2nnc(SCC(=O)NC3CC3)n2C)c1	nan
	1637639	26415	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	332	7	1	5	3.8	CC(=O)c1sc(NC(=O)CCCOc2ccccc2C)nc1C	nan
	CHEMBL1361423	26415	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	332	7	1	5	3.8	CC(=O)c1sc(NC(=O)CCCOc2ccccc2C)nc1C	nan
	16029936	26427	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	3	1	6	2.5	Cc1cc(C(=O)Nc2c(C)nc3ccccn3c2=O)ccc1[N+](=O)[O-]	nan
	CHEMBL1361527	26427	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	3	1	6	2.5	Cc1cc(C(=O)Nc2c(C)nc3ccccn3c2=O)ccc1[N+](=O)[O-]	nan
	16021826	26443	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	4	1	4	5.1	CSc1ncc(C(=O)Nc2cc(Cl)ccc2C)c(-c2ccccc2)n1	nan
	CHEMBL1361623	26443	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	4	1	4	5.1	CSc1ncc(C(=O)Nc2cc(Cl)ccc2C)c(-c2ccccc2)n1	nan
	135399263	26566	15	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	4	2	5	3.7	Cc1cccc(C)c1NC(=O)CSc1nc(O)c2ccccc2n1	nan
	CHEMBL1362620	26566	15	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	4	2	5	3.7	Cc1cccc(C)c1NC(=O)CSc1nc(O)c2ccccc2n1	nan
	5225696	26679	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	2	2	3	2.3	CC1=C(C#N)C(NC(=O)c2ccccc2Cl)(C(F)(F)F)C(=O)N1	nan
	CHEMBL1363628	26679	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	2	2	3	2.3	CC1=C(C#N)C(NC(=O)c2ccccc2Cl)(C(F)(F)F)C(=O)N1	nan
	1300378	26731	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	7	2	5	3.9	CC(=O)c1ccc(NC(=O)COc2ccccc2C(=O)Nc2ccc(C)cn2)cc1	nan
	CHEMBL1364136	26731	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	7	2	5	3.9	CC(=O)c1ccc(NC(=O)COc2ccccc2C(=O)Nc2ccc(C)cn2)cc1	nan
	1207158	26755	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	6	2	5	4.7	O=C(CSc1nc(-c2ccccc2)nc2ccccc12)Nc1cccc(C(=O)O)c1	nan
	CHEMBL1364382	26755	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	6	2	5	4.7	O=C(CSc1nc(-c2ccccc2)nc2ccccc12)Nc1cccc(C(=O)O)c1	nan
	658008	26757	6	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	347	6	1	5	3.7	CCN(CC)C(=O)CSC1=C(C#N)C(c2cccs2)C=C(C)N1	nan
	CHEMBL1364397	26757	6	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	347	6	1	5	3.7	CCN(CC)C(=O)CSC1=C(C#N)C(c2cccs2)C=C(C)N1	nan
	1071060	26976	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	5	2	6	3.1	COC(=O)c1c(NC(C)=O)sc(C(=O)Nc2ccccc2OC)c1C	nan
	CHEMBL1366254	26976	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	5	2	6	3.1	COC(=O)c1c(NC(C)=O)sc(C(=O)Nc2ccccc2OC)c1C	nan
	711643	27025	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	325	5	1	5	3.7	Cc1ccc(C(=O)Nc2nnc(COc3ccccc3)s2)cc1	nan
	CHEMBL1366637	27025	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	325	5	1	5	3.7	Cc1ccc(C(=O)Nc2nnc(COc3ccccc3)s2)cc1	nan
	16030455	27026	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	6	1	4	6.0	O=C(CSc1nc2ccccc2nc1Cc1ccccc1)Nc1ccccc1C(F)(F)F	nan
	CHEMBL1366645	27026	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	6	1	4	6.0	O=C(CSc1nc2ccccc2nc1Cc1ccccc1)Nc1ccccc1C(F)(F)F	nan
	16010113	27034	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	6	1	6	3.3	CC(C)Oc1ccc(CNC(=O)C2CCN(c3nc4ccccc4n(C)c3=O)CC2)cc1	nan
	CHEMBL1366755	27034	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	6	1	6	3.3	CC(C)Oc1ccc(CNC(=O)C2CCN(c3nc4ccccc4n(C)c3=O)CC2)cc1	nan
	2115552	27059	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	4	1	6	3.2	Cc1[nH]c2ccccc2c1C(=O)COC(=O)c1ccc2c(=O)n3c(nc2c1)CCC3	nan
	CHEMBL1366975	27059	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	4	1	6	3.2	Cc1[nH]c2ccccc2c1C(=O)COC(=O)c1ccc2c(=O)n3c(nc2c1)CCC3	nan
	868037	27160	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	275	4	1	4	3.4	COc1cccc2c(S)c(CCC(C)=O)c(C)nc12	nan
	CHEMBL1367790	27160	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	275	4	1	4	3.4	COc1cccc2c(S)c(CCC(C)=O)c(C)nc12	nan
	1086871	27297	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	8	1	8	3.4	COc1ccc(Cc2nnc(NC(=O)c3ccc(OC)c(OC)c3)s2)cc1OC	nan
	CHEMBL1368875	27297	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	8	1	8	3.4	COc1ccc(Cc2nnc(NC(=O)c3ccc(OC)c(OC)c3)s2)cc1OC	nan
	2054025	27583	10	None	-1	3	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	4	0	7	4.0	COC(=O)c1ccc(CSc2ncnc3c2oc2ccccc23)o1	nan
	CHEMBL1370794	27583	10	None	-1	3	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	4	0	7	4.0	COC(=O)c1ccc(CSc2ncnc3c2oc2ccccc23)o1	nan
	2951249	27645	18	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	7	1	7	3.5	COc1ccc(OC)c(C2C(C(=O)c3ccco3)=C(O)C(=O)N2Cc2cccnc2)c1	nan
	4590179	27645	18	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	7	1	7	3.5	COc1ccc(OC)c(C2C(C(=O)c3ccco3)=C(O)C(=O)N2Cc2cccnc2)c1	nan
	CHEMBL1371319	27645	18	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	7	1	7	3.5	COc1ccc(OC)c(C2C(C(=O)c3ccco3)=C(O)C(=O)N2Cc2cccnc2)c1	nan
	1520515	27735	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	3	0	7	4.4	COc1ccc(-c2nc3ccccc3n3c(-c4ccccc4)c4c(=O)n(C)c(=O)n(C)c4c23)cc1	nan
	CHEMBL1372041	27735	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	3	0	7	4.4	COc1ccc(-c2nc3ccccc3n3c(-c4ccccc4)c4c(=O)n(C)c(=O)n(C)c4c23)cc1	nan
	15988500	27796	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	584	13	2	9	3.7	CCCCCNC(=O)C1CCC(Cn2c(=O)c3sccc3n(CC(=O)NCc3cccc(OC)c3OC)c2=O)CC1	nan
	CHEMBL1372455	27796	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	584	13	2	9	3.7	CCCCCNC(=O)C1CCC(Cn2c(=O)c3sccc3n(CC(=O)NCc3cccc(OC)c3OC)c2=O)CC1	nan
	16030415	27878	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	5	1	5	4.0	Cc1ccc2nc(COc3ccccc3NC(=O)c3ccccc3F)cc(=O)n2c1	nan
	CHEMBL1372965	27878	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	5	1	5	4.0	Cc1ccc2nc(COc3ccccc3NC(=O)c3ccccc3F)cc(=O)n2c1	nan
	3141921	27904	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	295	3	0	4	4.1	N#CCSc1nc(-c2ccccc2)nc2ccc(F)cc12	nan
	CHEMBL1373143	27904	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	295	3	0	4	4.1	N#CCSc1nc(-c2ccccc2)nc2ccc(F)cc12	nan
	5740603	28015	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	319	4	2	4	3.3	COc1ccc2[nH]c(/C(C#N)=C\c3ccc(C(=O)O)cc3)nc2c1	nan
	CHEMBL1373830	28015	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	319	4	2	4	3.3	COc1ccc2[nH]c(/C(C#N)=C\c3ccc(C(=O)O)cc3)nc2c1	nan
	4965542	28044	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	6	1	11	0.2	C=CCSc1nnc(NC(=O)Cn2cnc3c2c(=O)n(C)c(=O)n3C)s1	nan
	CHEMBL1374122	28044	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	6	1	11	0.2	C=CCSc1nnc(NC(=O)Cn2cnc3c2c(=O)n(C)c(=O)n3C)s1	nan
	3496625	28045	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	7	1	7	5.2	Cc1cc(N2C(=O)C(O)=C(C(=O)c3ccc(C)o3)C2c2ccc(OCc3ccccc3)cc2)no1	nan
	CHEMBL1374123	28045	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	7	1	7	5.2	Cc1cc(N2C(=O)C(O)=C(C(=O)c3ccc(C)o3)C2c2ccc(OCc3ccccc3)cc2)no1	nan
	2945949	28140	18	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	335	4	1	5	2.5	O=C(CCN1C(=O)c2cccc3cccc(c23)C1=O)Nc1ccon1	nan
	CHEMBL1374764	28140	18	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	335	4	1	5	2.5	O=C(CCN1C(=O)c2cccc3cccc(c23)C1=O)Nc1ccon1	nan
	15989514	28180	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	535	8	1	7	3.7	O=C(Cn1c(=O)n(CCCS(=O)(=O)C2CCCCC2)c(=O)c2ccccc21)Nc1ccc(F)c(Cl)c1	nan
	CHEMBL1375013	28180	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	535	8	1	7	3.7	O=C(Cn1c(=O)n(CCCS(=O)(=O)C2CCCCC2)c(=O)c2ccccc21)Nc1ccc(F)c(Cl)c1	nan
	2212703	28246	10	None	-4	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	285	4	1	4	3.0	O=C(O)Cn1cc(C(=O)c2cccs2)c2ccccc21	nan
	CHEMBL1375453	28246	10	None	-4	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	285	4	1	4	3.0	O=C(O)Cn1cc(C(=O)c2cccs2)c2ccccc21	nan
	2471579	28270	9	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	521	9	2	7	5.5	COc1ccc(-c2nc(NC(=O)c3ccc(OCC(=O)Nc4ccc(F)cc4)c(OC)c3)sc2C)cc1	nan
	CHEMBL1375669	28270	9	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	521	9	2	7	5.5	COc1ccc(-c2nc(NC(=O)c3ccc(OCC(=O)Nc4ccc(F)cc4)c(OC)c3)sc2C)cc1	nan
	3167528	28286	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	6	2	7	2.9	Cc1ccc(OCC(=O)NNC(=O)CSc2ncnc3sc(C)c(C)c23)cc1	nan
	CHEMBL1375776	28286	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	6	2	7	2.9	Cc1ccc(OCC(=O)NNC(=O)CSc2ncnc3sc(C)c(C)c23)cc1	nan
	2397772	28318	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	9	1	10	1.1	COc1cc(C(=O)OCC(=O)c2c(N)n(C)c(=O)n(C)c2=O)ccc1OCCC(C)C	nan
	CHEMBL1376204	28318	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	9	1	10	1.1	COc1cc(C(=O)OCC(=O)c2c(N)n(C)c(=O)n(C)c2=O)ccc1OCCC(C)C	nan
	1767629	28382	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	2	0	4	5.0	O=c1oc2c3c(ccc2c2ccccc12)OCN(Cc1ccccc1Cl)C3	nan
	CHEMBL1376703	28382	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	2	0	4	5.0	O=c1oc2c3c(ccc2c2ccccc12)OCN(Cc1ccccc1Cl)C3	nan
	16024679	28468	1	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	441	7	1	6	3.3	COc1cccc(C(=O)c2cn(CC(=O)NCc3ccccc3)c3nc(C)ccc3c2=O)c1	nan
	CHEMBL1377672	28468	1	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	441	7	1	6	3.3	COc1cccc(C(=O)c2cn(CC(=O)NCc3ccccc3)c3nc(C)ccc3c2=O)c1	nan
	135520779	28484	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	313	2	1	6	3.3	CCCc1nc2oc3c(O)ncnc3c2c2c1COC(C)(C)C2	nan
	CHEMBL1377764	28484	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	313	2	1	6	3.3	CCCc1nc2oc3c(O)ncnc3c2c2c1COC(C)(C)C2	nan
	16194561	28492	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	5	1	10	2.1	Cc1nnc(NC(=O)CSc2ccc3nnc(-c4ccccn4)n3n2)s1	nan
	CHEMBL1377828	28492	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	5	1	10	2.1	Cc1nnc(NC(=O)CSc2ccc3nnc(-c4ccccn4)n3n2)s1	nan
	16025409	28498	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	5	1	6	2.6	NC(=O)CSc1ncc2c(n1)-c1ccccc1N(Cc1cccc(F)c1)S2(=O)=O	nan
	CHEMBL1377886	28498	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	5	1	6	2.6	NC(=O)CSc1ncc2c(n1)-c1ccccc1N(Cc1cccc(F)c1)S2(=O)=O	nan
	2816168	28531	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	3	0	8	1.2	CCOC(=O)c1nnn2c1nc(N1CCN(C)CC1)c1ccccc12	nan
	CHEMBL1378192	28531	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	3	0	8	1.2	CCOC(=O)c1nnn2c1nc(N1CCN(C)CC1)c1ccccc12	nan
	16021577	28558	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	356	4	1	6	2.3	CCCNC(=O)C1CCN(c2ncnc3c2nc2n3CCCCC2)CC1	nan
	CHEMBL1378416	28558	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	356	4	1	6	2.3	CCCNC(=O)C1CCN(c2ncnc3c2nc2n3CCCCC2)CC1	nan
	20886481	28699	0	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	356	5	1	4	3.9	CC(C)Oc1ccc(CNC(=O)c2ccc3c(c2)N(C)CCS3)cc1	nan
	CHEMBL1379683	28699	0	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	356	5	1	4	3.9	CC(C)Oc1ccc(CNC(=O)c2ccc3c(c2)N(C)CCS3)cc1	nan
	2731492	28700	6	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	287	3	2	3	3.7	COc1cccc(NC(S)=Nc2cc(C)cc(C)n2)c1	nan
	CHEMBL1379684	28700	6	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	287	3	2	3	3.7	COc1cccc(NC(S)=Nc2cc(C)cc(C)n2)c1	nan
	614385	28746	73	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	225	1	2	4	2.7	Nc1ccc(-c2nc3cc(N)ccc3o2)cc1	nan
	CHEMBL1380161	28746	73	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	225	1	2	4	2.7	Nc1ccc(-c2nc3cc(N)ccc3o2)cc1	nan
	16187343	28785	0	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	7	0	7	4.1	CC(=O)c1ccc(-c2nnc(CCC(=O)N(C)Cc3cccc4cnccc34)o2)s1	nan
	CHEMBL1380413	28785	0	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	7	0	7	4.1	CC(=O)c1ccc(-c2nnc(CCC(=O)N(C)Cc3cccc4cnccc34)o2)s1	nan
	705209	28787	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	2	2	6	2.7	N#Cc1c(N)n(-c2ccc(C(=O)O)cc2)c2nc3ccccc3nc12	nan
	CHEMBL1380440	28787	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	2	2	6	2.7	N#Cc1c(N)n(-c2ccc(C(=O)O)cc2)c2nc3ccccc3nc12	nan
	3724835	28813	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	454	9	1	7	3.3	CCCOc1cccc(C2C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2CCN2CCOCC2)c1	nan
	5033543	28813	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	454	9	1	7	3.3	CCCOc1cccc(C2C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2CCN2CCOCC2)c1	nan
	CHEMBL1380602	28813	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	454	9	1	7	3.3	CCCOc1cccc(C2C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2CCN2CCOCC2)c1	nan
	1445317	28817	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	203	1	1	2	3.4	CCc1cc2ccc(C)cc2nc1S	nan
	CHEMBL1380640	28817	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	203	1	1	2	3.4	CCc1cc2ccc(C)cc2nc1S	nan
	4430260	29008	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	270	4	0	6	2.2	O=[N+]([O-])c1cccc(OCc2cn3cccnc3n2)c1	nan
	CHEMBL1382302	29008	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	270	4	0	6	2.2	O=[N+]([O-])c1cccc(OCc2cn3cccnc3n2)c1	nan
	3785801	29104	8	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	8	1	6	4.6	CCCCN(CCCC)C(=O)c1sc2nc(N3CCOCC3)c3c(c2c1N)CCCC3	nan
	CHEMBL1383130	29104	8	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	8	1	6	4.6	CCCCN(CCCC)C(=O)c1sc2nc(N3CCOCC3)c3c(c2c1N)CCCC3	nan
	3151314	29111	15	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	5	2	8	1.6	N=c1c(C(=O)NCc2cccnc2)cc2c(=O)n3ccccc3nc2n1CC1CCCO1	nan
	CHEMBL1383245	29111	15	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	5	2	8	1.6	N=c1c(C(=O)NCc2cccnc2)cc2c(=O)n3ccccc3nc2n1CC1CCCO1	nan
	16241852	29169	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	3	1	7	2.6	CCc1ccc(-n2c(=O)c3ccccc3n3c(S)nnc23)cc1.CN(C)C=O	nan
	CHEMBL1383752	29169	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	3	1	7	2.6	CCc1ccc(-n2c(=O)c3ccccc3n3c(S)nnc23)cc1.CN(C)C=O	nan
	9550688	29203	2	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	347	2	0	6	3.2	O=c1sc(N2CCN(c3ccc(F)cc3)CC2)nc2ccsc12	nan
	CHEMBL1384034	29203	2	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	347	2	0	6	3.2	O=c1sc(N2CCN(c3ccc(F)cc3)CC2)nc2ccsc12	nan
	23004552	29227	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	3	0	8	0.5	CCOC(=O)N1CCN(S(=O)(=O)c2c(C)nc3sccn3c2=O)CC1	nan
	CHEMBL1384314	29227	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	3	0	8	0.5	CCOC(=O)N1CCN(S(=O)(=O)c2c(C)nc3sccn3c2=O)CC1	nan
	1830897	29300	11	None	-5	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	361	4	1	5	2.7	O=c1c(Cl)c(NS(=O)(=O)c2ccccc2)cnn1-c1ccccc1	nan
	CHEMBL1384824	29300	11	None	-5	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	361	4	1	5	2.7	O=c1c(Cl)c(NS(=O)(=O)c2ccccc2)cnn1-c1ccccc1	nan
	2488909	29425	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	344	5	1	7	1.6	COC(=O)CNC(=O)CSc1nnc2cc(C)c3ccccc3n12	nan
	CHEMBL1386026	29425	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	344	5	1	7	1.6	COC(=O)CNC(=O)CSc1nnc2cc(C)c3ccccc3n12	nan
	1301168	29587	9	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	4	1	6	4.6	Cc1ccc(S(=O)(=O)c2nc(Nc3ccccc3C#N)sc2Cl)cc1	nan
	CHEMBL1387246	29587	9	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	4	1	6	4.6	Cc1ccc(S(=O)(=O)c2nc(Nc3ccccc3C#N)sc2Cl)cc1	nan
	6264256	29600	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	550	11	1	8	4.1	CCCCOc1ccc(C2C(C(=O)c3ccc4c(c3)CC(C)O4)=C(O)C(=O)N2CCN2CCOCC2)cc1OC	nan
	CHEMBL1387384	29600	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	550	11	1	8	4.1	CCCCOc1ccc(C2C(C(=O)c3ccc4c(c3)CC(C)O4)=C(O)C(=O)N2CCN2CCOCC2)cc1OC	nan
	20904611	29685	0	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	10	1	9	1.8	COCCCn1c(=O)c2sccc2n2c(CCCC(=O)NCC3CCCO3)nnc12	nan
	CHEMBL1388050	29685	0	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	10	1	9	1.8	COCCCn1c(=O)c2sccc2n2c(CCCC(=O)NCC3CCCO3)nnc12	nan
	2819135	29763	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	310	3	0	6	3.3	COc1cccc(-c2c(C#N)c(SC)nc3cc(C)nn23)c1	nan
	CHEMBL1388609	29763	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	310	3	0	6	3.3	COc1cccc(-c2c(C#N)c(SC)nc3cc(C)nn23)c1	nan
	900107	29846	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	233	2	1	6	-1.0	NC(=O)Cn1cnc2nc3n(c2c1=O)CCC3	nan
	CHEMBL1389257	29846	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	233	2	1	6	-1.0	NC(=O)Cn1cnc2nc3n(c2c1=O)CCC3	nan
	1934247	29873	7	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	527	9	2	6	5.3	COCCCNC(=O)c1c(NC(=O)c2ccccc2Cl)n(Cc2ccccc2)c2nc3ccccc3nc12	nan
	CHEMBL1389486	29873	7	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	527	9	2	6	5.3	COCCCNC(=O)c1c(NC(=O)c2ccccc2Cl)n(Cc2ccccc2)c2nc3ccccc3nc12	nan
	2012798	29963	9	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	4	1	7	4.4	Cc1ccc(Cn2c(N)c(S(=O)(=O)c3cccs3)c3nc4ccccc4nc32)cc1	nan
	CHEMBL1390254	29963	9	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	4	1	7	4.4	Cc1ccc(Cn2c(N)c(S(=O)(=O)c3cccs3)c3nc4ccccc4nc32)cc1	nan
	6290194	30073	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	492	8	1	7	3.3	CCOc1cccc(C2C(C(=O)c3ccc4c(c3)CC(C)O4)=C(O)C(=O)N2CCN2CCOCC2)c1	nan
	CHEMBL1391210	30073	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	492	8	1	7	3.3	CCOc1cccc(C2C(C(=O)c3ccc4c(c3)CC(C)O4)=C(O)C(=O)N2CCN2CCOCC2)c1	nan
	16193052	30133	0	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	5	1	4	2.9	O=C(CCCN1C(=O)c2cccnc2C1=O)Nc1ccc(Br)cc1	nan
	CHEMBL1391769	30133	0	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	5	1	4	2.9	O=C(CCCN1C(=O)c2cccnc2C1=O)Nc1ccc(Br)cc1	nan
	886207	30288	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	310	3	1	5	2.3	CCNc1nc(C)c2cc(Br)c(=O)n(CC)c2n1	nan
	CHEMBL1393118	30288	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	310	3	1	5	2.3	CCNc1nc(C)c2cc(Br)c(=O)n(CC)c2n1	nan
	2889346	30303	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	3	1	4	3.5	CC(=O)C1=C(O)C(=O)N(c2ccc(Br)cn2)C1c1ccc(F)cc1	nan
	CHEMBL1393200	30303	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	3	1	4	3.5	CC(=O)C1=C(O)C(=O)N(c2ccc(Br)cn2)C1c1ccc(F)cc1	nan
	6622405	30307	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	6	0	6	2.9	CCn1c(=O)c2cc(C(=O)N(C)CC(OC)OC)sc2c2ccccc21	nan
	CHEMBL1393223	30307	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	6	0	6	2.9	CCn1c(=O)c2cc(C(=O)N(C)CC(OC)OC)sc2c2ccccc21	nan
	5181542	30335	18	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	4	1	6	4.0	Cc1cc(N2C(=O)C(O)=C(C(=O)c3ccco3)C2c2ccc(Cl)cc2)no1	nan
	CHEMBL1393467	30335	18	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	4	1	6	4.0	Cc1cc(N2C(=O)C(O)=C(C(=O)c3ccco3)C2c2ccc(Cl)cc2)no1	nan
	20917879	30342	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	6	0	6	2.4	CN(Cc1ccco1)S(=O)(=O)c1cc(F)ccc1CN1C(=O)c2cccnc2C1=O	nan
	CHEMBL1393505	30342	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	6	0	6	2.4	CN(Cc1ccco1)S(=O)(=O)c1cc(F)ccc1CN1C(=O)c2cccnc2C1=O	nan
	20888749	30375	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	5	0	8	2.7	CCS(=O)(=O)c1nc(S(=O)(=O)c2ccc(C)cc2)c(N2CC(C)OC(C)C2)s1	nan
	CHEMBL1393784	30375	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	5	0	8	2.7	CCS(=O)(=O)c1nc(S(=O)(=O)c2ccc(C)cc2)c(N2CC(C)OC(C)C2)s1	nan
	2135574	30445	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	528	9	1	8	4.4	CCOc1ccc(NC(=O)Cn2cc(C(=O)c3ccc(OCC)cc3)c(=O)c3cc4c(cc32)OCCO4)cc1	nan
	CHEMBL1394559	30445	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	528	9	1	8	4.4	CCOc1ccc(NC(=O)Cn2cc(C(=O)c3ccc(OCC)cc3)c(=O)c3cc4c(cc32)OCCO4)cc1	nan
	16033270	30446	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	4	1	5	5.3	Cc1ccc(NC(=O)c2sc3ncnc(N(C)C4CCCCC4)c3c2C)cc1	nan
	CHEMBL1394566	30446	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	4	1	5	5.3	Cc1ccc(NC(=O)c2sc3ncnc(N(C)C4CCCCC4)c3c2C)cc1	nan
	16025819	30451	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	471	6	1	4	5.4	CCc1ccc(CNC(=O)C2CCN(C(=O)c3ccc(-n4ccc5ccccc54)s3)CC2)cc1	nan
	CHEMBL1394644	30451	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	471	6	1	4	5.4	CCc1ccc(CNC(=O)C2CCN(C(=O)c3ccc(-n4ccc5ccccc54)s3)CC2)cc1	nan
	16018820	30459	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	460	7	1	8	4.7	CCc1nnc(SCC(=O)Nc2cc(Cl)c(OC)cc2OC)c2cc3oc(C)cc3n12	nan
	CHEMBL1394778	30459	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	460	7	1	8	4.7	CCc1nnc(SCC(=O)Nc2cc(Cl)c(OC)cc2OC)c2cc3oc(C)cc3n12	nan
	5144289	30482	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	6	2	4	3.4	O=C(NCCc1ccc(Cl)cc1)c1ccc(Cn2c(=O)[nH]c3ccccc3c2=O)cc1	nan
	CHEMBL1394997	30482	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	6	2	4	3.4	O=C(NCCc1ccc(Cl)cc1)c1ccc(Cn2c(=O)[nH]c3ccccc3c2=O)cc1	nan
	16031990	30495	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	5	1	6	4.7	Cc1nc(C)c(-c2ccc(SCC(=O)Nc3ccc(Br)cc3)nn2)s1	nan
	CHEMBL1395113	30495	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	5	1	6	4.7	Cc1nc(C)c(-c2ccc(SCC(=O)Nc3ccc(Br)cc3)nn2)s1	nan
	6200398	30514	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	315	6	1	7	2.8	CNc1oc(/C=C/c2cc(OC)c(OC)c(OC)c2)nc1C#N	nan
	CHEMBL1395288	30514	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	315	6	1	7	2.8	CNc1oc(/C=C/c2cc(OC)c(OC)c(OC)c2)nc1C#N	nan
	16033416	30523	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	496	8	2	5	5.8	CCOc1ccc(-c2cc(C(=O)NCc3ccc(OC)cc3)c3c(-c4ccc(F)cc4)[nH]nc3n2)cc1	nan
	CHEMBL1395414	30523	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	496	8	2	5	5.8	CCOc1ccc(-c2cc(C(=O)NCc3ccc(OC)cc3)c3c(-c4ccc(F)cc4)[nH]nc3n2)cc1	nan
	5323079	30549	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	6	1	4	5.2	CCOc1ccc(NC(=O)CSc2c3c(nc4ccccc24)CCCC3)cc1	nan
	CHEMBL1395837	30549	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	6	1	4	5.2	CCOc1ccc(NC(=O)CSc2c3c(nc4ccccc24)CCCC3)cc1	nan
	16024553	30552	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	6	1	5	4.2	Cc1ccc(CNC(=O)Cn2cc(C(=O)c3ccc(Cl)cc3)c(=O)c3ccc(C)nc32)cc1	nan
	CHEMBL1395881	30552	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	6	1	5	4.2	Cc1ccc(CNC(=O)Cn2cc(C(=O)c3ccc(Cl)cc3)c(=O)c3ccc(C)nc32)cc1	nan
	5296856	30574	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	1	1	4	2.6	Cc1cccn2c3c(c(=O)nc12)C(c1cccc(F)c1)CC(=O)N3	nan
	CHEMBL1396255	30574	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	1	1	4	2.6	Cc1cccn2c3c(c(=O)nc12)C(c1cccc(F)c1)CC(=O)N3	nan
	1730979	30577	15	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	3	1	3	6.9	O=C(Nc1cc(C(F)(F)F)ccc1Cl)c1cc(-c2cccs2)nc2ccccc12	nan
	CHEMBL1396294	30577	15	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	3	1	3	6.9	O=C(Nc1cc(C(F)(F)F)ccc1Cl)c1cc(-c2cccs2)nc2ccccc12	nan
	16019329	30581	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	442	4	0	9	2.6	CCN1CCN(c2nc3c(S(=O)(=O)c4ccc(C)cc4)nnn3c3ccsc23)CC1	nan
	CHEMBL1396323	30581	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	442	4	0	9	2.6	CCN1CCN(c2nc3c(S(=O)(=O)c4ccc(C)cc4)nnn3c3ccsc23)CC1	nan
	16018658	30592	0	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	6	1	6	4.9	CCc1cccc(C)c1NC(=O)C(CC)Sc1nncn2c1cc1occc12	nan
	CHEMBL1396473	30592	0	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	6	1	6	4.9	CCc1cccc(C)c1NC(=O)C(CC)Sc1nncn2c1cc1occc12	nan
	20885686	30658	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	6	1	6	1.4	Cc1nn(CCCC(=O)NCc2ccc(F)cc2)c(=O)c2nccn12	nan
	CHEMBL1397376	30658	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	6	1	6	1.4	Cc1nn(CCCC(=O)NCc2ccc(F)cc2)c(=O)c2nccn12	nan
	4904384	30676	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	324	5	1	3	3.5	COc1cc2cc(C(=O)N(C)Cc3ccccc3)[nH]c2cc1OC	nan
	CHEMBL1397630	30676	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	324	5	1	3	3.5	COc1cc2cc(C(=O)N(C)Cc3ccccc3)[nH]c2cc1OC	nan
	22517504	30727	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	366	4	1	6	2.3	Cc1ccccc1C(=O)Nc1nnc(S(=O)(=O)N2CCCCC2)s1	nan
	CHEMBL1398370	30727	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	366	4	1	6	2.3	Cc1ccccc1C(=O)Nc1nnc(S(=O)(=O)N2CCCCC2)s1	nan
	15989335	30742	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	576	13	2	7	4.4	CCOc1ccc(NC(=O)Cn2c(=O)n(CCCCC(=O)NCCc3ccc(Cl)cc3)c(=O)c3ccccc32)cc1	nan
	CHEMBL1398481	30742	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	576	13	2	7	4.4	CCOc1ccc(NC(=O)Cn2c(=O)n(CCCCC(=O)NCCc3ccc(Cl)cc3)c(=O)c3ccccc32)cc1	nan
	16022088	30751	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	477	4	0	6	4.8	COc1ccc2c(c1)c1c(c(=O)n(-c3cc(Cl)ccc3C)c(=O)n1Cc1ccc(F)cc1)n2C	nan
	CHEMBL1398563	30751	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	477	4	0	6	4.8	COc1ccc2c(c1)c1c(c(=O)n(-c3cc(Cl)ccc3C)c(=O)n1Cc1ccc(F)cc1)n2C	nan
	3594054	30846	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	497	5	1	5	6.2	N#Cc1c(C(F)(F)F)cc(-c2cccs2)nc1SCC(=O)Nc1cccc(Br)c1	nan
	CHEMBL1399458	30846	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	497	5	1	5	6.2	N#Cc1c(C(F)(F)F)cc(-c2cccs2)nc1SCC(=O)Nc1cccc(Br)c1	nan
	16017733	30859	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	4	1	5	2.8	O=C(Cn1ccn(-c2ccc(F)cc2)c(=O)c1=O)Nc1ccccc1C(F)(F)F	nan
	CHEMBL1399598	30859	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	4	1	5	2.8	O=C(Cn1ccn(-c2ccc(F)cc2)c(=O)c1=O)Nc1ccccc1C(F)(F)F	nan
	16023027	30969	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	6	1	6	2.8	CN(Cc1ccc(F)cc1)S(=O)(=O)c1nnc(NC(=O)c2ccccc2)s1	nan
	CHEMBL1400601	30969	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	6	1	6	2.8	CN(Cc1ccc(F)cc1)S(=O)(=O)c1nnc(NC(=O)c2ccccc2)s1	nan
	2992172	31110	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	348	5	1	7	2.8	CCOC(=O)c1sc(NC(=O)c2ccc(OC(C)=O)cc2)nc1C	nan
	CHEMBL1401867	31110	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	348	5	1	7	2.8	CCOC(=O)c1sc(NC(=O)c2ccc(OC(C)=O)cc2)nc1C	nan
	3124205	31164	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	4	1	4	3.3	COc1ccc(C2C(C(C)=O)=C(O)C(=O)N2c2ccc(F)cc2)cc1	nan
	CHEMBL1402337	31164	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	4	1	4	3.3	COc1ccc(C2C(C(C)=O)=C(O)C(=O)N2c2ccc(F)cc2)cc1	nan
	3833466	31205	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	5	1	8	4.3	COC(=O)c1ccc(C2C(C(=O)c3cc4ccccc4o3)=C(O)C(=O)N2c2cc(C)on2)cc1	nan
	CHEMBL1402650	31205	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	5	1	8	4.3	COC(=O)c1ccc(C2C(C(=O)c3cc4ccccc4o3)=C(O)C(=O)N2c2cc(C)on2)cc1	nan
	1451311	31218	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	290	5	0	5	3.4	CCOC(=O)CSc1nc(C(C)C)nc2ccccc12	nan
	CHEMBL1402735	31218	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	290	5	0	5	3.4	CCOC(=O)CSc1nc(C(C)C)nc2ccccc12	nan
	698553	31244	31	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	319	3	1	4	3.1	O=S(=O)(Nc1nc2ccccc2nc1Cl)c1ccccc1	nan
	CHEMBL1403001	31244	31	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	319	3	1	4	3.1	O=S(=O)(Nc1nc2ccccc2nc1Cl)c1ccccc1	nan
	2679217	31294	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	288	3	1	5	3.5	COc1ccc2oc(C(=O)Nc3nccs3)c(C)c2c1	nan
	CHEMBL1403552	31294	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	288	3	1	5	3.5	COc1ccc2oc(C(=O)Nc3nccs3)c(C)c2c1	nan
	3705005	31382	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	325	0	0	1	4.2	Brc1cc(Br)c2nc3c(cc2c1)CCC3	nan
	CHEMBL1404252	31382	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	325	0	0	1	4.2	Brc1cc(Br)c2nc3c(cc2c1)CCC3	nan
	738260	31443	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	3	1	3	4.1	COc1cc2ccccc2cc1C(=O)Nc1ccc(Cl)cn1	nan
	CHEMBL1404986	31443	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	3	1	3	4.1	COc1cc2ccccc2cc1C(=O)Nc1ccc(Cl)cn1	nan
	16406961	31454	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	440	2	1	6	2.8	Cc1c(CC(=O)N2C[C@@H]3C[C@H](C2)Cn2c3cccc2=O)c(=O)oc2cc(O)c(Cl)cc12	nan
	CHEMBL1405140	31454	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	440	2	1	6	2.8	Cc1c(CC(=O)N2C[C@@H]3C[C@H](C2)Cn2c3cccc2=O)c(=O)oc2cc(O)c(Cl)cc12	nan
	1277429	31515	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	3	0	7	3.5	c1ccc(-c2cc3c(N4CCN(c5ncccn5)CC4)ncnc3s2)cc1	nan
	CHEMBL1405710	31515	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	3	0	7	3.5	c1ccc(-c2cc3c(N4CCN(c5ncccn5)CC4)ncnc3s2)cc1	nan
	135681062	31530	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	330	5	2	6	0.1	O=C(NCCCN1CCCC1=O)c1c(O)nc2ccccn2c1=O	nan
	CHEMBL1405883	31530	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	330	5	2	6	0.1	O=C(NCCCN1CCCC1=O)c1c(O)nc2ccccn2c1=O	nan
	2479912	31541	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	4	1	7	1.2	Cn1c(N)c(C(=O)COc2ccc(Cl)cc2Cl)c(=O)n(C)c1=O	nan
	CHEMBL1405949	31541	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	4	1	7	1.2	Cn1c(N)c(C(=O)COc2ccc(Cl)cc2Cl)c(=O)n(C)c1=O	nan
	665818	31703	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	242	2	1	5	2.2	CNc1ncnc2c3cc(OC)ccc3n(C)c12	nan
	CHEMBL1407387	31703	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	242	2	1	5	2.2	CNc1ncnc2c3cc(OC)ccc3n(C)c12	nan
	2956880	31708	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	4	1	4	2.7	O=C(Nc1ccc(N2CCOCC2)cc1)C1CC(=O)N(c2ccc(F)cc2)C1	nan
	CHEMBL1407427	31708	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	4	1	4	2.7	O=C(Nc1ccc(N2CCOCC2)cc1)C1CC(=O)N(c2ccc(F)cc2)C1	nan
	7080333	31755	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	4	1	4	3.9	Cc1c(-c2cccc(NC(=O)Cc3ccccc3)c2)nc2ncccn12	nan
	CHEMBL1407681	31755	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	4	1	4	3.9	Cc1c(-c2cccc(NC(=O)Cc3ccccc3)c2)nc2ncccn12	nan
	16016996	31860	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	3	0	6	2.4	Cc1ccc(Cl)cc1N1CCN(C(=O)C(C)n2ncn3cccc3c2=O)CC1	nan
	CHEMBL1408470	31860	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	3	0	6	2.4	Cc1ccc(Cl)cc1N1CCN(C(=O)C(C)n2ncn3cccc3c2=O)CC1	nan
	236431	31889	62	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	263	1	1	1	3.6	CC(=O)Nc1ccc(Br)c2ccccc12	nan
	CHEMBL1408731	31889	62	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	263	1	1	1	3.6	CC(=O)Nc1ccc(Br)c2ccccc12	nan
	16019396	31989	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	499	5	1	10	4.2	O=S(=O)(c1ccc(Cl)cc1)c1nnn2c1nc(NCc1ccc3c(c1)OCO3)c1sccc12	nan
	CHEMBL1409519	31989	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	499	5	1	10	4.2	O=S(=O)(c1ccc(Cl)cc1)c1nnn2c1nc(NCc1ccc3c(c1)OCO3)c1sccc12	nan
	6625357	32004	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	7	1	6	1.3	Cc1nn(CCCC(=O)NCCc2ccccc2)c(=O)c2nccn12	nan
	CHEMBL1409636	32004	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	7	1	6	1.3	Cc1nn(CCCC(=O)NCCc2ccccc2)c(=O)c2nccn12	nan
	302041	32357	19	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	4	0	7	1.9	Cn1c2ccccc2c2nnc(SCCN3CCOCC3)nc21	nan
	CHEMBL1412491	32357	19	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	4	0	7	1.9	Cn1c2ccccc2c2nnc(SCCN3CCOCC3)nc21	nan
	2100500	32369	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	3	1	3	4.1	Cc1c(Cl)cccc1NC(=O)Cn1cc(C(F)(F)F)cc(Cl)c1=O	nan
	CHEMBL1412600	32369	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	3	1	3	4.1	Cc1c(Cl)cccc1NC(=O)Cn1cc(C(F)(F)F)cc(Cl)c1=O	nan
	2059848	32491	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	447	7	2	8	3.2	Cc1cc(C)nc(SCC(=O)Nc2ccc(S(=O)(=O)Nc3onc(C)c3C)cc2)n1	nan
	CHEMBL1413582	32491	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	447	7	2	8	3.2	Cc1cc(C)nc(SCC(=O)Nc2ccc(S(=O)(=O)Nc3onc(C)c3C)cc2)n1	nan
	16017166	32550	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	7	1	6	4.0	COc1cccc(CNC(=O)CCCn2nc(C)c3sc4ccccc4c3c2=O)c1	nan
	CHEMBL1414014	32550	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	7	1	6	4.0	COc1cccc(CNC(=O)CCCn2nc(C)c3sc4ccccc4c3c2=O)c1	nan
	2919306	32580	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	7	1	5	4.0	COCCCN1C(=O)C(O)=C(C(=O)c2ccc(C)o2)C1c1cccc(Br)c1	nan
	CHEMBL1414306	32580	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	7	1	5	4.0	COCCCN1C(=O)C(O)=C(C(=O)c2ccc(C)o2)C1c1cccc(Br)c1	nan
	16015068	32587	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	5	1	4	4.8	Cc1c(Cl)cccc1NC(=O)CSc1cc(-c2ccccc2)ncn1	nan
	CHEMBL1414379	32587	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	5	1	4	4.8	Cc1c(Cl)cccc1NC(=O)CSc1cc(-c2ccccc2)ncn1	nan
	16010393	32598	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	2	0	3	5.9	Cc1cccc2c1-c1sc(C(=O)N(C)c3cccc(C(F)(F)F)c3)cc1CO2	nan
	CHEMBL1414451	32598	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	2	0	3	5.9	Cc1cccc2c1-c1sc(C(=O)N(C)c3cccc(C(F)(F)F)c3)cc1CO2	nan
	3245690	32918	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	2	1	7	4.2	Cc1nc2ccc3nc(NC(=O)c4ccc5c(c4)OCCO5)sc3c2s1	nan
	CHEMBL1417231	32918	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	2	1	7	4.2	Cc1nc2ccc3nc(NC(=O)c4ccc5c(c4)OCCO5)sc3c2s1	nan
	24792497	33003	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	5	1	8	2.5	COc1ccc2cc(C#N)c(SCC(=O)Nc3nonc3C)nc2c1	nan
	CHEMBL1417975	33003	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	5	1	8	2.5	COc1ccc2cc(C#N)c(SCC(=O)Nc3nonc3C)nc2c1	nan
	2473907	33162	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	5	1	6	3.1	CCOC(=O)c1cc(-c2ccc(F)cc2)nc2c1c(=O)[nH]c(=O)n2Cc1ccccc1	nan
	CHEMBL1419339	33162	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	5	1	6	3.1	CCOC(=O)c1cc(-c2ccc(F)cc2)nc2c1c(=O)[nH]c(=O)n2Cc1ccccc1	nan
	2980984	33254	9	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	2	1	6	4.3	CC1(C)Cc2c(sc3c2c(N)nc(=S)n3Cc2ccccc2)CO1	nan
	CHEMBL1420144	33254	9	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	2	1	6	4.3	CC1(C)Cc2c(sc3c2c(N)nc(=S)n3Cc2ccccc2)CO1	nan
	16745931	33399	0	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	3	2	6	3.9	Cc1ccc(-c2csc3nc4cc(C(=O)NC5CCC(O)CC5)ccc4c(=O)n23)cc1	nan
	CHEMBL1421354	33399	0	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	3	2	6	3.9	Cc1ccc(-c2csc3nc4cc(C(=O)NC5CCC(O)CC5)ccc4c(=O)n23)cc1	nan
	2138543	33476	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	6	2	7	3.6	Cc1cccc(-c2nnn3c2nc(NCCc2ccc(S(N)(=O)=O)cc2)c2ccccc23)c1	nan
	CHEMBL1422079	33476	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	6	2	7	3.6	Cc1cccc(-c2nnn3c2nc(NCCc2ccc(S(N)(=O)=O)cc2)c2ccccc23)c1	nan
	6045016	33637	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	487	9	1	7	4.3	CCOc1cccc(C2C(C(=O)c3ccc4c(c3)CC(C)O4)=C(O)C(=O)N2CCCn2ccnc2)c1	nan
	CHEMBL1423355	33637	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	487	9	1	7	4.3	CCOc1cccc(C2C(C(=O)c3ccc4c(c3)CC(C)O4)=C(O)C(=O)N2CCCn2ccnc2)c1	nan
	3725185	33674	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	7	1	4	5.2	CN(C)c1ccc(P(=O)(OCc2ccccc2)C(O)c2ccc(Cl)cc2)cc1	nan
	CHEMBL1423606	33674	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	7	1	4	5.2	CN(C)c1ccc(P(=O)(OCc2ccccc2)C(O)c2ccc(Cl)cc2)cc1	nan
	135420429	33678	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	6	2	9	3.4	CCC(Sc1nc(O)c(C#N)c(-c2ccccc2)n1)C(=O)Nc1nnc(C)s1	nan
	CHEMBL1423657	33678	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	6	2	9	3.4	CCC(Sc1nc(O)c(C#N)c(-c2ccccc2)n1)C(=O)Nc1nnc(C)s1	nan
	950417	33824	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	334	2	0	7	1.2	Cc1cccn2c(=O)c(C=C(C#N)C#N)c(N3CCN(C)CC3)nc12	nan
	CHEMBL1424893	33824	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	334	2	0	7	1.2	Cc1cccn2c(=O)c(C=C(C#N)C#N)c(N3CCN(C)CC3)nc12	nan
	4008202	34144	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	6	1	9	1.9	CCOC(=O)c1sc2nc(C)nc(SCC(=O)NC3CCS(=O)(=O)C3)c2c1C	nan
	CHEMBL1427679	34144	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	6	1	9	1.9	CCOC(=O)c1sc2nc(C)nc(SCC(=O)NC3CCS(=O)(=O)C3)c2c1C	nan
	2810151	34172	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	334	2	1	4	3.7	O=C(Nc1nc2ccccc2c(=O)s1)c1ccc(F)cc1Cl	nan
	CHEMBL1427961	34172	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	334	2	1	4	3.7	O=C(Nc1nc2ccccc2c(=O)s1)c1ccc(F)cc1Cl	nan
	4603734	34367	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	6	1	7	2.3	O=C(COc1ncnc2ccccc12)Nc1cc(S(=O)(=O)N2CCOCC2)ccc1Cl	nan
	CHEMBL1429555	34367	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	6	1	7	2.3	O=C(COc1ncnc2ccccc12)Nc1cc(S(=O)(=O)N2CCOCC2)ccc1Cl	nan
	2369101	34374	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	4	0	5	3.2	CCN1C(=O)C(=C2C=C(C)N(Cc3ccco3)C(C)=C2)C(=O)N(CC)C1=S	nan
	CHEMBL1429586	34374	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	4	0	5	3.2	CCN1C(=O)C(=C2C=C(C)N(Cc3ccco3)C(C)=C2)C(=O)N(CC)C1=S	nan
	6110891	34384	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	498	7	1	7	3.4	O=C(C1=C(O)C(=O)N(CCCN2CCOCC2)C1c1ccc(Cl)cc1)c1ccc2c(c1)OCCO2	nan
	CHEMBL1429670	34384	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	498	7	1	7	3.4	O=C(C1=C(O)C(=O)N(CCCN2CCOCC2)C1c1ccc(Cl)cc1)c1ccc2c(c1)OCCO2	nan
	3186593	34606	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	3	0	8	0.3	CC1CCN(C(=O)CSc2nc3c(c(=O)n(C)c(=O)n3C)n2C)CC1	nan
	CHEMBL1431426	34606	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	3	0	8	0.3	CC1CCN(C(=O)CSc2nc3c(c(=O)n(C)c(=O)n3C)n2C)CC1	nan
	4836291	34706	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	454	4	0	3	4.9	CCC1CCCCN1C(=O)COc1c(Br)cc(Br)c2cccnc12	nan
	CHEMBL1432322	34706	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	454	4	0	3	4.9	CCC1CCCCN1C(=O)COc1c(Br)cc(Br)c2cccnc12	nan
	3236746	34723	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	344	7	2	4	3.9	CCOc1ccc(OCC)c(NC(=O)c2[nH]c(C)c(C(C)=O)c2C)c1	nan
	CHEMBL1432463	34723	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	344	7	2	4	3.9	CCOc1ccc(OCC)c(NC(=O)c2[nH]c(C)c(C(C)=O)c2C)c1	nan
	5186080	34807	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	3	0	5	3.1	CC1(C(=O)OCc2cc(=O)n3cc(Br)ccc3n2)CC1(Cl)Cl	nan
	CHEMBL1433143	34807	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	3	0	5	3.1	CC1(C(=O)OCc2cc(=O)n3cc(Br)ccc3n2)CC1(Cl)Cl	nan
	16025762	34845	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	4	0	5	4.1	CCOC(=O)C1CCCN(C(=O)c2ccc(-n3ccc4ccccc43)s2)C1	nan
	CHEMBL1433427	34845	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	4	0	5	4.1	CCOC(=O)C1CCCN(C(=O)c2ccc(-n3ccc4ccccc43)s2)C1	nan
	16031695	34915	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	306	4	1	5	2.7	CC(=O)c1ccc(NC(=O)c2ccc(-n3cnnc3)cc2)cc1	nan
	CHEMBL1434575	34915	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	306	4	1	5	2.7	CC(=O)c1ccc(NC(=O)c2ccc(-n3cnnc3)cc2)cc1	nan
	1003863	34932	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	4	2	5	5.6	COc1cccc(-c2ccc3c(N)c(C(=O)Nc4ccc(Cl)cc4F)sc3n2)c1	nan
	CHEMBL1434727	34932	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	4	2	5	5.6	COc1cccc(-c2ccc3c(N)c(C(=O)Nc4ccc(Cl)cc4F)sc3n2)c1	nan
	16404473	34963	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	545	8	1	8	3.7	COc1cc(OC)c(OC)cc1/C=C1\Oc2cc(OCC(=O)N3Cc4ccccc4C[C@H]3C(=O)O)ccc2C1=O	nan
	CHEMBL1435093	34963	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	545	8	1	8	3.7	COc1cc(OC)c(OC)cc1/C=C1\Oc2cc(OCC(=O)N3Cc4ccccc4C[C@H]3C(=O)O)ccc2C1=O	nan
	24891925	34982	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	6	1	7	2.3	O=C(CSc1nnc2ccc(-c3ccc(F)cc3)nn12)NCC1CCCO1	nan
	CHEMBL1435281	34982	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	6	1	7	2.3	O=C(CSc1nnc2ccc(-c3ccc(F)cc3)nn12)NCC1CCCO1	nan
	16416480	34986	17	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	4	1	6	3.0	COc1ccc(-c2cc3ccc(O)c(CN4CCOCC4)c3oc2=O)cc1	nan
	5457481	34986	17	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	4	1	6	3.0	COc1ccc(-c2cc3ccc(O)c(CN4CCOCC4)c3oc2=O)cc1	nan
	CHEMBL1435346	34986	17	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	4	1	6	3.0	COc1ccc(-c2cc3ccc(O)c(CN4CCOCC4)c3oc2=O)cc1	nan
	16034509	34990	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	7	1	6	4.6	CN(C)c1ccc(NC(=O)Cn2c(SCc3ccc(F)cc3)nc3cccnc32)cc1	nan
	CHEMBL1435377	34990	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	7	1	6	4.6	CN(C)c1ccc(NC(=O)Cn2c(SCc3ccc(F)cc3)nc3cccnc32)cc1	nan
	15989215	35003	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	461	7	1	8	2.8	COc1ccc(NC(=O)Cn2c(=O)n(-c3ccc(OC)c(OC)c3)c(=O)c3ccccc32)cc1	nan
	CHEMBL1435575	35003	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	461	7	1	8	2.8	COc1ccc(NC(=O)Cn2c(=O)n(-c3ccc(OC)c(OC)c3)c(=O)c3ccccc32)cc1	nan
	4281326	35061	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	6	1	4	5.3	Cc1cccc(C)c1OCC(=O)Nc1c(C(=O)c2ccccc2)oc2ccccc12	nan
	CHEMBL1436278	35061	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	6	1	4	5.3	Cc1cccc(C)c1OCC(=O)Nc1c(C(=O)c2ccccc2)oc2ccccc12	nan
	16009492	35152	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	5	1	6	4.0	Cc1csc2nc(COc3cccc(NC(=O)c4ccccc4F)c3)cc(=O)n12	nan
	CHEMBL1437588	35152	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	5	1	6	4.0	Cc1csc2nc(COc3cccc(NC(=O)c4ccccc4F)c3)cc(=O)n12	nan
	16015683	35154	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	479	5	1	5	5.9	O=C(Nc1ccc2nc(SCC(=O)N3CCc4ccccc43)sc2c1)c1ccc(Cl)cc1	nan
	CHEMBL1437631	35154	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	479	5	1	5	5.9	O=C(Nc1ccc2nc(SCC(=O)N3CCc4ccccc43)sc2c1)c1ccc(Cl)cc1	nan
	16025792	35166	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	6	1	5	4.9	COc1ccc(CNC(=O)C2CCN(C(=O)c3ccc(-n4ccc5ccccc54)s3)CC2)cc1	nan
	CHEMBL1437725	35166	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	6	1	5	4.9	COc1ccc(CNC(=O)C2CCN(C(=O)c3ccc(-n4ccc5ccccc54)s3)CC2)cc1	nan
	4523316	35270	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	2	0	5	2.6	CN(C(=O)c1cc2c(=O)n3ccccc3nc2n1C)C1CCCCC1	nan
	CHEMBL1438580	35270	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	2	0	5	2.6	CN(C(=O)c1cc2c(=O)n3ccccc3nc2n1C)C1CCCCC1	nan
	16012068	35329	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	4	1	7	2.6	Cc1cc(=O)n2nc(N3CCC(C(=O)NCc4ccc(Cl)cc4)CC3)sc2n1	nan
	CHEMBL1439177	35329	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	4	1	7	2.6	Cc1cc(=O)n2nc(N3CCC(C(=O)NCc4ccc(Cl)cc4)CC3)sc2n1	nan
	3846910	35350	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	3	2	6	4.2	Cc1ccccc1NC(=O)c1sc2nc(N3CCOCC3)c3c(c2c1N)CCCC3	nan
	CHEMBL1439341	35350	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	3	2	6	4.2	Cc1ccccc1NC(=O)c1sc2nc(N3CCOCC3)c3c(c2c1N)CCCC3	nan
	4246549	35513	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	440	4	1	4	5.2	Cc1ccc(NC(=O)c2oc3ccc(S(=O)(=O)N4CCCCCC4)cc3c2C)c(C)c1	nan
	CHEMBL1440777	35513	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	440	4	1	4	5.2	Cc1ccc(NC(=O)c2oc3ccc(S(=O)(=O)N4CCCCCC4)cc3c2C)c(C)c1	nan
	4230097	35532	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	490	9	1	9	4.1	O=C(O)CCCCCn1c(SCc2cc(=O)n3cc(Cl)ccc3n2)nc2ccsc2c1=O	nan
	CHEMBL1440951	35532	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	490	9	1	9	4.1	O=C(O)CCCCCn1c(SCc2cc(=O)n3cc(Cl)ccc3n2)nc2ccsc2c1=O	nan
	3272255	35665	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	7	2	7	0.7	Cc1sc2ncn(CC(=O)NCCCC(=O)N3CCC(C(N)=O)CC3)c(=O)c2c1C	nan
	CHEMBL1442168	35665	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	7	2	7	0.7	Cc1sc2ncn(CC(=O)NCCCC(=O)N3CCC(C(N)=O)CC3)c(=O)c2c1C	nan
	1077468	35694	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	464	6	2	8	1.8	Cc1cccn2c(=O)c3cc(C(=O)NC4CCCC4)c(=N)n(CCCN4CCOCC4)c3nc12	nan
	CHEMBL1442429	35694	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	464	6	2	8	1.8	Cc1cccn2c(=O)c3cc(C(=O)NC4CCCC4)c(=N)n(CCCN4CCOCC4)c3nc12	nan
	20876076	35708	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	460	6	1	8	0.8	COc1ccc(C)cc1NC(=O)CN(C)S(=O)(=O)c1ccc2c(c1)n(C)c(=O)c(=O)n2C	nan
	CHEMBL1442544	35708	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	460	6	1	8	0.8	COc1ccc(C)cc1NC(=O)CN(C)S(=O)(=O)c1ccc2c(c1)n(C)c(=O)c(=O)n2C	nan
	7217841	35753	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	319	3	1	6	2.9	Cc1nnc2ccc(-c3ccc(NC(=O)c4ccco4)cc3)nn12	nan
	CHEMBL1442956	35753	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	319	3	1	6	2.9	Cc1nnc2ccc(-c3ccc(NC(=O)c4ccco4)cc3)nn12	nan
	2975734	35762	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	3	0	7	2.3	CCOC(=O)C1CCCN(C(=O)c2cc3c(=O)n4ccccc4nc3s2)C1	nan
	CHEMBL1443010	35762	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	3	0	7	2.3	CCOC(=O)C1CCCN(C(=O)c2cc3c(=O)n4ccccc4nc3s2)C1	nan
	4611621	35918	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	7	1	6	4.8	COc1ccc(C2=NN(c3ccc(C(=O)O)cc3)C(c3ccc(OC)c(OC)c3)C2)cc1	nan
	CHEMBL1444507	35918	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	7	1	6	4.8	COc1ccc(C2=NN(c3ccc(C(=O)O)cc3)C(c3ccc(OC)c(OC)c3)C2)cc1	nan
	817359	35935	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	346	4	2	3	3.6	CC(=O)c1ccc(NC(=S)NC(=O)Cc2ccc(Cl)cc2)cc1	nan
	CHEMBL1444699	35935	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	346	4	2	3	3.6	CC(=O)c1ccc(NC(=S)NC(=O)Cc2ccc(Cl)cc2)cc1	nan
	4051948	35938	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	5	1	5	4.6	Cc1ccc(C(=O)C2=C(O)C(=O)N(Cc3ccco3)C2c2cccc(Cl)c2)o1	nan
	CHEMBL1444743	35938	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	5	1	5	4.6	Cc1ccc(C(=O)C2=C(O)C(=O)N(Cc3ccco3)C2c2cccc(Cl)c2)o1	nan
	3186591	35975	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	3	0	8	0.5	CC1CCCCN1C(=O)CSc1nc2c(c(=O)n(C)c(=O)n2C)n1C	nan
	CHEMBL1445043	35975	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	3	0	8	0.5	CC1CCCCN1C(=O)CSc1nc2c(c(=O)n(C)c(=O)n2C)n1C	nan
	16187836	36069	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	471	7	1	10	1.1	COc1ccccc1-c1nc(SCC(=O)NCC2CCCO2)c2c(=O)n(C)c(=O)n(C)c2n1	nan
	CHEMBL1445914	36069	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	471	7	1	10	1.1	COc1ccccc1-c1nc(SCC(=O)NCC2CCCO2)c2c(=O)n(C)c(=O)n(C)c2n1	nan
	16017757	36184	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	5	1	5	2.9	CCc1ccc(NC(=O)Cn2ccn(-c3cccc(Cl)c3)c(=O)c2=O)cc1	nan
	CHEMBL1446963	36184	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	5	1	5	2.9	CCc1ccc(NC(=O)Cn2ccn(-c3cccc(Cl)c3)c(=O)c2=O)cc1	nan
	2769301	36341	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	4	1	4	3.7	COc1ccc(-c2cc(C(=O)Nc3ccccc3F)on2)cc1	nan
	CHEMBL1448341	36341	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	4	1	4	3.7	COc1ccc(-c2cc(C(=O)Nc3ccccc3F)on2)cc1	nan
	3658309	36495	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	548	11	1	8	4.8	COc1cc(C2C(C(=O)c3cc4ccccc4o3)=C(O)C(=O)N2CCN2CCOCC2)ccc1OCCC(C)C	nan
	CHEMBL1449439	36495	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	548	11	1	8	4.8	COc1cc(C2C(C(=O)c3cc4ccccc4o3)=C(O)C(=O)N2CCN2CCOCC2)ccc1OCCC(C)C	nan
	3652194	36559	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	1	0	2	5.5	Brc1cc(Br)c2nc(-c3cccs3)ccc2c1	nan
	CHEMBL1449966	36559	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	1	0	2	5.5	Brc1cc(Br)c2nc(-c3cccs3)ccc2c1	nan
	3244704	36667	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	6	2	7	3.3	COc1ccc(C2C=C(c3cccs3)Nc3nc(CCCO)nn32)cc1	nan
	CHEMBL1450888	36667	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	6	2	7	3.3	COc1ccc(C2C=C(c3cccs3)Nc3nc(CCCO)nn32)cc1	nan
	1774540	36844	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	2	0	4	5.0	O=c1oc2c3c(ccc2c2ccccc12)OCN(Cc1cccc(Cl)c1)C3	nan
	CHEMBL1452222	36844	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	2	0	4	5.0	O=c1oc2c3c(ccc2c2ccccc12)OCN(Cc1cccc(Cl)c1)C3	nan
	649434	36932	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	410	6	1	7	4.2	CCOc1cccc(C2C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2c2nccs2)c1	nan
	CHEMBL1452945	36932	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	410	6	1	7	4.2	CCOc1cccc(C2C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2c2nccs2)c1	nan
	16187616	37081	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	426	7	1	10	2.8	COc1ccc(-c2nnc3ccc(SCC(=O)Nc4cc(C)on4)nn23)cc1OC	nan
	CHEMBL1454124	37081	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	426	7	1	10	2.8	COc1ccc(-c2nnc3ccc(SCC(=O)Nc4cc(C)on4)nn23)cc1OC	nan
	17580690	37118	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	1	1	2	3.5	Cc1c(C(=O)N2CC(C)OC(C)C2)[nH]c2ccc(Br)cc12	nan
	CHEMBL1454451	37118	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	1	1	2	3.5	Cc1c(C(=O)N2CC(C)OC(C)C2)[nH]c2ccc(Br)cc12	nan
	18204435	37212	6	None	-48	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	423	4	2	6	3.5	CNC(=O)c1ccc(NC(=O)C2CCN(c3ncnc4sc(C)c(C)c34)CC2)cc1	nan
	CHEMBL1455259	37212	6	None	-48	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	423	4	2	6	3.5	CNC(=O)c1ccc(NC(=O)C2CCN(c3ncnc4sc(C)c(C)c34)CC2)cc1	nan
	1265180	37319	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	6	1	8	1.0	CCCn1c(SCC(=O)NC2CCCC2)nc2c1c(=O)n(C)c(=O)n2C	nan
	CHEMBL1456231	37319	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	6	1	8	1.0	CCCn1c(SCC(=O)NC2CCCC2)nc2c1c(=O)n(C)c(=O)n2C	nan
	24793479	37437	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	410	6	2	6	3.3	COc1ccc(C(=O)NNC(=O)CSc2nc(C(C)C)nc3ccccc23)cc1	nan
	CHEMBL1457367	37437	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	410	6	2	6	3.3	COc1ccc(C(=O)NNC(=O)CSc2nc(C(C)C)nc3ccccc23)cc1	nan
	24819691	37529	0	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	5	3	4	3.2	COc1ccc2cc(OCC(=O)NNC(=O)Nc3ccc(F)cc3)ccc2c1	nan
	CHEMBL1458070	37529	0	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	5	3	4	3.2	COc1ccc2cc(OCC(=O)NNC(=O)Nc3ccc(F)cc3)ccc2c1	nan
	675984	37634	15	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	347	3	0	2	4.0	O=C(COc1ccc2ccccc2c1Br)N1CCCCC1	nan
	CHEMBL1458979	37634	15	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	347	3	0	2	4.0	O=C(COc1ccc2ccccc2c1Br)N1CCCCC1	nan
	866601	37766	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	2	1	5	3.4	O=C(NC1CCCCCC1)c1cc2c(=O)n3ccccc3nc2s1	nan
	CHEMBL1460115	37766	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	2	1	5	3.4	O=C(NC1CCCCCC1)c1cc2c(=O)n3ccccc3nc2s1	nan
	20912606	37954	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	475	7	0	7	3.4	CN(C)CCN(Cc1ccccc1)C(=O)C1CCN(c2ncnc3c2nc2n3CCCCC2)CC1	nan
	CHEMBL1461808	37954	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	475	7	0	7	3.4	CN(C)CCN(Cc1ccccc1)C(=O)C1CCN(c2ncnc3c2nc2n3CCCCC2)CC1	nan
	2745719	38177	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	280	3	1	5	2.8	CC(=O)Nc1nccc(-c2cc(-c3ccccc3)no2)n1	nan
	CHEMBL1463690	38177	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	280	3	1	5	2.8	CC(=O)Nc1nccc(-c2cc(-c3ccccc3)no2)n1	nan
	741378	38333	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	2	0	6	3.4	COC(=O)Sc1nnc(-c2ccc(Br)cc2)o1	nan
	CHEMBL1464821	38333	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	2	0	6	3.4	COC(=O)Sc1nnc(-c2ccc(Br)cc2)o1	nan
	203396	38364	77	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	1	0	3	2.8	O=c1c(Br)c(Br)cnn1-c1ccccc1	nan
	CHEMBL1465040	38364	77	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	1	0	3	2.8	O=c1c(Br)c(Br)cnn1-c1ccccc1	nan
	3518230	38384	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	466	6	1	6	4.0	O=C(C1=C(O)C(=O)N(CCN2CCOCC2)C1c1ccc(Cl)cc1)c1cc2ccccc2o1	nan
	4024784	38384	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	466	6	1	6	4.0	O=C(C1=C(O)C(=O)N(CCN2CCOCC2)C1c1ccc(Cl)cc1)c1cc2ccccc2o1	nan
	CHEMBL1465171	38384	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	466	6	1	6	4.0	O=C(C1=C(O)C(=O)N(CCN2CCOCC2)C1c1ccc(Cl)cc1)c1cc2ccccc2o1	nan
	24791767	38436	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	7	0	6	3.5	CCN(Cc1cnn(C)c1)C(=O)c1cc(COc2ccc3c(c2)CCCC3)on1	nan
	CHEMBL1465549	38436	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	7	0	6	3.5	CCN(Cc1cnn(C)c1)C(=O)c1cc(COc2ccc3c(c2)CCCC3)on1	nan
	16241464	38649	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	6	0	8	2.7	CN(C)C=O.O=[N+]([O-])c1cccc(COc2ncnc3cc([N+](=O)[O-])ccc23)c1	nan
	CHEMBL1467247	38649	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	6	0	8	2.7	CN(C)C=O.O=[N+]([O-])c1cccc(COc2ncnc3cc([N+](=O)[O-])ccc23)c1	nan
	1244301	38748	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	283	3	1	2	3.8	Cc1c(C(=O)NCc2ccccc2F)oc2ccccc12	nan
	CHEMBL1468217	38748	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	283	3	1	2	3.8	Cc1c(C(=O)NCc2ccccc2F)oc2ccccc12	nan
	18561646	38796	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	7	1	9	0.6	CC(C)Cc1nc(SCC(=O)NCC2CCCO2)c2c(=O)n(C)c(=O)n(C)c2n1	nan
	CHEMBL1468525	38796	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	7	1	9	0.6	CC(C)Cc1nc(SCC(=O)NCC2CCCO2)c2c(=O)n(C)c(=O)n(C)c2n1	nan
	4257704	38854	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	496	8	1	7	3.4	CCN(CC)S(=O)(=O)c1ccc(N2CCOCC2)c(NC(=O)c2cc([N+](=O)[O-])ccc2Cl)c1	nan
	CHEMBL1468952	38854	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	496	8	1	7	3.4	CCN(CC)S(=O)(=O)c1ccc(N2CCOCC2)c(NC(=O)c2cc([N+](=O)[O-])ccc2Cl)c1	nan
	20957237	38989	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	7	1	9	1.7	COc1ccc(CNC(=O)CCc2nnc3ccc(N4CCC5(CC4)OCCO5)nn23)cc1	nan
	CHEMBL1470126	38989	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	7	1	9	1.7	COc1ccc(CNC(=O)CCc2nnc3ccc(N4CCC5(CC4)OCCO5)nn23)cc1	nan
	1261892	38992	9	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	510	6	2	5	3.7	NS(=O)(=O)c1ccc(CCNC(=O)c2cc(-c3ccccn3)nc3ccc(Br)cc23)cc1	nan
	CHEMBL1470208	38992	9	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	510	6	2	5	3.7	NS(=O)(=O)c1ccc(CCNC(=O)c2cc(-c3ccccn3)nc3ccc(Br)cc23)cc1	nan
	2725142	39104	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	332	5	1	7	2.4	COc1nc(N)c(C#N)c(-c2ccc(N(C)CCC#N)cc2)c1C#N	nan
	CHEMBL1471123	39104	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	332	5	1	7	2.4	COc1nc(N)c(C#N)c(-c2ccc(N(C)CCC#N)cc2)c1C#N	nan
	15988569	39289	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	5	0	6	5.5	Cc1ccc(-c2nc(-c3cc4cccc(OCc5ccc(F)cc5)c4oc3=O)no2)cc1	nan
	CHEMBL1472849	39289	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	5	0	6	5.5	Cc1ccc(-c2nc(-c3cc4cccc(OCc5ccc(F)cc5)c4oc3=O)no2)cc1	nan
	1166244	39300	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	475	6	1	6	5.6	Cc1cccc(C)c1NC(=O)CCSc1nc(-c2ccc3c(c2)OCO3)cc(C(F)(F)F)n1	nan
	CHEMBL1472996	39300	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	475	6	1	6	5.6	Cc1cccc(C)c1NC(=O)CCSc1nc(-c2ccc3c(c2)OCO3)cc(C(F)(F)F)n1	nan
	16025417	39317	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	546	8	1	7	5.3	CCOc1ccc(NC(=O)CSc2ncc3c(n2)-c2ccccc2N(Cc2ccccc2C)S3(=O)=O)cc1	nan
	CHEMBL1473284	39317	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	546	8	1	7	5.3	CCOc1ccc(NC(=O)CSc2ncc3c(n2)-c2ccccc2N(Cc2ccccc2C)S3(=O)=O)cc1	nan
	16009695	39383	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	467	4	1	6	4.5	O=C(Cn1c(=O)n(-c2ccccc2Cl)c(=O)c2sc3ccccc3c21)NC1CCCCC1	nan
	CHEMBL1474245	39383	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	467	4	1	6	4.5	O=C(Cn1c(=O)n(-c2ccccc2Cl)c(=O)c2sc3ccccc3c21)NC1CCCCC1	nan
	2158398	39389	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	3	1	6	3.8	COc1ccc(Cl)cc1NC(=O)c1cc2c(=O)n3ccccc3nc2s1	nan
	CHEMBL1474329	39389	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	3	1	6	3.8	COc1ccc(Cl)cc1NC(=O)c1cc2c(=O)n3ccccc3nc2s1	nan
	16009720	39394	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	5	1	6	4.9	COc1ccc(CNc2nc3c(-c4ccc(C)cc4)nnn3c3ccccc23)cc1	nan
	CHEMBL1474419	39394	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	5	1	6	4.9	COc1ccc(CNc2nc3c(-c4ccc(C)cc4)nnn3c3ccccc23)cc1	nan
	16016110	39432	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	6	1	7	4.8	Cc1ccc(CNc2ccc(-c3nc(-c4ccco4)no3)cc2[N+](=O)[O-])cc1	nan
	CHEMBL1474896	39432	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	6	1	7	4.8	Cc1ccc(CNc2ccc(-c3nc(-c4ccco4)no3)cc2[N+](=O)[O-])cc1	nan
	16033296	39434	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	5	1	5	5.0	Cc1ccccc1CNC(=O)c1sc2ncnc(N(C)C3CCCCC3)c2c1C	nan
	CHEMBL1474937	39434	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	5	1	5	5.0	Cc1ccccc1CNC(=O)c1sc2ncnc(N(C)C3CCCCC3)c2c1C	nan
	3155029	39485	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	7	1	5	2.1	COc1ccc(CCNC(=O)CN2C(=O)COc3ccc(C)cc32)cc1OC	nan
	CHEMBL1475587	39485	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	7	1	5	2.1	COc1ccc(CCNC(=O)CN2C(=O)COc3ccc(C)cc32)cc1OC	nan
	16020275	39488	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	576	9	2	7	4.6	CCc1ccc(NC(=O)Cn2c(=O)n(-c3ccc(OC)cc3)c(=O)c3ccc(C(=O)NCc4ccc(C)cc4)cc32)cc1	nan
	CHEMBL1475630	39488	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	576	9	2	7	4.6	CCc1ccc(NC(=O)Cn2c(=O)n(-c3ccc(OC)cc3)c(=O)c3ccc(C(=O)NCc4ccc(C)cc4)cc32)cc1	nan
	16415433	39490	17	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	5	1	7	3.0	COc1ccc(-c2cc3ccc(O)c(CN4CCOCC4)c3oc2=O)cc1OC	nan
	5513689	39490	17	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	5	1	7	3.0	COc1ccc(-c2cc3ccc(O)c(CN4CCOCC4)c3oc2=O)cc1OC	nan
	CHEMBL1475648	39490	17	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	5	1	7	3.0	COc1ccc(-c2cc3ccc(O)c(CN4CCOCC4)c3oc2=O)cc1OC	nan
	3646895	39508	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	471	9	1	7	4.9	CCOCCCn1c(SCC(=O)Nc2ccc(F)cc2)nc2c(sc3ccccc32)c1=O	nan
	CHEMBL1475830	39508	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	471	9	1	7	4.9	CCOCCCn1c(SCC(=O)Nc2ccc(F)cc2)nc2c(sc3ccccc32)c1=O	nan
	16020214	39512	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	644	7	2	8	4.4	O=C(Cn1c(=O)n(-c2ccccc2)c(=O)c2ccc(C(=O)NCc3ccc4c(c3)OCO4)cc21)Nc1ccc(Br)cc1F	nan
	CHEMBL1475923	39512	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	644	7	2	8	4.4	O=C(Cn1c(=O)n(-c2ccccc2)c(=O)c2ccc(C(=O)NCc3ccc4c(c3)OCO4)cc21)Nc1ccc(Br)cc1F	nan
	15990518	39525	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	5	1	6	4.9	CCOC(=O)c1cccc(NC(=O)c2cc3cc4cc(OC)ccc4nc3s2)c1	nan
	CHEMBL1476197	39525	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	5	1	6	4.9	CCOC(=O)c1cccc(NC(=O)c2cc3cc4cc(OC)ccc4nc3s2)c1	nan
	16018050	39564	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	9	1	6	3.6	COc1ccc(CCNC(=O)CCCn2c(=O)c3cccn3c3ccc(F)cc32)cc1OC	nan
	CHEMBL1476725	39564	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	9	1	6	3.6	COc1ccc(CCNC(=O)CCCn2c(=O)c3cccn3c3ccc(F)cc32)cc1OC	nan
	18572231	39587	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	8	1	8	2.6	CCOc1ccc(-c2ccc3nnc(SCC(=O)NCC4CCCO4)n3n2)cc1	nan
	CHEMBL1477019	39587	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	8	1	8	2.6	CCOc1ccc(-c2ccc3nnc(SCC(=O)NCC4CCCO4)n3n2)cc1	nan
	5294687	39619	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	8	2	4	5.3	CCCOc1ccc(C(CC(=O)O)NC(=O)c2sc3ccccc3c2Cl)cc1	nan
	CHEMBL1477360	39619	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	8	2	4	5.3	CCCOc1ccc(C(CC(=O)O)NC(=O)c2sc3ccccc3c2Cl)cc1	nan
	3096467	39691	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	495	8	0	5	4.2	CCn1c(/C=C/N(C(C)=O)c2ccccc2)[n+](CCCS(=O)(=O)[O-])c2cc(Cl)c(Cl)cc21	nan
	5751261	39691	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	495	8	0	5	4.2	CCn1c(/C=C/N(C(C)=O)c2ccccc2)[n+](CCCS(=O)(=O)[O-])c2cc(Cl)c(Cl)cc21	nan
	CHEMBL1477993	39691	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	495	8	0	5	4.2	CCn1c(/C=C/N(C(C)=O)c2ccccc2)[n+](CCCS(=O)(=O)[O-])c2cc(Cl)c(Cl)cc21	nan
	2027019	39758	8	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	5	1	7	5.3	CSc1nc(SCC(=O)O)c2sc3nc(-c4ccccc4)c4c(c3c2n1)CCC4	nan
	CHEMBL1478587	39758	8	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	5	1	7	5.3	CSc1nc(SCC(=O)O)c2sc3nc(-c4ccccc4)c4c(c3c2n1)CCC4	nan
	2487220	39873	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	5	1	6	3.8	CCn1cc(C(=O)OCC(=O)Nc2cccc(Cl)c2Cl)c(=O)c2ccc(C)nc21	nan
	CHEMBL1479594	39873	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	5	1	6	3.8	CCn1cc(C(=O)OCC(=O)Nc2cccc(Cl)c2Cl)c(=O)c2ccc(C)nc21	nan
	16024523	39934	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	6	1	5	3.6	Cc1ccc(C(=O)c2cn(CC(=O)NCc3ccccc3)c3nc(C)ccc3c2=O)cc1	nan
	CHEMBL1480079	39934	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	6	1	5	3.6	Cc1ccc(C(=O)c2cn(CC(=O)NCc3ccccc3)c3nc(C)ccc3c2=O)cc1	nan
	16019201	39948	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	483	6	1	7	4.2	COc1ccc(Cn2c(=O)c3oc4ccccc4c3n(CC(=O)Nc3cc(C)cc(C)c3)c2=O)cc1	nan
	CHEMBL1480191	39948	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	483	6	1	7	4.2	COc1ccc(Cn2c(=O)c3oc4ccccc4c3n(CC(=O)Nc3cc(C)cc(C)c3)c2=O)cc1	nan
	5925055	40142	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	6	1	7	3.0	O=C(C1=C(O)C(=O)N(CCN2CCOCC2)C1c1cccc(Cl)c1)c1ccc2c(c1)OCCO2	nan
	CHEMBL1481881	40142	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	6	1	7	3.0	O=C(C1=C(O)C(=O)N(CCN2CCOCC2)C1c1cccc(Cl)c1)c1ccc2c(c1)OCCO2	nan
	7258994	40150	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	4	1	8	1.9	Cc1ccc2nc(SCC(=O)Nc3ccc4c(c3)OCCO4)nc(=O)n2c1	nan
	CHEMBL1481935	40150	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	4	1	8	1.9	Cc1ccc2nc(SCC(=O)Nc3ccc4c(c3)OCCO4)nc(=O)n2c1	nan
	1470918	40232	17	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	3	1	4	3.7	Cc1ccccc1C(=O)NN(C)c1nc2ccccc2nc1C(F)(F)F	nan
	CHEMBL1482653	40232	17	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	3	1	4	3.7	Cc1ccccc1C(=O)NN(C)c1nc2ccccc2nc1C(F)(F)F	nan
	3122172	40276	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	3	1	3	4.6	CC(=O)C1=C(O)C(=O)N(c2cccc(Br)c2)C1c1ccccc1Cl	nan
	CHEMBL1483069	40276	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	3	1	3	4.6	CC(=O)C1=C(O)C(=O)N(c2cccc(Br)c2)C1c1ccccc1Cl	nan
	1093408	40326	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	4	2	5	4.3	COCc1cc(C)nc2sc(C(=O)Nc3ccccc3Br)c(N)c12	nan
	CHEMBL1483523	40326	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	4	2	5	4.3	COCc1cc(C)nc2sc(C(=O)Nc3ccccc3Br)c(N)c12	nan
	1868051	40358	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	356	4	1	7	3.4	CSc1nc(SCC(=O)O)c2c3c(sc2n1)COC(C)(C)C3	nan
	CHEMBL1483727	40358	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	356	4	1	7	3.4	CSc1nc(SCC(=O)O)c2c3c(sc2n1)COC(C)(C)C3	nan
	4968512	40457	8	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	209	1	2	5	2.1	Nc1ccccc1-c1nnc(S)s1	nan
	CHEMBL1484500	40457	8	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	209	1	2	5	2.1	Nc1ccccc1-c1nnc(S)s1	nan
	1130974	40492	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	6	2	6	3.5	CCOc1ccc(NC(=O)c2sc(NC(C)=O)c(C(=O)OC)c2C)cc1	nan
	CHEMBL1484851	40492	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	6	2	6	3.5	CCOc1ccc(NC(=O)c2sc(NC(C)=O)c(C(=O)OC)c2C)cc1	nan
	16023029	40624	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	6	1	6	2.9	CN(Cc1ccc(F)cc1)S(=O)(=O)c1nnc(NC(=O)c2ccc(F)cc2)s1	nan
	CHEMBL1486082	40624	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	6	1	6	2.9	CN(Cc1ccc(F)cc1)S(=O)(=O)c1nnc(NC(=O)c2ccc(F)cc2)s1	nan
	2122608	40648	7	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	346	6	1	5	4.1	CC(=O)c1sc(NC(=O)COc2ccc(C(C)C)c(C)c2)nc1C	nan
	CHEMBL1486351	40648	7	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	346	6	1	5	4.1	CC(=O)c1sc(NC(=O)COc2ccc(C(C)C)c(C)c2)nc1C	nan
	15988496	40690	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	521	6	0	6	5.2	CCN(Cc1ccccc1)C(=O)Cn1c(=O)n(-c2ccc(F)c(Cl)c2)c(=O)c2sc3ccccc3c21	nan
	CHEMBL1486634	40690	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	521	6	0	6	5.2	CCN(Cc1ccccc1)C(=O)Cn1c(=O)n(-c2ccc(F)c(Cl)c2)c(=O)c2sc3ccccc3c21	nan
	5058050	40796	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	7	0	5	4.0	CCCCN(CCCC)C(=O)c1cc2c(=O)n3ccccc3nc2s1	nan
	CHEMBL1487547	40796	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	7	0	5	4.0	CCCCN(CCCC)C(=O)c1cc2c(=O)n3ccccc3nc2s1	nan
	1120443	40920	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	7	1	7	5.9	CCOc1cc(-c2nc3c(c(CC)nn3-c3ccccc3)c3cc(OC)c(OC)cc23)ccc1O	nan
	CHEMBL1488401	40920	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	7	1	7	5.9	CCOc1cc(-c2nc3c(c(CC)nn3-c3ccccc3)c3cc(OC)c(OC)cc23)ccc1O	nan
	1415522	40999	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	441	5	1	5	6.4	CCN(CC)C(=O)c1sc2nc(-c3cccs3)cc(-c3ccc(Cl)cc3)c2c1N	nan
	CHEMBL1488995	40999	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	441	5	1	5	6.4	CCN(CC)C(=O)c1sc2nc(-c3cccs3)cc(-c3ccc(Cl)cc3)c2c1N	nan
	2014552	41115	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	7	2	9	2.0	CCOc1cc(C2C(C#N)=C(N)SC(N)=C2C#N)ccc1OCCN1CCOCC1	nan
	CHEMBL1489906	41115	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	7	2	9	2.0	CCOc1cc(C2C(C#N)=C(N)SC(N)=C2C#N)ccc1OCCN1CCOCC1	nan
	2873834	41190	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	4	1	7	4.3	CC1=C(C(=O)OCC2CCCO2)C(c2coc3ccccc3c2=O)C2=C(O)CCCC2=N1	nan
	CHEMBL1490473	41190	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	4	1	7	4.3	CC1=C(C(=O)OCC2CCCO2)C(c2coc3ccccc3c2=O)C2=C(O)CCCC2=N1	nan
	1536777	41433	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	4	1	5	4.4	Cc1sc2ncnc(NC3CCN(Cc4ccccc4)CC3)c2c1C	nan
	CHEMBL1492096	41433	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	4	1	5	4.4	Cc1sc2ncnc(NC3CCN(Cc4ccccc4)CC3)c2c1C	nan
	2419865	41532	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	322	5	0	5	3.7	COc1ccc(C(C)=O)cc1COc1nc(C)nc2ccccc12	nan
	CHEMBL1492888	41532	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	322	5	0	5	3.7	COc1ccc(C(C)=O)cc1COc1nc(C)nc2ccccc12	nan
	1102906	41540	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	361	3	2	4	3.0	O=C(O)c1ccc(N2C(=O)c3cccc4c(C(=O)O)ccc(c34)C2=O)cc1	nan
	CHEMBL1492995	41540	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	361	3	2	4	3.0	O=C(O)c1ccc(N2C(=O)c3cccc4c(C(=O)O)ccc(c34)C2=O)cc1	nan
	3467703	41619	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	315	2	0	2	3.4	C=CCN1C(=O)c2cccc3c(Br)ccc(c23)C1=O	nan
	CHEMBL1493801	41619	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	315	2	0	2	3.4	C=CCN1C(=O)c2cccc3c(Br)ccc(c23)C1=O	nan
	7711621	41640	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	366	5	2	7	-0.5	CC(=O)Nc1ccc(S(=O)(=O)NCc2cc(=O)n(C)c(=O)n2C)cc1	nan
	CHEMBL1494013	41640	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	366	5	2	7	-0.5	CC(=O)Nc1ccc(S(=O)(=O)NCc2cc(=O)n(C)c(=O)n2C)cc1	nan
	681202	41709	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	3	3	3	3.6	Cc1sc(N=C(S)Nc2ccc(F)cc2)c(C(N)=O)c1C	nan
	CHEMBL1494694	41709	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	3	3	3	3.6	Cc1sc(N=C(S)Nc2ccc(F)cc2)c(C(N)=O)c1C	nan
	2451170	41788	15	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	268	2	1	6	2.8	CCOC(=O)c1sc2nc(C)nc(S)c2c1C	nan
	CHEMBL1495560	41788	15	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	268	2	1	6	2.8	CCOC(=O)c1sc2nc(C)nc(S)c2c1C	nan
	16017877	41830	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	3	0	4	2.6	Cc1ccccc1Cn1ccn(-c2ccc(F)c(F)c2)c(=O)c1=O	nan
	CHEMBL1495957	41830	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	3	0	4	2.6	Cc1ccccc1Cn1ccn(-c2ccc(F)c(F)c2)c(=O)c1=O	nan
	2917647	41953	15	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	4	1	6	3.5	O=C(C1=C(O)C(=O)N(c2ncccn2)C1c1ccc(Cl)cc1)c1ccco1	nan
	CHEMBL1497016	41953	15	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	4	1	6	3.5	O=C(C1=C(O)C(=O)N(c2ncccn2)C1c1ccc(Cl)cc1)c1ccco1	nan
	3493986	41974	8	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	539	8	1	6	5.3	CCOc1ccc(S(=O)(=O)[N-]c2nc3ccccc3nc2-[n+]2ccc(NC(=O)c3ccccc3C)cc2)cc1	nan
	CHEMBL1497174	41974	8	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	539	8	1	6	5.3	CCOc1ccc(S(=O)(=O)[N-]c2nc3ccccc3nc2-[n+]2ccc(NC(=O)c3ccccc3C)cc2)cc1	nan
	4260589	42011	6	None	-5	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	505	9	2	6	4.8	CCCC1(c2ccccc2)NC(=O)N(CC(=O)Nc2sc(-c3ccccc3)cc2C(=O)OCC)C1=O	nan
	CHEMBL1497431	42011	6	None	-5	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	505	9	2	6	4.8	CCCC1(c2ccccc2)NC(=O)N(CC(=O)Nc2sc(-c3ccccc3)cc2C(=O)OCC)C1=O	nan
	1234241	42072	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	274	1	1	5	2.9	Cc1nnc(S)c2nn(-c3ccccc3F)c(C)c12	nan
	CHEMBL1498110	42072	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	274	1	1	5	2.9	Cc1nnc(S)c2nn(-c3ccccc3F)c(C)c12	nan
	4056802	42275	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	6	1	6	2.8	Cc1cccn2c(=O)c3cc(C(=O)NCCCOC(C)C)sc3nc12	nan
	CHEMBL1499876	42275	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	6	1	6	2.8	Cc1cccn2c(=O)c3cc(C(=O)NCCCOC(C)C)sc3nc12	nan
	2908462	42280	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	7	1	6	3.1	O=C(C1=C(O)C(=O)N(CCCn2ccnc2)C1c1ccccc1)c1ccco1	nan
	CHEMBL1499902	42280	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	7	1	6	3.1	O=C(C1=C(O)C(=O)N(CCCn2ccnc2)C1c1ccccc1)c1ccco1	nan
	2551439	42412	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	6	0	8	1.7	COc1ccc(OCCOC(=O)c2nc3nccc(C)n3n2)cc1	nan
	CHEMBL1501099	42412	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	6	0	8	1.7	COc1ccc(OCCOC(=O)c2nc3nccc(C)n3n2)cc1	nan
	716763	42436	27	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	317	2	1	3	3.3	O=C(O)c1ccc(N2C(=O)c3cccc4cccc(c34)C2=O)cc1	nan
	CHEMBL1501298	42436	27	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	317	2	1	3	3.3	O=C(O)c1ccc(N2C(=O)c3cccc4cccc(c34)C2=O)cc1	nan
	5012247	42487	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	441	6	0	11	-2.0	CCN(C(=O)COC(=O)Cn1cnc2c1c(=O)n(C)c(=O)n2C)C1CCS(=O)(=O)C1	nan
	CHEMBL1501780	42487	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	441	6	0	11	-2.0	CCN(C(=O)COC(=O)Cn1cnc2c1c(=O)n(C)c(=O)n2C)C1CCS(=O)(=O)C1	nan
	2816746	42825	9	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	447	6	2	6	4.1	CCOC(=O)c1c(N=C(S)NCc2ccccc2)sc2c1CCN(C(=O)OCC)C2	nan
	CHEMBL1504775	42825	9	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	447	6	2	6	4.1	CCOC(=O)c1c(N=C(S)NCc2ccccc2)sc2c1CCN(C(=O)OCC)C2	nan
	2363951	42839	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	7	1	9	0.2	Cn1c(N)c(C(=O)COC(=O)CCC(=O)c2ccc(F)cc2)c(=O)n(C)c1=O	nan
	CHEMBL1504909	42839	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	7	1	9	0.2	Cn1c(N)c(C(=O)COC(=O)CCC(=O)c2ccc(F)cc2)c(=O)n(C)c1=O	nan
	3238944	42886	12	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	308	2	1	6	3.4	Cc1cccc(Nc2nn3c(=O)c4ccccc4nc3s2)c1	nan
	CHEMBL1505300	42886	12	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	308	2	1	6	3.4	Cc1cccc(Nc2nn3c(=O)c4ccccc4nc3s2)c1	nan
	7190519	42932	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	5	1	9	2.4	O=C(CSc1ccc2nnc(-c3ccccn3)n2n1)Nc1nccs1	nan
	CHEMBL1505657	42932	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	5	1	9	2.4	O=C(CSc1ccc2nnc(-c3ccccn3)n2n1)Nc1nccs1	nan
	3154081	43145	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	7	1	8	4.0	CCCOc1cccc(C2C(C(=O)c3ccco3)=C(O)C(=O)N2c2nnc(C)s2)c1	nan
	CHEMBL1507529	43145	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	7	1	8	4.0	CCCOc1cccc(C2C(C(=O)c3ccco3)=C(O)C(=O)N2c2nnc(C)s2)c1	nan
	1803037	43331	9	None	-4	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	521	7	1	5	6.1	Cc1cccc(NC(=O)CSc2nc(C)c(CC(=O)c3ccc(Br)cc3)c(C)c2C#N)c1C	nan
	CHEMBL1509120	43331	9	None	-4	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	521	7	1	5	6.1	Cc1cccc(NC(=O)CSc2nc(C)c(CC(=O)c3ccc(Br)cc3)c(C)c2C#N)c1C	nan
	3772923	43343	21	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	204	0	1	3	2.4	Cc1nc(S)c(C#N)c2c1CCCC2	nan
	CHEMBL1509207	43343	21	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	204	0	1	3	2.4	Cc1nc(S)c(C#N)c2c1CCCC2	nan
	3150659	43476	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	5	1	6	3.3	Cc1nc(SCC(=O)NCC2CCCO2)c2c3c(sc2n1)CCCC3	nan
	CHEMBL1510456	43476	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	5	1	6	3.3	Cc1nc(SCC(=O)NCC2CCCO2)c2c3c(sc2n1)CCCC3	nan
	2318166	43510	7	None	-4	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	5	1	6	4.7	CC(C)c1ccc(-c2c(C#N)c(N)nc(SCC(=O)N3CCCCCC3)c2C#N)cc1	nan
	CHEMBL1510689	43510	7	None	-4	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	5	1	6	4.7	CC(C)c1ccc(-c2c(C#N)c(N)nc(SCC(=O)N3CCCCCC3)c2C#N)cc1	nan
	4382156	43583	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	5	1	4	2.2	O=C(CCCN1C(=O)c2cccnc2C1=O)Nc1ccccc1F	nan
	CHEMBL1511309	43583	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	5	1	4	2.2	O=C(CCCN1C(=O)c2cccnc2C1=O)Nc1ccccc1F	nan
	5825936	43640	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	520	10	1	8	3.3	C=CCOc1ccc(C2C(C(=O)c3ccc4c(c3)OCCO4)=C(O)C(=O)N2CCCN2CCOCC2)cc1	nan
	CHEMBL1511801	43640	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	520	10	1	8	3.3	C=CCOc1ccc(C2C(C(=O)c3ccc4c(c3)OCCO4)=C(O)C(=O)N2CCCN2CCOCC2)cc1	nan
	1234706	43669	15	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	426	7	2	6	3.5	CCOc1ccccc1C(=O)Nc1ccc(S(=O)(=O)Nc2nc(C)cc(C)n2)cc1	nan
	CHEMBL1512389	43669	15	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	426	7	2	6	3.5	CCOc1ccccc1C(=O)Nc1ccc(S(=O)(=O)Nc2nc(C)cc(C)n2)cc1	nan
	18572258	43680	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	447	6	1	7	2.9	O=C(CSc1nnc2ccc(-c3ccc(Br)cc3)nn12)NCC1CCCO1	nan
	CHEMBL1512477	43680	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	447	6	1	7	2.9	O=C(CSc1nnc2ccc(-c3ccc(Br)cc3)nn12)NCC1CCCO1	nan
	7205055	43709	17	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	5	1	6	3.3	CCN1CCN(Cc2c(O)ccc3cc(-c4ccc(OC)cc4)c(=O)oc23)CC1	nan
	CHEMBL1512819	43709	17	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	5	1	6	3.3	CCN1CCN(Cc2c(O)ccc3cc(-c4ccc(OC)cc4)c(=O)oc23)CC1	nan
	53229784	43711	21	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	351	4	1	5	3.8	COc1ccc(-c2cc3ccc(O)c(CN4CCCC4)c3oc2=O)cc1	nan
	5457315	43711	21	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	351	4	1	5	3.8	COc1ccc(-c2cc3ccc(O)c(CN4CCCC4)c3oc2=O)cc1	nan
	CHEMBL1512839	43711	21	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	351	4	1	5	3.8	COc1ccc(-c2cc3ccc(O)c(CN4CCCC4)c3oc2=O)cc1	nan
	16026424	43745	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	5	0	7	3.4	COC(=O)c1sc2ccccc2c1S(=O)(=O)N1CCN(c2ccc(C(C)=O)cc2)CC1	nan
	CHEMBL1513424	43745	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	5	0	7	3.4	COC(=O)c1sc2ccccc2c1S(=O)(=O)N1CCN(c2ccc(C(C)=O)cc2)CC1	nan
	16019493	43760	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	8	1	7	3.6	Cc1ccc(S(=O)(=O)NCCc2nnc3ccc(SCc4ccccc4C)nn23)cc1	nan
	CHEMBL1513611	43760	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	8	1	7	3.6	Cc1ccc(S(=O)(=O)NCCc2nnc3ccc(SCc4ccccc4C)nn23)cc1	nan
	15989126	43764	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	552	11	2	7	4.7	Cc1ccccc1NC(=O)Cn1c(=O)n(CCCCCC(=O)NCc2ccccc2Cl)c(=O)c2sccc21	nan
	CHEMBL1513634	43764	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	552	11	2	7	4.7	Cc1ccccc1NC(=O)Cn1c(=O)n(CCCCCC(=O)NCc2ccccc2Cl)c(=O)c2sccc21	nan
	1252356	43780	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	478	7	1	6	5.5	Cc1cc(C)cc(NC(=O)CSc2oc(-c3ccccc3)nc2S(=O)(=O)c2ccccc2)c1	nan
	CHEMBL1513969	43780	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	478	7	1	6	5.5	Cc1cc(C)cc(NC(=O)CSc2oc(-c3ccccc3)nc2S(=O)(=O)c2ccccc2)c1	nan
	16406807	43784	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	8	3	6	2.7	CC[C@@H](C)[C@H](NC(=O)CNC(=O)Cc1c(C)c2c(cc(C)c3c(C)coc32)oc1=O)C(=O)O	nan
	CHEMBL1514043	43784	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	8	3	6	2.7	CC[C@@H](C)[C@H](NC(=O)CNC(=O)Cc1c(C)c2c(cc(C)c3c(C)coc32)oc1=O)C(=O)O	nan
	2135573	43815	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	514	8	1	8	4.1	CCOc1ccc(C(=O)c2cn(CC(=O)Nc3ccc(OC)cc3)c3cc4c(cc3c2=O)OCCO4)cc1	nan
	CHEMBL1514550	43815	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	514	8	1	8	4.1	CCOc1ccc(C(=O)c2cn(CC(=O)Nc3ccc(OC)cc3)c3cc4c(cc3c2=O)OCCO4)cc1	nan
	16018084	43857	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	9	1	6	3.6	COc1ccc(OC)c(CCNC(=O)CCCn2c(=O)c3cccn3c3ccc(F)cc32)c1	nan
	CHEMBL1515147	43857	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	9	1	6	3.6	COc1ccc(OC)c(CCNC(=O)CCCn2c(=O)c3cccn3c3ccc(F)cc32)c1	nan
	4302940	43858	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	5	1	4	5.4	CCn1cc(CNC(=O)c2cc(-c3ccc(C)cc3)nc3ccc(Br)cc23)c(C)n1	nan
	CHEMBL1515178	43858	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	5	1	4	5.4	CCn1cc(CNC(=O)c2cc(-c3ccc(C)cc3)nc3ccc(Br)cc23)c(C)n1	nan
	15989010	43873	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	477	7	1	8	3.0	Cc1cccc(Cn2c(=O)n(CCC(=O)NCc3ccc4c(c3)OCO4)c(=O)c3sccc32)c1	nan
	CHEMBL1515330	43873	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	477	7	1	8	3.0	Cc1cccc(Cn2c(=O)n(CCC(=O)NCc3ccc4c(c3)OCO4)c(=O)c3sccc32)c1	nan
	20885696	44033	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	9	1	8	1.4	COc1ccc(CCNC(=O)CCCn2nc(C)n3ccnc3c2=O)cc1OC	nan
	CHEMBL1517314	44033	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	9	1	8	1.4	COc1ccc(CCNC(=O)CCCn2nc(C)n3ccnc3c2=O)cc1OC	nan
	1488779	44257	21	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	320	4	0	4	4.6	COc1ccc(Oc2nccc(-c3ccc(F)cc3)c2C#N)cc1	nan
	CHEMBL1519391	44257	21	None	-1	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	320	4	0	4	4.6	COc1ccc(Oc2nccc(-c3ccc(F)cc3)c2C#N)cc1	nan
	3154197	44258	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	363	5	2	8	0.6	Cn1c(=O)c2c(ncn2CC(O)CNc2cccc(Cl)c2)n(C)c1=O	nan
	CHEMBL1519401	44258	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	363	5	2	8	0.6	Cn1c(=O)c2c(ncn2CC(O)CNc2cccc(Cl)c2)n(C)c1=O	nan
	5309980	44300	1	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	318	4	1	6	2.5	CC(Sc1ccc2nnc(-c3ccc(F)cc3)n2n1)C(=O)O	nan
	CHEMBL1519790	44300	1	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	318	4	1	6	2.5	CC(Sc1ccc2nnc(-c3ccc(F)cc3)n2n1)C(=O)O	nan
	20873023	44388	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	7	1	10	-0.3	CCOC(=O)CNC(=O)Cn1cnc2c(nnn2-c2ccc(OC)cc2)c1=O	nan
	CHEMBL1520622	44388	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	7	1	10	-0.3	CCOC(=O)CNC(=O)Cn1cnc2c(nnn2-c2ccc(OC)cc2)c1=O	nan
	135407280	44416	32	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	243	2	1	5	2.4	CSc1nc(O)c(C#N)c(-c2ccccc2)n1	nan
	CHEMBL1520797	44416	32	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	243	2	1	5	2.4	CSc1nc(O)c(C#N)c(-c2ccccc2)n1	nan
	2868262	44480	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	3	1	3	4.7	CC(=O)C1=C(O)C(=O)N(c2ccc(Br)cc2)C1c1ccc(Br)cc1	nan
	CHEMBL1521342	44480	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	3	1	3	4.7	CC(=O)C1=C(O)C(=O)N(c2ccc(Br)cc2)C1c1ccc(Br)cc1	nan
	646901	44530	3	None	-4	3	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	5	1	7	3.6	CCc1cc2cc3c(cc2nc1SCC(=O)Nc1cc(C)on1)OCO3	nan
	CHEMBL1521729	44530	3	None	-4	3	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	5	1	7	3.6	CCc1cc2cc3c(cc2nc1SCC(=O)Nc1cc(C)on1)OCO3	nan
	16012248	44546	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	4	1	5	5.0	Cc1cc(C)c2c(n1)nn1c(C)c(CCC(=O)Nc3ccc(C)c(Cl)c3)c(C)nc21	nan
	CHEMBL1521906	44546	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	4	1	5	5.0	Cc1cc(C)c2c(n1)nn1c(C)c(CCC(=O)Nc3ccc(C)c(Cl)c3)c(C)nc21	nan
	5086217	44568	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	4	2	4	4.6	CCOC(=O)c1c(N=C(S)Nc2ccc(F)cc2)sc2c1CCC2	nan
	CHEMBL1522109	44568	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	4	2	4	4.6	CCOC(=O)c1c(N=C(S)Nc2ccc(F)cc2)sc2c1CCC2	nan
	2929681	44639	17	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	457	6	2	7	2.6	Cc1cccn2c(=O)c3cc(C(=O)NCC4CCCO4)c(=N)n(CCc4ccccc4)c3nc12	nan
	CHEMBL1522811	44639	17	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	457	6	2	7	2.6	Cc1cccn2c(=O)c3cc(C(=O)NCC4CCCO4)c(=N)n(CCc4ccccc4)c3nc12	nan
	352022	44681	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	268	3	0	7	0.5	CCCSc1nc2c(c(=O)n(C)c(=O)n2C)n1C	nan
	CHEMBL1523163	44681	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	268	3	0	7	0.5	CCCSc1nc2c(c(=O)n(C)c(=O)n2C)n1C	nan
	861889	44691	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	4	1	3	4.0	Cc1ccc2nc(SCC(=O)NC3CCCC3)c(C)cc2c1	nan
	CHEMBL1523239	44691	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	4	1	3	4.0	Cc1ccc2nc(SCC(=O)NC3CCCC3)c(C)cc2c1	nan
	4099138	44696	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	510	9	2	8	3.5	O=C(CCCCCn1c(=S)[nH]c2ccc(N3CCOCC3)cc2c1=O)NCc1ccc2c(c1)OCO2	nan
	CHEMBL1523295	44696	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	510	9	2	8	3.5	O=C(CCCCCn1c(=S)[nH]c2ccc(N3CCOCC3)cc2c1=O)NCc1ccc2c(c1)OCO2	nan
	5760985	44976	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	4	1	4	4.8	O=C(C1=C(O)C(=O)N(c2ccccn2)C1c1ccc(F)cc1)c1ccc(Br)cc1	nan
	CHEMBL1525962	44976	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	4	1	4	4.8	O=C(C1=C(O)C(=O)N(c2ccccn2)C1c1ccc(F)cc1)c1ccc(Br)cc1	nan
	3186625	45198	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	5	2	9	0.7	CC(=O)Nc1cccc(NC(=O)CSc2nc3c(c(=O)n(C)c(=O)n3C)n2C)c1	nan
	CHEMBL1527889	45198	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	5	2	9	0.7	CC(=O)Nc1cccc(NC(=O)CSc2nc3c(c(=O)n(C)c(=O)n3C)n2C)c1	nan
	1166606	45270	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	463	8	1	6	5.3	COc1ccc(NC(=O)CCSc2nc(-c3ccc(OC)cc3)cc(C(F)(F)F)n2)cc1	nan
	CHEMBL1528550	45270	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	463	8	1	6	5.3	COc1ccc(NC(=O)CCSc2nc(-c3ccc(OC)cc3)cc(C(F)(F)F)n2)cc1	nan
	1109837	45351	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	5	1	5	4.2	Cc1ccccc1OCC(=O)Nc1ccc(-c2nc3ncccc3o2)cc1	nan
	CHEMBL1529226	45351	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	5	1	5	4.2	Cc1ccccc1OCC(=O)Nc1ccc(-c2nc3ncccc3o2)cc1	nan
	4413149	45374	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	5	1	4	3.1	Cc1ccc(Cl)cc1NC(=O)CCCN1C(=O)c2cccnc2C1=O	nan
	CHEMBL1529453	45374	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	5	1	4	3.1	Cc1ccc(Cl)cc1NC(=O)CCCN1C(=O)c2cccnc2C1=O	nan
	6086754	45437	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	8	1	7	3.9	COc1cccc(C2C(C(=O)c3ccc4c(c3)CC(C)O4)=C(O)C(=O)N2CCCn2ccnc2)c1	nan
	CHEMBL1529980	45437	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	8	1	7	3.9	COc1cccc(C2C(C(=O)c3ccc4c(c3)CC(C)O4)=C(O)C(=O)N2CCCn2ccnc2)c1	nan
	4881121	45476	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	5	0	7	2.0	CCc1cc2c(SCC(=O)N(C)C3CCS(=O)(=O)C3)ncnc2s1	nan
	CHEMBL1530432	45476	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	5	0	7	2.0	CCc1cc2c(SCC(=O)N(C)C3CCS(=O)(=O)C3)ncnc2s1	nan
	15988929	45529	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	534	12	2	8	3.7	COc1ccccc1NC(=O)Cn1c(=O)n(CCCCCC(=O)NCc2ccccc2)c(=O)c2sccc21	nan
	CHEMBL1530799	45529	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	534	12	2	8	3.7	COc1ccccc1NC(=O)Cn1c(=O)n(CCCCCC(=O)NCc2ccccc2)c(=O)c2sccc21	nan
	2956077	45594	21	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	5	1	3	3.4	COc1ccc2cc(Br)ccc2c1CC(=O)NCC1CCCO1	nan
	CHEMBL1531449	45594	21	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	5	1	3	3.4	COc1ccc2cc(Br)ccc2c1CC(=O)NCC1CCCO1	nan
	646794	46012	5	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	5	1	6	2.4	O=C(C1=C(O)C(=O)N(CC2CCCO2)C1c1cccnc1)c1ccco1	nan
	CHEMBL1535358	46012	5	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	5	1	6	2.4	O=C(C1=C(O)C(=O)N(CC2CCCO2)C1c1cccnc1)c1ccco1	nan
	9551120	46147	0	None	-14	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	3	1	6	3.0	CCOC(=O)Cn1c(=S)[nH]c2c(oc3ccc(Cl)cc32)c1=O	nan
	CHEMBL1536779	46147	0	None	-14	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	3	1	6	3.0	CCOC(=O)Cn1c(=S)[nH]c2c(oc3ccc(Cl)cc32)c1=O	nan
	5297702	46247	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	295	1	1	3	4.2	Nc1c2c(nc3cccc(Cl)c13)N(c1ccccc1)CC2	nan
	CHEMBL1537611	46247	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	295	1	1	3	4.2	Nc1c2c(nc3cccc(Cl)c13)N(c1ccccc1)CC2	nan
	5069161	46441	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	6	2	6	3.5	O=C(CCCn1c(=S)[nH]c2cc3c(cc2c1=O)OCO3)NCc1ccccc1Cl	nan
	CHEMBL1539200	46441	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	6	2	6	3.5	O=C(CCCn1c(=S)[nH]c2cc3c(cc2c1=O)OCO3)NCc1ccccc1Cl	nan
	1373674	46511	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	351	4	1	8	0.1	Cn1c(=O)c2c(nc(SCC(=O)NC3CCCC3)n2C)n(C)c1=O	nan
	CHEMBL1539818	46511	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	351	4	1	8	0.1	Cn1c(=O)c2c(nc(SCC(=O)NC3CCCC3)n2C)n(C)c1=O	nan
	20888840	46552	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	6	0	8	2.2	CCCS(=O)(=O)c1nc(S(=O)(=O)c2ccc(C)cc2)c(N2CCN(C)CC2)s1	nan
	CHEMBL1540109	46552	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	6	0	8	2.2	CCCS(=O)(=O)c1nc(S(=O)(=O)c2ccc(C)cc2)c(N2CCN(C)CC2)s1	nan
	2823604	46632	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	267	3	0	4	3.2	COC(=O)CSc1ccnc2cc(Cl)ccc12	nan
	CHEMBL1540846	46632	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	267	3	0	4	3.2	COC(=O)CSc1ccnc2cc(Cl)ccc12	nan
	2502748	46666	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	7	0	7	3.0	COc1cc(CN(C)Cc2cc(=O)n3ccsc3n2)ccc1OC(F)F	nan
	CHEMBL1541111	46666	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	7	0	7	3.0	COc1cc(CN(C)Cc2cc(=O)n3ccsc3n2)ccc1OC(F)F	nan
	3119316	46724	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	4	1	4	3.9	COc1ccc(C2C(C(C)=O)=C(O)C(=O)N2c2ccc(Br)cc2)cc1	nan
	CHEMBL1541516	46724	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	4	1	4	3.9	COc1ccc(C2C(C(C)=O)=C(O)C(=O)N2c2ccc(Br)cc2)cc1	nan
	4885704	46777	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	3	1	7	2.5	O=c1c2ccccc2cnn1Cc1nnc(S)n1-c1ccccc1F	nan
	CHEMBL1541978	46777	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	3	1	7	2.5	O=c1c2ccccc2cnn1Cc1nnc(S)n1-c1ccccc1F	nan
	20884256	46959	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	5	1	8	0.5	Cc1nn(CC(=O)NCCN2CCOCC2)c(=O)c2cc3sccc3n12	nan
	CHEMBL1543621	46959	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	5	1	8	0.5	Cc1nn(CC(=O)NCCN2CCOCC2)c(=O)c2cc3sccc3n12	nan
	1451421	47060	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	7	0	6	3.9	CCOC(=O)CSc1nc(COc2ccccc2)nc2ccccc12	nan
	CHEMBL1544289	47060	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	7	0	6	3.9	CCOC(=O)CSc1nc(COc2ccccc2)nc2ccccc12	nan
	7120054	47136	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	324	2	1	5	3.8	COc1cccc(-n2c(=S)[nH]c3c(oc4ccccc43)c2=O)c1	nan
	CHEMBL1544911	47136	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	324	2	1	5	3.8	COc1cccc(-n2c(=S)[nH]c3c(oc4ccccc43)c2=O)c1	nan
	3192298	47156	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	215	2	0	5	1.3	Cc1nc2ccccn2c1C(=O)OCC#N	nan
	CHEMBL1545062	47156	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	215	2	0	5	1.3	Cc1nc2ccccn2c1C(=O)OCC#N	nan
	976399	47164	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	283	2	0	4	4.1	Cc1ccc(OC(=O)c2ccc3nc(C)sc3c2)cc1	nan
	CHEMBL1545103	47164	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	283	2	0	4	4.1	Cc1ccc(OC(=O)c2ccc3nc(C)sc3c2)cc1	nan
	3455851	47262	25	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	3	1	4	3.2	O=S(=O)(Nc1nc2ccccc2nc1Cl)c1ccc(F)cc1	nan
	CHEMBL1545899	47262	25	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	3	1	4	3.2	O=S(=O)(Nc1nc2ccccc2nc1Cl)c1ccc(F)cc1	nan
	2431161	47471	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	491	6	1	6	3.6	CC(C)[C@H](NC(=O)c1ccccc1Cl)C(=O)OCc1cc(=O)n2cc(Br)ccc2n1	nan
	CHEMBL1547817	47471	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	491	6	1	6	3.6	CC(C)[C@H](NC(=O)c1ccccc1Cl)C(=O)OCc1cc(=O)n2cc(Br)ccc2n1	nan
	3111438	47527	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	4	0	4	3.2	CC(=O)OCCCN1C(=O)c2cccc3cc(Br)cc(c23)C1=O	nan
	CHEMBL1548381	47527	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	4	0	4	3.2	CC(=O)OCCCN1C(=O)c2cccc3cc(Br)cc(c23)C1=O	nan
	24792694	47528	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	313	4	1	6	1.9	Cn1c2ccccc2c2nnc(SCC(=O)NC3CC3)nc21	nan
	CHEMBL1548382	47528	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	313	4	1	6	1.9	Cn1c2ccccc2c2nnc(SCC(=O)NC3CC3)nc21	nan
	664646	47543	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	4	1	5	3.6	COc1ccc(C(=O)OCc2cc3cccc(C)c3nc2O)cc1	nan
	CHEMBL1548510	47543	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	4	1	5	3.6	COc1ccc(C(=O)OCc2cc3cccc(C)c3nc2O)cc1	nan
	839503	47564	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	324	5	3	3	3.0	O=C(Nc1ccccc1C(=O)O)c1ccc(NC(=O)C2CC2)cc1	nan
	CHEMBL1548673	47564	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	324	5	3	3	3.0	O=C(Nc1ccccc1C(=O)O)c1ccc(NC(=O)C2CC2)cc1	nan
	4839425	47657	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	6	0	10	0.2	CN(C)S(=O)(=O)c1cc(C(=O)OCCn2cnc3c2c(=O)n(C)c(=O)n3C)ccc1Cl	nan
	CHEMBL1549482	47657	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	6	0	10	0.2	CN(C)S(=O)(=O)c1cc(C(=O)OCCn2cnc3c2c(=O)n(C)c(=O)n3C)ccc1Cl	nan
	838258	47740	24	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	238	1	1	3	3.6	Sc1nc(-c2ccccc2)nc2ccccc12	nan
	CHEMBL1550135	47740	24	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	238	1	1	3	3.6	Sc1nc(-c2ccccc2)nc2ccccc12	nan
	2794423	47769	15	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	195	0	1	2	2.3	NC1=CC(=O)c2cccc3cccc1c23	nan
	CHEMBL1550366	47769	15	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	195	0	1	2	2.3	NC1=CC(=O)c2cccc3cccc1c23	nan
	16187761	47793	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	5	1	7	2.2	Cc1cc(C)n2nc(C(=O)N3CCCC(CNS(=O)(=O)c4cccs4)C3)cc2n1	nan
	CHEMBL1550610	47793	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	5	1	7	2.2	Cc1cc(C)n2nc(C(=O)N3CCCC(CNS(=O)(=O)c4cccs4)C3)cc2n1	nan
	4969856	47868	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	282	3	2	6	2.1	CC(=O)Nc1ccc(Nc2ncnc3c2cnn3C)cc1	nan
	CHEMBL1551291	47868	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	282	3	2	6	2.1	CC(=O)Nc1ccc(Nc2ncnc3c2cnn3C)cc1	nan
	16009663	47871	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	487	6	1	7	4.8	CSc1cccc(NC(=O)Cn2c(=O)n(Cc3ccccc3)c(=O)c3sc4ccccc4c32)c1	nan
	CHEMBL1551326	47871	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	487	6	1	7	4.8	CSc1cccc(NC(=O)Cn2c(=O)n(Cc3ccccc3)c(=O)c3sc4ccccc4c32)c1	nan
	7184893	47947	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	6	1	8	3.7	CCCCNc1nc2c(S(=O)(=O)c3ccc(C)cc3)nnn2c2ccsc12	nan
	CHEMBL1552371	47947	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	6	1	8	3.7	CCCCNc1nc2c(S(=O)(=O)c3ccc(C)cc3)nnn2c2ccsc12	nan
	1003444	47958	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	3	2	5	5.7	Nc1c(C(=O)Nc2ccc(Cl)cc2F)sc2nc(-c3cccs3)ccc12	nan
	CHEMBL1552586	47958	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	3	2	5	5.7	Nc1c(C(=O)Nc2ccc(Cl)cc2F)sc2nc(-c3cccs3)ccc12	nan
	1841026	47988	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	5	0	8	1.6	CCOC(=O)/C(C#N)=C/c1c(N2CCN(CC)CC2)nc2c(C)cccn2c1=O	nan
	CHEMBL1553005	47988	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	5	0	8	1.6	CCOC(=O)/C(C#N)=C/c1c(N2CCN(CC)CC2)nc2c(C)cccn2c1=O	nan
	15988107	47990	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	510	8	0	7	3.8	CCN(Cc1ccccc1)C(=O)Cn1c(=O)n(Cc2ccccc2)c(=O)c2c1c1cc(OC)ccc1n2C	nan
	CHEMBL1553031	47990	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	510	8	0	7	3.8	CCN(Cc1ccccc1)C(=O)Cn1c(=O)n(Cc2ccccc2)c(=O)c2c1c1cc(OC)ccc1n2C	nan
	16009750	47994	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	4	1	5	4.9	Cc1cccc(-c2nnn3c2nc(NCc2ccccc2)c2ccccc23)c1	nan
	CHEMBL1553063	47994	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	4	1	5	4.9	Cc1cccc(-c2nnn3c2nc(NCc2ccccc2)c2ccccc23)c1	nan
	15988172	48012	1	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	5	2	4	2.2	CCCCNC(=O)c1ccc2c(=O)n(-c3ccccc3)c(=O)[nH]c2c1	nan
	CHEMBL1553275	48012	1	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	5	2	4	2.2	CCCCNC(=O)c1ccc2c(=O)n(-c3ccccc3)c(=O)[nH]c2c1	nan
	135697665	48022	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	5	1	9	1.8	O=C(OCc1nc(O)c2sccc2n1)c1cccc(S(=O)(=O)N2CCOCC2)c1	nan
	CHEMBL1553392	48022	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	5	1	9	1.8	O=C(OCc1nc(O)c2sccc2n1)c1cccc(S(=O)(=O)N2CCOCC2)c1	nan
	5927505	48216	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	523	7	1	7	4.1	O=C(C1=C(O)C(=O)N(CCCn2ccnc2)C1c1cccc(Br)c1)c1ccc2c(c1)OCCO2	nan
	CHEMBL1556043	48216	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	523	7	1	7	4.1	O=C(C1=C(O)C(=O)N(CCCn2ccnc2)C1c1cccc(Br)c1)c1ccc2c(c1)OCCO2	nan
	2195056	48249	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	5	1	2	4.7	O=C(Nc1ccc(F)cc1)c1ccc(COc2ccccc2)cc1	nan
	CHEMBL1556330	48249	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	5	1	2	4.7	O=C(Nc1ccc(F)cc1)c1ccc(COc2ccccc2)cc1	nan
	5301777	48266	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	493	5	2	6	5.9	COC(=O)c1ccccc1NC(=O)c1sc2nc(C)cc(C)c2c1NC(=O)c1ccccc1Cl	nan
	CHEMBL1556556	48266	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	493	5	2	6	5.9	COC(=O)c1ccccc1NC(=O)c1sc2nc(C)cc(C)c2c1NC(=O)c1ccccc1Cl	nan
	3404081	48289	24	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	189	0	1	2	3.1	Cc1ccc2c(C)cc(S)nc2c1	nan
	CHEMBL1556798	48289	24	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	189	0	1	2	3.1	Cc1ccc2c(C)cc(S)nc2c1	nan
	1348154	48296	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	396	4	1	4	4.9	O=C(Cc1ccc(Cl)cc1)Nc1ccc2nn(-c3ccc(Cl)cc3)nc2c1	nan
	CHEMBL1556858	48296	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	396	4	1	4	4.9	O=C(Cc1ccc(Cl)cc1)Nc1ccc2nn(-c3ccc(Cl)cc3)nc2c1	nan
	3708288	48308	7	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	1	4	7	2.3	N#Cc1c(N)nc2c3c(sc(=N)c2c1N)NC(=O)CC3c1ccccc1	nan
	CHEMBL1556915	48308	7	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	1	4	7	2.3	N#Cc1c(N)nc2c3c(sc(=N)c2c1N)NC(=O)CC3c1ccccc1	nan
	285470	48349	24	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	4	1	5	4.6	CCNc1nc(Cl)nc(-c2cn(-c3ccccc3)c3ccccc23)n1	nan
	CHEMBL1557270	48349	24	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	4	1	5	4.6	CCNc1nc(Cl)nc(-c2cn(-c3ccccc3)c3ccccc23)n1	nan
	16009846	48394	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	5	1	8	1.7	COc1ccc(NC(=O)Cn2c(=O)c3ccccc3n3nncc23)c(OC)c1	nan
	CHEMBL1557614	48394	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	5	1	8	1.7	COc1ccc(NC(=O)Cn2c(=O)c3ccccc3n3nncc23)c(OC)c1	nan
	16010737	48403	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	6	1	6	3.1	CCc1ccc(NC(=O)Cn2c(=O)n(Cc3ccc(C)cc3)c(=O)c3cccnc32)cc1	nan
	CHEMBL1557693	48403	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	6	1	6	3.1	CCc1ccc(NC(=O)Cn2c(=O)n(Cc3ccc(C)cc3)c(=O)c3cccnc32)cc1	nan
	3333649	48562	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	5	1	5	3.2	COc1ccc(S(=O)(=O)N2CCCCC2)cc1NC(=O)c1cccs1	nan
	CHEMBL1559037	48562	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	5	1	5	3.2	COc1ccc(S(=O)(=O)N2CCCCC2)cc1NC(=O)c1cccs1	nan
	1166246	48617	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	475	6	1	6	5.6	Cc1ccc(NC(=O)CCSc2nc(-c3ccc4c(c3)OCO4)cc(C(F)(F)F)n2)c(C)c1	nan
	CHEMBL1559537	48617	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	475	6	1	6	5.6	Cc1ccc(NC(=O)CCSc2nc(-c3ccc4c(c3)OCO4)cc(C(F)(F)F)n2)c(C)c1	nan
	16009080	48819	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	569	7	1	7	6.7	CCOc1ccc(-c2cc3nc(C4CCN(C(=O)OC(C)(C)C)CC4)c(C(=O)Nc4cccc(CC)c4)cn3n2)cc1	nan
	CHEMBL1561508	48819	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	569	7	1	7	6.7	CCOc1ccc(-c2cc3nc(C4CCN(C(=O)OC(C)(C)C)CC4)c(C(=O)Nc4cccc(CC)c4)cn3n2)cc1	nan
	3141845	48877	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	4	1	4	6.0	COc1cc(NC(=O)c2ccc(Cl)cc2Cl)ccc1-c1cc2ccccc2oc1=O	nan
	CHEMBL1562003	48877	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	4	1	4	6.0	COc1cc(NC(=O)c2ccc(Cl)cc2Cl)ccc1-c1cc2ccccc2oc1=O	nan
	2510921	48983	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	6	1	5	2.8	O=C(CNC(=O)C1CCCCC1)OCC(=O)c1ccc(Cl)s1	nan
	CHEMBL1562941	48983	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	6	1	5	2.8	O=C(CNC(=O)C1CCCCC1)OCC(=O)c1ccc(Cl)s1	nan
	4800554	49105	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	6	1	6	3.8	COc1cc(C(C)=O)ccc1OCC(=O)Nc1ccc2nc(C)sc2c1	nan
	CHEMBL1563979	49105	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	6	1	6	3.8	COc1cc(C(C)=O)ccc1OCC(=O)Nc1ccc2nc(C)sc2c1	nan
	16009343	49124	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	348	4	0	5	4.3	Cc1ccccc1OCc1cc(=O)n2c(-c3ccccc3)csc2n1	nan
	CHEMBL1564149	49124	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	348	4	0	5	4.3	Cc1ccccc1OCc1cc(=O)n2c(-c3ccccc3)csc2n1	nan
	4911790	49235	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	306	2	1	2	3.4	COc1ccc2cc(C(=O)N3CCc4ccccc4C3)[nH]c2c1	nan
	CHEMBL1565220	49235	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	306	2	1	2	3.4	COc1ccc2cc(C(=O)N3CCc4ccccc4C3)[nH]c2c1	nan
	974361	49290	12	None	-1	3	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	336	3	1	6	3.9	Cc1onc(-c2ccccc2)c1C(=O)Nc1cccc2nsnc12	nan
	CHEMBL1565576	49290	12	None	-1	3	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	336	3	1	6	3.9	Cc1onc(-c2ccccc2)c1C(=O)Nc1cccc2nsnc12	nan
	15989682	49317	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	509	8	1	8	3.5	COc1ccc(NC(=O)Cn2c(=O)n(Cc3ccccc3Cl)c(=O)c3cc(OC)c(OC)cc32)cc1	nan
	CHEMBL1565778	49317	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	509	8	1	8	3.5	COc1ccc(NC(=O)Cn2c(=O)n(Cc3ccccc3Cl)c(=O)c3cc(OC)c(OC)cc32)cc1	nan
	1977639	49320	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	515	6	1	5	5.2	O=C(Nc1cc[n+](-c2nc3ccccc3nc2[N-]S(=O)(=O)c2ccccc2)cc1)c1ccccc1Cl	nan
	CHEMBL1565785	49320	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	515	6	1	5	5.2	O=C(Nc1cc[n+](-c2nc3ccccc3nc2[N-]S(=O)(=O)c2ccccc2)cc1)c1ccccc1Cl	nan
	789538	49455	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	210	0	1	4	2.0	CC1=C(C)C(C)=C(C#N)C(=C(C#N)C#N)N1	nan
	CHEMBL1566885	49455	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	210	0	1	4	2.0	CC1=C(C)C(C)=C(C#N)C(=C(C#N)C#N)N1	nan
	3442888	49559	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	1	0	5	3.1	Cc1cccn2c(=O)c3cc(C(=O)N4CCCC(C)C4)sc3nc12	nan
	CHEMBL1567700	49559	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	1	0	5	3.1	Cc1cccn2c(=O)c3cc(C(=O)N4CCCC(C)C4)sc3nc12	nan
	16009353	49871	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	4	0	5	4.6	Cc1cccc(OCc2cc(=O)n3c(-c4ccccc4)csc3n2)c1C	nan
	CHEMBL1570398	49871	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	4	0	5	4.6	Cc1cccc(OCc2cc(=O)n3c(-c4ccccc4)csc3n2)c1C	nan
	16019299	49885	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	5	1	5	4.2	Cc1cc(C)c(NC(=O)CSc2ccc(-c3ccccn3)nn2)c(C)c1	nan
	CHEMBL1570518	49885	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	5	1	5	4.2	Cc1cc(C)c(NC(=O)CSc2ccc(-c3ccccn3)nn2)c(C)c1	nan
	4917201	49957	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	261	4	1	6	1.4	CC(C(=O)Nc1cccnc1)n1cc([N+](=O)[O-])cn1	nan
	CHEMBL1571073	49957	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	261	4	1	6	1.4	CC(C(=O)Nc1cccnc1)n1cc([N+](=O)[O-])cn1	nan
	15990163	49959	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	7	2	7	3.3	COc1ccc(S(=O)(=O)Nc2cc3c(cc2NCc2ccccc2)n(C)c(=O)n3C)cc1	nan
	CHEMBL1571094	49959	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	7	2	7	3.3	COc1ccc(S(=O)(=O)Nc2cc3c(cc2NCc2ccccc2)n(C)c(=O)n3C)cc1	nan
	16194623	50044	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	5	0	8	1.8	CC(=O)C(Sc1ccc2nnc(-c3cccnc3)n2n1)C(C)=O	nan
	CHEMBL1572020	50044	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	5	0	8	1.8	CC(=O)C(Sc1ccc2nnc(-c3cccnc3)n2n1)C(C)=O	nan
	135408736	50099	38	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	228	1	1	5	2.1	Sc1ncnc2c1cnn2-c1ccccc1	nan
	CHEMBL1572500	50099	38	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	228	1	1	5	2.1	Sc1ncnc2c1cnn2-c1ccccc1	nan
	2769007	50415	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	293	4	0	7	1.4	CCOC(=O)C(C)Sc1nc(=O)n2cc(C)ccc2n1	nan
	CHEMBL1575703	50415	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	293	4	0	7	1.4	CCOC(=O)C(C)Sc1nc(=O)n2cc(C)ccc2n1	nan
	2808306	50431	21	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	297	5	2	4	3.1	CC(=O)c1sc(C(C)(C)C)cc1NC(=O)CCC(=O)O	nan
	CHEMBL1575844	50431	21	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	297	5	2	4	3.1	CC(=O)c1sc(C(C)(C)C)cc1NC(=O)CCC(=O)O	nan
	4356534	50534	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	441	7	1	6	4.4	COc1ccc2nc(Cl)c(C3CC(c4ccco4)=NN3C(=O)CCCC(=O)O)cc2c1	nan
	CHEMBL1576687	50534	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	441	7	1	6	4.4	COc1ccc2nc(Cl)c(C3CC(c4ccco4)=NN3C(=O)CCCC(=O)O)cc2c1	nan
	22517522	50657	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	396	6	1	7	2.1	CC(Oc1ccccc1)C(=O)Nc1nnc(S(=O)(=O)N2CCCCC2)s1	nan
	CHEMBL1577822	50657	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	396	6	1	7	2.1	CC(Oc1ccccc1)C(=O)Nc1nnc(S(=O)(=O)N2CCCCC2)s1	nan
	20856926	50847	0	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	336	5	2	4	3.0	CC(=O)c1cccc(NC(=O)CNC(=O)c2cc3ccccc3o2)c1	nan
	CHEMBL1579387	50847	0	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	336	5	2	4	3.0	CC(=O)c1cccc(NC(=O)CNC(=O)c2cc3ccccc3o2)c1	nan
	4368409	50938	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	8	1	8	4.7	CCCCOc1cccc(C2C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2c2nnc(C)s2)c1	nan
	CHEMBL1580198	50938	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	8	1	8	4.7	CCCCOc1cccc(C2C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2c2nnc(C)s2)c1	nan
	990451	51003	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	5	0	7	3.2	Cc1ccc(-n2nc3c(SCCN4CCOCC4)nnc(C)c3c2C)cc1	nan
	CHEMBL1580766	51003	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	5	0	7	3.2	Cc1ccc(-n2nc3c(SCCN4CCOCC4)nnc(C)c3c2C)cc1	nan
	661914	51090	18	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	6	1	8	3.7	COc1ccc(C2C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2c2cc(C)on2)cc1OC	nan
	CHEMBL1581469	51090	18	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	6	1	8	3.7	COc1ccc(C2C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2c2cc(C)on2)cc1OC	nan
	679340	51102	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	258	1	2	6	1.8	Cc1ccc(C2C(C#N)=C(N)SC(N)=C2C#N)o1	nan
	CHEMBL1581638	51102	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	258	1	2	6	1.8	Cc1ccc(C2C(C#N)=C(N)SC(N)=C2C#N)o1	nan
	990454	51121	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	5	0	7	3.0	Cc1nnc(SCCN2CCOCC2)c2nn(-c3ccccc3F)c(C)c12	nan
	CHEMBL1581794	51121	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	5	0	7	3.0	Cc1nnc(SCCN2CCOCC2)c2nn(-c3ccccc3F)c(C)c12	nan
	2666708	51167	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	5	1	7	3.3	COc1cc(C(=O)Nc2nc3ccc(S(C)(=O)=O)cc3s2)cc(OC)c1C	nan
	CHEMBL1582108	51167	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	5	1	7	3.3	COc1cc(C(=O)Nc2nc3ccc(S(C)(=O)=O)cc3s2)cc(OC)c1C	nan
	1943119	51442	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	8	0	10	2.9	COCCn1c(-c2cc(OC)c(OC)c(OC)c2)nc2oc3cc(OC)ccc3c(=O)c2c1=O	nan
	CHEMBL1584456	51442	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	8	0	10	2.9	COCCn1c(-c2cc(OC)c(OC)c(OC)c2)nc2oc3cc(OC)ccc3c(=O)c2c1=O	nan
	5923696	51621	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	4	1	9	-0.3	N#C/C(=C\c1c(N2CCOCC2)nc2ccccn2c1=O)C(=O)NC1CCS(=O)(=O)C1	nan
	CHEMBL1585817	51621	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	4	1	9	-0.3	N#C/C(=C\c1c(N2CCOCC2)nc2ccccn2c1=O)C(=O)NC1CCS(=O)(=O)C1	nan
	11957204	51668	10	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	373	4	1	5	5.1	O=C(Nc1nccs1)c1cc2sccc2n1Cc1ccc(Cl)cc1	nan
	CHEMBL1586282	51668	10	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	373	4	1	5	5.1	O=C(Nc1nccs1)c1cc2sccc2n1Cc1ccc(Cl)cc1	nan
	2534667	51680	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	300	5	0	6	2.4	COc1ccc(C(C)=O)cc1COC(=O)c1cnc(C)cn1	nan
	CHEMBL1586370	51680	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	300	5	0	6	2.4	COc1ccc(C(C)=O)cc1COC(=O)c1cnc(C)cn1	nan
	2048070	51684	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	4	2	4	4.0	Cc1ccc(NC(=O)CSc2nc3cc(Br)c[nH]c-3n2)cc1C	nan
	CHEMBL1586414	51684	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	4	2	4	4.0	Cc1ccc(NC(=O)CSc2nc3cc(Br)c[nH]c-3n2)cc1C	nan
	4382155	51730	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	6	1	4	2.7	CCc1ccccc1NC(=O)CCCN1C(=O)c2cccnc2C1=O	nan
	CHEMBL1586776	51730	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	6	1	4	2.7	CCc1ccccc1NC(=O)CCCN1C(=O)c2cccnc2C1=O	nan
	3548898	51764	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	440	4	2	6	1.7	CC(=O)N1CCc2c(sc(NC(=O)c3cccc(N4C(=O)CCC4=O)c3)c2C(N)=O)C1	nan
	CHEMBL1587022	51764	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	440	4	2	6	1.7	CC(=O)N1CCc2c(sc(NC(=O)c3cccc(N4C(=O)CCC4=O)c3)c2C(N)=O)C1	nan
	3565925	51835	18	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	310	3	1	5	2.9	COCCn1c(=S)[nH]c2sc3c(c2c1=O)CCC(C)C3	nan
	CHEMBL1587609	51835	18	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	310	3	1	5	2.9	COCCn1c(=S)[nH]c2sc3c(c2c1=O)CCC(C)C3	nan
	661736	51854	14	None	-1	3	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	4	0	6	3.5	Cc1ccccc1N1C(=O)CC(Sc2nnc(-c3ccccc3)o2)C1=O	nan
	CHEMBL1587764	51854	14	None	-1	3	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	4	0	6	3.5	Cc1ccccc1N1C(=O)CC(Sc2nnc(-c3ccccc3)o2)C1=O	nan
	5919084	51907	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	482	7	1	7	2.9	O=C(C1=C(O)C(=O)N(CCCN2CCOCC2)C1c1ccc(F)cc1)c1ccc2c(c1)OCCO2	nan
	CHEMBL1588231	51907	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	482	7	1	7	2.9	O=C(C1=C(O)C(=O)N(CCCN2CCOCC2)C1c1ccc(F)cc1)c1ccc2c(c1)OCCO2	nan
	859793	51935	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	4	0	9	-0.6	Cn1c(=O)c2c(nc(SCCN3CCOCC3)n2C)n(C)c1=O	nan
	CHEMBL1588519	51935	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	4	0	9	-0.6	Cn1c(=O)c2c(nc(SCCN3CCOCC3)n2C)n(C)c1=O	nan
	4203923	52005	15	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	454	9	1	7	4.4	CCN(CC)CCN1C(=O)C(O)=C(C(=O)c2cc3cccc(OC)c3o2)C1c1cccs1	nan
	4573010	52005	15	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	454	9	1	7	4.4	CCN(CC)CCN1C(=O)C(O)=C(C(=O)c2cc3cccc(OC)c3o2)C1c1cccs1	nan
	CHEMBL1589149	52005	15	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	454	9	1	7	4.4	CCN(CC)CCN1C(=O)C(O)=C(C(=O)c2cc3cccc(OC)c3o2)C1c1cccs1	nan
	16016946	52086	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	3	1	5	4.5	Cc1c(Cl)cccc1NC(=O)Cn1nc(C)c2sc3ccccc3c2c1=O	nan
	CHEMBL1589855	52086	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	3	1	5	4.5	Cc1c(Cl)cccc1NC(=O)Cn1nc(C)c2sc3ccccc3c2c1=O	nan
	16014998	52088	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	332	4	1	5	4.8	CSc1nc(Nc2ccc(C)cc2)c(C#N)c(-c2ccccc2)n1	nan
	CHEMBL1589876	52088	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	332	4	1	5	4.8	CSc1nc(Nc2ccc(C)cc2)c(C#N)c(-c2ccccc2)n1	nan
	16017572	52100	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	6	1	6	1.7	CCC(=O)Nc1nnc(S(=O)(=O)N(C)Cc2ccccc2)s1	nan
	CHEMBL1589962	52100	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	6	1	6	1.7	CCC(=O)Nc1nnc(S(=O)(=O)N(C)Cc2ccccc2)s1	nan
	16019870	52105	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	481	8	1	6	4.8	COc1ccc(OC)c(NC(=O)CSc2cn(CC(=O)N3CCCCCC3)c3ccccc23)c1	nan
	CHEMBL1590046	52105	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	481	8	1	6	4.8	COc1ccc(OC)c(NC(=O)CSc2cn(CC(=O)N3CCCCCC3)c3ccccc23)c1	nan
	8070199	52117	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	8	1	7	3.5	Cn1nnnc1SCCCNCc1ccc(-c2ccc(Br)cc2)o1	nan
	CHEMBL1590182	52117	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	8	1	7	3.5	Cn1nnnc1SCCCNCc1ccc(-c2ccc(Br)cc2)o1	nan
	1252599	52136	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	356	4	1	7	1.9	COC(=O)c1cc(CN2C(=O)c3ccccc3C2=O)c(O)c([N+](=O)[O-])c1	nan
	CHEMBL1590469	52136	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	356	4	1	7	1.9	COC(=O)c1cc(CN2C(=O)c3ccccc3C2=O)c(O)c([N+](=O)[O-])c1	nan
	3438312	52155	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	5	2	5	3.3	COc1ccccc1Cn1c(=S)[nH]c2cc(C(=O)NC(C)C)ccc2c1=O	nan
	CHEMBL1590737	52155	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	5	2	5	3.3	COc1ccccc1Cn1c(=S)[nH]c2cc(C(=O)NC(C)C)ccc2c1=O	nan
	8391566	52183	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	304	3	0	7	2.5	Cc1nnc(SCc2cc(=O)n3c(C)cccc3n2)s1	nan
	CHEMBL1590986	52183	7	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	304	3	0	7	2.5	Cc1nnc(SCc2cc(=O)n3c(C)cccc3n2)s1	nan
	16017932	52210	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	477	4	1	6	5.8	CCN(CC)c1ccc2cc(-c3nc4sc5c(c4c(=O)[nH]3)CCC(C(C)(C)C)C5)c(=O)oc2c1	nan
	CHEMBL1591378	52210	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	477	4	1	6	5.8	CCN(CC)c1ccc2cc(-c3nc4sc5c(c4c(=O)[nH]3)CCC(C(C)(C)C)C5)c(=O)oc2c1	nan
	7152123	52308	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	6	1	6	4.3	COc1ccc(-c2cn3nc(SCC(=O)Nc4ccccc4F)ccc3n2)cc1	nan
	CHEMBL1592684	52308	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	6	1	6	4.3	COc1ccc(-c2cn3nc(SCC(=O)Nc4ccccc4F)ccc3n2)cc1	nan
	20885677	52332	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	325	6	1	6	1.3	Cc1nn(CCCC(=O)NCc2ccccc2)c(=O)c2nccn12	nan
	CHEMBL1592977	52332	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	325	6	1	6	1.3	Cc1nn(CCCC(=O)NCc2ccccc2)c(=O)c2nccn12	nan
	16403621	52335	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	467	7	1	7	3.0	COc1ccc(OC)c(/C=C2\Oc3cc(OCC(=O)N4CCC(C(=O)O)CC4)ccc3C2=O)c1	nan
	CHEMBL1593051	52335	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	467	7	1	7	3.0	COc1ccc(OC)c(/C=C2\Oc3cc(OCC(=O)N4CCC(C(=O)O)CC4)ccc3C2=O)c1	nan
	20893093	52344	0	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	3	1	7	3.0	Cc1cc(=O)n2nc(N3CCCC3C(=O)Nc3cccc(Cl)c3C)sc2n1	nan
	CHEMBL1593179	52344	0	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	3	1	7	3.0	Cc1cc(=O)n2nc(N3CCCC3C(=O)Nc3cccc(Cl)c3C)sc2n1	nan
	16018628	52404	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	396	4	0	7	5.4	Cc1oc(-c2ccccc2Cl)nc1CSc1nncn2c1cc1occc12	nan
	CHEMBL1594061	52404	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	396	4	0	7	5.4	Cc1oc(-c2ccccc2Cl)nc1CSc1nncn2c1cc1occc12	nan
	16025303	52555	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	550	7	1	6	5.2	Cc1ccc(CNC(=O)CSc2ncc3c(n2)-c2ccc(Cl)cc2N(Cc2ccccc2)S3(=O)=O)cc1	nan
	CHEMBL1595335	52555	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	550	7	1	6	5.2	Cc1ccc(CNC(=O)CSc2ncc3c(n2)-c2ccc(Cl)cc2N(Cc2ccccc2)S3(=O)=O)cc1	nan
	5310070	52563	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	315	5	0	8	1.8	CCOC(=O)CSc1ccc2nnc(-c3cccnc3)n2n1	nan
	CHEMBL1595390	52563	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	315	5	0	8	1.8	CCOC(=O)CSc1ccc2nnc(-c3cccnc3)n2n1	nan
	15991139	52595	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	363	5	0	4	5.2	CCC(C)OC(=O)/C(C#N)=C\c1ccc(-c2cccc(C(F)(F)F)c2)o1	nan
	CHEMBL1595672	52595	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	363	5	0	4	5.2	CCC(C)OC(=O)/C(C#N)=C\c1ccc(-c2cccc(C(F)(F)F)c2)o1	nan
	5135766	52687	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	4	1	3	5.0	O=C(COc1ccc2oc3c(c2c1)CCCC3)Nc1ccc(Cl)cc1	nan
	CHEMBL1596555	52687	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	4	1	3	5.0	O=C(COc1ccc2oc3c(c2c1)CCCC3)Nc1ccc(Cl)cc1	nan
	3653425	52776	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	8	1	7	3.7	COC(=O)c1ccc(C2C(C(=O)c3cc4ccccc4o3)=C(O)C(=O)N2CCCN(C)C)cc1	nan
	661006	52776	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	8	1	7	3.7	COC(=O)c1ccc(C2C(C(=O)c3cc4ccccc4o3)=C(O)C(=O)N2CCCN(C)C)cc1	nan
	CHEMBL1597383	52776	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	8	1	7	3.7	COC(=O)c1ccc(C2C(C(=O)c3cc4ccccc4o3)=C(O)C(=O)N2CCCN(C)C)cc1	nan
	2991609	52780	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	7	2	4	1.6	Cc1ccc(OCC(=O)NCCNC(=O)c2cccnc2)cc1C	nan
	CHEMBL1597415	52780	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	7	2	4	1.6	Cc1ccc(OCC(=O)NCCNC(=O)c2cccnc2)cc1C	nan
	20893092	52839	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	3	1	7	2.4	Cc1cc(=O)n2nc(N3CCCC3C(=O)Nc3ccccc3C)sc2n1	nan
	CHEMBL1597947	52839	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	3	1	7	2.4	Cc1cc(=O)n2nc(N3CCCC3C(=O)Nc3ccccc3C)sc2n1	nan
	44666769	52861	20	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	318	4	2	6	0.9	Cc1cc(=O)oc2c(CN3CCN(CCO)CC3)c(O)ccc12	nan
	5289738	52861	20	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	318	4	2	6	0.9	Cc1cc(=O)oc2c(CN3CCN(CCO)CC3)c(O)ccc12	nan
	CHEMBL1598157	52861	20	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	318	4	2	6	0.9	Cc1cc(=O)oc2c(CN3CCN(CCO)CC3)c(O)ccc12	nan
	5310246	52872	9	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	4	1	6	4.0	COc1ccc(-c2cn3c(C)c(C(=O)Nc4ccncc4)sc3n2)cc1	nan
	CHEMBL1598249	52872	9	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	4	1	6	4.0	COc1ccc(-c2cn3c(C)c(C(=O)Nc4ccncc4)sc3n2)cc1	nan
	2807627	52927	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	217	1	0	5	1.4	CC1CCCN(c2ccc3nncn3n2)C1	nan
	CHEMBL1598761	52927	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	217	1	0	5	1.4	CC1CCCN(c2ccc3nncn3n2)C1	nan
	22514515	53011	1	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	5	0	7	0.9	CCOC(=O)C1CCN(C(=O)Cn2nc(CC)n3cccc3c2=O)CC1	nan
	CHEMBL1599442	53011	1	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	5	0	7	0.9	CCOC(=O)C1CCN(C(=O)Cn2nc(CC)n3cccc3c2=O)CC1	nan
	2913046	53197	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	442	5	1	5	5.1	Cc1ccc(C(=O)C2=C(O)C(=O)N(Cc3cccnc3)C2c2ccc(Cl)c(Cl)c2)o1	nan
	CHEMBL1601179	53197	14	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	442	5	1	5	5.1	Cc1ccc(C(=O)C2=C(O)C(=O)N(Cc3cccnc3)C2c2ccc(Cl)c(Cl)c2)o1	nan
	3152554	53224	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	5	1	5	4.3	O=C(C1=C(O)C(=O)N(CC2CCCO2)C1c1ccc(Cl)cc1Cl)c1ccco1	nan
	CHEMBL1601448	53224	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	5	1	5	4.3	O=C(C1=C(O)C(=O)N(CC2CCCO2)C1c1ccc(Cl)cc1Cl)c1ccco1	nan
	3733422	53270	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	5	1	6	4.2	COc1ccc(C2C(C(=O)c3cccs3)=C(O)C(=O)N2c2cccc(C)n2)cc1	nan
	CHEMBL1602024	53270	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	5	1	6	4.2	COc1ccc(C2C(C(=O)c3cccs3)=C(O)C(=O)N2c2cccc(C)n2)cc1	nan
	3185717	53273	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	550	9	3	8	3.2	Cc1cccc(N(C(=O)c2snc(C(N)=O)c2N)C(C(=O)NCC2CCCO2)c2ccc(N(C)C)cc2)c1C	nan
	CHEMBL1602063	53273	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	550	9	3	8	3.2	Cc1cccc(N(C(=O)c2snc(C(N)=O)c2N)C(C(=O)NCC2CCCO2)c2ccc(N(C)C)cc2)c1C	nan
	1541054	53600	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	6	1	5	4.3	CCOc1cccc(NC(=O)CSc2nc(C)c3c(c2C#N)CCCC3)c1	nan
	CHEMBL1604887	53600	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	6	1	5	4.3	CCOc1cccc(NC(=O)CSc2nc(C)c3c(c2C#N)CCCC3)c1	nan
	20885689	53665	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	7	1	7	1.3	COc1ccc(CNC(=O)CCCn2nc(C)n3ccnc3c2=O)cc1	nan
	CHEMBL1605440	53665	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	7	1	7	1.3	COc1ccc(CNC(=O)CCCn2nc(C)n3ccnc3c2=O)cc1	nan
	2890303	53764	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	3	1	4	2.7	CC(=O)C1=C(O)C(=O)N(c2ccccn2)C1c1cccc(F)c1	nan
	CHEMBL1606210	53764	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	3	1	4	2.7	CC(=O)C1=C(O)C(=O)N(c2ccccn2)C1c1cccc(F)c1	nan
	16030495	53805	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	6	1	4	5.9	Cc1ccc(Cl)cc1NC(=O)CSc1nc2ccccc2nc1Cc1ccccc1	nan
	CHEMBL1606531	53805	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	6	1	4	5.9	Cc1ccc(Cl)cc1NC(=O)CSc1nc2ccccc2nc1Cc1ccccc1	nan
	855274	53937	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	269	2	0	5	2.0	COc1ccc2cc(C#N)c(N3CCOCC3)nc2c1	nan
	CHEMBL1607471	53937	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	269	2	0	5	2.0	COc1ccc2cc(C#N)c(N3CCOCC3)nc2c1	nan
	3663093	53961	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	490	6	2	8	4.6	CCc1nnc(NC(=O)CSc2nc3c([nH]c4ccccc43)c(=O)n2-c2cc(C)cc(C)c2)s1	nan
	CHEMBL1607685	53961	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	490	6	2	8	4.6	CCc1nnc(NC(=O)CSc2nc3c([nH]c4ccccc43)c(=O)n2-c2cc(C)cc(C)c2)s1	nan
	889917	54062	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	275	5	1	3	3.7	CCc1c(SCCC(=O)O)nc2ccccc2c1C	nan
	CHEMBL1608598	54062	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	275	5	1	3	3.7	CCc1c(SCCC(=O)O)nc2ccccc2c1C	nan
	7120053	54213	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	308	1	1	4	4.1	Cc1cccc(-n2c(=S)[nH]c3c(oc4ccccc43)c2=O)c1	nan
	CHEMBL1609827	54213	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	308	1	1	4	4.1	Cc1cccc(-n2c(=S)[nH]c3c(oc4ccccc43)c2=O)c1	nan
	2371304	54252	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	5	1	6	2.8	O=C(CSc1ncnc2ccccc12)NCc1ccc2c(c1)OCO2	nan
	CHEMBL1610145	54252	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	5	1	6	2.8	O=C(CSc1ncnc2ccccc12)NCc1ccc2c(c1)OCO2	nan
	4380426	54299	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	3	1	4	4.3	O=C(Nc1nnc(-c2ccccc2Cl)s1)c1ccccc1F	nan
	CHEMBL1610533	54299	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	3	1	4	4.3	O=C(Nc1nnc(-c2ccccc2Cl)s1)c1ccccc1F	nan
	2813334	54383	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	4	0	6	3.2	CCOC(=O)C1CCCN(C(=O)c2csc(-c3ccc4c(c3)CCO4)n2)C1	nan
	CHEMBL1611317	54383	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	4	0	6	3.2	CCOC(=O)C1CCCN(C(=O)c2csc(-c3ccc4c(c3)CCO4)n2)C1	nan
	16014906	54429	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	292	3	1	2	3.7	Cc1ccc(CNC(=O)c2cc3cc(C)ccc3n2C)cc1	nan
	CHEMBL1611737	54429	5	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	292	3	1	2	3.7	Cc1ccc(CNC(=O)c2cc3cc(C)ccc3n2C)cc1	nan
	4853715	54440	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	3	1	5	3.6	CC(=O)c1sc(NC(=O)c2cnc(Cl)c(Cl)c2)nc1C	nan
	CHEMBL1611812	54440	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	3	1	5	3.6	CC(=O)c1sc(NC(=O)c2cnc(Cl)c(Cl)c2)nc1C	nan
	16009370	54453	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	4	0	5	5.3	O=c1cc(COc2ccc(Cl)cc2Cl)nc2scc(-c3ccccc3)n12	nan
	CHEMBL1611935	54453	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	4	0	5	5.3	O=c1cc(COc2ccc(Cl)cc2Cl)nc2scc(-c3ccccc3)n12	nan
	24892471	54750	0	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	9	1	5	6.4	CCCCNc1c(-c2ccc(SC(C)CC)c(OC)c2)nc2ccc(C)cn12	nan
	CHEMBL1356182	54750	0	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	9	1	5	6.4	CCCCNc1c(-c2ccc(SC(C)CC)c(OC)c2)nc2ccc(C)cn12	nan
	CHEMBL1616404	54750	0	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	9	1	5	6.4	CCCCNc1c(-c2ccc(SC(C)CC)c(OC)c2)nc2ccc(C)cn12	nan
	24789689	55108	0	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	325	4	2	4	3.3	CC(=O)Nc1ccc(-c2sc(Nc3ccccc3)n[n+]2C)cc1	nan
	CHEMBL1395742	55108	0	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	325	4	2	4	3.3	CC(=O)Nc1ccc(-c2sc(Nc3ccccc3)n[n+]2C)cc1	nan
	CHEMBL1619301	55108	0	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	325	4	2	4	3.3	CC(=O)Nc1ccc(-c2sc(Nc3ccccc3)n[n+]2C)cc1	nan
	6489920	55254	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	264	3	0	2	3.1	CCn1c(/C=C/c2cc[n+](C)cc2)nc2ccccc21	nan
	CHEMBL1428082	55254	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	264	3	0	2	3.1	CCn1c(/C=C/c2cc[n+](C)cc2)nc2ccccc21	nan
	CHEMBL1620517	55254	4	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	264	3	0	2	3.1	CCn1c(/C=C/c2cc[n+](C)cc2)nc2ccccc21	nan
	5064206	55301	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	4	0	4	4.9	Cc1cc[n+]2cc(-c3cccc([N+](=O)[O-])c3)c(-c3cccc([N+](=O)[O-])c3)cc2c1	nan
	CHEMBL1455685	55301	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	4	0	4	4.9	Cc1cc[n+]2cc(-c3cccc([N+](=O)[O-])c3)c(-c3cccc([N+](=O)[O-])c3)cc2c1	nan
	CHEMBL1621049	55301	6	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	4	0	4	4.9	Cc1cc[n+]2cc(-c3cccc([N+](=O)[O-])c3)c(-c3cccc([N+](=O)[O-])c3)cc2c1	nan
	820476	55554	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	195	0	1	1	2.2	Nc1ccc2ccc3cccc[n+]3c2c1	nan
	CHEMBL1522563	55554	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	195	0	1	1	2.2	Nc1ccc2ccc3cccc[n+]3c2c1	nan
	CHEMBL1623170	55554	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	195	0	1	1	2.2	Nc1ccc2ccc3cccc[n+]3c2c1	nan
	1560419	55558	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	7	2	4	3.4	O=C(O)CCCCCNc1ncnc2ccc(Br)cc12	nan
	CHEMBL1517106	55558	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	7	2	4	3.4	O=C(O)CCCCCNc1ncnc2ccc(Br)cc12	nan
	CHEMBL1623202	55558	16	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	7	2	4	3.4	O=C(O)CCCCCNc1ncnc2ccc(Br)cc12	nan
	1567753	55570	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	336	7	1	5	3.7	COc1ccc(-c2nc(NCCCN(C)C)c3ccccc3n2)cc1	nan
	CHEMBL1534121	55570	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	336	7	1	5	3.7	COc1ccc(-c2nc(NCCCN(C)C)c3ccccc3n2)cc1	nan
	CHEMBL1623318	55570	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	336	7	1	5	3.7	COc1ccc(-c2nc(NCCCN(C)C)c3ccccc3n2)cc1	nan
	818329	55734	28	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	331	2	1	4	4.0	Sc1nnc(-c2ccc(Br)cc2)n1-c1ccccc1	nan
	CHEMBL1568356	55734	28	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	331	2	1	4	4.0	Sc1nnc(-c2ccc(Br)cc2)n1-c1ccccc1	nan
	CHEMBL1624703	55734	28	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	331	2	1	4	4.0	Sc1nnc(-c2ccc(Br)cc2)n1-c1ccccc1	nan
	3146476	69468	5	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	2	0	2	4.9	CCN1C(=Cc2sc3ccccc3[n+]2C)C=Cc2cccc(C)c21	nan
	5767654	69468	5	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	2	0	2	4.9	CCN1C(=Cc2sc3ccccc3[n+]2C)C=Cc2cccc(C)c21	nan
	6248042	69468	5	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	2	0	2	4.9	CCN1C(=Cc2sc3ccccc3[n+]2C)C=Cc2cccc(C)c21	nan
	CHEMBL193627	69468	5	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	2	0	2	4.9	CCN1C(=Cc2sc3ccccc3[n+]2C)C=Cc2cccc(C)c21	nan
	CHEMBL584458	69468	5	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	2	0	2	4.9	CCN1C(=Cc2sc3ccccc3[n+]2C)C=Cc2cccc(C)c21	nan
	2152519	71643	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	512	7	0	9	3.6	CCOC(=O)c1cc2c(=O)n3ccccc3nc2n(Cc2ccco2)/c1=N/C(=O)c1ccccc1OCC	nan
	CHEMBL1973861	71643	11	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	512	7	0	9	3.6	CCOC(=O)c1cc2c(=O)n3ccccc3nc2n(Cc2ccco2)/c1=N/C(=O)c1ccccc1OCC	nan
	2003230	71897	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	398	5	0	8	1.2	CCOC(=O)c1cc2c(=O)n3cccc(C)c3nc2n(CCOC)/c1=N\C(C)=O	nan
	CHEMBL1981685	71897	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	398	5	0	8	1.2	CCOC(=O)c1cc2c(=O)n3cccc(C)c3nc2n(CCOC)/c1=N\C(C)=O	nan
	9580624	72045	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	302	6	1	7	2.5	COc1cccc(/C=N/Nc2ncccc2[N+](=O)[O-])c1OC	nan
	CHEMBL1986514	72045	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	302	6	1	7	2.5	COc1cccc(/C=N/Nc2ncccc2[N+](=O)[O-])c1OC	nan
	9564678	72189	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	5	1	9	-0.4	COc1ccc(/C=N/NC(=O)Cn2cnc3c2c(=O)n(C)c(=O)n3C)cc1	nan
	CHEMBL1991163	72189	12	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	5	1	9	-0.4	COc1ccc(/C=N/NC(=O)Cn2cnc3c2c(=O)n(C)c(=O)n3C)cc1	nan
	135406177	72213	5	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	279	2	2	4	3.6	Cc1ccc(O)c(/N=C/C2=C(O)c3ccccc3C2=O)c1	nan
	CHEMBL1991885	72213	5	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	279	2	2	4	3.6	Cc1ccc(O)c(/N=C/C2=C(O)c3ccccc3C2=O)c1	nan
	9583975	72300	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	5	2	6	5.8	Nc1c(C(=O)N/N=C/c2ccccc2Cl)oc2nc(-c3ccccc3)cc(-c3ccco3)c12	nan
	CHEMBL1995041	72300	2	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	5	2	6	5.8	Nc1c(C(=O)N/N=C/c2ccccc2Cl)oc2nc(-c3ccccc3)cc(-c3ccco3)c12	nan
	5936993	72471	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	6	0	2	6.9	CCN(CC)c1ccc(/C=C/c2cc(-c3ccccc3)c3ccccc3n2)cc1	nan
	CHEMBL2001294	72471	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	6	0	2	6.9	CCN(CC)c1ccc(/C=C/c2cc(-c3ccccc3)c3ccccc3n2)cc1	nan
	735993	87582	36	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	253	2	1	4	3.1	CN(C)c1ccc(-c2nc3cc(N)ccc3o2)cc1	nan
	CHEMBL234378	87582	36	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	253	2	1	4	3.1	CN(C)c1ccc(-c2nc3cc(N)ccc3o2)cc1	nan
	9638128	107267	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	330	7	0	5	3.4	CCN(CC)c1ccc(C(=O)c2cnc(/N=C/N(C)C)s2)cc1	nan
	CHEMBL3191439	107267	13	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	330	7	0	5	3.4	CCN(CC)c1ccc(C(=O)c2cnc(/N=C/N(C)C)s2)cc1	nan
	24892228	107371	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	464	9	0	8	2.7	COCCn1/c(=N\C(=O)CCS(=O)(=O)c2ccccc2)sc2c(OC)ccc(OC)c21	nan
	CHEMBL3192568	107371	8	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	464	9	0	8	2.7	COCCn1/c(=N\C(=O)CCS(=O)(=O)c2ccccc2)sc2c(OC)ccc(OC)c21	nan
	46497908	107531	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	6	1	10	0.2	Cn1c(=O)c2c(ncn2CC(=O)N/N=C/C=C\c2ccccc2[N+](=O)[O-])n(C)c1=O	nan
	CHEMBL3194459	107531	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	6	1	10	0.2	Cn1c(=O)c2c(ncn2CC(=O)N/N=C/C=C\c2ccccc2[N+](=O)[O-])n(C)c1=O	nan
	135412189	107756	9	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	320	5	3	10	1.0	COc1cc(/C=N/Nc2nc(O)nnc2C)cc([N+](=O)[O-])c1O	nan
	CHEMBL3197005	107756	9	None	-2	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	320	5	3	10	1.0	COc1cc(/C=N/Nc2nc(O)nnc2C)cc([N+](=O)[O-])c1O	nan
	4122444	108020	11	None	-8	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	310	3	0	6	2.4	CCOC(=O)c1s/c(=N\C(=O)c2cccs2)n(C)c1C	nan
	CHEMBL3199794	108020	11	None	-8	2	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	310	3	0	6	2.4	CCOC(=O)c1s/c(=N\C(=O)c2cccs2)n(C)c1C	nan
	5343366	108025	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	263	4	0	7	1.8	CSc1nncn1/N=C/c1ccc([N+](=O)[O-])cc1	nan
	CHEMBL3199842	108025	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	263	4	0	7	1.8	CSc1nncn1/N=C/c1ccc([N+](=O)[O-])cc1	nan
	135411619	108035	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	331	4	1	8	1.5	Cc1nn(-c2ccc([N+](=O)[O-])cc2)c(O)c1/C=N/N1CCOCC1	nan
	CHEMBL3199911	108035	9	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	331	4	1	8	1.5	Cc1nn(-c2ccc([N+](=O)[O-])cc2)c(O)c1/C=N/N1CCOCC1	nan
	9955	141805	95	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	135	0	2	4	-0.1	Nc1nc2ncnc-2c[nH]1	nan
	CHEMBL1356616	141805	95	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	135	0	2	4	-0.1	Nc1nc2ncnc-2c[nH]1	nan
	CHEMBL388594	141805	95	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	135	0	2	4	-0.1	Nc1nc2ncnc-2c[nH]1	nan
	154730799	167115	40	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	558	8	1	7	4.0	CCN(CC)c1ccc2c(-c3ccc(S(=O)(=O)O)cc3S(=O)(=O)[O-])c3ccc(=[N+](CC)CC)cc-3oc2c1	nan
	65191	167115	40	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	558	8	1	7	4.0	CCN(CC)c1ccc2c(-c3ccc(S(=O)(=O)O)cc3S(=O)(=O)[O-])c3ccc(=[N+](CC)CC)cc-3oc2c1	nan
	CHEMBL1306565	167115	40	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	558	8	1	7	4.0	CCN(CC)c1ccc2c(-c3ccc(S(=O)(=O)O)cc3S(=O)(=O)[O-])c3ccc(=[N+](CC)CC)cc-3oc2c1	nan
	CHEMBL4302011	167115	40	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	558	8	1	7	4.0	CCN(CC)c1ccc2c(-c3ccc(S(=O)(=O)O)cc3S(=O)(=O)[O-])c3ccc(=[N+](CC)CC)cc-3oc2c1	nan
	21551	183668	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	284	2	0	6	0.6	Cn1c(=O)c2c(nc(Cc3ccccc3)n2C)n(C)c1=O	nan
	CHEMBL483661	183668	3	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	284	2	0	6	0.6	Cn1c(=O)c2c(nc(Cc3ccccc3)n2C)n(C)c1=O	nan
	4380636	199321	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	4	1	4	5.3	CC(C)c1ccc(Nc2c(-c3ccccn3)nc3ccccn23)cc1	nan
	CHEMBL602150	199321	10	None	-	1	Human	4.6	pPotency	=	4.6	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	4	1	4	5.3	CC(C)c1ccc(Nc2c(-c3ccccn3)nc3ccccn23)cc1	nan
	1499	2060	43	None	-31622	36	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	211	4	4	4	1.1	CC(NCC(c1ccc(c(c1)O)O)O)C	nan
	3779	2060	43	None	-31622	36	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	211	4	4	4	1.1	CC(NCC(c1ccc(c(c1)O)O)O)C	nan
	536	2060	43	None	-31622	36	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	211	4	4	4	1.1	CC(NCC(c1ccc(c(c1)O)O)O)C	nan
	CHEMBL434	2060	43	None	-31622	36	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	211	4	4	4	1.1	CC(NCC(c1ccc(c(c1)O)O)O)C	nan
	DB01064	2060	43	None	-31622	36	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	211	4	4	4	1.1	CC(NCC(c1ccc(c(c1)O)O)O)C	nan
	3762	14331	24	None	1	2	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	239	5	4	4	1.9	CCC(NC(C)C)C(O)c1ccc(O)c(O)c1	nan
	CHEMBL1201153	14331	24	None	1	2	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	239	5	4	4	1.9	CCC(NC(C)C)C(O)c1ccc(O)c(O)c1	nan
	CHEMBL1201213	14331	24	None	1	2	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	239	5	4	4	1.9	CCC(NC(C)C)C(O)c1ccc(O)c(O)c1	nan
	1214032	19562	13	None	-2	2	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	526	6	1	7	6.1	CC1(C)Cc2nc3sc4c(SCC(=O)NC(c5ccccc5)c5ccccc5)ncnc4c3cc2CO1	nan
	CHEMBL1301335	19562	13	None	-2	2	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	526	6	1	7	6.1	CC1(C)Cc2nc3sc4c(SCC(=O)NC(c5ccccc5)c5ccccc5)ncnc4c3cc2CO1	nan
	15990933	21573	6	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	5	2	3	6.2	CC(C)c1ccc(Nc2cc(C(=O)NC3CCCCC3)c3ccccc3n2)cc1	nan
	CHEMBL1319127	21573	6	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	5	2	3	6.2	CC(C)c1ccc(Nc2cc(C(=O)NC3CCCCC3)c3ccccc3n2)cc1	nan
	1716420	21872	14	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	558	4	1	5	6.5	COc1ccc(-c2cc(C(F)(F)F)n3nc(C(=O)Nc4cccc(C(F)(F)F)c4)c(Br)c3n2)cc1	nan
	CHEMBL1321710	21872	14	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	558	4	1	5	6.5	COc1ccc(-c2cc(C(F)(F)F)n3nc(C(=O)Nc4cccc(C(F)(F)F)c4)c(Br)c3n2)cc1	nan
	2919028	24169	15	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	498	7	1	10	3.9	COC(=O)c1sc(N2C(=O)C(O)=C(C(=O)c3ccc(C)o3)C2c2ccc(OC)c(OC)c2)nc1C	nan
	CHEMBL1341127	24169	15	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	498	7	1	10	3.9	COC(=O)c1sc(N2C(=O)C(O)=C(C(=O)c3ccc(C)o3)C2c2ccc(OC)c(OC)c2)nc1C	nan
	16019314	30684	12	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	485	5	1	9	4.9	COc1ccc(C)cc1Nc1nc2c(S(=O)(=O)c3cccc(Cl)c3)nnn2c2ccsc12	nan
	CHEMBL1397774	30684	12	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	485	5	1	9	4.9	COc1ccc(C)cc1Nc1nc2c(S(=O)(=O)c3cccc(Cl)c3)nnn2c2ccsc12	nan
	944832	31345	9	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	235	0	2	3	3.0	Sc1[nH]cnc2c3cc(Cl)ccc3nc1-2	nan
	CHEMBL1404042	31345	9	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	235	0	2	3	3.0	Sc1[nH]cnc2c3cc(Cl)ccc3nc1-2	nan
	4024853	31486	7	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	7	1	5	5.6	CCCOc1ccc(C(=O)Nc2ccc3oc(-c4ccc(N(C)C)cc4)nc3c2)cc1	nan
	CHEMBL1405437	31486	7	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	7	1	5	5.6	CCCOc1ccc(C(=O)Nc2ccc3oc(-c4ccc(N(C)C)cc4)nc3c2)cc1	nan
	24892224	33882	5	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	6	1	9	0.5	CC(C)c1nc(SCC(=O)NCC2CCCO2)c2c(=O)n(C)c(=O)n(C)c2n1	nan
	CHEMBL1425449	33882	5	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	6	1	9	0.5	CC(C)c1nc(SCC(=O)NCC2CCCO2)c2c(=O)n(C)c(=O)n(C)c2n1	nan
	16033262	36044	0	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	4	1	5	5.9	Cc1c(C(=O)Nc2ccc(Br)cc2F)sc2ncnc(N(C)C3CCCCC3)c12	nan
	CHEMBL1445708	36044	0	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	4	1	5	5.9	Cc1c(C(=O)Nc2ccc(Br)cc2F)sc2ncnc(N(C)C3CCCCC3)c12	nan
	4179349	39357	11	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	515	8	1	7	5.6	CCOC(=O)c1ccc(NC(=O)CSc2nc(-c3ccc(OC)cc3)cc(C(F)(F)F)c2C#N)cc1	nan
	CHEMBL1473745	39357	11	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	515	8	1	7	5.6	CCOC(=O)c1ccc(NC(=O)CSc2nc(-c3ccc(OC)cc3)cc(C(F)(F)F)c2C#N)cc1	nan
	2810065	42713	6	None	1	2	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	2	1	5	4.0	O=C(Nc1nc2c(Br)cc(Br)cc2c(=O)s1)c1ccco1	nan
	CHEMBL1503612	42713	6	None	1	2	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	2	1	5	4.0	O=C(Nc1nc2c(Br)cc(Br)cc2c(=O)s1)c1ccco1	nan
	16019583	43838	5	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	506	4	0	9	3.1	CCN1CCN(c2nc3c(S(=O)(=O)c4ccc(Br)cc4)nnn3c3ccsc23)CC1	nan
	CHEMBL1514816	43838	5	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	506	4	0	9	3.1	CCN1CCN(c2nc3c(S(=O)(=O)c4ccc(Br)cc4)nnn3c3ccsc23)CC1	nan
	16023031	44370	5	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	6	1	6	3.1	Cc1ccc(C(=O)Nc2nnc(S(=O)(=O)N(C)Cc3ccc(F)cc3)s2)cc1	nan
	CHEMBL1520434	44370	5	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	6	1	6	3.1	Cc1ccc(C(=O)Nc2nnc(S(=O)(=O)N(C)Cc3ccc(F)cc3)s2)cc1	nan
	16030551	47858	5	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	8	1	4	5.1	CC(C)CCNC(=O)CSc1nc2ccccc2nc1Cc1ccc(Cl)cc1	nan
	CHEMBL1551173	47858	5	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	8	1	4	5.1	CC(C)CCNC(=O)CSc1nc2ccccc2nc1Cc1ccc(Cl)cc1	nan
	16009713	53694	6	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	5	1	6	4.9	COc1ccc(-c2nnn3c2nc(NCc2ccc(C)cc2)c2ccccc23)cc1	nan
	CHEMBL1605623	53694	6	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	5	1	6	4.9	COc1ccc(-c2nnn3c2nc(NCc2ccc(C)cc2)c2ccccc23)cc1	nan
	49858523	89104	0	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	426	5	0	5	5.0	CCCC[C@]12Cc3cc(C#N)ccc3[C@H](O1)c1c(cc(C)n(Cc3ccccc3)c1=O)O2	nan
	CHEMBL2373613	89104	0	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	426	5	0	5	5.0	CCCC[C@]12Cc3cc(C#N)ccc3[C@H](O1)c1c(cc(C)n(Cc3ccccc3)c1=O)O2	nan
	16010255	5895	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	463	4	1	7	5.1	Cc1ccc(Nc2nc3c(S(=O)(=O)c4ccccc4)nnn3c3ccc(Cl)cc23)c(C)c1	nan
	CHEMBL1079970	5895	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	463	4	1	7	5.1	Cc1ccc(Nc2nc3c(S(=O)(=O)c4ccccc4)nnn3c3ccc(Cl)cc23)c(C)c1	nan
	16010278	6054	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	5	1	7	4.4	O=S(=O)(c1ccccc1)c1nnn2c1nc(NCc1ccccc1)c1cc(Cl)ccc12	nan
	CHEMBL1080898	6054	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	5	1	7	4.4	O=S(=O)(c1ccccc1)c1nnn2c1nc(NCc1ccccc1)c1cc(Cl)ccc12	nan
	18560284	6269	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	528	7	1	8	3.3	O=C1CCCN1CCCNc1nc2c(S(=O)(=O)c3ccc(Br)cc3)nnn2c2ccccc12	nan
	CHEMBL1082027	6269	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	528	7	1	8	3.3	O=C1CCCN1CCCNc1nc2c(S(=O)(=O)c3ccc(Br)cc3)nnn2c2ccccc12	nan
	16010337	6307	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	5	1	7	4.1	CCc1ccc(S(=O)(=O)c2nnn3c2nc(NC(C)C)c2cc(Cl)ccc23)cc1	nan
	CHEMBL1082207	6307	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	5	1	7	4.1	CCc1ccc(S(=O)(=O)c2nnn3c2nc(NC(C)C)c2cc(Cl)ccc23)cc1	nan
	7185123	10577	7	None	-851	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	4	1	8	3.9	O=S(=O)(c1ccccc1)c1nnn2c1nc(NC1CCCCC1)c1sccc12	nan
	CHEMBL1170673	10577	7	None	-851	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	4	1	8	3.9	O=S(=O)(c1ccccc1)c1nnn2c1nc(NC1CCCCC1)c1sccc12	nan
	16019553	10606	7	None	-912	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	479	6	1	8	4.4	CC(C)CCNc1nc2c(S(=O)(=O)c3ccc(Br)cc3)nnn2c2ccsc12	nan
	CHEMBL1170871	10606	7	None	-912	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	479	6	1	8	4.4	CC(C)CCNc1nc2c(S(=O)(=O)c3ccc(Br)cc3)nnn2c2ccsc12	nan
	16019312	10797	0	None	-144	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	441	5	1	9	4.2	Cc1ccc(S(=O)(=O)c2nnn3c2nc(NCc2cccs2)c2sccc23)cc1	nan
	CHEMBL1172727	10797	0	None	-144	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	441	5	1	9	4.2	Cc1ccc(S(=O)(=O)c2nnn3c2nc(NCc2cccs2)c2sccc23)cc1	nan
	4968664	19499	7	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	519	8	2	6	6.2	COc1cc(C(=O)Nc2nc(-c3cc(C)ccc3C)c(C)s2)ccc1OCC(=O)Nc1ccc(F)cc1	nan
	CHEMBL1300883	19499	7	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	519	8	2	6	6.2	COc1cc(C(=O)Nc2nc(-c3cc(C)ccc3C)c(C)s2)ccc1OCC(=O)Nc1ccc(F)cc1	nan
	16435505	19535	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	5	2	8	1.5	Cc1ccc2nc3c(cc(C(=O)NCC4CCCO4)c(=N)n3CC3CCCO3)c(=O)n2c1	nan
	CHEMBL1301161	19535	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	5	2	8	1.5	Cc1ccc2nc3c(cc(C(=O)NCC4CCCO4)c(=N)n3CC3CCCO3)c(=O)n2c1	nan
	1451395	19561	4	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	7	1	5	5.6	Cc1cccc(NC(=O)CSc2nc(COc3ccccc3)nc3ccccc23)c1C	nan
	CHEMBL1301326	19561	4	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	7	1	5	5.6	Cc1cccc(NC(=O)CSc2nc(COc3ccccc3)nc3ccccc23)c1C	nan
	1019237	19722	14	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	6	2	5	3.6	COc1ccccc1C(=O)Nc1cccc(NC(=O)c2ccccc2OC)n1	nan
	CHEMBL1302646	19722	14	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	6	2	5	3.6	COc1ccccc1C(=O)Nc1cccc(NC(=O)c2ccccc2OC)n1	nan
	1176215	19905	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	6	1	7	3.7	CCc1nnc(NC(=O)CSc2nc3cc(OC)ccc3cc2C)s1	nan
	CHEMBL1304139	19905	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	6	1	7	3.7	CCc1nnc(NC(=O)CSc2nc3cc(OC)ccc3cc2C)s1	nan
	706653	19911	12	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	309	1	1	5	3.5	N#Cc1c(-c2ccccc2)c(C#N)c2nc3ccccc3n2c1N	nan
	CHEMBL1304187	19911	12	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	309	1	1	5	3.5	N#Cc1c(-c2ccccc2)c(C#N)c2nc3ccccc3n2c1N	nan
	2060107	19957	7	None	-5	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	7	1	7	4.7	COc1ccc(NC(=O)CSc2nnc(-c3cccs3)n2-c2ccccc2)cc1	nan
	CHEMBL1304585	19957	7	None	-5	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	7	1	7	4.7	COc1ccc(NC(=O)CSc2nnc(-c3cccs3)n2-c2ccccc2)cc1	nan
	16034541	20168	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	6	1	6	3.5	CN(Cc1ccc(F)cc1)S(=O)(=O)c1nnc(NC(=O)c2ccccc2Br)s1	nan
	CHEMBL1306241	20168	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	6	1	6	3.5	CN(Cc1ccc(F)cc1)S(=O)(=O)c1nnc(NC(=O)c2ccccc2Br)s1	nan
	12005386	20250	6	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	7	1	6	4.7	CCCCOc1ccc(C(=O)Nn2c(-c3cccs3)nc3ccccc3c2=O)cc1	nan
	CHEMBL1306967	20250	6	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	7	1	6	4.7	CCCCOc1ccc(C(=O)Nn2c(-c3cccs3)nc3ccccc3c2=O)cc1	nan
	24818410	20502	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	6	0	6	4.2	COc1cccc(COC(=O)c2c(C)nn(-c3ccccc3)c2Cl)c1OC	nan
	CHEMBL1308959	20502	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	6	0	6	4.2	COc1cccc(COC(=O)c2c(C)nn(-c3ccccc3)c2Cl)c1OC	nan
	2081889	20775	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	7	1	7	4.1	Cc1sc2nc(SCC(=O)NCc3ccco3)n(Cc3ccccc3)c(=O)c2c1C	nan
	CHEMBL1311321	20775	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	7	1	7	4.1	Cc1sc2nc(SCC(=O)NCc3ccco3)n(Cc3ccccc3)c(=O)c2c1C	nan
	2102674	20801	5	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	6	1	7	3.6	Cc1cc(NC(=O)CSc2nc3ccccc3c(=O)n2Cc2ccc(F)cc2)no1	nan
	CHEMBL1311532	20801	5	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	6	1	7	3.6	Cc1cc(NC(=O)CSc2nc3ccccc3c(=O)n2Cc2ccc(F)cc2)no1	nan
	651309	21139	2	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	5	1	5	2.8	Cc1ccc2cc(C#N)c(SCC(=O)NCC3CCCO3)nc2c1	nan
	CHEMBL1314039	21139	2	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	5	1	5	2.8	Cc1ccc2cc(C#N)c(SCC(=O)NCC3CCCO3)nc2c1	nan
	16028453	21206	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	472	8	3	4	5.4	CCc1ccccc1NC(=O)Nc1cc(C(=O)NCc2ccc(OC)cc2)ccc1N1CCCC1	nan
	CHEMBL1314777	21206	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	472	8	3	4	5.4	CCc1ccccc1NC(=O)Nc1cc(C(=O)NCc2ccc(OC)cc2)ccc1N1CCCC1	nan
	15990013	21219	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	6	2	8	3.4	COc1ccccc1CNC(=O)c1cccc(Nc2nc3ccccc3n3nnnc23)c1	nan
	CHEMBL1314976	21219	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	6	2	8	3.4	COc1ccccc1CNC(=O)c1cccc(Nc2nc3ccccc3n3nnnc23)c1	nan
	16025439	21240	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	516	7	1	6	4.6	Cc1ccccc1CN1c2ccccc2-c2nc(SCC(=O)NCc3ccccc3)ncc2S1(=O)=O	nan
	CHEMBL1315303	21240	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	516	7	1	6	4.6	Cc1ccccc1CN1c2ccccc2-c2nc(SCC(=O)NCc3ccccc3)ncc2S1(=O)=O	nan
	18579745	21262	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	7	1	7	2.9	CCOC(=O)c1nn(-c2ccc(F)cc2)c(=O)cc1OCC(=O)Nc1cccc(C)c1	nan
	CHEMBL1315496	21262	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	7	1	7	2.9	CCOC(=O)c1nn(-c2ccc(F)cc2)c(=O)cc1OCC(=O)Nc1cccc(C)c1	nan
	135455826	21313	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	2	1	5	4.9	Cc1ccc(-c2cc(C(F)F)nc3sc4c(O)ncnc4c23)cc1	nan
	CHEMBL1316104	21313	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	2	1	5	4.9	Cc1ccc(-c2cc(C(F)F)nc3sc4c(O)ncnc4c23)cc1	nan
	16008870	21327	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	2	1	4	3.9	Cn1c(C(=O)Nc2cccc(Cl)c2)cc2c(=O)n(C)c3ccccc3c21	nan
	CHEMBL1316241	21327	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	2	1	4	3.9	Cn1c(C(=O)Nc2cccc(Cl)c2)cc2c(=O)n(C)c3ccccc3c21	nan
	16024585	21332	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	5	1	5	3.5	Cc1ccc2c(=O)c(C(=O)c3ccc(F)cc3)cn(CC(=O)NC3CCCCC3)c2n1	nan
	CHEMBL1316336	21332	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	5	1	5	3.5	Cc1ccc2c(=O)c(C(=O)c3ccc(F)cc3)cn(CC(=O)NC3CCCCC3)c2n1	nan
	16023032	21336	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	4	2	5	4.7	CC(=O)c1ccc(NC(=O)c2cccc(NC(=O)N3CCSc4ncccc43)c2)cc1	nan
	CHEMBL1316423	21336	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	4	2	5	4.7	CC(=O)c1ccc(NC(=O)c2cccc(NC(=O)N3CCSc4ncccc43)c2)cc1	nan
	937929	21349	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	286	2	1	4	3.6	Cc1nc(N)c(C#N)c(-c2cccnc2)c1-c1ccccc1	nan
	CHEMBL1316609	21349	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	286	2	1	4	3.6	Cc1nc(N)c(C#N)c(-c2cccnc2)c1-c1ccccc1	nan
	16009522	21386	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	7	1	7	3.7	Cc1csc2nc(COc3ccc(NC(=O)COc4ccccc4)cc3)cc(=O)n12	nan
	CHEMBL1317126	21386	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	7	1	7	3.7	Cc1csc2nc(COc3ccc(NC(=O)COc4ccccc4)cc3)cc(=O)n12	nan
	16020239	21451	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	527	6	1	5	5.2	Cc1ccc(-n2c(=O)c3ccc(C(=O)NCc4ccccc4Cl)cc3n(Cc3cccc(F)c3)c2=O)cc1	nan
	CHEMBL1317963	21451	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	527	6	1	5	5.2	Cc1ccc(-n2c(=O)c3ccc(C(=O)NCc4ccccc4Cl)cc3n(Cc3cccc(F)c3)c2=O)cc1	nan
	16022974	21452	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	492	5	1	6	4.8	Cc1nnc(N2CCC(C(=O)NCc3ccc(F)cc3)CC2)c2nn(-c3ccc(Cl)cc3)c(C)c12	nan
	CHEMBL1317977	21452	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	492	5	1	6	4.8	Cc1nnc(N2CCC(C(=O)NCc3ccc(F)cc3)CC2)c2nn(-c3ccc(Cl)cc3)c(C)c12	nan
	3450154	21488	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	5	1	6	2.6	CC(=O)c1sc(NC(=O)C2CCCN2S(=O)(=O)c2ccccc2F)nc1C	nan
	CHEMBL1318435	21488	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	5	1	6	2.6	CC(=O)c1sc(NC(=O)C2CCCN2S(=O)(=O)c2ccccc2F)nc1C	nan
	15988872	21489	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	5	1	6	5.4	CCOC(=O)c1c(NC(=O)c2cc(-c3ccc(Cl)cc3)on2)sc2c1CCCC2	nan
	CHEMBL1318439	21489	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	5	1	6	5.4	CCOC(=O)c1c(NC(=O)c2cc(-c3ccc(Cl)cc3)on2)sc2c1CCCC2	nan
	16008607	21492	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	398	5	1	6	1.6	Cc1nc2c(c(C)c1CCC(=O)NCc1ccc(F)cc1)c(=O)n(C)c(=O)n2C	nan
	CHEMBL1318457	21492	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	398	5	1	6	1.6	Cc1nc2c(c(C)c1CCC(=O)NCc1ccc(F)cc1)c(=O)n(C)c(=O)n2C	nan
	15991398	21510	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	4	1	4	6.3	Cc1ccc(NC(=O)c2cc3c(-c4ccccc4)nn(-c4ccccc4)c3s2)cc1	nan
	CHEMBL1318575	21510	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	4	1	4	6.3	Cc1ccc(NC(=O)c2cc3c(-c4ccccc4)nn(-c4ccccc4)c3s2)cc1	nan
	3144686	21537	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	6	1	4	4.3	CCC(C)NC(=O)CSc1nc(-c2ccc(F)cc2)cc(C(F)(F)F)n1	nan
	CHEMBL1318807	21537	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	6	1	4	4.3	CCC(C)NC(=O)CSc1nc(-c2ccc(F)cc2)cc(C(F)(F)F)n1	nan
	1329083	21583	7	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	6	2	4	4.7	Cc1cccc(C)c1NC(=O)COc1ccccc1C(=O)Nc1ccc(Br)cn1	nan
	CHEMBL1319204	21583	7	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	6	2	4	4.7	Cc1cccc(C)c1NC(=O)COc1ccccc1C(=O)Nc1ccc(Br)cn1	nan
	1983515	21611	8	None	-5	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	521	6	1	6	5.3	O=C(Nc1cc[n+](-c2nc3ccccc3nc2[N-]S(=O)(=O)c2ccc(Cl)cc2)cc1)c1cccs1	nan
	CHEMBL1319447	21611	8	None	-5	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	521	6	1	6	5.3	O=C(Nc1cc[n+](-c2nc3ccccc3nc2[N-]S(=O)(=O)c2ccc(Cl)cc2)cc1)c1cccs1	nan
	20889080	21657	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	4	1	5	4.1	CC(CNc1nc2ccc(Cl)cc2n2cnnc12)c1ccccc1	nan
	CHEMBL1319804	21657	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	4	1	5	4.1	CC(CNc1nc2ccc(Cl)cc2n2cnnc12)c1ccccc1	nan
	16017559	21763	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	4	1	6	2.5	Cc1cccc(C(=O)Nc2nnc(S(=O)(=O)N3CCC(C)CC3)s2)c1	nan
	CHEMBL1320668	21763	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	4	1	6	2.5	Cc1cccc(C(=O)Nc2nnc(S(=O)(=O)N3CCC(C)CC3)s2)c1	nan
	16029569	21901	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	5	1	5	4.5	Cc1cc2c(=O)c(C(=O)c3ccncc3)cn(CC(=O)Nc3cccc(C)c3C)c2cc1C	nan
	CHEMBL1321921	21901	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	5	1	5	4.5	Cc1cc2c(=O)c(C(=O)c3ccncc3)cn(CC(=O)Nc3cccc(C)c3C)c2cc1C	nan
	15989030	21933	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	518	9	2	7	3.9	Cc1ccc(CNC(=O)CCCn2c(=O)c3sccc3n(CC(=O)Nc3c(C)cccc3C)c2=O)cc1	nan
	CHEMBL1322214	21933	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	518	9	2	7	3.9	Cc1ccc(CNC(=O)CCCn2c(=O)c3sccc3n(CC(=O)Nc3c(C)cccc3C)c2=O)cc1	nan
	4412940	21998	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	488	9	1	7	5.1	CCOc1ccc(-n2cc(C(=O)Nc3ccccc3OCC)c3cc(OC)c(OC)cc3c2=O)cc1	nan
	CHEMBL1322786	21998	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	488	9	1	7	5.1	CCOc1ccc(-n2cc(C(=O)Nc3ccccc3OCC)c3cc(OC)c(OC)cc3c2=O)cc1	nan
	3197538	22046	5	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	5	0	5	5.3	CCCc1nc(SCC(=O)N2c3ccccc3CC2C)c2c(C)c(C)sc2n1	nan
	CHEMBL1323376	22046	5	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	5	0	5	5.3	CCCc1nc(SCC(=O)N2c3ccccc3CC2C)c2c(C)c(C)sc2n1	nan
	3223224	22175	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	4	1	4	2.5	Cc1ccnc(N2CCC(C(=O)NCc3ccccc3F)CC2)n1	nan
	CHEMBL1324395	22175	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	4	1	4	2.5	Cc1ccnc(N2CCC(C(=O)NCc3ccccc3F)CC2)n1	nan
	16025301	22186	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	594	8	1	8	5.4	CCOC(=O)c1cccc(NC(=O)CSc2ncc3c(n2)-c2ccc(Cl)cc2N(Cc2ccccc2)S3(=O)=O)c1	nan
	CHEMBL1324479	22186	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	594	8	1	8	5.4	CCOC(=O)c1cccc(NC(=O)CSc2ncc3c(n2)-c2ccc(Cl)cc2N(Cc2ccccc2)S3(=O)=O)c1	nan
	24818748	22229	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	6	3	5	3.9	COc1ccc(NC(=O)NNC(=O)COc2ccc3cc(Br)ccc3c2)c(OC)c1	nan
	CHEMBL1324786	22229	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	6	3	5	3.9	COc1ccc(NC(=O)NNC(=O)COc2ccc3cc(Br)ccc3c2)c(OC)c1	nan
	15991180	22304	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	5	1	4	6.4	CCOc1ccc(C(=O)Nc2ccc(Cl)c(-c3nc4cc(C)cc(C)c4o3)c2)cc1	nan
	CHEMBL1325481	22304	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	5	1	4	6.4	CCOc1ccc(C(=O)Nc2ccc(Cl)c(-c3nc4cc(C)cc(C)c4o3)c2)cc1	nan
	794333	22428	52	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	290	3	0	2	3.7	COc1ccc(C(=O)c2ccc(Br)cc2)cc1	nan
	CHEMBL1326786	22428	52	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	290	3	0	2	3.7	COc1ccc(C(=O)c2ccc(Br)cc2)cc1	nan
	16012102	22449	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	4	1	7	3.2	CCc1cccc(C)c1NC(=O)C1CCN(c2nn3c(=O)cc(C)nc3s2)CC1	nan
	CHEMBL1326931	22449	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	4	1	7	3.2	CCc1cccc(C)c1NC(=O)C1CCN(c2nn3c(=O)cc(C)nc3s2)CC1	nan
	2097459	22465	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	3	1	3	4.1	Cc1ccc(NC(=O)Cn2cc(C(F)(F)F)cc(Cl)c2=O)cc1Cl	nan
	CHEMBL1327066	22465	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	3	1	3	4.1	Cc1ccc(NC(=O)Cn2cc(C(F)(F)F)cc(Cl)c2=O)cc1Cl	nan
	15988236	22486	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	7	1	7	2.1	CCC(C)NC(=O)Cn1c(=O)n(-c2cc(OC)cc(OC)c2)c(=O)c2ccccc21	nan
	CHEMBL1327218	22486	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	7	1	7	2.1	CCC(C)NC(=O)Cn1c(=O)n(-c2cc(OC)cc(OC)c2)c(=O)c2ccccc21	nan
	6825246	22523	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	581	8	2	8	1.9	CCOc1ccc(-n2c([S-])c(C(=O)Nc3ccc(S(=O)(=O)N4CCOCC4)cc3)[n+]3cc(C(N)=O)ccc23)cc1	nan
	CHEMBL1327580	22523	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	581	8	2	8	1.9	CCOc1ccc(-n2c([S-])c(C(=O)Nc3ccc(S(=O)(=O)N4CCOCC4)cc3)[n+]3cc(C(N)=O)ccc23)cc1	nan
	3192843	22555	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	6	2	6	2.8	O=C(Cn1nnc(-c2ccccc2NC(=O)c2ccccc2F)n1)NC1CCCC1	nan
	CHEMBL1327798	22555	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	6	2	6	2.8	O=C(Cn1nnc(-c2ccccc2NC(=O)c2ccccc2F)n1)NC1CCCC1	nan
	2816102	22616	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	259	2	0	5	3.3	CCOc1ncnc2c1sc1nc(C)cc(C)c12	nan
	CHEMBL1328179	22616	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	259	2	0	5	3.3	CCOc1ncnc2c1sc1nc(C)cc(C)c12	nan
	16009635	22762	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	491	7	1	8	4.5	COc1ccc(C(=O)Nc2cccc(OCc3cc(=O)n4c5c(sc4n3)CCCC5)c2)cc1OC	nan
	CHEMBL1329536	22762	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	491	7	1	8	4.5	COc1ccc(C(=O)Nc2cccc(OCc3cc(=O)n4c5c(sc4n3)CCCC5)c2)cc1OC	nan
	753116	22823	49	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	331	2	1	3	4.3	Cc1ccc(-c2cc(C(=O)O)c3cc(Br)ccc3n2)o1	nan
	CHEMBL1330042	22823	49	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	331	2	1	3	4.3	Cc1ccc(-c2cc(C(=O)O)c3cc(Br)ccc3n2)o1	nan
	4246541	22932	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	482	6	1	4	4.9	CCN(CC)S(=O)(=O)c1ccc2oc(C(=O)Nc3ccc(Br)cc3F)c(C)c2c1	nan
	CHEMBL1330918	22932	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	482	6	1	4	4.9	CCN(CC)S(=O)(=O)c1ccc2oc(C(=O)Nc3ccc(Br)cc3F)c(C)c2c1	nan
	701957	22997	17	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	258	2	0	3	3.4	CCOc1cc(C)cc2oc(=O)c3c(c12)CCCC3	nan
	CHEMBL1331353	22997	17	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	258	2	0	3	3.4	CCOc1cc(C)cc2oc(=O)c3c(c12)CCCC3	nan
	16014559	22998	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	4	1	6	4.9	COc1ccc(-c2nc3nc(C)cc(Nc4cccc(C(F)(F)F)c4)n3n2)cc1	nan
	CHEMBL1331359	22998	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	4	1	6	4.9	COc1ccc(-c2nc3nc(C)cc(Nc4cccc(C(F)(F)F)c4)n3n2)cc1	nan
	16009329	23073	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	480	5	1	7	3.3	O=C(Cn1cc(S(=O)(=O)c2ccc(F)cc2)c(=O)c2cc3c(cc21)OCO3)Nc1ccccc1	nan
	CHEMBL1331963	23073	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	480	5	1	7	3.3	O=C(Cn1cc(S(=O)(=O)c2ccc(F)cc2)c(=O)c2cc3c(cc21)OCO3)Nc1ccccc1	nan
	2151601	23120	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	5	1	6	5.5	Cc1ccc(-n2c(SCC(=O)Nc3cccc(C)c3)nc3c(oc4ccccc43)c2=O)cc1	nan
	CHEMBL1332323	23120	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	5	1	6	5.5	Cc1ccc(-n2c(SCC(=O)Nc3cccc(C)c3)nc3c(oc4ccccc43)c2=O)cc1	nan
	5310234	23213	11	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	366	6	1	8	2.2	O=C(CSc1ccc2nnc(-c3cccnc3)n2n1)NCc1ccco1	nan
	CHEMBL1333013	23213	11	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	366	6	1	8	2.2	O=C(CSc1ccc2nnc(-c3cccnc3)n2n1)NCc1ccco1	nan
	16018028	23332	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	345	5	1	4	2.6	O=C(Cn1c(=O)c2cccn2c2ccccc21)NCCc1ccccc1	nan
	CHEMBL1333957	23332	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	345	5	1	4	2.6	O=C(Cn1c(=O)c2cccn2c2ccccc21)NCCc1ccccc1	nan
	3174233	23390	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	10	3	7	3.1	CCCCOc1ccc(N(CC(=O)NC2CCCCC2)C(=O)c2snc(C(N)=O)c2N)cc1	nan
	CHEMBL1334365	23390	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	10	3	7	3.1	CCCCOc1ccc(N(CC(=O)NC2CCCCC2)C(=O)c2snc(C(N)=O)c2N)cc1	nan
	2237458	23398	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	6	1	8	2.3	COCc1cc(C)nc(SCC(=O)Nc2ccc3c(c2)n(C)c(=O)n3C)c1C#N	nan
	CHEMBL1334406	23398	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	6	1	8	2.3	COCc1cc(C)nc(SCC(=O)Nc2ccc3c(c2)n(C)c(=O)n3C)c1C#N	nan
	16030555	23453	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	5	0	4	5.9	O=C(CSc1nc2ccccc2nc1Cc1ccc(Cl)cc1)N1CCCc2ccccc21	nan
	CHEMBL1334948	23453	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	5	0	4	5.9	O=C(CSc1nc2ccccc2nc1Cc1ccc(Cl)cc1)N1CCCc2ccccc21	nan
	1257917	23473	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	2	1	4	3.0	O=C(Nc1ccc(F)cc1F)c1cc2ncc(Br)cn2n1	nan
	CHEMBL1335101	23473	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	2	1	4	3.0	O=C(Nc1ccc(F)cc1F)c1cc2ncc(Br)cn2n1	nan
	16010812	23505	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	3	0	7	3.8	Fc1ccc(N2CCN(c3nc4ccccc4c4nc(-c5cccnc5)nn34)CC2)cc1	nan
	CHEMBL1335280	23505	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	3	0	7	3.8	Fc1ccc(N2CCN(c3nc4ccccc4c4nc(-c5cccnc5)nn34)CC2)cc1	nan
	16015336	23534	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	6	1	7	5.4	CCc1ccc(NC(=O)c2sc(-n3nc(C)c(Cc4ccc5c(c4)OCO5)c3C)nc2C)cc1	nan
	CHEMBL1335512	23534	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	6	1	7	5.4	CCc1ccc(NC(=O)c2sc(-n3nc(C)c(Cc4ccc5c(c4)OCO5)c3C)nc2C)cc1	nan
	1450291	23611	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	4	1	6	3.8	Cc1cc(C)c2cc(C#N)c(SCC(=O)Nc3cc(C)on3)nc2c1	nan
	CHEMBL1336163	23611	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	4	1	6	3.8	Cc1cc(C)c2cc(C#N)c(SCC(=O)Nc3cc(C)on3)nc2c1	nan
	5115564	23615	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	467	5	3	7	5.7	N#Cc1ccccc1NC(=O)C1SC(Nc2ccccc2)=C(c2nc3ccccc3s2)C1=N	nan
	CHEMBL1336187	23615	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	467	5	3	7	5.7	N#Cc1ccccc1NC(=O)C1SC(Nc2ccccc2)=C(c2nc3ccccc3s2)C1=N	nan
	1366812	23954	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	5	1	4	5.3	Cc1ccc(-c2nc3ccccc3s2)cc1NC(=O)COc1ccccc1	nan
	CHEMBL1339140	23954	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	5	1	4	5.3	Cc1ccc(-c2nc3ccccc3s2)cc1NC(=O)COc1ccccc1	nan
	1860843	24081	11	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	3	2	5	5.2	Nc1c(C(=O)Nc2ccc(Br)cc2)sc2nc(-c3ccco3)ccc12	nan
	CHEMBL1340363	24081	11	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	3	2	5	5.2	Nc1c(C(=O)Nc2ccc(Br)cc2)sc2nc(-c3ccco3)ccc12	nan
	1258323	24147	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	436	5	2	6	3.6	Nc1c(C(=O)NCCc2ccccc2)sc2nc(N3CCOCC3)c3c(c12)CCCC3	nan
	CHEMBL1340956	24147	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	436	5	2	6	3.6	Nc1c(C(=O)NCCc2ccccc2)sc2nc(N3CCOCC3)c3c(c12)CCCC3	nan
	1248113	24159	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	5	0	7	3.3	CCOC(=O)c1cc(OC(=O)c2cccs2)n(-c2ccccc2)n1	nan
	CHEMBL1341066	24159	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	5	0	7	3.3	CCOC(=O)c1cc(OC(=O)c2cccs2)n(-c2ccccc2)n1	nan
	2478762	24407	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	5	2	6	3.3	Cc1c(C(=O)OCC(=O)Nc2ccc(S(N)(=O)=O)cc2)oc2c1ccc1ccccc12	nan
	CHEMBL1343023	24407	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	5	2	6	3.3	Cc1c(C(=O)OCC(=O)Nc2ccc(S(N)(=O)=O)cc2)oc2c1ccc1ccccc12	nan
	3243891	24420	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	290	3	1	6	2.6	Cc1ccc(CNc2nc3ccccc3n3nnnc23)cc1	nan
	CHEMBL1343134	24420	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	290	3	1	6	2.6	Cc1ccc(CNc2nc3ccccc3n3nnnc23)cc1	nan
	2242090	24613	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	3	2	5	3.5	CS(=O)(=O)c1ccc2nc(NC(=O)Nc3ccccc3F)sc2c1	nan
	CHEMBL1344848	24613	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	3	2	5	3.5	CS(=O)(=O)c1ccc2nc(NC(=O)Nc3ccccc3F)sc2c1	nan
	665134	24649	7	None	-1	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	4	1	5	3.7	O=C1CC(c2ccc(F)cc2)Cc2nc(NCc3ccco3)ncc21	nan
	CHEMBL1345142	24649	7	None	-1	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	4	1	5	3.7	O=C1CC(c2ccc(F)cc2)Cc2nc(NCc3ccco3)ncc21	nan
	1096895	24698	45	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	241	3	2	5	0.6	O=C(O)c1nn2cc(CCO)cnc2c1Cl	nan
	CHEMBL1345601	24698	45	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	241	3	2	5	0.6	O=C(O)c1nn2cc(CCO)cnc2c1Cl	nan
	3640616	24769	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	3	0	6	3.4	O=C(OC1CCOC1=O)c1cc(-c2cccs2)nc2ccccc12	nan
	CHEMBL1346240	24769	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	3	0	6	3.4	O=C(OC1CCOC1=O)c1cc(-c2cccs2)nc2ccccc12	nan
	4846975	24941	21	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	286	2	1	3	4.5	Sc1ncc(-c2ccc(Cl)cc2)n1-c1ccccc1	nan
	CHEMBL1347553	24941	21	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	286	2	1	3	4.5	Sc1ncc(-c2ccc(Cl)cc2)n1-c1ccccc1	nan
	5219047	24987	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	285	5	2	4	2.1	CCC(C)NC(=O)COC(=O)c1ccc(Cl)cc1O	nan
	CHEMBL1347937	24987	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	285	5	2	4	2.1	CCC(C)NC(=O)COC(=O)c1ccc(Cl)cc1O	nan
	16193959	25023	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	563	11	2	9	2.0	NS(=O)(=O)c1ccc(CCNC(=O)CCCn2c(SCC(=O)N3CCCC3)nc3ccsc3c2=O)cc1	nan
	CHEMBL1348274	25023	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	563	11	2	9	2.0	NS(=O)(=O)c1ccc(CCNC(=O)CCCn2c(SCC(=O)N3CCCC3)nc3ccsc3c2=O)cc1	nan
	3342394	25268	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	398	7	1	5	3.3	C=CCN1C(=O)c2ccccc2Sc2ccc(C(=O)NCC(OC)OC)cc21	nan
	CHEMBL1350401	25268	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	398	7	1	5	3.3	C=CCN1C(=O)c2ccccc2Sc2ccc(C(=O)NCC(OC)OC)cc21	nan
	16011056	25769	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	472	7	1	6	4.1	CCc1cc2c(cc3c(=O)n(CCCC(=O)NCc4cccc(Br)c4)ncn32)s1	nan
	CHEMBL1354311	25769	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	472	7	1	6	4.1	CCc1cc2c(cc3c(=O)n(CCCC(=O)NCc4cccc(Br)c4)ncn32)s1	nan
	16025634	25778	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	478	4	1	6	4.1	Cc1ccc(NC(=O)CSc2ncc3c(n2)-c2ccc(Cl)cc2N(C)S3(=O)=O)cc1F	nan
	CHEMBL1354359	25778	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	478	4	1	6	4.1	Cc1ccc(NC(=O)CSc2ncc3c(n2)-c2ccc(Cl)cc2N(C)S3(=O)=O)cc1F	nan
	16009946	25812	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	472	7	1	7	1.6	CCc1cccc(CC)c1NC(=O)CN(C)S(=O)(=O)c1ccc2c(c1)n(C)c(=O)c(=O)n2C	nan
	CHEMBL1354862	25812	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	472	7	1	7	1.6	CCc1cccc(CC)c1NC(=O)CN(C)S(=O)(=O)c1ccc2c(c1)n(C)c(=O)c(=O)n2C	nan
	16018892	25836	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	5	0	7	5.9	CCc1nnc(SCc2nc(-c3ccccc3F)oc2C)c2cc3sccc3n12	nan
	CHEMBL1355121	25836	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	5	0	7	5.9	CCc1nnc(SCc2nc(-c3ccccc3F)oc2C)c2cc3sccc3n12	nan
	4363763	25907	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	528	5	0	8	4.0	CCOC(=O)c1cc2c(=O)n3ccccc3nc2n(CC2CCCO2)/c1=N\C(=O)c1ccc(C(C)(C)C)cc1	nan
	CHEMBL1356044	25907	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	528	5	0	8	4.0	CCOC(=O)c1cc2c(=O)n3ccccc3nc2n(CC2CCCO2)/c1=N\C(=O)c1ccc(C(C)(C)C)cc1	nan
	16024946	25923	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	4	1	4	4.1	O=C(NCc1ccccc1Cl)c1ccc2c(c1)nnn2C1CCCC1	nan
	CHEMBL1356218	25923	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	4	1	4	4.1	O=C(NCc1ccccc1Cl)c1ccc2c(c1)nnn2C1CCCC1	nan
	15990261	25926	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	4	0	7	4.1	Cc1nnc2c(N3CCN(c4ccccc4)CC3)nc3ccc(C(=O)c4ccccc4)cc3n12	nan
	CHEMBL1356236	25926	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	4	0	7	4.1	Cc1nnc2c(N3CCN(c4ccccc4)CC3)nc3ccc(C(=O)c4ccccc4)cc3n12	nan
	16031511	25930	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	6	1	6	4.1	COc1ccc(-c2nnc(SCC(=O)Nc3ccc(F)cc3)s2)cc1	nan
	CHEMBL1356303	25930	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	6	1	6	4.1	COc1ccc(-c2nnc(SCC(=O)Nc3ccc(F)cc3)s2)cc1	nan
	16030397	25946	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	8	1	5	3.4	COCCNC(=O)CSc1nc2ccccc2nc1Cc1ccc(C)cc1	nan
	CHEMBL1356573	25946	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	8	1	5	3.4	COCCNC(=O)CSc1nc2ccccc2nc1Cc1ccc(C)cc1	nan
	16009450	25963	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	7	1	7	3.5	O=C(COc1ccc(F)cc1)Nc1ccc(OCc2cc(=O)n3ccsc3n2)cc1	nan
	CHEMBL1356791	25963	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	7	1	7	3.5	O=C(COc1ccc(F)cc1)Nc1ccc(OCc2cc(=O)n3ccsc3n2)cc1	nan
	756766	25975	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	3	1	4	3.8	Cn1c(SCc2cccc(F)c2)nc2c([nH]c3ccccc32)c1=O	nan
	CHEMBL1356946	25975	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	3	1	4	3.8	Cn1c(SCc2cccc(F)c2)nc2c([nH]c3ccccc32)c1=O	nan
	2141078	25987	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	5	1	6	4.7	COc1ccc(CNc2nc3c(-c4cccc(F)c4)nnn3c3ccccc23)cc1	nan
	CHEMBL1357087	25987	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	5	1	6	4.7	COc1ccc(CNc2nc3c(-c4cccc(F)c4)nnn3c3ccccc23)cc1	nan
	15988374	26018	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	569	6	0	6	5.7	O=C(CSc1ncc2c(n1)-c1ccccc1N(Cc1ccc(F)cc1)S2(=O)=O)c1ccc(Br)cc1	nan
	CHEMBL1357521	26018	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	569	6	0	6	5.7	O=C(CSc1ncc2c(n1)-c1ccccc1N(Cc1ccc(F)cc1)S2(=O)=O)c1ccc(Br)cc1	nan
	16020301	26032	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	566	8	2	7	4.2	COc1ccc(-n2c(=O)c3ccc(C(=O)NCc4ccc(C)cc4)cc3n(CC(=O)Nc3ccc(F)cc3)c2=O)cc1	nan
	CHEMBL1357758	26032	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	566	8	2	7	4.2	COc1ccc(-n2c(=O)c3ccc(C(=O)NCc4ccc(C)cc4)cc3n(CC(=O)Nc3ccc(F)cc3)c2=O)cc1	nan
	16024673	26042	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	475	7	1	6	3.9	COc1cccc(C(=O)c2cn(CC(=O)NCc3ccccc3Cl)c3nc(C)ccc3c2=O)c1	nan
	CHEMBL1357949	26042	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	475	7	1	6	3.9	COc1cccc(C(=O)c2cn(CC(=O)NCc3ccccc3Cl)c3nc(C)ccc3c2=O)c1	nan
	16016274	26060	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	4	0	6	4.2	Cc1cccc(-c2noc(-c3ccc(N4CCCC4)c([N+](=O)[O-])c3)n2)c1	nan
	CHEMBL1358183	26060	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	4	0	6	4.2	Cc1cccc(-c2noc(-c3ccc(N4CCCC4)c([N+](=O)[O-])c3)n2)c1	nan
	20880782	26072	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	472	8	1	7	3.0	CC1CCCCN1CCNC(=O)CCc1nnc2n(Cc3ccccc3)c(=O)c3ccccc3n12	nan
	CHEMBL1358259	26072	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	472	8	1	7	3.0	CC1CCCCN1CCNC(=O)CCc1nnc2n(Cc3ccccc3)c(=O)c3ccccc3n12	nan
	15988865	26088	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	322	3	1	5	3.6	Cc1ccc(NC(=O)c2cc(-c3ccc4c(c3)OCO4)on2)cc1	nan
	CHEMBL1358506	26088	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	322	3	1	5	3.6	Cc1ccc(NC(=O)c2cc(-c3ccc4c(c3)OCO4)on2)cc1	nan
	16009824	26105	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	496	6	2	7	4.0	NS(=O)(=O)c1ccc(CCNc2nc3c(-c4cccc(F)c4)nnn3c3ccc(Cl)cc23)cc1	nan
	CHEMBL1358725	26105	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	496	6	2	7	4.0	NS(=O)(=O)c1ccc(CCNc2nc3c(-c4cccc(F)c4)nnn3c3ccc(Cl)cc23)cc1	nan
	1231059	26108	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	293	3	1	4	3.7	CC(=O)Nc1cccc(-c2nnc(-c3ccc(C)cc3)o2)c1	nan
	CHEMBL1358793	26108	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	293	3	1	4	3.7	CC(=O)Nc1cccc(-c2nnc(-c3ccc(C)cc3)o2)c1	nan
	1317893	26152	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	5	1	5	5.2	Cc1cc(OCC(=O)Nc2cc(-c3nc4ncccc4o3)ccc2C)ccc1Cl	nan
	CHEMBL1359048	26152	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	5	1	5	5.2	Cc1cc(OCC(=O)Nc2cc(-c3nc4ncccc4o3)ccc2C)ccc1Cl	nan
	3410425	26266	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	7	0	7	3.7	CCOCCn1/c(=N/C(=O)c2ccc3c(c2)OCCO3)sc2cc(OCC)ccc21	nan
	CHEMBL1360046	26266	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	7	0	7	3.7	CCOCCn1/c(=N/C(=O)c2ccc3c(c2)OCCO3)sc2cc(OCC)ccc21	nan
	2335932	26348	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	4	1	5	2.8	Cc1cccc(C)c1NC(=O)COC(=O)c1ccc2c(c1)OCO2	nan
	CHEMBL1360771	26348	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	4	1	5	2.8	Cc1cccc(C)c1NC(=O)COC(=O)c1ccc2c(c1)OCO2	nan
	16009752	26411	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	331	5	1	5	4.5	CCCCNc1nc2c(-c3cccc(C)c3)nnn2c2ccccc12	nan
	CHEMBL1361402	26411	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	331	5	1	5	4.5	CCCCNc1nc2c(-c3cccc(C)c3)nnn2c2ccccc12	nan
	16022921	26424	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	498	7	1	7	4.7	CCOc1ccccc1CNC(=O)C1CCN(c2nnc(C)c3c(C)n(-c4ccc(C)cc4)nc23)CC1	nan
	CHEMBL1361507	26424	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	498	7	1	7	4.7	CCOc1ccccc1CNC(=O)C1CCN(c2nnc(C)c3c(C)n(-c4ccc(C)cc4)nc23)CC1	nan
	2345644	26496	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	6	1	7	3.5	COc1cccc(C(=O)Nc2nnc(-c3ccc(OC)cc3OC)s2)c1	nan
	CHEMBL1362103	26496	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	6	1	7	3.5	COc1cccc(C(=O)Nc2nnc(-c3ccc(OC)cc3OC)s2)c1	nan
	16022913	26539	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	6	1	6	4.3	Cc1ccc(-n2nc3c(N4CCC(C(=O)NCCc5ccccc5)CC4)nnc(C)c3c2C)cc1	nan
	CHEMBL1362452	26539	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	6	1	6	4.3	Cc1ccc(-n2nc3c(N4CCC(C(=O)NCCc5ccccc5)CC4)nnc(C)c3c2C)cc1	nan
	1313404	26553	10	None	-1	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	479	6	1	7	4.0	CCOc1cc(C2C(C(=O)OC)=CN(C3CCCC3)C=C2C(=O)OC)cc(Br)c1O	nan
	CHEMBL1362550	26553	10	None	-1	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	479	6	1	7	4.0	CCOc1cc(C2C(C(=O)OC)=CN(C3CCCC3)C=C2C(=O)OC)cc(Br)c1O	nan
	3448294	26574	23	None	-19	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	313	4	0	3	5.0	O=Cc1cc2ccccc2nc1SCc1ccc(Cl)cc1	nan
	CHEMBL1362687	26574	23	None	-19	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	313	4	0	3	5.0	O=Cc1cc2ccccc2nc1SCc1ccc(Cl)cc1	nan
	16026537	26698	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	5	1	6	4.2	CC(=O)c1cccc(NC(=O)C(C)n2c(=O)cc(C)c3c(C)nn(-c4ccccc4)c32)c1	nan
	CHEMBL1363862	26698	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	5	1	6	4.2	CC(=O)c1cccc(NC(=O)C(C)n2c(=O)cc(C)c3c(C)nn(-c4ccccc4)c32)c1	nan
	16009886	26708	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	471	5	1	7	4.3	COc1cccc(-n2c(=O)c3sc4ccccc4c3n(CC(=O)Nc3ccccc3C)c2=O)c1	nan
	CHEMBL1363941	26708	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	471	5	1	7	4.3	COc1cccc(-n2c(=O)c3sc4ccccc4c3n(CC(=O)Nc3ccccc3C)c2=O)c1	nan
	3359750	26776	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	5	1	4	5.2	O=C(CSc1nc(-c2ccccc2)c2ccccc2n1)Nc1ccc(F)cc1	nan
	CHEMBL1364552	26776	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	5	1	4	5.2	O=C(CSc1nc(-c2ccccc2)c2ccccc2n1)Nc1ccc(F)cc1	nan
	16019445	26830	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	477	5	1	8	5.7	Cc1ccc(C)c(Nc2nc3c(S(=O)(=O)c4ccc(C(C)C)cc4)nnn3c3ccsc23)c1	nan
	CHEMBL1365021	26830	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	477	5	1	8	5.7	Cc1ccc(C)c(Nc2nc3c(S(=O)(=O)c4ccc(C(C)C)cc4)nnn3c3ccsc23)c1	nan
	1152421	27029	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	7	1	6	5.4	CCOc1ccccc1NC(=O)CSc1nc(-c2cccs2)cc(C(F)(F)F)n1	nan
	CHEMBL1366693	27029	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	7	1	6	5.4	CCOc1ccccc1NC(=O)CSc1nc(-c2cccs2)cc(C(F)(F)F)n1	nan
	1080694	27057	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	3	1	5	3.2	CC1(C)CC(=O)c2sc(NS(=O)(=O)c3ccc(F)cc3)nc2C1	nan
	CHEMBL1366962	27057	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	3	1	5	3.2	CC1(C)CC(=O)c2sc(NS(=O)(=O)c3ccc(F)cc3)nc2C1	nan
	16022984	27131	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	7	1	7	4.0	COc1ccc(-n2nc3c(N4CCC(C(=O)NCCc5ccccc5)CC4)nnc(C)c3c2C)cc1	nan
	CHEMBL1367585	27131	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	7	1	7	4.0	COc1ccc(-n2nc3c(N4CCC(C(=O)NCCc5ccccc5)CC4)nnc(C)c3c2C)cc1	nan
	16015654	27284	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	358	6	1	5	4.7	CC(=O)Nc1ccc2nc(SCCOc3ccc(C)cc3)sc2c1	nan
	CHEMBL1368731	27284	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	358	6	1	5	4.7	CC(=O)Nc1ccc2nc(SCCOc3ccc(C)cc3)sc2c1	nan
	2918354	27578	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	7	1	5	3.7	COCCCN1C(=O)C(O)=C(C(=O)c2ccco2)C1c1cccc(Br)c1	nan
	CHEMBL1370753	27578	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	7	1	5	3.7	COCCCN1C(=O)C(O)=C(C(=O)c2ccco2)C1c1cccc(Br)c1	nan
	1005238	27614	18	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	5	1	7	3.5	Cc1cc(NC(=O)CSc2nc3c(c(-c4cccnc4)c2C#N)CCC3)no1	nan
	CHEMBL1371055	27614	18	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	5	1	7	3.5	Cc1cc(NC(=O)CSc2nc3c(c(-c4cccnc4)c2C#N)CCC3)no1	nan
	1442423	27910	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	356	4	1	6	4.0	Cc1cc(NC(=O)CSc2nc(C(C)(C)C)nc3ccccc23)no1	nan
	CHEMBL1373175	27910	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	356	4	1	6	4.0	Cc1cc(NC(=O)CSc2nc(C(C)(C)C)nc3ccccc23)no1	nan
	6615570	27966	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	4	1	7	3.7	COc1ccc(C)cc1NC(=O)c1sc2nc(C)nc(N3CCOCC3)c2c1C	nan
	CHEMBL1373530	27966	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	4	1	7	3.7	COc1ccc(C)cc1NC(=O)c1sc2nc(C)nc(N3CCOCC3)c2c1C	nan
	2410746	27986	35	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	4	2	5	3.0	CC(=O)Nc1ccc(S(=O)(=O)Nc2nc3ccccc3nc2Cl)cc1	nan
	CHEMBL1373647	27986	35	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	4	2	5	3.0	CC(=O)Nc1ccc(S(=O)(=O)Nc2nc3ccccc3nc2Cl)cc1	nan
	16009969	28112	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	5	1	7	1.3	CN(CC(=O)Nc1ccc(Cl)cc1F)S(=O)(=O)c1ccc2c(c1)n(C)c(=O)c(=O)n2C	nan
	CHEMBL1374581	28112	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	5	1	7	1.3	CN(CC(=O)Nc1ccc(Cl)cc1F)S(=O)(=O)c1ccc2c(c1)n(C)c(=O)c(=O)n2C	nan
	9547710	28114	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	4	1	9	0.3	Cn1c(N)c(C(=O)COC(=O)c2ccnc3ccccc23)c(=O)n(C)c1=O	nan
	CHEMBL1374591	28114	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	4	1	9	0.3	Cn1c(N)c(C(=O)COC(=O)c2ccnc3ccccc23)c(=O)n(C)c1=O	nan
	4414022	28144	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	7	1	6	4.0	CCOC(=O)c1c(NC(=O)C(C)Oc2ccccc2F)sc(C(C)=O)c1C	nan
	CHEMBL1374782	28144	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	7	1	6	4.0	CCOC(=O)c1c(NC(=O)C(C)Oc2ccccc2F)sc(C(C)=O)c1C	nan
	679950	28207	12	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	5	1	6	2.9	CCN(CC)c1ccc(-c2c(C#N)c(N)nc(OC)c2C#N)cc1	nan
	CHEMBL1375207	28207	12	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	5	1	6	2.9	CCN(CC)c1ccc(-c2c(C#N)c(N)nc(OC)c2C#N)cc1	nan
	5297522	28218	20	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	4	2	7	4.0	CCOC(=O)c1ccc(NC(=O)c2sc3nc4c(cc3c2N)N2CCC4CC2)cc1	nan
	CHEMBL1375280	28218	20	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	4	2	7	4.0	CCOC(=O)c1ccc(NC(=O)c2sc3nc4c(cc3c2N)N2CCC4CC2)cc1	nan
	16022988	28265	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	5	1	7	2.8	CCNC(=O)C1CCN(c2nnc(C)c3c(C)n(-c4ccc(OC)cc4)nc23)CC1	nan
	CHEMBL1375625	28265	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	5	1	7	2.8	CCNC(=O)C1CCN(c2nnc(C)c3c(C)n(-c4ccc(OC)cc4)nc23)CC1	nan
	1224964	28269	16	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	4	2	3	4.2	O=C(Nc1ccc(C(=O)NC2CCCCC2)cc1)c1cncc(Br)c1	nan
	CHEMBL1375663	28269	16	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	4	2	3	4.2	O=C(Nc1ccc(C(=O)NC2CCCCC2)cc1)c1cncc(Br)c1	nan
	16009514	28352	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	5	1	6	4.2	Cc1ccc(C(=O)Nc2ccc(OCc3cc(=O)n4c(C)csc4n3)cc2)cc1	nan
	CHEMBL1376473	28352	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	5	1	6	4.2	Cc1ccc(C(=O)Nc2ccc(OCc3cc(=O)n4c(C)csc4n3)cc2)cc1	nan
	16010769	28425	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	4	0	5	3.6	Cc1ccc(Cn2c(=O)n(Cc3ccccc3Cl)c(=O)c3cccnc32)cc1	nan
	CHEMBL1377217	28425	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	4	0	5	3.6	Cc1ccc(Cn2c(=O)n(Cc3ccccc3Cl)c(=O)c3cccnc32)cc1	nan
	16024487	28479	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	5	1	5	4.2	Cc1cc(C)cc(NC(=O)Cn2cc(C(=O)c3ccccc3)c(=O)c3ccc(C)nc32)c1	nan
	CHEMBL1377738	28479	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	5	1	5	4.2	Cc1cc(C)cc(NC(=O)Cn2cc(C(=O)c3ccccc3)c(=O)c3ccc(C)nc32)c1	nan
	20887350	28771	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	2	0	7	1.3	Cc1nn(CC(=O)N2CCC3(CC2)OCCO3)c(=O)c2cc3ccccc3n12	nan
	CHEMBL1380351	28771	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	2	0	7	1.3	Cc1nn(CC(=O)N2CCC3(CC2)OCCO3)c(=O)c2cc3ccccc3n12	nan
	1943710	28930	8	None	-6	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	8	1	7	5.1	CCCCc1nc2sc3c(SCC(=O)NCc4ccco4)ncnc3c2c2c1CCC2	nan
	CHEMBL1381564	28930	8	None	-6	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	8	1	7	5.1	CCCCc1nc2sc3c(SCC(=O)NCc4ccco4)ncnc3c2c2c1CCC2	nan
	2220993	28967	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	3	1	5	4.5	Cc1cc(NC(=O)c2cc(-c3ccccn3)nc3c(Cl)cccc23)no1	nan
	CHEMBL1381905	28967	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	3	1	5	4.5	Cc1cc(NC(=O)c2cc(-c3ccccn3)nc3c(Cl)cccc23)no1	nan
	2551678	28975	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	5	1	5	5.3	Cc1[nH]c2ccccc2c1C(=O)CSc1nc2ccccc2c(=O)n1-c1ccccc1F	nan
	CHEMBL1381998	28975	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	5	1	5	5.3	Cc1[nH]c2ccccc2c1C(=O)CSc1nc2ccccc2c(=O)n1-c1ccccc1F	nan
	15997541	29245	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	492	7	2	7	3.4	COc1ccc(-n2nc(C(=O)NCC(=O)Nc3cccc(Cl)c3)c3ccccc3c2=O)cc1OC	nan
	CHEMBL1384419	29245	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	492	7	2	7	3.4	COc1ccc(-n2nc(C(=O)NCC(=O)Nc3cccc(Cl)c3)c3ccccc3c2=O)cc1OC	nan
	2412434	29318	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	5	2	6	2.0	NS(=O)(=O)c1ccc(NC(=O)CSc2ncnc3ccccc23)cc1	nan
	CHEMBL1385049	29318	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	5	2	6	2.0	NS(=O)(=O)c1ccc(NC(=O)CSc2ncnc3ccccc23)cc1	nan
	1490540	29325	14	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	299	4	1	4	3.9	COc1ccccc1CNc1ncnc2cc(Cl)ccc12	nan
	CHEMBL1385084	29325	14	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	299	4	1	4	3.9	COc1ccccc1CNc1ncnc2cc(Cl)ccc12	nan
	1442725	29368	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	5	1	4	3.9	CC(C)c1nc(SCC(=O)NC2CCCC2)c2ccccc2n1	nan
	CHEMBL1385478	29368	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	5	1	4	3.9	CC(C)c1nc(SCC(=O)NC2CCCC2)c2ccccc2n1	nan
	660521	29447	13	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	4	1	6	4.4	N#Cc1cc2c(nc1SCC(=O)Nc1sc3c(c1C#N)CCC3)CCCCC2	nan
	CHEMBL1386214	29447	13	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	4	1	6	4.4	N#Cc1cc2c(nc1SCC(=O)Nc1sc3c(c1C#N)CCC3)CCCCC2	nan
	658023	29772	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	5	2	7	2.7	CCOc1ccc(C2C(C#N)=C(N)SC(N)=C2C#N)c(OCC)c1	nan
	CHEMBL1388744	29772	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	5	2	7	2.7	CCOc1ccc(C2C(C#N)=C(N)SC(N)=C2C#N)c(OCC)c1	nan
	5913531	29825	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	475	8	1	8	3.3	COc1cccc(C2C(C(=O)c3ccc4c(c3)OCCO4)=C(O)C(=O)N2CCCn2ccnc2)c1	nan
	CHEMBL1389094	29825	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	475	8	1	8	3.3	COc1cccc(C2C(C(=O)c3ccc4c(c3)OCCO4)=C(O)C(=O)N2CCCn2ccnc2)c1	nan
	135749817	29970	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	335	2	2	4	4.9	N#C/C(=C(\O)c1cc(Cl)sc1Cl)c1nc2ccccc2[nH]1	nan
	CHEMBL1390333	29970	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	335	2	2	4	4.9	N#C/C(=C(\O)c1cc(Cl)sc1Cl)c1nc2ccccc2[nH]1	nan
	135468428	30148	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	516	5	2	7	5.1	Cc1cc(-n2c(SCC(=O)Nc3ccc(Br)cc3)nc3nnc(C)c-3c2N)ccc1Cl	nan
	CHEMBL1391897	30148	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	516	5	2	7	5.1	Cc1cc(-n2c(SCC(=O)Nc3ccc(Br)cc3)nc3nnc(C)c-3c2N)ccc1Cl	nan
	5393174	30174	38	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	268	2	1	4	3.2	COc1ccc(-c2cc3ccc(O)cc3oc2=O)cc1	nan
	CHEMBL1392132	30174	38	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	268	2	1	4	3.2	COc1ccc(-c2cc3ccc(O)cc3oc2=O)cc1	nan
	738837	30200	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	269	2	1	2	3.9	Cc1occc1C(=O)Nc1cccc(C(F)(F)F)c1	nan
	CHEMBL1392331	30200	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	269	2	1	2	3.9	Cc1occc1C(=O)Nc1cccc(C(F)(F)F)c1	nan
	16194581	30268	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	4	1	9	0.9	CC(Sc1nc(-c2ccco2)nc2c1c(=O)n(C)c(=O)n2C)C(=O)O	nan
	CHEMBL1392938	30268	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	4	1	9	0.9	CC(Sc1nc(-c2ccco2)nc2c1c(=O)n(C)c(=O)n2C)C(=O)O	nan
	16029022	30491	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	5	1	6	2.5	COC(=O)c1ccc(NC(=O)c2cc(S(=O)(=O)N3CCC(C)CC3)cn2C)cc1	nan
	CHEMBL1395073	30491	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	5	1	6	2.5	COC(=O)c1ccc(NC(=O)c2cc(S(=O)(=O)N3CCC(C)CC3)cn2C)cc1	nan
	16024525	30539	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	6	1	5	4.2	Cc1ccc(C(=O)c2cn(CC(=O)NCc3ccccc3Cl)c3nc(C)ccc3c2=O)cc1	nan
	CHEMBL1395642	30539	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	6	1	5	4.2	Cc1ccc(C(=O)c2cn(CC(=O)NCc3ccccc3Cl)c3nc(C)ccc3c2=O)cc1	nan
	16009355	30545	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	5	0	5	5.1	CC(C)c1ccc(OCc2cc(=O)n3c(-c4ccccc4)csc3n2)cc1	nan
	CHEMBL1395773	30545	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	5	0	5	5.1	CC(C)c1ccc(OCc2cc(=O)n3c(-c4ccccc4)csc3n2)cc1	nan
	16012262	30598	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	5	1	7	1.7	Cc1cccc(NC(=O)CCS(=O)(=O)c2ccc3c(c2)n(C)c(=O)c(=O)n3C)c1C	nan
	CHEMBL1396597	30598	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	5	1	7	1.7	Cc1cccc(NC(=O)CCS(=O)(=O)c2ccc3c(c2)n(C)c(=O)c(=O)n3C)c1C	nan
	16425494	30617	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	3	1	5	2.9	CN1CCN(Cc2c(O)ccc3cc(-c4ccccc4)c(=O)oc23)CC1	nan
	5522461	30617	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	3	1	5	2.9	CN1CCN(Cc2c(O)ccc3cc(-c4ccccc4)c(=O)oc23)CC1	nan
	CHEMBL1396834	30617	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	3	1	5	2.9	CN1CCN(Cc2c(O)ccc3cc(-c4ccccc4)c(=O)oc23)CC1	nan
	15988387	30621	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	3	2	4	2.2	COc1cccc(C(=O)NC2=NC(c3ccccc3F)CC(=O)N2)c1	nan
	CHEMBL1396902	30621	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	3	2	4	2.2	COc1cccc(C(=O)NC2=NC(c3ccccc3F)CC(=O)N2)c1	nan
	16030463	30641	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	5	0	4	4.6	CC1CCN(C(=O)CSc2nc3ccccc3nc2Cc2ccccc2)CC1	nan
	CHEMBL1397149	30641	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	5	0	4	4.6	CC1CCN(C(=O)CSc2nc3ccccc3nc2Cc2ccccc2)CC1	nan
	16011758	30651	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	8	1	7	2.8	COc1ccc(OC)c(CNC(=O)CCCn2c(=O)c3cccn3c3cccnc32)c1	nan
	CHEMBL1397253	30651	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	8	1	7	2.8	COc1ccc(OC)c(CNC(=O)CCCn2c(=O)c3cccn3c3cccnc32)c1	nan
	15988254	30709	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	5	0	7	3.1	COc1cc(OC)cc(-n2c(=O)c3ccccc3n(Cc3ccccc3C#N)c2=O)c1	nan
	CHEMBL1398033	30709	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	5	0	7	3.1	COc1cc(OC)cc(-n2c(=O)c3ccccc3n(Cc3ccccc3C#N)c2=O)c1	nan
	5089883	30718	17	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	487	7	0	6	5.9	O=C(CSc1oc(-c2ccc(F)cc2)nc1S(=O)(=O)c1ccccc1)c1ccc(Cl)cc1	nan
	CHEMBL1398184	30718	17	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	487	7	0	6	5.9	O=C(CSc1oc(-c2ccc(F)cc2)nc1S(=O)(=O)c1ccccc1)c1ccc(Cl)cc1	nan
	16020303	30723	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	566	8	2	7	4.2	COc1ccc(-n2c(=O)c3ccc(C(=O)NCc4ccc(C)cc4)cc3n(CC(=O)Nc3cccc(F)c3)c2=O)cc1	nan
	CHEMBL1398259	30723	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	566	8	2	7	4.2	COc1ccc(-n2c(=O)c3ccc(C(=O)NCc4ccc(C)cc4)cc3n(CC(=O)Nc3cccc(F)c3)c2=O)cc1	nan
	16025636	30729	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	482	4	1	6	3.9	CN1c2cc(Cl)ccc2-c2nc(SCC(=O)Nc3ccc(F)cc3F)ncc2S1(=O)=O	nan
	CHEMBL1398402	30729	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	482	4	1	6	3.9	CN1c2cc(Cl)ccc2-c2nc(SCC(=O)Nc3ccc(F)cc3F)ncc2S1(=O)=O	nan
	16030333	30738	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	9	1	6	4.6	COc1ccc(CNC(=O)CSc2nc3ccccc3nc2Cc2ccccc2OC)cc1	nan
	CHEMBL1398464	30738	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	9	1	6	4.6	COc1ccc(CNC(=O)CSc2nc3ccccc3nc2Cc2ccccc2OC)cc1	nan
	16022444	30764	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	6	2	7	4.8	CCc1ccccc1Nc1nn2c(=O)c3ccc(C(=O)NCc4ccc(C)cc4)cc3nc2s1	nan
	CHEMBL1398653	30764	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	6	2	7	4.8	CCc1ccccc1Nc1nn2c(=O)c3ccc(C(=O)NCc4ccc(C)cc4)cc3nc2s1	nan
	4135187	30817	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	7	1	6	4.4	Cc1ccc(CNC(=O)CSc2nc3ccsc3c(=O)n2Cc2ccccc2F)cc1	nan
	CHEMBL1399236	30817	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	7	1	6	4.4	Cc1ccc(CNC(=O)CSc2nc3ccsc3c(=O)n2Cc2ccccc2F)cc1	nan
	2135591	30821	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	518	7	1	7	4.7	CCOc1ccc(C(=O)c2cn(CC(=O)Nc3ccc(Cl)cc3)c3cc4c(cc3c2=O)OCCO4)cc1	nan
	CHEMBL1399275	30821	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	518	7	1	7	4.7	CCOc1ccc(C(=O)c2cn(CC(=O)Nc3ccc(Cl)cc3)c3cc4c(cc3c2=O)OCCO4)cc1	nan
	135546815	30828	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	5	2	5	4.0	Cc1ccc(NC(=O)C(C)Sc2nc(-c3ccccc3)c(C#N)c(=O)[nH]2)c(C)c1	nan
	CHEMBL1399310	30828	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	5	2	5	4.0	Cc1ccc(NC(=O)C(C)Sc2nc(-c3ccccc3)c(C#N)c(=O)[nH]2)c(C)c1	nan
	135513990	30875	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	4	2	5	4.4	Cc1c(Br)ccc(NC(=O)CSc2nc(O)c3ccccc3n2)c1C	nan
	CHEMBL1399762	30875	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	4	2	5	4.4	Cc1c(Br)ccc(NC(=O)CSc2nc(O)c3ccccc3n2)c1C	nan
	6484563	30951	33	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	232	0	2	2	3.4	SC1=NC2(CCCCC2)Nc2ccccc21	nan
	CHEMBL1400466	30951	33	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	232	0	2	2	3.4	SC1=NC2(CCCCC2)Nc2ccccc21	nan
	16011170	30973	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	400	4	1	5	4.6	COC(=O)c1cc2oc3ccccc3c2n1CC(=O)Nc1ccc(Cl)cc1F	nan
	CHEMBL1400646	30973	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	400	4	1	5	4.6	COC(=O)c1cc2oc3ccccc3c2n1CC(=O)Nc1ccc(Cl)cc1F	nan
	2404851	30999	18	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	3	1	7	1.0	O=S(=O)(c1cccc(-c2nnc(S)o2)c1)N1CCOCC1	nan
	CHEMBL1400922	30999	18	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	3	1	7	1.0	O=S(=O)(c1cccc(-c2nnc(S)o2)c1)N1CCOCC1	nan
	659778	31024	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	3	1	4	4.3	O=C(Nc1ccc2oc(-c3ccncc3)nc2c1)c1ccccc1F	nan
	CHEMBL1401137	31024	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	3	1	4	4.3	O=C(Nc1ccc2oc(-c3ccncc3)nc2c1)c1ccccc1F	nan
	4852309	31039	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	361	6	1	3	4.5	COc1cc(C(=O)NC(c2ccccc2)c2ccccc2)cc(OC)c1C	nan
	CHEMBL1401266	31039	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	361	6	1	3	4.5	COc1cc(C(=O)NC(c2ccccc2)c2ccccc2)cc(OC)c1C	nan
	1994854	31042	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	466	6	1	8	3.6	CCn1c(SCC(=O)Nc2ccc(C(C)=O)cc2)nc2nc3c(cc2c1=O)COC(C)(C)C3	nan
	CHEMBL1401292	31042	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	466	6	1	8	3.6	CCn1c(SCC(=O)Nc2ccc(C(C)=O)cc2)nc2nc3c(cc2c1=O)COC(C)(C)C3	nan
	16011439	31342	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	508	9	1	6	6.3	COc1ccc(Cn2c(SCc3ccc(C(=O)NC(C)c4ccccc4)cc3)nc3cccnc32)cc1	nan
	CHEMBL1404015	31342	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	508	9	1	6	6.3	COc1ccc(Cn2c(SCc3ccc(C(=O)NC(C)c4ccccc4)cc3)nc3cccnc32)cc1	nan
	2456084	31347	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	493	8	2	8	4.0	COc1cc(NC(=O)c2ccco2)c(C(=O)OCC(=O)Nc2ncc(Cl)cc2Cl)cc1OC	nan
	CHEMBL1404053	31347	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	493	8	2	8	4.0	COc1cc(NC(=O)c2ccco2)c(C(=O)OCC(=O)Nc2ncc(Cl)cc2Cl)cc1OC	nan
	2826390	31439	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	4	2	5	2.9	COC(=O)c1sccc1NC(=O)C1CC(C)=C(C)CC1C(=O)O	nan
	CHEMBL1404933	31439	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	4	2	5	2.9	COC(=O)c1sccc1NC(=O)C1CC(C)=C(C)CC1C(=O)O	nan
	16007508	31451	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	6	1	3	5.7	CCc1ccc(CNC(=O)CSc2c3c(nc4ccc(Cl)cc24)CCCC3)cc1	nan
	CHEMBL1405105	31451	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	6	1	3	5.7	CCc1ccc(CNC(=O)CSc2c3c(nc4ccc(Cl)cc24)CCCC3)cc1	nan
	1930124	31542	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	534	8	1	7	5.3	CCCCn1c(NS(=O)(=O)c2ccccc2)c(S(=O)(=O)c2ccc(C)cc2)c2nc3ccccc3nc21	nan
	CHEMBL1405964	31542	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	534	8	1	7	5.3	CCCCn1c(NS(=O)(=O)c2ccccc2)c(S(=O)(=O)c2ccc(C)cc2)c2nc3ccccc3nc21	nan
	135464462	31696	20	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	3	1	6	3.1	CN(C)Cc1c(O)ccc2cc(-c3nc4ccccc4n3C)c(=O)oc12	nan
	CHEMBL1407344	31696	20	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	3	1	6	3.1	CN(C)Cc1c(O)ccc2cc(-c3nc4ccccc4n3C)c(=O)oc12	nan
	3221573	31727	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	8	3	5	3.0	COCCCN=C(S)NCCNc1nc2c(C)c(C)ccc2cc1C#N	nan
	CHEMBL1407546	31727	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	8	3	5	3.0	COCCCN=C(S)NCCNc1nc2c(C)c(C)ccc2cc1C#N	nan
	266900	31741	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	304	1	1	3	4.3	COC(=O)c1cc(C)nc2c(C)cc3[nH]c4ccccc4c3c12	nan
	CHEMBL1407610	31741	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	304	1	1	3	4.3	COC(=O)c1cc(C)nc2c(C)cc3[nH]c4ccccc4c3c12	nan
	16018228	31804	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	330	5	1	5	1.1	CN(C)CCNC(=O)Cn1c(=O)c2cccn2c2ccc(F)cc21	nan
	CHEMBL1408060	31804	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	330	5	1	5	1.1	CN(C)CCNC(=O)Cn1c(=O)c2cccn2c2ccc(F)cc21	nan
	800213	31836	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	3	1	4	4.8	CC(C)(C)c1ccc(-c2nnc(NC(=O)c3ccccc3)s2)cc1	nan
	CHEMBL1408281	31836	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	3	1	4	4.8	CC(C)(C)c1ccc(-c2nnc(NC(=O)c3ccccc3)s2)cc1	nan
	4837904	31900	16	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	7	1	6	4.1	COc1ccc(CCNC(=O)Cc2c(C)c3cc4c(C)coc4cc3oc2=O)cc1OC	nan
	CHEMBL1408806	31900	16	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	7	1	6	4.1	COc1ccc(CCNC(=O)Cc2c(C)c3cc4c(C)coc4cc3oc2=O)cc1OC	nan
	915456	31903	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	4	2	4	4.6	Oc1ccccc1-c1nc(NCc2ccccc2)c2ccccc2n1	nan
	CHEMBL1408828	31903	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	4	2	4	4.6	Oc1ccccc1-c1nc(NCc2ccccc2)c2ccccc2n1	nan
	15988127	32033	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	570	6	3	6	7.6	COc1ccccc1NC(=O)c1sc2nc(C)c(C(=O)Nc3ccc(C)cc3C)c(-c3ccccc3Cl)c2c1N	nan
	CHEMBL1409862	32033	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	570	6	3	6	7.6	COc1ccccc1NC(=O)c1sc2nc(C)c(C(=O)Nc3ccc(C)cc3C)c(-c3ccccc3Cl)c2c1N	nan
	649505	32036	5	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	5	1	7	2.3	O=C(Nc1ccc2c(c1)OCO2)C1CCN(c2ccc(S(=O)(=O)N3CCOCC3)cc2)CC1	nan
	CHEMBL1409886	32036	5	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	5	1	7	2.3	O=C(Nc1ccc2c(c1)OCO2)C1CCN(c2ccc(S(=O)(=O)N3CCOCC3)cc2)CC1	nan
	688670	32054	26	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	282	3	0	4	3.5	COc1ccc(-c2cc(=O)c3cc(OC)ccc3o2)cc1	nan
	CHEMBL1410006	32054	26	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	282	3	0	4	3.5	COc1ccc(-c2cc(=O)c3cc(OC)ccc3o2)cc1	nan
	4137223	32162	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	3	1	5	5.2	Cc1nc(N2CCC(C)CC2)c2c(C)c(C(=O)Nc3ccc(C)c(F)c3)sc2n1	nan
	CHEMBL1410912	32162	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	3	1	5	5.2	Cc1nc(N2CCC(C)CC2)c2c(C)c(C(=O)Nc3ccc(C)c(F)c3)sc2n1	nan
	1088392	32353	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	5	1	7	3.0	COC(=O)c1sc(NC(=O)c2c(OC)cccc2OC)c(C#N)c1C	nan
	CHEMBL1412474	32353	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	5	1	7	3.0	COC(=O)c1sc(NC(=O)c2c(OC)cccc2OC)c(C#N)c1C	nan
	790792	32511	36	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	233	2	1	3	3.4	CCc1c(C)nc2ccc(OC)cc2c1S	nan
	CHEMBL1413735	32511	36	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	233	2	1	3	3.4	CCc1c(C)nc2ccc(OC)cc2c1S	nan
	16015840	32544	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	5	1	4	5.0	Cc1cccc(-c2nc3cc(NC(=O)COc4ccccc4F)ccc3o2)c1	nan
	CHEMBL1413987	32544	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	5	1	4	5.0	Cc1cccc(-c2nc3cc(NC(=O)COc4ccccc4F)ccc3o2)c1	nan
	655034	32640	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	479	8	2	7	2.4	COc1cc(CC(NC(C)=O)C(=O)NC2CCN(c3nc(C)cc(C)c3C#N)CC2)cc(OC)c1	nan
	CHEMBL1414774	32640	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	479	8	2	7	2.4	COc1cc(CC(NC(C)=O)C(=O)NC2CCN(c3nc(C)cc(C)c3C#N)CC2)cc(OC)c1	nan
	16016268	32642	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	471	6	0	8	5.0	COc1ccccc1N1CCN(c2ccc(-c3nc(-c4ccccc4C)no3)cc2[N+](=O)[O-])CC1	nan
	CHEMBL1414801	32642	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	471	6	0	8	5.0	COc1ccccc1N1CCN(c2ccc(-c3nc(-c4ccccc4C)no3)cc2[N+](=O)[O-])CC1	nan
	2156145	32739	11	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	461	6	2	9	4.3	COc1ccc(-n2c(SCC(=O)Nc3cc(C)on3)nc3c4ccccc4nc-3c2O)cc1	nan
	CHEMBL1415709	32739	11	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	461	6	2	9	4.3	COc1ccc(-n2c(SCC(=O)Nc3cc(C)on3)nc3c4ccccc4nc-3c2O)cc1	nan
	7190669	32800	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	5	1	7	3.1	O=C(CSc1ccc2nnc(-c3cccnc3)n2n1)Nc1ccc(F)cc1	nan
	CHEMBL1416264	32800	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	5	1	7	3.1	O=C(CSc1ccc2nnc(-c3cccnc3)n2n1)Nc1ccc(F)cc1	nan
	16012962	32815	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	2	0	6	3.9	Fc1cccc(-n2ncc3c2ncn2nc(-c4ccccc4Cl)nc32)c1	nan
	CHEMBL1416375	32815	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	2	0	6	3.9	Fc1cccc(-n2ncc3c2ncn2nc(-c4ccccc4Cl)nc32)c1	nan
	4808145	32972	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	4	0	7	1.3	Cn1c(=O)c2c(ncn2CCOc2ccc(Br)cc2)n(C)c1=O	nan
	CHEMBL1417778	32972	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	4	0	7	1.3	Cn1c(=O)c2c(ncn2CCOc2ccc(Br)cc2)n(C)c1=O	nan
	16009664	33051	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	5	1	6	4.6	COc1ccc(CNc2nc3c(-c4ccccc4)nnn3c3ccccc23)cc1	nan
	CHEMBL1418446	33051	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	5	1	6	4.6	COc1ccc(CNc2nc3c(-c4ccccc4)nnn3c3ccccc23)cc1	nan
	4625060	33122	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	356	3	2	4	2.2	O=C(CC1N=C2c3ccccc3NC(=S)N2C1=O)NC1CCCCC1	nan
	CHEMBL1419028	33122	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	356	3	2	4	2.2	O=C(CC1N=C2c3ccccc3NC(=S)N2C1=O)NC1CCCCC1	nan
	665236	33168	8	None	-1	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	5	1	7	4.4	CCc1nc(SCC(=O)Nc2ccc3c(c2)OCCO3)c2oc3ccccc3c2n1	nan
	CHEMBL1419387	33168	8	None	-1	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	5	1	7	4.4	CCc1nc(SCC(=O)Nc2ccc3c(c2)OCCO3)c2oc3ccccc3c2n1	nan
	20927027	33185	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	4	1	7	2.0	O=S(=O)(c1ccc(-c2ccc(O)nn2)o1)N1CCN(c2ccccc2)CC1	nan
	CHEMBL1419593	33185	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	4	1	7	2.0	O=S(=O)(c1ccc(-c2ccc(O)nn2)o1)N1CCN(c2ccccc2)CC1	nan
	16024782	33344	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	454	4	0	5	3.9	O=S(=O)(c1ccc2nc(N3CCN(c4ccccc4F)CC3)ccc2c1)N1CCCCC1	nan
	CHEMBL1420848	33344	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	454	4	0	5	3.9	O=S(=O)(c1ccc2nc(N3CCN(c4ccccc4F)CC3)ccc2c1)N1CCCCC1	nan
	3185701	33367	3	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	541	10	3	8	3.0	CCOc1ccc(C(C(=O)NCC2CCCO2)N(C(=O)c2snc(C(N)=O)c2N)c2ccccc2F)cc1	nan
	CHEMBL1421091	33367	3	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	541	10	3	8	3.0	CCOc1ccc(C(C(=O)NCC2CCCO2)N(C(=O)c2snc(C(N)=O)c2N)c2ccccc2F)cc1	nan
	1078539	33618	20	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	351	2	0	7	2.5	Cc1cccc(-n2ncc3c(N4CCC5(CC4)OCCO5)ncnc32)c1	nan
	CHEMBL1423202	33618	20	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	351	2	0	7	2.5	Cc1cccc(-n2ncc3c(N4CCC5(CC4)OCCO5)ncnc32)c1	nan
	993322	33657	15	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	6	1	7	4.2	COc1ccc(-c2cc(C(F)(F)F)nc(SCC(=O)Nc3cc(C)on3)n2)cc1	nan
	CHEMBL1423477	33657	15	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	6	1	7	4.2	COc1ccc(-c2cc(C(F)(F)F)nc(SCC(=O)Nc3cc(C)on3)n2)cc1	nan
	16194711	33867	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	497	8	1	9	1.5	CCOC(=O)N1CCN(C(=O)CSc2ccc3nnc(CCNC(=O)c4ccccc4)n3n2)CC1	nan
	CHEMBL1425185	33867	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	497	8	1	9	1.5	CCOC(=O)N1CCN(C(=O)CSc2ccc3nnc(CCNC(=O)c4ccccc4)n3n2)CC1	nan
	661193	34050	8	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	5	1	7	1.9	Cc1cccc(-n2ncc3c(NCCN4CCOCC4)ncnc32)c1	nan
	CHEMBL1426726	34050	8	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	5	1	7	1.9	Cc1cccc(-n2ncc3c(NCCN4CCOCC4)ncnc32)c1	nan
	2999700	34195	3	None	-1	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	4	1	5	4.6	Cn1c(/C(C#N)=C(\O)COc2ccc3ccccc3c2)nc2ccccc21	nan
	CHEMBL1428087	34195	3	None	-1	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	4	1	5	4.6	Cn1c(/C(C#N)=C(\O)COc2ccc3ccccc3c2)nc2ccccc21	nan
	1371384	34318	10	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	225	1	1	4	2.7	Cc1ccc(/C=C2/SC(=O)NC2=S)o1	nan
	CHEMBL1429158	34318	10	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	225	1	1	4	2.7	Cc1ccc(/C=C2/SC(=O)NC2=S)o1	nan
	2815019	34614	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	317	2	1	8	0.7	Cn1c(=O)c2c(nc(Sc3ccccc3N)n2C)n(C)c1=O	nan
	CHEMBL1431497	34614	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	317	2	1	8	0.7	Cn1c(=O)c2c(nc(Sc3ccccc3N)n2C)n(C)c1=O	nan
	2114663	34657	6	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	4	1	5	5.3	Cc1onc(-c2ccccc2)c1C(=O)Nc1nc(-c2cc(F)ccc2F)cs1	nan
	CHEMBL1431887	34657	6	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	4	1	5	5.3	Cc1onc(-c2ccccc2)c1C(=O)Nc1nc(-c2cc(F)ccc2F)cs1	nan
	650995	34760	13	None	-3	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	4	1	6	4.2	Cc1nonc1NC(=O)CSc1nc2cc(Cl)ccc2c2c1CCCC2	nan
	CHEMBL1432773	34760	13	None	-3	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	4	1	6	4.2	Cc1nonc1NC(=O)CSc1nc2cc(Cl)ccc2c2c1CCCC2	nan
	15989049	34848	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	529	8	1	8	3.9	O=C(CCCn1c(=O)c2sccc2n(Cc2ccc(F)cc2Cl)c1=O)NCc1ccc2c(c1)OCO2	nan
	CHEMBL1433448	34848	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	529	8	1	8	3.9	O=C(CCCn1c(=O)c2sccc2n(Cc2ccc(F)cc2Cl)c1=O)NCc1ccc2c(c1)OCO2	nan
	16009658	34862	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	5	1	6	4.6	O=C(Nc1ccc(OCc2cc(=O)n3c4c(sc3n2)CCCC4)cc1)c1cccc(F)c1	nan
	CHEMBL1433649	34862	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	5	1	6	4.6	O=C(Nc1ccc(OCc2cc(=O)n3c4c(sc3n2)CCCC4)cc1)c1cccc(F)c1	nan
	16030989	34868	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	5	0	7	4.3	COC(=O)c1c(-c2ccc(Cl)cc2)noc1N1CCN(c2ccc(C(C)=O)cc2)CC1	nan
	CHEMBL1433722	34868	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	5	0	7	4.3	COC(=O)c1c(-c2ccc(Cl)cc2)noc1N1CCN(c2ccc(C(C)=O)cc2)CC1	nan
	15990910	34881	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	5	2	4	5.8	CSc1cccc(Nc2cc(C(=O)NC3CCCCC3)c3ccccc3n2)c1	nan
	CHEMBL1433922	34881	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	5	2	4	5.8	CSc1cccc(Nc2cc(C(=O)NC3CCCCC3)c3ccccc3n2)c1	nan
	16008787	34922	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	4	1	5	4.3	COc1ccccc1CNC(=O)c1cc2c(=O)oc3ccc(C)cc3c2s1	nan
	CHEMBL1434647	34922	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	4	1	5	4.3	COc1ccccc1CNC(=O)c1cc2c(=O)oc3ccc(C)cc3c2s1	nan
	16022785	34923	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	481	6	1	8	3.5	Cc1ccc(NC(=O)Cn2c(=O)n(Cc3nc(-c4ccccc4)no3)c(=O)c3ccccc32)c(C)c1	nan
	CHEMBL1434648	34923	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	481	6	1	8	3.5	Cc1ccc(NC(=O)Cn2c(=O)n(Cc3nc(-c4ccccc4)no3)c(=O)c3ccccc32)c(C)c1	nan
	24819144	34928	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	5	0	6	6.0	COC(=O)c1ccc(/C=C/c2c(-c3ccsc3)oc3ccc(N4CCOCC4)cc23)cc1	nan
	CHEMBL1434681	34928	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	5	0	6	6.0	COC(=O)c1ccc(/C=C/c2c(-c3ccsc3)oc3ccc(N4CCOCC4)cc23)cc1	nan
	135546816	34934	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	7	2	6	3.8	CCOc1ccccc1NC(=O)C(C)Sc1nc(-c2ccccc2)c(C#N)c(=O)[nH]1	nan
	CHEMBL1434743	34934	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	7	2	6	3.8	CCOc1ccccc1NC(=O)C(C)Sc1nc(-c2ccccc2)c(C#N)c(=O)[nH]1	nan
	16024519	34952	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	5	1	7	3.7	Cc1ccc(C(=O)c2cn(CC(=O)Nc3ccc4c(c3)OCCO4)c3nc(C)ccc3c2=O)cc1	nan
	CHEMBL1435013	34952	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	5	1	7	3.7	Cc1ccc(C(=O)c2cn(CC(=O)Nc3ccc4c(c3)OCCO4)c3nc(C)ccc3c2=O)cc1	nan
	16018510	34956	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	4	1	5	5.3	COc1cccc(-c2cn3c(n2)sc2cc(C(=O)NC4CCCCC4)ccc23)c1	nan
	CHEMBL1435044	34956	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	4	1	5	5.3	COc1cccc(-c2cn3c(n2)sc2cc(C(=O)NC4CCCCC4)ccc23)c1	nan
	15988487	34966	3	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	2	1	4	4.3	CC1(C)CC(=O)c2cc(-c3nc(-c4ccccc4)cs3)c(=O)[nH]c2C1	nan
	CHEMBL1435109	34966	3	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	2	1	4	4.3	CC1(C)CC(=O)c2cc(-c3nc(-c4ccccc4)cs3)c(=O)[nH]c2C1	nan
	6225711	35031	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	4	2	4	3.6	Cc1cc(O)c2c(C)c(CC(=O)NCc3ccccc3Cl)c(=O)oc2c1	nan
	CHEMBL1435970	35031	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	4	2	4	3.6	Cc1cc(O)c2c(C)c(CC(=O)NCc3ccccc3Cl)c(=O)oc2c1	nan
	15987771	35035	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	519	5	0	5	3.5	CCC(=O)N1CCc2cc(Br)cc(S(=O)(=O)N3CCN(c4ccc(C(C)=O)cc4)CC3)c21	nan
	CHEMBL1436008	35035	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	519	5	0	5	3.5	CCC(=O)N1CCc2cc(Br)cc(S(=O)(=O)N3CCN(c4ccc(C(C)=O)cc4)CC3)c21	nan
	5059361	35054	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	446	2	0	6	4.7	Cc1cccc(-c2nc3ccccc3n3c(-c4ccccc4)c4c(=O)n(C)c(=O)n(C)c4c23)c1	nan
	CHEMBL1436184	35054	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	446	2	0	6	4.7	Cc1cccc(-c2nc3ccccc3n3c(-c4ccccc4)c4c(=O)n(C)c(=O)n(C)c4c23)c1	nan
	4230972	35125	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	543	9	2	7	4.8	CC(C)c1ccc(NC(=O)CSC2=Nc3ccccc3C3=NC(CCC(=O)NCc4ccco4)C(=O)N23)cc1	nan
	CHEMBL1437178	35125	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	543	9	2	7	4.8	CC(C)c1ccc(NC(=O)CSC2=Nc3ccccc3C3=NC(CCC(=O)NCc4ccco4)C(=O)N23)cc1	nan
	16007712	35126	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	530	6	0	6	3.5	CCN(CC)S(=O)(=O)c1ccc2c(c1)c(=O)c(C(=O)N1CCN(c3cc(Cl)ccc3C)CC1)cn2C	nan
	CHEMBL1437207	35126	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	530	6	0	6	3.5	CCN(CC)S(=O)(=O)c1ccc2c(c1)c(=O)c(C(=O)N1CCN(c3cc(Cl)ccc3C)CC1)cn2C	nan
	15988469	35206	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	6	1	6	4.8	COc1ccc(NC(=O)C2CCN(c3ccc(Sc4ccc(C)cc4)nn3)CC2)cc1	nan
	CHEMBL1438027	35206	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	6	1	6	4.8	COc1ccc(NC(=O)C2CCN(c3ccc(Sc4ccc(C)cc4)nn3)CC2)cc1	nan
	3230795	35220	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	3	0	6	4.6	CN(C(=O)CSC1=NC2C(N=N1)c1cc(Br)ccc1N2C)C1CCCCC1	nan
	CHEMBL1438136	35220	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	3	0	6	4.6	CN(C(=O)CSC1=NC2C(N=N1)c1cc(Br)ccc1N2C)C1CCCCC1	nan
	16017737	35431	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	4	1	5	1.9	O=C(Cn1ccn(-c2ccc(F)cc2)c(=O)c1=O)Nc1ccc(F)cc1	nan
	CHEMBL1440044	35431	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	4	1	5	1.9	O=C(Cn1ccn(-c2ccc(F)cc2)c(=O)c1=O)Nc1ccc(F)cc1	nan
	16024943	35476	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	348	4	1	5	4.0	CC(=O)c1ccc(NC(=O)c2ccc3c(c2)nnn3C2CCCC2)cc1	nan
	CHEMBL1440442	35476	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	348	4	1	5	4.0	CC(=O)c1ccc(NC(=O)c2ccc3c(c2)nnn3C2CCCC2)cc1	nan
	16195917	35549	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	5	1	8	0.2	Cn1c(N)c(C(=O)COC(=O)CC2CC3CCC2C3)c(=O)n(C)c1=O	nan
	CHEMBL1441131	35549	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	5	1	8	0.2	Cn1c(N)c(C(=O)COC(=O)CC2CC3CCC2C3)c(=O)n(C)c1=O	nan
	16009208	35644	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	6	1	6	3.2	CCOc1ccc(CNC(=O)Cn2ncc3c(=O)oc4ccc(C)cc4c32)cc1	nan
	CHEMBL1441997	35644	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	6	1	6	3.2	CCOc1ccc(CNC(=O)Cn2ncc3c(=O)oc4ccc(C)cc4c32)cc1	nan
	2980137	35856	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	5	0	7	2.7	COc1ccc(-n2c(SC(C)C(=O)N3CCOCC3)nc3ccccc3c2=O)cc1	nan
	CHEMBL1443960	35856	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	5	0	7	2.7	COc1ccc(-n2c(SC(C)C(=O)N3CCOCC3)nc3ccccc3c2=O)cc1	nan
	2421482	35923	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	491	8	1	9	3.0	CCOC(=O)c1cc(-c2cc(OC)c(OC)c(OC)c2)nc2c1c(=O)[nH]c(=O)n2Cc1ccccc1	nan
	CHEMBL1444560	35923	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	491	8	1	9	3.0	CCOC(=O)c1cc(-c2cc(OC)c(OC)c(OC)c2)nc2c1c(=O)[nH]c(=O)n2Cc1ccccc1	nan
	2136705	35968	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	492	7	1	7	3.8	COc1cc2c(=O)c(S(=O)(=O)c3ccccc3)cn(CC(=O)Nc3ccccc3C)c2cc1OC	nan
	CHEMBL1444994	35968	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	492	7	1	7	3.8	COc1cc2c(=O)c(S(=O)(=O)c3ccccc3)cn(CC(=O)Nc3ccccc3C)c2cc1OC	nan
	4154281	35990	5	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	4	1	5	5.3	O=C(CSc1ncnc2c1sc1ccccc12)Nc1ccc(Br)cc1	nan
	CHEMBL1445182	35990	5	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	4	1	5	5.3	O=C(CSc1ncnc2c1sc1ccccc12)Nc1ccc(Br)cc1	nan
	738863	36017	14	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	316	2	1	4	3.6	O=C(Nc1nc(=O)c2ccccc2s1)c1ccc(Cl)cc1	nan
	CHEMBL1445436	36017	14	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	316	2	1	4	3.6	O=C(Nc1nc(=O)c2ccccc2s1)c1ccc(Cl)cc1	nan
	3151463	36377	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	6	2	7	1.8	COCCCn1c(=N)c(C(=O)NC2CCCC2)cc2c(=O)n3ccccc3nc21	nan
	CHEMBL1448581	36377	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	6	2	7	1.8	COCCCn1c(=N)c(C(=O)NC2CCCC2)cc2c(=O)n3ccccc3nc21	nan
	20903711	36449	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	346	7	1	7	1.1	COCCNC(=O)CCc1nnc2ccc(N3CCC(C)CC3)nn12	nan
	CHEMBL1449064	36449	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	346	7	1	7	1.1	COCCNC(=O)CCc1nnc2ccc(N3CCC(C)CC3)nn12	nan
	9550466	36461	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	426	6	1	4	5.5	Cc1ccc(-n2nc(C)c3c(C)c(CCC(=O)NC(C)c4ccccc4)c(C)nc32)cc1	nan
	CHEMBL1449158	36461	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	426	6	1	4	5.5	Cc1ccc(-n2nc(C)c3c(C)c(CCC(=O)NC(C)c4ccccc4)c(C)nc32)cc1	nan
	1440341	36467	4	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	348	4	1	3	4.8	Cc1cc2cc3c(cc2nc1SCC(=O)Nc1ccccc1)CCC3	nan
	CHEMBL1449215	36467	4	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	348	4	1	3	4.8	Cc1cc2cc3c(cc2nc1SCC(=O)Nc1ccccc1)CCC3	nan
	1034641	36584	10	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	2	1	5	3.8	Cc1ccc(-n2c(N)c(C#N)c(-c3ccc(Cl)cc3)c(C#N)c2=O)cc1	nan
	CHEMBL1450150	36584	10	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	2	1	5	3.8	Cc1ccc(-n2c(N)c(C#N)c(-c3ccc(Cl)cc3)c(C#N)c2=O)cc1	nan
	16009195	36604	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	5	0	5	3.5	CCN(Cc1ccccc1)C(=O)Cn1ncc2c(=O)oc3ccc(C)cc3c21	nan
	CHEMBL1450283	36604	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	5	0	5	3.5	CCN(Cc1ccccc1)C(=O)Cn1ncc2c(=O)oc3ccc(C)cc3c21	nan
	1341628	36666	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	5	1	4	5.8	CC(=O)c1ccc(NC(=O)c2cn(-c3ccccc3)nc2-c2ccc(Br)cc2)cc1	nan
	CHEMBL1450882	36666	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	5	1	4	5.8	CC(=O)c1ccc(NC(=O)c2cn(-c3ccccc3)nc2-c2ccc(Br)cc2)cc1	nan
	16019140	37078	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	497	5	1	8	3.9	Cc1cc(C)cc(NC(=O)Cn2c(=O)n(Cc3ccc4c(c3)OCO4)c(=O)c3oc4ccccc4c32)c1	nan
	CHEMBL1454100	37078	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	497	5	1	8	3.9	Cc1cc(C)cc(NC(=O)Cn2c(=O)n(Cc3ccc4c(c3)OCO4)c(=O)c3oc4ccccc4c32)c1	nan
	16009221	37122	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	498	8	1	7	4.6	CCOc1ccc(NC(=O)Cn2cc(C(=O)c3ccc(CC)cc3)c(=O)c3cc4c(cc32)OCO4)cc1	nan
	CHEMBL1454484	37122	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	498	8	1	7	4.6	CCOc1ccc(NC(=O)Cn2cc(C(=O)c3ccc(CC)cc3)c(=O)c3cc4c(cc32)OCO4)cc1	nan
	16026522	37150	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	6	1	5	4.3	CCOC(=O)c1sc2cccc(F)c2c1S(=O)(=O)NCc1ccccc1Cl	nan
	CHEMBL1454707	37150	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	6	1	5	4.3	CCOC(=O)c1sc2cccc(F)c2c1S(=O)(=O)NCc1ccccc1Cl	nan
	6011252	37192	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	564	12	1	8	4.5	CCCCOc1ccc(C2C(C(=O)c3ccc4c(c3)CC(C)O4)=C(O)C(=O)N2CCCN2CCOCC2)cc1OC	nan
	CHEMBL1455062	37192	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	564	12	1	8	4.5	CCCCOc1ccc(C2C(C(=O)c3ccc4c(c3)CC(C)O4)=C(O)C(=O)N2CCCN2CCOCC2)cc1OC	nan
	16026066	37208	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	465	4	1	4	4.7	CCc1ccccc1NC(=O)C1CCN(C2=NS(=O)(=O)C(c3ccc(C)c(C)c3)=C2C)CC1	nan
	CHEMBL1455235	37208	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	465	4	1	4	4.7	CCc1ccccc1NC(=O)C1CCN(C2=NS(=O)(=O)C(c3ccc(C)c(C)c3)=C2C)CC1	nan
	24819160	37317	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	6	0	6	5.9	COC(=O)c1ccc(/C=C/c2c(-c3ccc(OC)cc3)oc3ccc(N4CCOCC4)cc23)cc1	nan
	CHEMBL1456226	37317	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	6	0	6	5.9	COC(=O)c1ccc(/C=C/c2c(-c3ccc(OC)cc3)oc3ccc(N4CCOCC4)cc23)cc1	nan
	135520065	37512	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	8	2	8	2.5	COC(=O)C(CC(C)C)NC(=O)CSc1nc(O)c(C#N)c(-c2ccccc2)n1	nan
	CHEMBL1457936	37512	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	8	2	8	2.5	COC(=O)C(CC(C)C)NC(=O)CSc1nc(O)c(C#N)c(-c2ccccc2)n1	nan
	2125831	37559	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	308	3	2	2	3.9	CC(=O)c1c(C)[nH]c(C(=O)Nc2ccc(Cl)cc2F)c1C	nan
	CHEMBL1458351	37559	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	308	3	2	2	3.9	CC(=O)c1c(C)[nH]c(C(=O)Nc2ccc(Cl)cc2F)c1C	nan
	1110886	37829	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	479	6	3	5	5.4	CC(=O)Nc1ccc(-c2cc(-c3ccc(NC(C)=O)cc3)nc(-c3ccc(NC(C)=O)cc3)n2)cc1	nan
	CHEMBL1460618	37829	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	479	6	3	5	5.4	CC(=O)Nc1ccc(-c2cc(-c3ccc(NC(C)=O)cc3)nc(-c3ccc(NC(C)=O)cc3)n2)cc1	nan
	17255621	37884	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	5	2	6	3.7	CCOc1ccc(NC(=O)Nc2nc3ccc(S(C)(=O)=O)cc3s2)cc1	nan
	CHEMBL1461095	37884	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	5	2	6	3.7	CCOc1ccc(NC(=O)Nc2nc3ccc(S(C)(=O)=O)cc3s2)cc1	nan
	4437250	37887	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	6	2	2	4.2	CCN=C(S)N(CCc1c(C)[nH]c2ccccc12)Cc1cccnc1	nan
	CHEMBL1461107	37887	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	6	2	2	4.2	CCN=C(S)N(CCc1c(C)[nH]c2ccccc12)Cc1cccnc1	nan
	2784799	38013	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	241	1	1	4	2.5	O=C1C([N+](=O)[O-])=C(O)c2cccc3cccc1c23	nan
	CHEMBL1462267	38013	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	241	1	1	4	2.5	O=C1C([N+](=O)[O-])=C(O)c2cccc3cccc1c23	nan
	1442463	38178	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	3	1	5	4.0	CC(C)(C)c1nc(SCC(=O)N2CC(=O)Nc3ccccc32)c2ccccc2n1	nan
	CHEMBL1463696	38178	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	3	1	5	4.0	CC(C)(C)c1nc(SCC(=O)N2CC(=O)Nc3ccccc32)c2ccccc2n1	nan
	664194	38206	9	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	302	2	0	7	2.7	c1ccc(-n2ncc3c2ncn2nc(-c4ccco4)nc32)cc1	nan
	CHEMBL1463869	38206	9	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	302	2	0	7	2.7	c1ccc(-n2ncc3c2ncn2nc(-c4ccco4)nc32)cc1	nan
	2370579	38271	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	309	4	1	8	-0.4	Cn1c(N)c(C(=O)COC(=O)C2CCCC2)c(=O)n(C)c1=O	nan
	CHEMBL1464368	38271	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	309	4	1	8	-0.4	Cn1c(N)c(C(=O)COC(=O)C2CCCC2)c(=O)n(C)c1=O	nan
	4230513	38313	14	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	5	0	9	0.6	CC(C)Cn1c(CN2CCN(C(=O)c3ccco3)CC2)nc2c1c(=O)n(C)c(=O)n2C	nan
	CHEMBL1464655	38313	14	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	5	0	9	0.6	CC(C)Cn1c(CN2CCN(C(=O)c3ccco3)CC2)nc2c1c(=O)n(C)c(=O)n2C	nan
	1214727	38449	3	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	351	2	1	5	4.2	Cc1c(-c2ccc(Cl)cc2)oc(=O)c2c(N)n(-c3ccccc3)nc12	nan
	CHEMBL1465659	38449	3	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	351	2	1	5	4.2	Cc1c(-c2ccc(Cl)cc2)oc(=O)c2c(N)n(-c3ccccc3)nc12	nan
	4225516	38554	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	363	4	1	5	3.5	O=C(O)c1cccnc1SCc1cn2cc(Br)ccc2n1	nan
	CHEMBL1466534	38554	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	363	4	1	5	3.5	O=C(O)c1cccnc1SCc1cn2cc(Br)ccc2n1	nan
	16020097	38665	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	461	9	1	7	3.3	CCCCN(C)CCNC(=O)c1nn(-c2ccc(OC)cc2)c(=O)c2c1c1ccccc1n2C	nan
	CHEMBL1467366	38665	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	461	9	1	7	3.3	CCCCN(C)CCNC(=O)c1nn(-c2ccc(OC)cc2)c(=O)c2c1c1ccccc1n2C	nan
	3137696	38681	20	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	316	3	0	7	-0.2	COCCn1c(Br)nc2c1c(=O)n(C)c(=O)n2C	nan
	CHEMBL1467508	38681	20	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	316	3	0	7	-0.2	COCCn1c(Br)nc2c1c(=O)n(C)c(=O)n2C	nan
	2396532	38780	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	5	2	9	-0.1	CC(=O)c1c(C)[nH]c(C(=O)OCC(=O)c2c(N)n(C)c(=O)n(C)c2=O)c1C	nan
	CHEMBL1468416	38780	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	5	2	9	-0.1	CC(=O)c1c(C)[nH]c(C(=O)OCC(=O)c2c(N)n(C)c(=O)n(C)c2=O)c1C	nan
	4994172	38905	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	3	2	5	4.0	Nc1cc(C(=O)Nc2ccc(Cl)cc2)ccc1N1CC2CC(C1)c1cccc(=O)n1C2	nan
	CHEMBL1469442	38905	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	3	2	5	4.0	Nc1cc(C(=O)Nc2ccc(Cl)cc2)ccc1N1CC2CC(C1)c1cccc(=O)n1C2	nan
	2517516	39057	7	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	4	1	5	2.7	CC(C)COc1ccc(C(=O)N2C(=O)c3ccc(N)cc3C2=O)cc1	nan
	CHEMBL1470757	39057	7	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	4	1	5	2.7	CC(C)COc1ccc(C(=O)N2C(=O)c3ccc(N)cc3C2=O)cc1	nan
	4968659	39186	7	None	-5	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	519	9	2	6	6.1	CCc1ccc(-c2nc(NC(=O)c3ccc(OCC(=O)Nc4ccc(F)cc4)c(OC)c3)sc2C)cc1	nan
	CHEMBL1471857	39186	7	None	-5	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	519	9	2	6	6.1	CCc1ccc(-c2nc(NC(=O)c3ccc(OCC(=O)Nc4ccc(F)cc4)c(OC)c3)sc2C)cc1	nan
	16032187	39296	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	6	2	8	2.7	Cc1cc(NC(=O)CSc2ncc(C(=O)Nc3ccc(Cl)cc3)c(=O)n2C)no1	nan
	CHEMBL1472946	39296	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	6	2	8	2.7	Cc1cc(NC(=O)CSc2ncc(C(=O)Nc3ccc(Cl)cc3)c(=O)n2C)no1	nan
	16416626	39338	15	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	5	2	6	2.3	O=c1oc2c(CN3CCN(CCO)CC3)c(O)ccc2cc1-c1ccccc1	nan
	7205030	39338	15	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	5	2	6	2.3	O=c1oc2c(CN3CCN(CCO)CC3)c(O)ccc2cc1-c1ccccc1	nan
	CHEMBL1473511	39338	15	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	5	2	6	2.3	O=c1oc2c(CN3CCN(CCO)CC3)c(O)ccc2cc1-c1ccccc1	nan
	16022561	39340	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	489	6	2	7	5.0	Cc1c(Cl)cccc1Nc1nn2c(=O)c3ccc(C(=O)NCCc4ccccc4)cc3nc2s1	nan
	CHEMBL1473551	39340	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	489	6	2	7	5.0	Cc1c(Cl)cccc1Nc1nn2c(=O)c3ccc(C(=O)NCCc4ccccc4)cc3nc2s1	nan
	16025981	39376	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	4	1	5	4.3	O=c1cc2nc(-c3ccccc3F)nc(SCc3ccc(Br)cc3)n2[nH]1	nan
	CHEMBL1474099	39376	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	4	1	5	4.3	O=c1cc2nc(-c3ccccc3F)nc(SCc3ccc(Br)cc3)n2[nH]1	nan
	5302625	39407	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	6	2	5	6.0	CCc1ccc(NC(=O)c2sc3nc(C)cc(C)c3c2NC(=O)c2ccccc2OC)cc1	nan
	CHEMBL1474507	39407	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	6	2	5	6.0	CCc1ccc(NC(=O)c2sc3nc(C)cc(C)c3c2NC(=O)c2ccccc2OC)cc1	nan
	20893081	39445	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	4	1	8	2.1	COc1ccc(NC(=O)C2CCCN2c2nn3c(=O)cc(C)nc3s2)cc1	nan
	CHEMBL1475089	39445	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	4	1	8	2.1	COc1ccc(NC(=O)C2CCCN2c2nn3c(=O)cc(C)nc3s2)cc1	nan
	15988958	39463	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	550	11	2	7	4.5	Cc1ccc(CNC(=O)CCCCCn2c(=O)c3sccc3n(CC(=O)Nc3ccc(C)c(F)c3)c2=O)cc1	nan
	CHEMBL1475354	39463	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	550	11	2	7	4.5	Cc1ccc(CNC(=O)CCCCCn2c(=O)c3sccc3n(CC(=O)Nc3ccc(C)c(F)c3)c2=O)cc1	nan
	16020297	39484	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	557	7	1	6	5.2	COc1ccc(-n2c(=O)c3ccc(C(=O)NCc4ccc(C)cc4)cc3n(Cc3ccc(F)cc3Cl)c2=O)cc1	nan
	CHEMBL1475582	39484	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	557	7	1	6	5.2	COc1ccc(-n2c(=O)c3ccc(C(=O)NCc4ccc(C)cc4)cc3n(Cc3ccc(F)cc3Cl)c2=O)cc1	nan
	16015655	39537	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	489	6	1	6	5.6	COc1ccccc1C(=O)Nc1ccc2nc(SCC(=O)N3CCCc4ccccc43)sc2c1	nan
	CHEMBL1476387	39537	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	489	6	1	6	5.6	COc1ccccc1C(=O)Nc1ccc2nc(SCC(=O)N3CCCc4ccccc43)sc2c1	nan
	15988828	39569	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	3	1	5	4.0	O=C(Nc1cccc(Cl)c1)c1cc(-c2ccc3c(c2)OCO3)on1	nan
	CHEMBL1476787	39569	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	3	1	5	4.0	O=C(Nc1cccc(Cl)c1)c1cc(-c2ccc3c(c2)OCO3)on1	nan
	15988909	39609	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	5	0	7	3.4	COc1cc(OC)cc(-n2c(=O)c3sccc3n(Cc3ccc(F)cc3)c2=O)c1	nan
	CHEMBL1477251	39609	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	5	0	7	3.4	COc1cc(OC)cc(-n2c(=O)c3sccc3n(Cc3ccc(F)cc3)c2=O)c1	nan
	16027484	39625	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	464	6	1	8	3.8	O=C(Nc1ccc(C(=O)OCc2cc(=O)n3nc(C4CC4)sc3n2)cc1)c1cccc(F)c1	nan
	CHEMBL1477385	39625	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	464	6	1	8	3.8	O=C(Nc1ccc(C(=O)OCc2cc(=O)n3nc(C4CC4)sc3n2)cc1)c1cccc(F)c1	nan
	16009837	39633	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	491	5	1	7	4.7	COc1cccc(NC(=O)Cn2c(=O)n(-c3ccc(Cl)cc3)c(=O)c3sc4ccccc4c32)c1	nan
	CHEMBL1477435	39633	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	491	5	1	7	4.7	COc1cccc(NC(=O)Cn2c(=O)n(-c3ccc(Cl)cc3)c(=O)c3sc4ccccc4c32)c1	nan
	663717	39688	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	6	0	7	4.0	CCOCCCn1cnc2c(c1=O)c1nc3ccccc3nc1n2-c1ccc(C)cc1	nan
	CHEMBL1477914	39688	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	6	0	7	4.0	CCOCCCn1cnc2c(c1=O)c1nc3ccccc3nc1n2-c1ccc(C)cc1	nan
	16018985	39703	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	6	1	5	4.3	O=C(NCCc1ccc(Cl)cc1)c1ccc(Cn2c(=O)c3cccn3c3cccnc32)cc1	nan
	CHEMBL1478117	39703	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	6	1	5	4.3	O=C(NCCc1ccc(Cl)cc1)c1ccc(Cn2c(=O)c3cccn3c3cccnc32)cc1	nan
	15988423	39783	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	3	2	4	2.8	COc1ccccc1NC(=O)c1cc2c([nH]c1=O)CC(C)(C)CC2=O	nan
	CHEMBL1478841	39783	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	3	2	4	2.8	COc1ccccc1NC(=O)c1cc2c([nH]c1=O)CC(C)(C)CC2=O	nan
	24819115	39834	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	4	5	6	2.9	Nc1c(Cl)cc(-c2nc3cc(C(=O)NCCO)ccc3c(O)c2O)cc1Cl	nan
	CHEMBL1479302	39834	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	4	5	6	2.9	Nc1c(Cl)cc(-c2nc3cc(C(=O)NCCO)ccc3c(O)c2O)cc1Cl	nan
	2511800	39858	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	7	2	5	4.0	CCOc1ncccc1C(=O)Nc1ccc(C(=O)Nc2ccc(OC)cc2)cc1	nan
	CHEMBL1479469	39858	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	7	2	5	4.0	CCOc1ncccc1C(=O)Nc1ccc(C(=O)Nc2ccc(OC)cc2)cc1	nan
	3352626	40001	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	480	11	1	6	5.3	CCCC[S+]([O-])CC(O)CSc1nc(-c2ccc(OC)cc2)cc(-c2ccccc2)c1C#N	nan
	CHEMBL1480619	40001	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	480	11	1	6	5.3	CCCC[S+]([O-])CC(O)CSc1nc(-c2ccc(OC)cc2)cc(-c2ccccc2)c1C#N	nan
	20957489	40146	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	494	9	1	8	2.0	O=C1CCCN1CCCNc1ccc2nnc(CCC(=O)N3CCN(c4ccc(F)cc4)CC3)n2n1	nan
	CHEMBL1481894	40146	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	494	9	1	8	2.0	O=C1CCCN1CCCNc1ccc2nnc(CCC(=O)N3CCN(c4ccc(F)cc4)CC3)n2n1	nan
	16033868	40151	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	463	6	2	9	4.0	COc1ccccc1Nc1nn2c(=O)c3ccc(C(=O)NCc4cccs4)cc3nc2s1	nan
	CHEMBL1481939	40151	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	463	6	2	9	4.0	COc1ccccc1Nc1nn2c(=O)c3ccc(C(=O)NCc4cccs4)cc3nc2s1	nan
	5297519	40201	18	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	4	1	5	4.4	N#Cc1cc2c(nc1SCC(=O)Nc1ccc(C(F)(F)F)cc1)C1CCN2CC1	nan
	CHEMBL1482409	40201	18	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	4	1	5	4.4	N#Cc1cc2c(nc1SCC(=O)Nc1ccc(C(F)(F)F)cc1)C1CCN2CC1	nan
	16030774	40263	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	6	1	9	1.2	Cn1c(=O)c2c(SCC(=O)NCC3CCCO3)nc(-c3ccccc3F)nc2n(C)c1=O	nan
	CHEMBL1482929	40263	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	6	1	9	1.2	Cn1c(=O)c2c(SCC(=O)NCC3CCCO3)nc(-c3ccccc3F)nc2n(C)c1=O	nan
	16017755	40342	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	6	1	5	2.0	O=C(Cn1ccn(-c2cccc(Cl)c2)c(=O)c1=O)NCCc1ccccc1	nan
	CHEMBL1483603	40342	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	6	1	5	2.0	O=C(Cn1ccn(-c2cccc(Cl)c2)c(=O)c1=O)NCCc1ccccc1	nan
	16015423	40356	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	8	1	6	6.2	COc1cc(C)ccc1OCCSc1nc2ccc(NC(=O)c3ccccc3F)cc2s1	nan
	CHEMBL1483703	40356	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	8	1	6	6.2	COc1cc(C)ccc1OCCSc1nc2ccc(NC(=O)c3ccccc3F)cc2s1	nan
	1477383	40636	11	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	296	2	3	3	2.7	O=C(NC(=S)Nc1cccc2[nH]ncc12)c1ccccc1	nan
	CHEMBL1486203	40636	11	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	296	2	3	3	2.7	O=C(NC(=S)Nc1cccc2[nH]ncc12)c1ccccc1	nan
	16009820	40669	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	3	1	5	4.5	CC(C)Nc1nc2c(-c3cccc(Br)c3)nnn2c2ccccc12	nan
	CHEMBL1486479	40669	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	3	1	5	4.5	CC(C)Nc1nc2c(-c3cccc(Br)c3)nnn2c2ccccc12	nan
	646986	40754	13	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	6	1	5	3.5	O=C(C1=C(O)C(=O)N(CCc2ccccc2)C1c1cccnc1)c1ccco1	nan
	CHEMBL1487207	40754	13	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	6	1	5	3.5	O=C(C1=C(O)C(=O)N(CCc2ccccc2)C1c1cccnc1)c1ccco1	nan
	15996976	40853	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	457	5	2	4	3.0	CC1CCN(S(=O)(=O)c2ccc3[nH]cc(C(=O)NCc4ccc(F)cc4)c(=O)c3c2)CC1	nan
	CHEMBL1487954	40853	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	457	5	2	4	3.0	CC1CCN(S(=O)(=O)c2ccc3[nH]cc(C(=O)NCc4ccc(F)cc4)c(=O)c3c2)CC1	nan
	24260	41012	82	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	224	1	3	3	2.4	Nc1ccc(-c2nc3cc(N)ccc3[nH]2)cc1	nan
	CHEMBL1489074	41012	82	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	224	1	3	3	2.4	Nc1ccc(-c2nc3cc(N)ccc3[nH]2)cc1	nan
	3144653	41019	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	7	1	5	3.8	CCCNC(=O)CSc1nc(-c2ccc(OC)cc2)cc(C(F)(F)F)n1	nan
	CHEMBL1489101	41019	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	7	1	5	3.8	CCCNC(=O)CSc1nc(-c2ccc(OC)cc2)cc(C(F)(F)F)n1	nan
	5079958	41020	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	309	4	1	3	4.6	CCc1ccc(Sc2cc(C(=O)O)c3ccccc3n2)cc1	nan
	CHEMBL1489124	41020	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	309	4	1	3	4.6	CCc1ccc(Sc2cc(C(=O)O)c3ccccc3n2)cc1	nan
	16001343	41062	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	7	1	7	3.3	COc1cc(NC(=O)CSc2cc(=O)n(C)c3ccccc23)cc(OC)c1OC	nan
	CHEMBL1489463	41062	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	7	1	7	3.3	COc1cc(NC(=O)CSc2cc(=O)n(C)c3ccccc23)cc(OC)c1OC	nan
	1327191	41089	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	373	5	2	6	4.8	COc1ccc(OC)c(Nc2nc(-c3ccccc3O)nc3ccccc23)c1	nan
	CHEMBL1489694	41089	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	373	5	2	6	4.8	COc1ccc(OC)c(Nc2nc(-c3ccccc3O)nc3ccccc23)c1	nan
	3151460	41110	17	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	6	2	7	2.2	COCCCn1c(=N)c(C(=O)NC2CCCCC2)cc2c(=O)n3ccccc3nc21	nan
	CHEMBL1489888	41110	17	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	6	2	7	2.2	COCCCn1c(=N)c(C(=O)NC2CCCCC2)cc2c(=O)n3ccccc3nc21	nan
	4282213	41174	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	1	0	5	2.8	CC1CCCN(C(=O)c2cc3c(=O)n4ccccc4nc3s2)C1	nan
	CHEMBL1490341	41174	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	1	0	5	2.8	CC1CCCN(C(=O)c2cc3c(=O)n4ccccc4nc3s2)C1	nan
	28358990	41381	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	482	5	1	6	5.1	CCN1CCN(Cc2c(O)ccc3c(=O)c(Oc4ccccc4Cl)c(C(F)(F)F)oc23)CC1	nan
	5451590	41381	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	482	5	1	6	5.1	CCN1CCN(Cc2c(O)ccc3c(=O)c(Oc4ccccc4Cl)c(C(F)(F)F)oc23)CC1	nan
	CHEMBL1491733	41381	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	482	5	1	6	5.1	CCN1CCN(Cc2c(O)ccc3c(=O)c(Oc4ccccc4Cl)c(C(F)(F)F)oc23)CC1	nan
	16025965	41460	3	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	5	1	10	1.4	CCOC(=O)c1cccc(NC(=O)c2cnc3sc(N4CCOCC4)nn3c2=O)c1	nan
	CHEMBL1492345	41460	3	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	5	1	10	1.4	CCOC(=O)c1cccc(NC(=O)c2cnc3sc(N4CCOCC4)nn3c2=O)c1	nan
	6157069	41526	14	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	7	1	7	3.5	COc1ccc(C(=O)C2=C(O)C(=O)N(Cc3cccnc3)C2c2ccco2)cc1OC	nan
	CHEMBL1492815	41526	14	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	7	1	7	3.5	COc1ccc(C(=O)C2=C(O)C(=O)N(Cc3cccnc3)C2c2ccco2)cc1OC	nan
	12005902	41562	9	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	478	7	1	10	4.1	COc1ccc(-c2nnc3ccc(SCC(=O)Nc4nc5ccccc5s4)nn23)cc1OC	nan
	CHEMBL1493244	41562	9	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	478	7	1	10	4.1	COc1ccc(-c2nnc3ccc(SCC(=O)Nc4nc5ccccc5s4)nn23)cc1OC	nan
	16022789	41573	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	481	6	1	8	3.5	Cc1ccc(NC(=O)Cn2c(=O)n(Cc3nc(-c4ccccc4)no3)c(=O)c3ccccc32)cc1C	nan
	CHEMBL1493335	41573	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	481	6	1	8	3.5	Cc1ccc(NC(=O)Cn2c(=O)n(Cc3nc(-c4ccccc4)no3)c(=O)c3ccccc32)cc1C	nan
	2096572	41638	6	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	5	1	5	5.0	COc1ccc2c(C)cc(SCC(=O)Nc3ncc(Cl)cc3Cl)nc2c1	nan
	CHEMBL1493965	41638	6	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	5	1	5	5.0	COc1ccc2c(C)cc(SCC(=O)Nc3ncc(Cl)cc3Cl)nc2c1	nan
	16026311	41785	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	5	1	5	4.5	CCc1ccc(-n2nc(C)c3c(C)cc(=O)n(CC(=O)Nc4ccc(F)cc4C)c32)cc1	nan
	CHEMBL1495516	41785	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	5	1	5	4.5	CCc1ccc(-n2nc(C)c3c(C)cc(=O)n(CC(=O)Nc4ccc(F)cc4C)c32)cc1	nan
	4258482	41909	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	5	0	5	5.6	Cc1cccc(Cc2c(C)nc3nc(SCc4ccccc4Cl)nn3c2C)c1	nan
	CHEMBL1496672	41909	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	5	0	5	5.6	Cc1cccc(Cc2c(C)nc3nc(SCc4ccccc4Cl)nn3c2C)c1	nan
	17583888	41945	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	6	1	5	3.5	CCCc1cc(=O)oc2c(C)c(OCC(=O)Nc3ccccn3)ccc12	nan
	CHEMBL1496919	41945	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	6	1	5	3.5	CCCc1cc(=O)oc2c(C)c(OCC(=O)Nc3ccccn3)ccc12	nan
	3260315	42015	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	5	1	9	0.6	Cc1ccc(Cl)cc1NC(=O)COC(=O)Cn1cnc2c1c(=O)n(C)c(=O)n2C	nan
	CHEMBL1497548	42015	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	5	1	9	0.6	Cc1ccc(Cl)cc1NC(=O)COC(=O)Cn1cnc2c1c(=O)n(C)c(=O)n2C	nan
	1488204	42305	14	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	441	4	0	5	5.3	O=S(=O)(c1ccccc1)c1cnc(-c2cccnc2)nc1-c1ccc(Cl)c(Cl)c1	nan
	CHEMBL1500120	42305	14	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	441	4	0	5	5.3	O=S(=O)(c1ccccc1)c1cnc(-c2cccnc2)nc1-c1ccc(Cl)c(Cl)c1	nan
	5309910	42835	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	8	2	7	2.2	CCOc1ccc(Cn2nnc(C(=O)NCc3ccc(OC)cc3)c2N)cc1	nan
	CHEMBL1504868	42835	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	8	2	7	2.2	CCOc1ccc(Cn2nnc(C(=O)NCc3ccc(OC)cc3)c2N)cc1	nan
	135422740	42883	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	517	5	1	7	4.8	Nc1c2cnnc-2nc(SCC(=O)c2ccc(Br)cc2)n1-c1ccc(Br)cc1	nan
	CHEMBL1505277	42883	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	517	5	1	7	4.8	Nc1c2cnnc-2nc(SCC(=O)c2ccc(Br)cc2)n1-c1ccc(Br)cc1	nan
	4975174	43433	14	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	5	0	7	1.2	COCCCn1c(C(=O)N2CCOCC2)cc2c(=O)n3ccccc3nc21	nan
	CHEMBL1510079	43433	14	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	5	0	7	1.2	COCCCn1c(C(=O)N2CCOCC2)cc2c(=O)n3ccccc3nc21	nan
	6236457	43457	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	523	7	1	10	4.0	COc1cc(C2C(C(=O)c3ccc4c(c3)CC(C)O4)=C(O)C(=O)N2c2nnc(C)s2)cc(OC)c1OC	nan
	CHEMBL1510318	43457	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	523	7	1	10	4.0	COc1cc(C2C(C(=O)c3ccc4c(c3)CC(C)O4)=C(O)C(=O)N2c2nnc(C)s2)cc(OC)c1OC	nan
	135399378	43485	16	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	4	2	7	2.5	CCOc1ccc(N2CC(=O)C(c3nc(O)c4ccccc4n3)=C2N)cc1	nan
	CHEMBL1510511	43485	16	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	4	2	7	2.5	CCOc1ccc(N2CC(=O)C(c3nc(O)c4ccccc4n3)=C2N)cc1	nan
	16026527	43663	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	6	1	6	3.7	COc1ccc(CNC(=O)C(C)n2c(=O)cc(C)c3c(C)nn(-c4ccccc4)c32)cc1	nan
	CHEMBL1512255	43663	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	6	1	6	3.7	COc1ccc(CNC(=O)C(C)n2c(=O)cc(C)c3c(C)nn(-c4ccccc4)c32)cc1	nan
	16012611	43682	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	4	1	4	4.8	Cc1nc2c(c(C)nn2C(C)(C)C)c(C)c1CCC(=O)Nc1ccc(F)cc1	nan
	CHEMBL1512506	43682	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	4	1	4	4.8	Cc1nc2c(c(C)nn2C(C)(C)C)c(C)c1CCC(=O)Nc1ccc(F)cc1	nan
	4405319	43713	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	5	1	4	6.3	CCOc1ccc(C(=O)Nc2ccc3oc(-c4cccc5ccccc45)nc3c2)cc1	nan
	CHEMBL1512869	43713	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	5	1	4	6.3	CCOc1ccc(C(=O)Nc2ccc3oc(-c4cccc5ccccc45)nc3c2)cc1	nan
	16024551	43740	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	503	7	1	7	4.4	CCOC(=O)c1ccc(NC(=O)Cn2cc(C(=O)c3ccc(Cl)cc3)c(=O)c3ccc(C)nc32)cc1	nan
	CHEMBL1513333	43740	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	503	7	1	7	4.4	CCOC(=O)c1ccc(NC(=O)Cn2cc(C(=O)c3ccc(Cl)cc3)c(=O)c3ccc(C)nc32)cc1	nan
	135416471	43747	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	276	1	1	4	2.5	Cc1ccc(-c2nc3c4ccccc4[nH]c(=O)n3n2)cc1	nan
	CHEMBL1513443	43747	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	276	1	1	4	2.5	Cc1ccc(-c2nc3c4ccccc4[nH]c(=O)n3n2)cc1	nan
	1306158	43769	19	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	5	1	5	5.2	COc1cc(OC)cc(C(=O)Nc2ccccc2-c2nc3ccccc3s2)c1	nan
	CHEMBL1513732	43769	19	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	5	1	5	5.2	COc1cc(OC)cc(C(=O)Nc2ccccc2-c2nc3ccccc3s2)c1	nan
	1887235	43805	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	6	1	5	4.8	COc1ccc(NC(=O)CCn2nc(-c3ccc(Cl)cc3)c3ccccc3c2=O)cc1	nan
	CHEMBL1514436	43805	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	6	1	5	4.8	COc1ccc(NC(=O)CCn2nc(-c3ccc(Cl)cc3)c3ccccc3c2=O)cc1	nan
	2158481	43817	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	363	2	1	5	4.1	Cc1cccc(NC(=O)c2cc3c(=O)n4cccc(C)c4nc3s2)c1C	nan
	CHEMBL1514582	43817	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	363	2	1	5	4.1	Cc1cccc(NC(=O)c2cc3c(=O)n4cccc(C)c4nc3s2)c1C	nan
	2134751	43818	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	539	10	1	8	4.5	O=C(CCCCCn1c(=O)c2sccc2n(Cc2ccccc2Cl)c1=O)NCc1ccc2c(c1)OCO2	nan
	CHEMBL1514595	43818	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	539	10	1	8	4.5	O=C(CCCCCn1c(=O)c2sccc2n(Cc2ccccc2Cl)c1=O)NCc1ccc2c(c1)OCO2	nan
	7990486	43821	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	8	1	6	2.5	COc1cccc(CNC(=O)COC(=O)/C(C#N)=C/c2ccc(N(C)C)cc2)c1	nan
	CHEMBL1514625	43821	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	8	1	6	2.5	COc1cccc(CNC(=O)COC(=O)/C(C#N)=C/c2ccc(N(C)C)cc2)c1	nan
	16016989	43834	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	4	1	5	4.1	Cc1ccc(CNC(=O)C(C)n2nc(C)c3sc4ccccc4c3c2=O)cc1	nan
	CHEMBL1514781	43834	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	4	1	5	4.1	Cc1ccc(CNC(=O)C(C)n2nc(C)c3sc4ccccc4c3c2=O)cc1	nan
	4246910	43841	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	7	0	10	0.0	CCOCCn1c(CN2CCN(C(=O)c3ccco3)CC2)nc2c1c(=O)n(C)c(=O)n2C	nan
	CHEMBL1514858	43841	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	7	0	10	0.0	CCOCCn1c(CN2CCN(C(=O)c3ccco3)CC2)nc2c1c(=O)n(C)c(=O)n2C	nan
	16030776	43845	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	5	1	10	1.9	Cc1cc(NC(=O)CSc2nc(-c3ccccc3F)nc3c2c(=O)n(C)c(=O)n3C)no1	nan
	CHEMBL1514941	43845	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	5	1	10	1.9	Cc1cc(NC(=O)CSc2nc(-c3ccccc3F)nc3c2c(=O)n(C)c(=O)n3C)no1	nan
	16022121	43868	3	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	466	4	0	7	2.9	COc1ccc2c(c1)c1c(c(=O)n(-c3cccc(Cl)c3)c(=O)n1CC(=O)N1CCCC1)n2C	nan
	CHEMBL1515298	43868	3	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	466	4	0	7	2.9	COc1ccc2c(c1)c1c(c(=O)n(-c3cccc(Cl)c3)c(=O)n1CC(=O)N1CCCC1)n2C	nan
	6418314	43874	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	454	7	1	5	5.4	CCC(Sc1nnc(-c2ccc(F)cc2)c(-c2ccc(F)cc2)n1)C(=O)NC1CCCC1	nan
	CHEMBL1515335	43874	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	454	7	1	5	5.4	CCC(Sc1nnc(-c2ccc(F)cc2)c(-c2ccc(F)cc2)n1)C(=O)NC1CCCC1	nan
	16031608	43883	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	471	6	2	6	2.6	COc1ccc(NC(=O)C2CCN(S(=O)(=O)c3ccc4[nH]c(=O)ccc4c3)CC2)c(OC)c1	nan
	CHEMBL1515521	43883	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	471	6	2	6	2.6	COc1ccc(NC(=O)C2CCN(S(=O)(=O)c3ccc4[nH]c(=O)ccc4c3)CC2)c(OC)c1	nan
	16014254	43890	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	480	8	2	6	3.2	NS(=O)(=O)c1ccc(CCNC(=O)c2nc(SCc3ccccc3F)ncc2Cl)cc1	nan
	CHEMBL1515689	43890	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	480	8	2	6	3.2	NS(=O)(=O)c1ccc(CCNC(=O)c2nc(SCc3ccccc3F)ncc2Cl)cc1	nan
	16009753	43901	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	1	0	5	3.8	Cn1c(=O)n(-c2ccc(Br)cc2F)c(=O)c2sc3ccccc3c21	nan
	CHEMBL1515791	43901	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	1	0	5	3.8	Cn1c(=O)n(-c2ccc(Br)cc2F)c(=O)c2sc3ccccc3c21	nan
	16029066	43913	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	5	1	5	3.0	CC(=O)c1ccc(NC(=O)c2cc(S(=O)(=O)N3CCCCCC3)cn2C)cc1	nan
	CHEMBL1515983	43913	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	5	1	5	3.0	CC(=O)c1ccc(NC(=O)c2cc(S(=O)(=O)N3CCCCCC3)cn2C)cc1	nan
	16027656	43920	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	7	1	9	4.0	CC(C)Cc1nn2c(=O)cc(COC(=O)c3cccc(NC(=O)c4cccs4)c3)nc2s1	nan
	CHEMBL1516060	43920	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	7	1	9	4.0	CC(C)Cc1nn2c(=O)cc(COC(=O)c3cccc(NC(=O)c4cccs4)c3)nc2s1	nan
	16030468	43935	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	7	1	6	3.9	Cc1ccc(OCC(=O)Nc2ccccc2OCc2cc(=O)n3ccccc3n2)cc1C	nan
	CHEMBL1516233	43935	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	7	1	6	3.9	Cc1ccc(OCC(=O)Nc2ccccc2OCc2cc(=O)n3ccccc3n2)cc1C	nan
	15990035	43936	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	6	2	7	3.2	CC(C)CCNC(=O)c1cccc(Nc2nc3ccccc3n3nnnc23)c1	nan
	CHEMBL1516237	43936	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	6	2	7	3.2	CC(C)CCNC(=O)c1cccc(Nc2nc3ccccc3n3nnnc23)c1	nan
	6220215	43983	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	320	1	2	3	3.2	CC1=CC2=NC(=O)/C(=C/c3c(C)[nH]c4ccc(C)cc34)C(=N)N2O1	nan
	CHEMBL1516846	43983	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	320	1	2	3	3.2	CC1=CC2=NC(=O)/C(=C/c3c(C)[nH]c4ccc(C)cc34)C(=N)N2O1	nan
	3238933	44032	6	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	4	2	5	4.8	O=C(Nc1c(C(=O)Nc2cccc(F)c2)oc2ccccc12)c1ccc2c(c1)OCO2	nan
	CHEMBL1517304	44032	6	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	4	2	5	4.8	O=C(Nc1c(C(=O)Nc2cccc(F)c2)oc2ccccc12)c1ccc2c(c1)OCO2	nan
	24687299	44094	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	5	1	6	3.9	CC(=O)c1sc(NC(=O)c2cccc(N3C(=O)CCC3=O)c2)nc1-c1ccccc1	nan
	CHEMBL1517943	44094	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	5	1	6	3.9	CC(=O)c1sc(NC(=O)c2cccc(N3C(=O)CCC3=O)c2)nc1-c1ccccc1	nan
	16009652	44110	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	4	2	4	5.8	O=C(Nc1c(C(=O)Nc2ccccc2F)oc2ccccc12)c1cc2ccccc2o1	nan
	CHEMBL1518097	44110	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	4	2	4	5.8	O=C(Nc1c(C(=O)Nc2ccccc2F)oc2ccccc12)c1cc2ccccc2o1	nan
	3298558	44150	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	480	7	1	7	3.7	O=C(CCCCCn1c(=S)[nH]c2cc3c(cc2c1=O)OCO3)N1CCN(c2ccccc2)CC1	nan
	CHEMBL1518549	44150	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	480	7	1	7	3.7	O=C(CCCCCn1c(=S)[nH]c2cc3c(cc2c1=O)OCO3)N1CCN(c2ccccc2)CC1	nan
	5286935	44165	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	318	2	2	4	2.4	Cc1ccc(NC(=O)/C(C#N)=C(\N)C(Cl)(Cl)Cl)nc1	nan
	CHEMBL1518626	44165	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	318	2	2	4	2.4	Cc1ccc(NC(=O)/C(C#N)=C(\N)C(Cl)(Cl)Cl)nc1	nan
	16031509	44213	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	6	1	6	4.6	COc1ccc(-c2nnc(SCC(=O)Nc3ccc(Cl)cc3)s2)cc1	nan
	CHEMBL1519036	44213	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	6	1	6	4.6	COc1ccc(-c2nnc(SCC(=O)Nc3ccc(Cl)cc3)s2)cc1	nan
	938163	44253	12	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	317	2	1	5	3.2	CC(=O)Nc1cccc(-c2nnc3c4ccccc4c(C)nn23)c1	nan
	CHEMBL1519354	44253	12	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	317	2	1	5	3.2	CC(=O)Nc1cccc(-c2nnc3c4ccccc4c(C)nn23)c1	nan
	2473851	44254	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	9	2	6	2.5	COc1cc(C(=O)NCCNC(=O)c2cc(OC)c(C)c(OC)c2)cc(OC)c1C	nan
	CHEMBL1519363	44254	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	9	2	6	2.5	COc1cc(C(=O)NCCNC(=O)c2cc(OC)c(C)c(OC)c2)cc(OC)c1C	nan
	24687548	44345	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	7	1	10	2.1	COc1ccc(OC)c(-c2csc(NC(=O)CSc3nnnn3C)n2)c1	nan
	CHEMBL1520201	44345	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	7	1	10	2.1	COc1ccc(OC)c(-c2csc(NC(=O)CSc3nnnn3C)n2)c1	nan
	1142116	44349	11	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	5	1	4	4.7	O=C(CSc1nc2c(c(C(F)(F)F)n1)CCc1ccccc1-2)NCc1ccccc1	nan
	CHEMBL1520265	44349	11	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	5	1	4	4.7	O=C(CSc1nc2c(c(C(F)(F)F)n1)CCc1ccccc1-2)NCc1ccccc1	nan
	2577415	44609	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	7	0	8	2.4	CN(C)S(=O)(=O)c1ccc(C(=O)OCC(=O)c2csc(N3CCCCC3)n2)cc1	nan
	CHEMBL1522536	44609	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	7	0	8	2.4	CN(C)S(=O)(=O)c1ccc(C(=O)OCC(=O)c2csc(N3CCCCC3)n2)cc1	nan
	16027586	44774	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	8	1	8	3.6	CCc1nn2c(=O)cc(COC(=O)c3ccc(NC(=O)CCc4ccccc4)cc3)nc2s1	nan
	CHEMBL1524058	44774	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	8	1	8	3.6	CCc1nn2c(=O)cc(COC(=O)c3ccc(NC(=O)CCc4ccccc4)cc3)nc2s1	nan
	22581682	44799	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	396	6	1	6	3.9	COc1ccc(-c2cn3nc(SCC(=O)NC4CCCCC4)ccc3n2)cc1	nan
	CHEMBL1524339	44799	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	396	6	1	6	3.9	COc1ccc(-c2cn3nc(SCC(=O)NC4CCCCC4)ccc3n2)cc1	nan
	2814763	44811	14	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	288	2	2	1	4.2	O=C(Nc1ccc(F)cc1)c1cc2cc(Cl)ccc2[nH]1	nan
	CHEMBL1524425	44811	14	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	288	2	2	1	4.2	O=C(Nc1ccc(F)cc1)c1cc2cc(Cl)ccc2[nH]1	nan
	16012570	44878	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	5	1	5	4.4	Cc1cc(C)c2c(n1)nn1c(C)c(CCC(=O)NCc3ccccc3Cl)c(C)nc21	nan
	CHEMBL1525143	44878	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	5	1	5	4.4	Cc1cc(C)c2c(n1)nn1c(C)c(CCC(=O)NCc3ccccc3Cl)c(C)nc21	nan
	3119681	45182	15	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	5	2	3	6.1	O=C(Cc1ccccc1)Nc1sc2c(c1C(=O)Nc1cccc(Cl)c1)CCCCC2	nan
	CHEMBL1527765	45182	15	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	5	2	3	6.1	O=C(Cc1ccccc1)Nc1sc2c(c1C(=O)Nc1cccc(Cl)c1)CCCCC2	nan
	3370309	45363	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	9	2	7	3.5	CCN(CCCNC(=O)CCn1c(=S)[nH]c2cc3c(cc2c1=O)OCO3)c1cccc(C)c1	nan
	CHEMBL1529348	45363	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	9	2	7	3.5	CCN(CCCNC(=O)CCn1c(=S)[nH]c2cc3c(cc2c1=O)OCO3)c1cccc(C)c1	nan
	3178487	45418	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	4	0	8	0.8	CCn1c(SCC(=O)N2CCC(C)CC2)nc2c1c(=O)n(C)c(=O)n2C	nan
	CHEMBL1529806	45418	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	4	0	8	0.8	CCn1c(SCC(=O)N2CCC(C)CC2)nc2c1c(=O)n(C)c(=O)n2C	nan
	3161332	45668	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	4	1	4	5.4	COc1ccc(-c2nc3ccccc3s2)cc1NC(=O)c1ccccc1F	nan
	CHEMBL1532063	45668	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	4	1	4	5.4	COc1ccc(-c2nc3ccccc3s2)cc1NC(=O)c1ccccc1F	nan
	3787408	45771	9	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	534	8	1	7	5.3	CCCCn1c(NS(=O)(=O)c2ccc(C)cc2)c(S(=O)(=O)c2ccccc2)c2nc3ccccc3nc21	nan
	CHEMBL1532953	45771	9	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	534	8	1	7	5.3	CCCCn1c(NS(=O)(=O)c2ccc(C)cc2)c(S(=O)(=O)c2ccccc2)c2nc3ccccc3nc21	nan
	2105095	45772	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	6	1	7	3.7	Cc1cc(NC(=O)CSc2nc3cc(Cl)ccc3c(=O)n2CC(C)C)no1	nan
	CHEMBL1532957	45772	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	6	1	7	3.7	Cc1cc(NC(=O)CSc2nc3cc(Cl)ccc3c(=O)n2CC(C)C)no1	nan
	2965497	45775	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	536	4	0	5	4.2	O=C(c1cc(-c2ccccn2)nc2ccc(Br)cc12)N1CCN(S(=O)(=O)c2ccccc2)CC1	nan
	CHEMBL1532981	45775	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	536	4	0	5	4.2	O=C(c1cc(-c2ccccn2)nc2ccc(Br)cc12)N1CCN(S(=O)(=O)c2ccccc2)CC1	nan
	16019855	45828	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	304	2	0	5	3.8	Cc1ccccc1-c1noc(-c2cc3ccccc3oc2=O)n1	nan
	CHEMBL1533477	45828	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	304	2	0	5	3.8	Cc1ccccc1-c1noc(-c2cc3ccccc3oc2=O)n1	nan
	17374586	46288	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	373	4	0	4	3.5	CCC(Oc1cc(Cl)ccc1Cl)C(=O)N1CCC2(CC1)OCCO2	nan
	CHEMBL1537906	46288	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	373	4	0	4	3.5	CCC(Oc1cc(Cl)ccc1Cl)C(=O)N1CCC2(CC1)OCCO2	nan
	1078178	46594	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	7	2	6	3.2	COc1cc(OC)cc(C(=O)Nc2ccc(S(=O)(=O)Nc3ccccn3)cc2)c1	nan
	CHEMBL1540495	46594	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	7	2	6	3.2	COc1cc(OC)cc(C(=O)Nc2ccc(S(=O)(=O)Nc3ccccn3)cc2)c1	nan
	721260	46628	35	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	222	2	1	5	1.7	CCOC(=O)c1cc(C#N)c(S)nc1C	nan
	CHEMBL1540818	46628	35	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	222	2	1	5	1.7	CCOC(=O)c1cc(C#N)c(S)nc1C	nan
	657993	46640	14	None	-31	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	282	2	1	4	3.4	COc1ccc(-c2c(C#N)c(S)nc3c2CCC3)cc1	nan
	CHEMBL1540912	46640	14	None	-31	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	282	2	1	4	3.4	COc1ccc(-c2c(C#N)c(S)nc3c2CCC3)cc1	nan
	1356173	47087	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	4	2	4	4.8	CCOC(=O)c1c(N=C(S)Nc2ccc(C)cc2)sc2c1CCC2	nan
	CHEMBL1544543	47087	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	4	2	4	4.8	CCOC(=O)c1c(N=C(S)Nc2ccc(C)cc2)sc2c1CCC2	nan
	16195345	47217	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	500	8	2	8	0.4	Cn1c(=O)c2cc(S(=O)(=O)NC(Cc3ccccc3)C(=O)NCC3CCCO3)ccc2n(C)c1=O	nan
	CHEMBL1545503	47217	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	500	8	2	8	0.4	Cn1c(=O)c2cc(S(=O)(=O)NC(Cc3ccccc3)C(=O)NCC3CCCO3)ccc2n(C)c1=O	nan
	2868878	47232	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	3	1	3	4.1	CC(=O)C1=C(O)C(=O)N(c2ccc(Br)cc2)C1c1cccc(F)c1	nan
	CHEMBL1545607	47232	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	3	1	3	4.1	CC(=O)C1=C(O)C(=O)N(c2ccc(Br)cc2)C1c1cccc(F)c1	nan
	3186499	47252	4	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	5	1	8	3.5	CCc1nnc(NC(=O)CSc2nc3cc4c(cc3cc2C)OCCO4)s1	nan
	CHEMBL1545790	47252	4	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	5	1	8	3.5	CCc1nnc(NC(=O)CSc2nc3cc4c(cc3cc2C)OCCO4)s1	nan
	1485832	47320	12	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	2	1	4	4.6	O=C(Nc1ccccc1)c1cc2c(=O)c3ccccc3oc2nc1C(F)(F)F	nan
	CHEMBL1546403	47320	12	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	2	1	4	4.6	O=C(Nc1ccccc1)c1cc2c(=O)c3ccccc3oc2nc1C(F)(F)F	nan
	24892595	47499	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	426	7	2	7	3.8	COCCn1c(SCC(=O)Nc2cccc(F)c2)nc2c3ccccc3nc-2c1O	nan
	CHEMBL1548166	47499	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	426	7	2	7	3.8	COCCn1c(SCC(=O)Nc2cccc(F)c2)nc2c3ccccc3nc-2c1O	nan
	4223534	47519	3	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	300	3	1	2	4.5	CC1(C)C(CSc2nc3ccccc3[nH]2)C1(Cl)Cl	nan
	CHEMBL1548301	47519	3	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	300	3	1	2	4.5	CC1(C)C(CSc2nc3ccccc3[nH]2)C1(Cl)Cl	nan
	818439	47595	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	248	1	2	7	1.1	COC(=O)c1sc2nc(N)c(C#N)cc2c1N	nan
	CHEMBL1548988	47595	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	248	1	2	7	1.1	COC(=O)c1sc2nc(N)c(C#N)cc2c1N	nan
	1417035	47666	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	4	1	8	1.0	Cn1c(=O)c2c(nc(SCc3ccc(C(=O)O)cc3)n2C)n(C)c1=O	nan
	CHEMBL1549569	47666	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	4	1	8	1.0	Cn1c(=O)c2c(nc(SCc3ccc(C(=O)O)cc3)n2C)n(C)c1=O	nan
	1838684	47698	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	6	1	6	4.3	O=C(COc1ccc(Cl)cc1)NCc1nnc2c3ccccc3c(-c3ccccc3)nn12	nan
	CHEMBL1549821	47698	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	6	1	6	4.3	O=C(COc1ccc(Cl)cc1)NCc1nnc2c3ccccc3c(-c3ccccc3)nn12	nan
	1777240	47851	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	4	1	5	2.3	Cc1cc(OCC(=O)N2CCC(C(=O)O)CC2)c2c3c(c(=O)oc2c1)CCC3	nan
	CHEMBL1551078	47851	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	4	1	5	2.3	Cc1cc(OCC(=O)N2CCC(C(=O)O)CC2)c2c3c(c(=O)oc2c1)CCC3	nan
	16009855	47895	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	495	5	1	6	4.5	O=C(Cn1c(=O)n(Cc2ccc(F)cc2)c(=O)c2sc3ccccc3c21)Nc1ccc(F)cc1F	nan
	CHEMBL1551826	47895	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	495	5	1	6	4.5	O=C(Cn1c(=O)n(Cc2ccc(F)cc2)c(=O)c2sc3ccccc3c21)Nc1ccc(F)cc1F	nan
	16030710	47901	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	518	5	1	9	3.3	COC(=O)c1ccc(NC(=O)N2CCN(Cc3cc(=O)n4nc(-c5ccc(C)cc5)sc4n3)CC2)cc1	nan
	CHEMBL1551878	47901	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	518	5	1	9	3.3	COC(=O)c1ccc(NC(=O)N2CCN(Cc3cc(=O)n4nc(-c5ccc(C)cc5)sc4n3)CC2)cc1	nan
	1004076	47904	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	4	2	5	5.3	COc1ccc(-c2ccc3c(N)c(C(=O)Nc4cc(F)ccc4C)sc3n2)cc1	nan
	CHEMBL1551914	47904	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	4	2	5	5.3	COc1ccc(-c2ccc3c(N)c(C(=O)Nc4cc(F)ccc4C)sc3n2)cc1	nan
	7222625	47965	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	5	1	6	4.4	Cc1nc(C)c(-c2ccc(SCC(=O)Nc3ccc(C)c(F)c3)nn2)s1	nan
	CHEMBL1552706	47965	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	5	1	6	4.4	Cc1nc(C)c(-c2ccc(SCC(=O)Nc3ccc(C)c(F)c3)nn2)s1	nan
	16010352	48001	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	8	1	4	4.6	CCOC(=O)c1c(C)c(-c2ccccc2)n(CC(=O)NCCc2cccc(C)c2)c1C	nan
	CHEMBL1553141	48001	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	8	1	4	4.6	CCOC(=O)c1c(C)c(-c2ccccc2)n(CC(=O)NCCc2cccc(C)c2)c1C	nan
	16030832	48055	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	3	1	4	4.2	O=C(Nc1ccccc1C(=O)N1CCCCC1)c1nsc2ccccc12	nan
	CHEMBL1553983	48055	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	3	1	4	4.2	O=C(Nc1ccccc1C(=O)N1CCCCC1)c1nsc2ccccc12	nan
	16012075	48061	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	6	1	6	4.2	CC(=O)c1ccc(NC(=O)Cn2ncc3c4ccccc4n(Cc4ccccc4)c3c2=O)cc1	nan
	CHEMBL1554061	48061	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	6	1	6	4.2	CC(=O)c1ccc(NC(=O)Cn2ncc3c4ccccc4n(Cc4ccccc4)c3c2=O)cc1	nan
	16008778	48063	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	487	7	0	9	1.9	CCOC(=O)Cn1c(=O)oc2cc(S(=O)(=O)N3CCN(c4ccc(C(C)=O)cc4)CC3)ccc21	nan
	CHEMBL1554084	48063	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	487	7	0	9	1.9	CCOC(=O)Cn1c(=O)oc2cc(S(=O)(=O)N3CCN(c4ccc(C(C)=O)cc4)CC3)ccc21	nan
	3147967	48067	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	363	4	1	6	3.6	Cc1cccc(NC(=O)CSc2nnc3c4ccccc4n(C)c3n2)c1	nan
	CHEMBL1554132	48067	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	363	4	1	6	3.6	Cc1cccc(NC(=O)CSc2nnc3c4ccccc4n(C)c3n2)c1	nan
	1222858	48074	15	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	7	1	8	3.3	COC(=O)c1sc(NC(=O)/C=C/c2ccc(OC)c(OC)c2)c(C(=O)OC)c1C	nan
	CHEMBL1554200	48074	15	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	7	1	8	3.3	COC(=O)c1sc(NC(=O)/C=C/c2ccc(OC)c(OC)c2)c(C(=O)OC)c1C	nan
	16027476	48075	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	7	1	9	3.6	COc1ccccc1C(=O)Nc1ccc(C(=O)OCc2cc(=O)n3nc(C4CC4)sc3n2)cc1	nan
	CHEMBL1554206	48075	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	7	1	9	3.6	COc1ccccc1C(=O)Nc1ccc(C(=O)OCc2cc(=O)n3nc(C4CC4)sc3n2)cc1	nan
	15989095	48076	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	10	2	7	2.2	NC(=O)Cn1c(=O)n(CCCCCC(=O)NCc2ccccc2Cl)c(=O)c2sccc21	nan
	CHEMBL1554211	48076	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	10	2	7	2.2	NC(=O)Cn1c(=O)n(CCCCCC(=O)NCc2ccccc2Cl)c(=O)c2sccc21	nan
	15991109	48081	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	5	1	3	5.2	Cc1ccc2c(c1)c(=O)c1ccccc1n2CCCC(=O)Nc1ccc(F)cc1F	nan
	CHEMBL1554314	48081	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	5	1	3	5.2	Cc1ccc2c(c1)c(=O)c1ccccc1n2CCCC(=O)Nc1ccc(F)cc1F	nan
	3503858	48089	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	471	7	1	6	5.3	CCC(C)NC(=O)CSc1nc2c(sc3ccccc32)c(=O)n1Cc1ccccc1Cl	nan
	CHEMBL1554470	48089	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	471	7	1	6	5.3	CCC(C)NC(=O)CSc1nc2c(sc3ccccc32)c(=O)n1Cc1ccccc1Cl	nan
	16024920	48124	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	472	7	1	5	5.0	CCCOc1ccc(CNC(=O)C2CCN(c3nc4ccccc4nc3C(F)(F)F)CC2)cc1	nan
	CHEMBL1555031	48124	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	472	7	1	5	5.0	CCCOc1ccc(CNC(=O)C2CCN(c3nc4ccccc4nc3C(F)(F)F)CC2)cc1	nan
	16009072	48132	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	4	1	4	2.8	CCOc1ccc(S(=O)(=O)c2c[nH]c3ccccc3c2=O)cc1	nan
	CHEMBL1555115	48132	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	4	1	4	2.8	CCOc1ccc(S(=O)(=O)c2c[nH]c3ccccc3c2=O)cc1	nan
	16015125	48135	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	5	1	5	4.6	Cc1ccc(OCC(=O)Nc2nc(-c3ccc(Br)cc3)ns2)cc1C	nan
	CHEMBL1555140	48135	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	5	1	5	4.6	Cc1ccc(OCC(=O)Nc2nc(-c3ccc(Br)cc3)ns2)cc1C	nan
	9550626	48178	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	7	1	7	3.9	CCOC(=O)c1c(NC(=O)c2cc(CC(C)C)on2)sc(C(C)=O)c1C	nan
	CHEMBL1555685	48178	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	7	1	7	3.9	CCOC(=O)c1c(NC(=O)c2cc(CC(C)C)on2)sc(C(C)=O)c1C	nan
	2176795	48219	15	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	5	2	5	3.8	Cc1onc(-c2ccccc2Cl)c1C(=O)NC(=S)NCC(=O)c1ccccc1	nan
	CHEMBL1556085	48219	15	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	5	2	5	3.8	Cc1onc(-c2ccccc2Cl)c1C(=O)NC(=S)NCC(=O)c1ccccc1	nan
	16022893	48354	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	5	1	6	4.8	Cc1ccc(-n2nc3c(N4CCC(C(=O)NC(C)c5ccccc5)CC4)nnc(C)c3c2C)cc1	nan
	CHEMBL1557305	48354	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	5	1	6	4.8	Cc1ccc(-n2nc3c(N4CCC(C(=O)NC(C)c5ccccc5)CC4)nnc(C)c3c2C)cc1	nan
	16011715	48422	3	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	294	2	1	6	2.9	Cc1cc(F)ccc1Nc1nc2ccccc2n2nnnc12	nan
	CHEMBL1557862	48422	3	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	294	2	1	6	2.9	Cc1cc(F)ccc1Nc1nc2ccccc2n2nnnc12	nan
	15989730	48427	3	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	289	2	1	5	3.6	Cc1cc(C)cc(Nc2nc3ccccc3n3cnnc23)c1	nan
	CHEMBL1557912	48427	3	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	289	2	1	5	3.6	Cc1cc(C)cc(Nc2nc3ccccc3n3cnnc23)c1	nan
	16011441	48512	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	512	9	1	6	5.9	COc1ccc(Cn2c(SCc3ccc(C(=O)NCc4ccccc4F)cc3)nc3cccnc32)cc1	nan
	CHEMBL1558654	48512	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	512	9	1	6	5.9	COc1ccc(Cn2c(SCc3ccc(C(=O)NCc4ccccc4F)cc3)nc3cccnc32)cc1	nan
	16030801	48551	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	4	1	5	4.4	COc1ccc(-c2cc3ccc(O)c(CN4CCCC(C)C4)c3oc2=O)cc1	nan
	CHEMBL1558940	48551	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	4	1	5	4.4	COc1ccc(-c2cc3ccc(O)c(CN4CCCC(C)C4)c3oc2=O)cc1	nan
	1970873	48554	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	4	0	10	3.5	Cc1cccn2c(=O)c3cc(C#N)c(=O)n(-c4nnc(SCc5ccc(F)cc5)s4)c3nc12	nan
	CHEMBL1558965	48554	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	4	0	10	3.5	Cc1cccn2c(=O)c3cc(C#N)c(=O)n(-c4nnc(SCc5ccc(F)cc5)s4)c3nc12	nan
	16024619	48569	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	497	8	1	7	4.3	CCOC(=O)c1ccc(NC(=O)Cn2cc(C(=O)c3ccc(CC)cc3)c(=O)c3ccc(C)nc32)cc1	nan
	CHEMBL1559093	48569	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	497	8	1	7	4.3	CCOC(=O)c1ccc(NC(=O)Cn2cc(C(=O)c3ccc(CC)cc3)c(=O)c3ccc(C)nc32)cc1	nan
	135448823	48671	12	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	5	2	8	2.7	Cc1cc(NC(=O)CSc2nc(O)c(C#N)c(-c3ccccc3)n2)no1	nan
	CHEMBL1560048	48671	12	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	5	2	8	2.7	Cc1cc(NC(=O)CSc2nc(O)c(C#N)c(-c3ccccc3)n2)no1	nan
	20944767	48774	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	4	1	4	3.3	O=C(CN1c2ccccc2S(=O)(=O)c2ccccc21)NCc1ccccc1	nan
	CHEMBL1561113	48774	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	4	1	4	3.3	O=C(CN1c2ccccc2S(=O)(=O)c2ccccc21)NCc1ccccc1	nan
	938228	48801	8	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	302	3	1	5	3.3	COc1cccc(-c2cc(-c3cccnc3)nc(N)c2C#N)c1	nan
	CHEMBL1561334	48801	8	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	302	3	1	5	3.3	COc1cccc(-c2cc(-c3cccnc3)nc(N)c2C#N)c1	nan
	2136514	49030	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	498	7	1	7	4.2	CCc1ccc(C(=O)c2cn(CC(=O)Nc3ccc(OC)cc3)c3cc4c(cc3c2=O)OCCO4)cc1	nan
	CHEMBL1563400	49030	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	498	7	1	7	4.2	CCc1ccc(C(=O)c2cn(CC(=O)Nc3ccc(OC)cc3)c3cc4c(cc3c2=O)OCCO4)cc1	nan
	16195481	49073	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	7	3	8	2.2	COc1cc2nc(S)nc(NCCc3ccc(S(N)(=O)=O)cc3)c2cc1OC	nan
	CHEMBL1563755	49073	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	7	3	8	2.2	COc1cc2nc(S)nc(NCCc3ccc(S(N)(=O)=O)cc3)c2cc1OC	nan
	16010206	49218	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	5	1	7	1.6	CCc1ccc(NC(=O)C2CCCN2S(=O)(=O)c2ccc3c(c2)n(C)c(=O)c(=O)n3C)cc1	nan
	CHEMBL1565063	49218	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	5	1	7	1.6	CCc1ccc(NC(=O)C2CCCN2S(=O)(=O)c2ccc3c(c2)n(C)c(=O)c(=O)n3C)cc1	nan
	16017589	49437	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	4	1	7	1.5	O=C(Nc1nnc(S(=O)(=O)N2CCOCC2)s1)c1ccccc1Cl	nan
	CHEMBL1566733	49437	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	4	1	7	1.5	O=C(Nc1nnc(S(=O)(=O)N2CCOCC2)s1)c1ccccc1Cl	nan
	2764046	49441	46	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	4	1	3	4.8	O=C(O)Cc1sc(-c2ccccc2Cl)nc1-c1ccccc1	nan
	CHEMBL1566761	49441	46	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	4	1	3	4.8	O=C(O)Cc1sc(-c2ccccc2Cl)nc1-c1ccccc1	nan
	1419199	49460	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	516	6	1	5	4.6	O=C(O)CCCC(=O)N1CCN(c2nc(-c3ccccc3Cl)c3cc(Br)ccc3n2)CC1	nan
	1419200	49460	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	516	6	1	5	4.6	O=C(O)CCCC(=O)N1CCN(c2nc(-c3ccccc3Cl)c3cc(Br)ccc3n2)CC1	nan
	CHEMBL1566925	49460	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	516	6	1	5	4.6	O=C(O)CCCC(=O)N1CCN(c2nc(-c3ccccc3Cl)c3cc(Br)ccc3n2)CC1	nan
	1101443	49547	9	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	3	1	3	5.0	O=C(Nc1ccc2oc(-c3cccc(F)c3)nc2c1)c1ccccc1F	nan
	CHEMBL1567607	49547	9	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	3	1	3	5.0	O=C(Nc1ccc2oc(-c3cccc(F)c3)nc2c1)c1ccccc1F	nan
	663542	49659	15	None	-1	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	4	1	5	4.2	O=C(CSc1ncnc2c1oc1ccccc12)Nc1cccc(F)c1	nan
	CHEMBL1568508	49659	15	None	-1	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	4	1	5	4.2	O=C(CSc1ncnc2c1oc1ccccc12)Nc1cccc(F)c1	nan
	2837061	49664	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	4	2	3	4.9	O=C(Nc1cccc(NC(=O)c2ccc(Cl)cc2)n1)c1ccc(Cl)cc1	nan
	CHEMBL1568556	49664	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	4	2	3	4.9	O=C(Nc1cccc(NC(=O)c2ccc(Cl)cc2)n1)c1ccc(Cl)cc1	nan
	6618042	49675	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	5	0	6	3.5	CCCCn1c(=O)nc2n(-c3ccc(OC)cc3)c3ccccc3cc-2c1=O	nan
	CHEMBL1568603	49675	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	5	0	6	3.5	CCCCn1c(=O)nc2n(-c3ccc(OC)cc3)c3ccccc3cc-2c1=O	nan
	648080	49738	4	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	5	1	6	3.6	COc1ccc2cc(C)c(SCC(=O)Nc3cc(C)on3)nc2c1	nan
	CHEMBL1569235	49738	4	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	5	1	6	3.6	COc1ccc2cc(C)c(SCC(=O)Nc3cc(C)on3)nc2c1	nan
	2726812	49783	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	267	2	0	4	3.4	COC(=O)c1cc2cc(Cl)ccc2nc1SC	nan
	CHEMBL1569571	49783	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	267	2	0	4	3.4	COC(=O)c1cc2cc(Cl)ccc2nc1SC	nan
	802608	49927	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	3	1	2	4.3	COc1ccc(Br)cc1C(=O)Nc1cccc(C)c1C	nan
	CHEMBL1570796	49927	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	3	1	2	4.3	COc1ccc(Br)cc1C(=O)Nc1cccc(C)c1C	nan
	1247683	49948	12	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	3	1	6	3.2	Cc1cc(C(=O)Nc2nc3ccc(S(C)(=O)=O)cc3s2)c(C)o1	nan
	CHEMBL1570956	49948	12	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	3	1	6	3.2	Cc1cc(C(=O)Nc2nc3ccc(S(C)(=O)=O)cc3s2)c(C)o1	nan
	2874268	50000	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	307	5	1	5	3.0	Cc1cc(NCCCN(C)C)n2c(nc3ccccc32)c1C#N	nan
	CHEMBL1571576	50000	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	307	5	1	5	3.0	Cc1cc(NCCCN(C)C)n2c(nc3ccccc32)c1C#N	nan
	15988316	50014	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	7	1	8	2.7	CCOC(=O)c1ccc(NC(=O)COC(=O)c2cn(CC)c3nc(C)ccc3c2=O)cc1	nan
	CHEMBL1571739	50014	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	7	1	8	2.7	CCOC(=O)c1ccc(NC(=O)COC(=O)c2cn(CC)c3nc(C)ccc3c2=O)cc1	nan
	6037218	50084	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	6	1	7	3.6	COc1ccc(C2C(C(=O)c3ccc4c(c3)OCCO4)=C(O)C(=O)N2Cc2cccnc2)cc1	nan
	CHEMBL1572317	50084	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	6	1	7	3.6	COc1ccc(C2C(C(=O)c3ccc4c(c3)OCCO4)=C(O)C(=O)N2Cc2cccnc2)cc1	nan
	995077	50169	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	4	1	4	4.3	Cn1cc(CNC(=O)c2cc(-c3ccccc3)nc3ccc(Br)cc23)cn1	nan
	CHEMBL1573031	50169	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	4	1	4	4.3	Cn1cc(CNC(=O)c2cc(-c3ccccc3)nc3ccc(Br)cc23)cn1	nan
	1927600	50269	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	540	8	2	5	7.1	CCc1ccccc1NC(=O)CSc1nc(C)c(C(=O)Nc2ccccc2)c(-c2ccc(Cl)cc2)c1C#N	nan
	CHEMBL1574096	50269	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	540	8	2	5	7.1	CCc1ccccc1NC(=O)CSc1nc(C)c(C(=O)Nc2ccccc2)c(-c2ccc(Cl)cc2)c1C#N	nan
	857532	50278	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	5	1	3	4.3	CCc1cc2cccc(C)c2nc1SCC(=O)NC1CCCC1	nan
	CHEMBL1574178	50278	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	5	1	3	4.3	CCc1cc2cccc(C)c2nc1SCC(=O)NC1CCCC1	nan
	7206308	50301	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	5	1	8	3.1	O=C(CSc1ccc(-c2ccc3c(c2)OCO3)nn1)Nc1nccs1	nan
	CHEMBL1574382	50301	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	5	1	8	3.1	O=C(CSc1ccc(-c2ccc3c(c2)OCO3)nn1)Nc1nccs1	nan
	2906920	50471	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	3	1	4	4.3	O=C(Nc1ccc(N2C(=O)C3CCCCC3C2=O)cc1Cl)c1cccs1	nan
	CHEMBL1576225	50471	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	3	1	4	4.3	O=C(Nc1ccc(N2C(=O)C3CCCCC3C2=O)cc1Cl)c1cccs1	nan
	135444827	50480	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	3	1	6	3.0	COc1cccc(N2CC(=O)C(c3nc4ccccc4s3)=C2N)c1	nan
	CHEMBL1576321	50480	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	3	1	6	3.0	COc1cccc(N2CC(=O)C(c3nc4ccccc4s3)=C2N)c1	nan
	4099135	50548	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	500	9	2	6	4.4	O=C(CCCCCn1c(=S)[nH]c2ccc(N3CCOCC3)cc2c1=O)NCc1cccc(Cl)c1	nan
	CHEMBL1576790	50548	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	500	9	2	6	4.4	O=C(CCCCCn1c(=S)[nH]c2ccc(N3CCOCC3)cc2c1=O)NCc1cccc(Cl)c1	nan
	652081	50752	21	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	5	2	8	1.8	Cc1cccn2c(=O)c3cc(C(=O)NCC4CCCO4)c(=N)n(Cc4cccnc4)c3nc12	nan
	CHEMBL1578543	50752	21	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	5	2	8	1.8	Cc1cccn2c(=O)c3cc(C(=O)NCC4CCCO4)c(=N)n(Cc4cccnc4)c3nc12	nan
	2040375	50776	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	5	0	6	4.7	COc1cc2oc(=O)c3c(c2cc1OCC(=O)c1c(C)n(C)c2ccccc12)CCCC3	nan
	CHEMBL1578721	50776	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	5	0	6	4.7	COc1cc2oc(=O)c3c(c2cc1OCC(=O)c1c(C)n(C)c2ccccc12)CCCC3	nan
	5100816	50930	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	10	2	6	3.0	O=C(COC(=O)c1cccnc1SCC(=O)NCc1ccccc1)NCc1ccccc1	nan
	CHEMBL1580143	50930	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	10	2	6	3.0	O=C(COC(=O)c1cccnc1SCC(=O)NCc1ccccc1)NCc1ccccc1	nan
	2823757	51466	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	277	2	1	2	4.4	CC(C)(C)c1ccc(C(=O)Nc2ccc(F)cc2)s1	nan
	CHEMBL1584690	51466	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	277	2	1	2	4.4	CC(C)(C)c1ccc(C(=O)Nc2ccc(F)cc2)s1	nan
	1447358	51679	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	5	2	6	1.7	CC(C)C(=O)NNC(=O)CN1CCN(c2nc(-c3ccccc3)cs2)CC1	nan
	CHEMBL1586366	51679	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	5	2	6	1.7	CC(C)C(=O)NNC(=O)CN1CCN(c2nc(-c3ccccc3)cs2)CC1	nan
	2123807	51852	7	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	5	2	7	0.9	COc1ccc(C(=O)Nc2cccc3c2C(=O)NC3=O)cc1S(=O)(=O)N1CCOCC1	nan
	CHEMBL1587750	51852	7	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	5	2	7	0.9	COc1ccc(C(=O)Nc2cccc3c2C(=O)NC3=O)cc1S(=O)(=O)N1CCOCC1	nan
	2639566	52061	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	6	0	6	3.1	COc1ccc(C(=O)COc2ccc3ccc(=O)oc3c2)c(OC)c1	nan
	CHEMBL1589654	52061	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	6	0	6	3.1	COc1ccc(C(=O)COc2ccc3ccc(=O)oc3c2)c(OC)c1	nan
	16027668	52090	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	6	1	8	3.4	COc1ccccc1C(=O)Nc1cccc(C(=O)OCc2cc(=O)n3ccsc3n2)c1	nan
	CHEMBL1589886	52090	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	6	1	8	3.4	COc1ccccc1C(=O)Nc1cccc(C(=O)OCc2cc(=O)n3ccsc3n2)c1	nan
	16027394	52099	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	7	1	8	3.4	Cc1nn2c(=O)cc(COC(=O)c3ccc(NC(=O)CCc4ccccc4)cc3)nc2s1	nan
	CHEMBL1589930	52099	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	7	1	8	3.4	Cc1nn2c(=O)cc(COC(=O)c3ccc(NC(=O)CCc4ccccc4)cc3)nc2s1	nan
	16007616	52115	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	485	6	1	5	3.6	CN(C1CCCCC1)S(=O)(=O)c1ccc2c(c1)c(=O)c(C(=O)NCc1ccc(F)cc1)cn2C	nan
	CHEMBL1590166	52115	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	485	6	1	5	3.6	CN(C1CCCCC1)S(=O)(=O)c1ccc2c(c1)c(=O)c(C(=O)NCc1ccc(F)cc1)cn2C	nan
	16018888	52132	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	345	3	0	5	5.2	Cc1nnc(SCc2ccccc2Cl)c2cc3sccc3n12	nan
	CHEMBL1590393	52132	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	345	3	0	5	5.2	Cc1nnc(SCc2ccccc2Cl)c2cc3sccc3n12	nan
	2058614	52135	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	496	5	0	8	3.8	CCOC(=O)c1cc2c(=O)n3ccccc3nc2n(Cc2ccco2)/c1=N\C(=O)c1cc(C)cc(C)c1	nan
	CHEMBL1590410	52135	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	496	5	0	8	3.8	CCOC(=O)c1cc2c(=O)n3ccccc3nc2n(Cc2ccco2)/c1=N\C(=O)c1cc(C)cc(C)c1	nan
	16025295	52146	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	550	7	1	6	5.8	CCc1cccc(NC(=O)CSc2ncc3c(n2)-c2ccc(Cl)cc2N(Cc2ccccc2)S3(=O)=O)c1	nan
	CHEMBL1590637	52146	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	550	7	1	6	5.8	CCc1cccc(NC(=O)CSc2ncc3c(n2)-c2ccc(Cl)cc2N(Cc2ccccc2)S3(=O)=O)c1	nan
	16017896	52186	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	3	0	7	2.7	COc1ccc(N2CCN(C(=O)c3sc4nc5n(c(=O)c4c3C)CCC5)CC2)cc1	nan
	CHEMBL1591031	52186	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	3	0	7	2.7	COc1ccc(N2CCN(C(=O)c3sc4nc5n(c(=O)c4c3C)CCC5)CC2)cc1	nan
	16024829	52223	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	3	1	4	4.6	O=C(Nc1ccc(F)cc1)C1CCN(c2nc3ccccc3nc2C(F)(F)F)CC1	nan
	CHEMBL1591484	52223	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	3	1	4	4.6	O=C(Nc1ccc(F)cc1)C1CCN(c2nc3ccccc3nc2C(F)(F)F)CC1	nan
	16027514	52234	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	460	6	1	8	3.9	Cc1cccc(C(=O)Nc2cccc(C(=O)OCc3cc(=O)n4nc(C5CC5)sc4n3)c2)c1	nan
	CHEMBL1591656	52234	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	460	6	1	8	3.9	Cc1cccc(C(=O)Nc2cccc(C(=O)OCc3cc(=O)n4nc(C5CC5)sc4n3)c2)c1	nan
	16012296	52241	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	293	3	1	2	5.0	Cc1cccc(NC(=O)c2ccc(-c3ccccc3)s2)c1	nan
	CHEMBL1591740	52241	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	293	3	1	2	5.0	Cc1cccc(NC(=O)c2ccc(-c3ccccc3)s2)c1	nan
	16019608	52291	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	4	1	8	3.3	Cc1ccc(S(=O)(=O)c2nnn3c2nc(NC(C)C)c2sccc23)cc1	nan
	CHEMBL1592430	52291	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	4	1	8	3.3	Cc1ccc(S(=O)(=O)c2nnn3c2nc(NC(C)C)c2sccc23)cc1	nan
	135546866	52347	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	4	2	4	3.7	Cc1ccc(NC(=O)C(C)Sc2nc3c(c(=O)[nH]2)CCCC3)cc1Cl	nan
	CHEMBL1593216	52347	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	4	2	4	3.7	Cc1ccc(NC(=O)C(C)Sc2nc3c(c(=O)[nH]2)CCCC3)cc1Cl	nan
	3955100	52353	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	8	1	7	4.2	CCOc1ccc(-c2nnc(SCC(=O)Nc3cc(C)ccc3OC)o2)cc1	nan
	CHEMBL1593290	52353	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	8	1	7	4.2	CCOc1ccc(-c2nnc(SCC(=O)Nc3cc(C)ccc3OC)o2)cc1	nan
	16019825	52370	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	4	2	4	3.2	Cc1ccc(C)c(NC(=O)C2CCCN(S(=O)(=O)c3ccc4[nH]c(=O)ccc4c3)C2)c1	nan
	CHEMBL1593576	52370	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	4	2	4	3.2	Cc1ccc(C)c(NC(=O)C2CCCN(S(=O)(=O)c3ccc4[nH]c(=O)ccc4c3)C2)c1	nan
	7598919	52564	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	6	1	5	3.5	CCOC(=O)c1ccc(NC(=O)c2cccn(Cc3ccccc3F)c2=O)cc1	nan
	CHEMBL1595394	52564	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	6	1	5	3.5	CCOC(=O)c1ccc(NC(=O)c2cccn(Cc3ccccc3F)c2=O)cc1	nan
	2135415	52599	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	3	1	6	2.0	Cc1ccc(NC(=O)Cn2c(=O)c3ccccc3n3nncc23)cc1	nan
	CHEMBL1595713	52599	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	3	1	6	2.0	Cc1ccc(NC(=O)Cn2c(=O)c3ccccc3n3nncc23)cc1	nan
	15988650	52646	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	5	1	5	5.6	Cc1cc(NC(=O)c2cc(-c3ccc(Br)cc3)on2)nn1Cc1ccc(Cl)cc1	nan
	CHEMBL1596161	52646	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	5	1	5	5.6	Cc1cc(NC(=O)c2cc(-c3ccc(Br)cc3)on2)nn1Cc1ccc(Cl)cc1	nan
	16009387	52665	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	496	5	1	7	3.9	O=C(Cn1cc(S(=O)(=O)c2ccc(Cl)cc2)c(=O)c2ccccc21)Nc1ccc2c(c1)OCO2	nan
	CHEMBL1596294	52665	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	496	5	1	7	3.9	O=C(Cn1cc(S(=O)(=O)c2ccc(Cl)cc2)c(=O)c2ccccc21)Nc1ccc2c(c1)OCO2	nan
	16028259	52689	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	7	1	6	3.0	CCOc1ccc(-c2cc3c(=O)n(CC(=O)NCc4ccc(F)cc4)ccn3n2)cc1	nan
	CHEMBL1596560	52689	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	7	1	6	3.0	CCOc1ccc(-c2cc3c(=O)n(CC(=O)NCc4ccc(F)cc4)ccn3n2)cc1	nan
	1450700	52703	2	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	330	4	0	7	2.5	CCOC(=O)CSc1nc2cc3c(cc2cc1C#N)OCCO3	nan
	CHEMBL1596663	52703	2	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	330	4	0	7	2.5	CCOC(=O)CSc1nc2cc3c(cc2cc1C#N)OCCO3	nan
	859504	52721	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	319	4	0	6	3.3	Cc1cc2cc3c(cc2nc1SCC(=O)OC(C)C)OCO3	nan
	CHEMBL1596835	52721	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	319	4	0	6	3.3	Cc1cc2cc3c(cc2nc1SCC(=O)OC(C)C)OCO3	nan
	20903879	52733	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	6	1	8	1.7	CC(=O)c1cccc(NC(=O)CCc2nnc3ccc(N4CCN(C)CC4)nn23)c1	nan
	CHEMBL1596921	52733	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	6	1	8	1.7	CC(=O)c1cccc(NC(=O)CCc2nnc3ccc(N4CCN(C)CC4)nn23)c1	nan
	5922522	52795	10	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	457	9	1	6	4.7	CCCCOc1ccc(C(=O)C2=C(O)C(=O)N(Cc3cccnc3)C2c2ccncc2)c(C)c1	nan
	CHEMBL1597564	52795	10	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	457	9	1	6	4.7	CCCCOc1ccc(C(=O)C2=C(O)C(=O)N(Cc3cccnc3)C2c2ccncc2)c(C)c1	nan
	16031965	52800	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	7	2	6	4.1	COc1ccc(-c2nc(C)c(CCNC(=O)C(=O)Nc3c(C)cccc3C)s2)cc1OC	nan
	CHEMBL1597608	52800	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	7	2	6	4.1	COc1ccc(-c2nc(C)c(CCNC(=O)C(=O)Nc3c(C)cccc3C)s2)cc1OC	nan
	4656755	52820	5	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	3	1	5	3.9	COc1ccc(C(=O)Nc2cc(C)c3c(=O)oc4ccccc4c3n2)cc1	nan
	CHEMBL1597754	52820	5	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	3	1	5	3.9	COc1ccc(C(=O)Nc2cc(C)c3c(=O)oc4ccccc4c3n2)cc1	nan
	16030399	52840	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	5	0	4	4.9	Cc1ccc(Cc2nc3ccccc3nc2SCC(=O)N2CCC(C)CC2)cc1	nan
	CHEMBL1597953	52840	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	5	0	4	4.9	Cc1ccc(Cc2nc3ccccc3nc2SCC(=O)N2CCC(C)CC2)cc1	nan
	23603072	52983	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	4	0	7	0.7	CC1CCCN(C(=O)CCS(=O)(=O)c2ccc3c(c2)n(C)c(=O)c(=O)n3C)C1	nan
	CHEMBL1599245	52983	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	4	0	7	0.7	CC1CCCN(C(=O)CCS(=O)(=O)c2ccc3c(c2)n(C)c(=O)c(=O)n3C)C1	nan
	16009708	53134	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	7	2	5	5.0	COc1ccc(CC(=O)Nc2c(C(=O)Nc3ccc(F)cc3)oc3ccccc23)cc1OC	nan
	CHEMBL1600646	53134	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	7	2	5	5.0	COc1ccc(CC(=O)Nc2c(C(=O)Nc3ccc(F)cc3)oc3ccccc23)cc1OC	nan
	1093818	53207	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	3	1	4	4.3	O=C(Nc1cccnc1)c1cc(-c2ccc(Cl)cc2Cl)on1	nan
	CHEMBL1601278	53207	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	3	1	4	4.3	O=C(Nc1cccnc1)c1cc(-c2ccc(Cl)cc2Cl)on1	nan
	4327872	53290	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	1	0	6	1.4	CC1CN(C(=O)c2cc3c(=O)n4ccccc4nc3n2C)CC(C)O1	nan
	CHEMBL1602225	53290	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	1	0	6	1.4	CC1CN(C(=O)c2cc3c(=O)n4ccccc4nc3n2C)CC(C)O1	nan
	7199971	53444	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	5	1	8	3.5	Cc1ccc(-n2ncc3c(SCC(=O)Nc4cc(C)on4)ncnc32)c(C)c1	nan
	CHEMBL1603605	53444	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	5	1	8	3.5	Cc1ccc(-n2ncc3c(SCC(=O)Nc4cc(C)on4)ncnc32)c(C)c1	nan
	22522531	53452	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	345	4	1	4	3.5	CCc1cccc(NC(=O)Cn2c(=O)c3cccn3c3ccccc32)c1	nan
	CHEMBL1603663	53452	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	345	4	1	4	3.5	CCc1cccc(NC(=O)Cn2c(=O)c3cccn3c3ccccc32)c1	nan
	7763635	53541	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	7	0	7	1.7	COc1ccc(C(=O)COC(=O)CN2C(=O)c3ccccc3C2=O)c(OC)c1	nan
	CHEMBL1604328	53541	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	7	0	7	1.7	COc1ccc(C(=O)COC(=O)CN2C(=O)c3ccccc3C2=O)c(OC)c1	nan
	1072346	53654	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	5	1	6	4.5	O=C(CSc1nc(-c2ccccc2)nc2ccccc12)Nc1nccs1	nan
	CHEMBL1605363	53654	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	5	1	6	4.5	O=C(CSc1nc(-c2ccccc2)nc2ccccc12)Nc1nccs1	nan
	1005145	53690	13	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	4	1	6	3.6	N#Cc1cc2c(nc1SCC(=O)Nc1sc3c(c1C#N)CCC3)CCC2	nan
	CHEMBL1605614	53690	13	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	4	1	6	3.6	N#Cc1cc2c(nc1SCC(=O)Nc1sc3c(c1C#N)CCC3)CCC2	nan
	15991041	53743	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	7	2	3	5.7	CCCOc1ccc(C(=O)Nc2ccc(NC(=O)c3ccccc3)c(Br)c2)cc1	nan
	CHEMBL1606046	53743	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	7	2	3	5.7	CCCOc1ccc(C(=O)Nc2ccc(NC(=O)c3ccccc3)c(Br)c2)cc1	nan
	2934348	53903	18	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	5	2	6	3.4	O=C(C1=C(O)C(=O)N(Cc2ccco2)C1c1cccc(O)c1)c1ccco1	nan
	CHEMBL1607257	53903	18	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	5	2	6	3.4	O=C(C1=C(O)C(=O)N(Cc2ccco2)C1c1cccc(O)c1)c1ccco1	nan
	16027345	53969	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	6	1	5	4.4	CCCNC(=O)Cn1nc(-c2ccc(C)c(C)c2)c2cnc3ccc(OC)cc3c21	nan
	CHEMBL1607743	53969	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	6	1	5	4.4	CCCNC(=O)Cn1nc(-c2ccc(C)c(C)c2)c2cnc3ccc(OC)cc3c21	nan
	753354	53979	11	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	2	0	6	2.6	O=C1c2ccccc2C(=O)N1c1nc2nccc(-c3ccccc3)n2n1	nan
	CHEMBL1607842	53979	11	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	2	0	6	2.6	O=C1c2ccccc2C(=O)N1c1nc2nccc(-c3ccccc3)n2n1	nan
	3512516	54112	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	5	2	7	4.2	CCOc1ccc(NC(=O)c2sc3nc(N4CCOCC4)c4c(c3c2N)CCCC4)cc1	nan
	CHEMBL1609027	54112	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	5	2	7	4.2	CCOc1ccc(NC(=O)c2sc3nc(N4CCOCC4)c4c(c3c2N)CCCC4)cc1	nan
	16011054	54126	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	7	1	6	4.0	CCc1cc2c(cc3c(=O)n(CCCC(=O)NCc4cccc(Cl)c4)ncn32)s1	nan
	CHEMBL1609118	54126	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	7	1	6	4.0	CCc1cc2c(cc3c(=O)n(CCCC(=O)NCc4cccc(Cl)c4)ncn32)s1	nan
	2422324	54231	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	5	3	8	-0.1	COCCn1c(N)c(C(=S)NC(=O)c2cccs2)c(=O)[nH]c1=O	nan
	CHEMBL1609964	54231	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	5	3	8	-0.1	COCCn1c(N)c(C(=S)NC(=O)c2cccs2)c(=O)[nH]c1=O	nan
	16007504	54289	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	426	6	1	4	5.2	COc1ccc(CNC(=O)CSc2c3c(nc4ccc(Cl)cc24)CCCC3)cc1	nan
	CHEMBL1610456	54289	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	426	6	1	4	5.2	COc1ccc(CNC(=O)CSc2c3c(nc4ccc(Cl)cc24)CCCC3)cc1	nan
	2134793	54298	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	7	0	6	5.6	COCCCn1c(SCc2cccc(Cl)c2)nc2c(sc3ccccc32)c1=O	nan
	CHEMBL1610529	54298	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	7	0	6	5.6	COCCCn1c(SCc2cccc(Cl)c2)nc2c(sc3ccccc32)c1=O	nan
	3374134	54325	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	5	2	4	2.4	O=C(Cn1c(=S)[nH]c2ccccc2c1=O)NCCc1ccccc1	nan
	CHEMBL1610861	54325	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	5	2	4	2.4	O=C(Cn1c(=S)[nH]c2ccccc2c1=O)NCCc1ccccc1	nan
	3185781	54413	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	502	10	3	8	2.2	COCCN(C(=O)c1snc(C(N)=O)c1N)C(C(=O)NC1CCCCC1)c1ccc(N(C)C)cc1	nan
	CHEMBL1611537	54413	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	502	10	3	8	2.2	COCCN(C(=O)c1snc(C(N)=O)c1N)C(C(=O)NC1CCCCC1)c1ccc(N(C)C)cc1	nan
	3353363	54426	14	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	4	0	6	4.1	COc1ccc(C2CC(=O)c3cnc(N4CCc5ccccc54)nc3C2)cc1OC	nan
	CHEMBL1611722	54426	14	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	4	0	6	4.1	COc1ccc(C2CC(=O)c3cnc(N4CCc5ccccc54)nc3C2)cc1OC	nan
	2201483	55373	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	426	5	4	7	2.8	Cc1cc(C)nc(NC(=N)Nc2ccc(S(=O)(=O)Nc3nc(C)cc(C)n3)cc2)n1	nan
	5739455	55373	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	426	5	4	7	2.8	Cc1cc(C)nc(NC(=N)Nc2ccc(S(=O)(=O)Nc3nc(C)cc(C)n3)cc2)n1	nan
	9587736	55373	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	426	5	4	7	2.8	Cc1cc(C)nc(NC(=N)Nc2ccc(S(=O)(=O)Nc3nc(C)cc(C)n3)cc2)n1	nan
	CHEMBL1442349	55373	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	426	5	4	7	2.8	Cc1cc(C)nc(NC(=N)Nc2ccc(S(=O)(=O)Nc3nc(C)cc(C)n3)cc2)n1	nan
	CHEMBL1621693	55373	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	426	5	4	7	2.8	Cc1cc(C)nc(NC(=N)Nc2ccc(S(=O)(=O)Nc3nc(C)cc(C)n3)cc2)n1	nan
	354678	55557	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	3	1	8	1.6	CCC1(OC(=O)CN)C(=O)OCc2c1cc1n(c2=O)Cc2cc3ccccc3nc2-1	nan
	CHEMBL1518154	55557	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	3	1	8	1.6	CCC1(OC(=O)CN)C(=O)OCc2c1cc1n(c2=O)Cc2cc3ccccc3nc2-1	nan
	CHEMBL1623188	55557	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	3	1	8	1.6	CCC1(OC(=O)CN)C(=O)OCc2c1cc1n(c2=O)Cc2cc3ccccc3nc2-1	nan
	24792219	55688	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	454	7	1	4	6.5	Fc1ccc(-[n+]2nc(Nc3ccccc3)sc2-c2ccc(OCc3ccccc3)cc2)cc1	nan
	CHEMBL1551405	55688	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	454	7	1	4	6.5	Fc1ccc(-[n+]2nc(Nc3ccccc3)sc2-c2ccc(OCc3ccccc3)cc2)cc1	nan
	CHEMBL1624286	55688	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	454	7	1	4	6.5	Fc1ccc(-[n+]2nc(Nc3ccccc3)sc2-c2ccc(OCc3ccccc3)cc2)cc1	nan
	3490356	72113	11	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	322	3	0	5	2.2	C#CCn1/c(=N/C(=O)CSC(C)=O)sc2cc(F)ccc21	nan
	CHEMBL1988684	72113	11	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	322	3	0	5	2.2	C#CCn1/c(=N/C(=O)CSC(C)=O)sc2cc(F)ccc21	nan
	1522244	85068	69	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	164	0	1	3	1.9	Cn1c(S)nc2ccccc21	nan
	CHEMBL227086	85068	69	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	164	0	1	3	1.9	Cn1c(S)nc2ccccc21	nan
	25252625	107129	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	299	6	1	5	1.8	COc1ccc(CC(=O)N/N=C/c2cccnc2)cc1OC	nan
	CHEMBL3189886	107129	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	299	6	1	5	1.8	COc1ccc(CC(=O)N/N=C/c2cccnc2)cc1OC	nan
	9701594	107285	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	4	2	6	2.1	O=C(N/N=C1\C/C(=N\NC(=O)c2ccncc2)c2ccccc21)c1ccncc1	nan
	CHEMBL3191689	107285	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	4	2	6	2.1	O=C(N/N=C1\C/C(=N\NC(=O)c2ccncc2)c2ccccc21)c1ccncc1	nan
	4141152	108379	11	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	318	3	0	5	2.6	CCOC(=O)c1s/c(=N\C(=O)c2cccc(C)c2)n(C)c1C	nan
	CHEMBL3210377	108379	11	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	318	3	0	5	2.6	CCOC(=O)c1s/c(=N\C(=O)c2cccc(C)c2)n(C)c1C	nan
	2150923	108582	9	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	5	0	7	3.1	CCn1/c(=N/C(=O)c2cccc(N3C(=O)CCC3=O)c2)sc2c(OC)ccc(OC)c21	nan
	CHEMBL3212992	108582	9	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	5	0	7	3.1	CCn1/c(=N/C(=O)c2cccc(N3C(=O)CCC3=O)c2)sc2c(OC)ccc(OC)c21	nan
	1477780	197401	14	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	5	1	6	3.0	COc1cc(-c2nc3ccc(N4CCN(C)CC4)cc3[nH]2)cc(OC)c1OC	nan
	CHEMBL587856	197401	14	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	5	1	6	3.0	COc1cc(-c2nc3ccc(N4CCN(C)CC4)cc3[nH]2)cc(OC)c1OC	nan
	7190643	20856	10	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	5	1	7	3.2	Cc1ccc(NC(=O)CSc2ccc3nnc(-c4cccnc4)n3n2)cc1	nan
	CHEMBL1311897	20856	10	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	5	1	7	3.2	Cc1ccc(NC(=O)CSc2ccc3nnc(-c4cccnc4)n3n2)cc1	nan
	1739479	21201	11	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	5	0	4	6.0	Cc1cc(Br)cc2c(C(=O)OCC(=O)c3ccccc3)cc(-c3ccccc3)nc12	nan
	CHEMBL1314681	21201	11	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	5	0	4	6.0	Cc1cc(Br)cc2c(C(=O)OCC(=O)c3ccccc3)cc(-c3ccccc3)nc12	nan
	15988299	21598	9	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	5	1	7	2.9	Cn1c(=O)c2sccc2n2c(CCCC(=O)Nc3ccc(F)cc3F)nnc12	nan
	CHEMBL1319322	21598	9	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	5	1	7	2.9	Cn1c(=O)c2sccc2n2c(CCCC(=O)Nc3ccc(F)cc3F)nnc12	nan
	4146227	26694	11	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	491	7	1	7	5.6	CCOC(=O)c1ccc(NC(=O)CSc2nc(-c3cccs3)cc(C(F)(F)F)c2C#N)cc1	nan
	CHEMBL1363837	26694	11	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	491	7	1	7	5.6	CCOC(=O)c1ccc(NC(=O)CSc2nc(-c3cccs3)cc(C(F)(F)F)c2C#N)cc1	nan
	15988966	30644	6	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	501	10	1	4	6.5	CC(C)CN(CCCNC(=O)c1cc(-c2ccc(Br)s2)nc2ccccc12)CC(C)C	nan
	CHEMBL1397188	30644	6	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	501	10	1	4	6.5	CC(C)CN(CCCNC(=O)c1cc(-c2ccc(Br)s2)nc2ccccc12)CC(C)C	nan
	1398096	30985	9	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	7	2	5	2.8	CC(C)c1nnc(NC(=O)CCC(=O)NCc2ccc(F)cc2)s1	nan
	CHEMBL1400798	30985	9	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	7	2	5	2.8	CC(C)c1nnc(NC(=O)CCC(=O)NCc2ccc(F)cc2)s1	nan
	24792315	31321	2	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	5	1	9	1.9	CCc1nnc(NC(=O)CSc2nnc3nc(C)cc(C)n23)s1	nan
	CHEMBL1403815	31321	2	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	5	1	9	1.9	CCc1nnc(NC(=O)CSc2nnc3nc(C)cc(C)n23)s1	nan
	15991483	39341	6	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	493	8	0	6	6.1	CCOc1ccc(-c2nnc(SCC(=O)c3ccc(Br)cc3)n2-c2ccccc2)cc1	nan
	CHEMBL1473564	39341	6	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	493	8	0	6	6.1	CCOc1ccc(-c2nnc(SCC(=O)c3ccc(Br)cc3)n2-c2ccccc2)cc1	nan
	4299978	43608	7	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	463	7	1	9	1.5	COc1ccc(S(=O)(=O)N2CCOCC2)cc1NC(=O)CSc1nnc2ccccn12	nan
	CHEMBL1511455	43608	7	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	463	7	1	9	1.5	COc1ccc(S(=O)(=O)N2CCOCC2)cc1NC(=O)CSc1nnc2ccccn12	nan
	16019368	52397	9	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	495	6	1	10	4.5	COc1cc(Nc2nc3c(S(=O)(=O)c4ccc(C)c(C)c4)nnn3c3ccsc23)cc(OC)c1	nan
	CHEMBL1593977	52397	9	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	495	6	1	10	4.5	COc1cc(Nc2nc3c(S(=O)(=O)c4ccc(C)c(C)c4)nnn3c3ccsc23)cc(OC)c1	nan
	814542	52826	22	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	215	0	2	3	2.7	Cc1ccc2[nH]c3c(S)ncnc3c2c1	nan
	CHEMBL1597829	52826	22	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	215	0	2	3	2.7	Cc1ccc2[nH]c3c(S)ncnc3c2c1	nan
	9619102	72097	8	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	7	1	11	-0.4	COc1ccc(/C=N/NC(=O)Cn2cnc3c2c(=O)n(C)c(=O)n3C)c(OC)c1OC	nan
	CHEMBL1988156	72097	8	None	-	1	Human	5.5	pPotency	=	5.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	7	1	11	-0.4	COc1ccc(/C=N/NC(=O)Cn2cnc3c2c(=O)n(C)c(=O)n3C)c(OC)c1OC	nan
	16010435	6121	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	507	6	1	8	5.0	COc1ccccc1CNc1nc2c(S(=O)(=O)c3ccc(C)c(C)c3)nnn2c2ccc(Cl)cc12	nan
	CHEMBL1081265	6121	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	507	6	1	8	5.0	COc1ccccc1CNc1nc2c(S(=O)(=O)c3ccc(C)c(C)c3)nnn2c2ccc(Cl)cc12	nan
	1375940	7475	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	289	3	1	5	1.0	COc1ccccc1NC=C1C(=O)N(C)C(=O)N(C)C1=O	nan
	CHEMBL1087646	7475	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	289	3	1	5	1.0	COc1ccccc1NC=C1C(=O)N(C)C(=O)N(C)C1=O	nan
	16019310	10659	10	None	-47	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	5	1	8	4.2	Cc1ccc(S(=O)(=O)c2nnn3c2nc(NCc2ccc(F)cc2)c2sccc23)cc1	nan
	CHEMBL1171436	10659	10	None	-47	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	5	1	8	4.2	Cc1ccc(S(=O)(=O)c2nnn3c2nc(NCc2ccc(F)cc2)c2sccc23)cc1	nan
	16019394	10764	8	None	-37	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	447	4	1	8	4.6	O=S(=O)(c1ccc(Cl)cc1)c1nnn2c1nc(NC1CCCCC1)c1sccc12	nan
	CHEMBL1172405	10764	8	None	-37	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	447	4	1	8	4.6	O=S(=O)(c1ccc(Cl)cc1)c1nnn2c1nc(NC1CCCCC1)c1sccc12	nan
	16019397	10857	11	None	-54	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	461	5	1	9	4.5	O=S(=O)(c1ccc(Cl)cc1)c1nnn2c1nc(NCc1cccs1)c1sccc12	nan
	CHEMBL1173286	10857	11	None	-54	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	461	5	1	9	4.5	O=S(=O)(c1ccc(Cl)cc1)c1nnn2c1nc(NCc1cccs1)c1sccc12	nan
	684664	15266	23	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	289	2	1	5	2.7	N#Cc1c(N)nc(N2CCCC2)c(C#N)c1-c1ccccc1	nan
	CHEMBL1215029	15266	23	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	289	2	1	5	2.7	N#Cc1c(N)nc(N2CCCC2)c(C#N)c1-c1ccccc1	nan
	34768	16224	55	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	347	4	5	10	-1.9	Nc1ncnc2c1ncn2[C@@H]1O[C@H](COP(=O)(O)O)[C@@H](O)[C@@H]1O	nan
	CHEMBL1230732	16224	55	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	347	4	5	10	-1.9	Nc1ncnc2c1ncn2[C@@H]1O[C@H](COP(=O)(O)O)[C@@H](O)[C@@H]1O	nan
	CHEMBL3392220	16224	55	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	347	4	5	10	-1.9	Nc1ncnc2c1ncn2[C@@H]1O[C@H](COP(=O)(O)O)[C@@H](O)[C@@H]1O	nan
	3733180	19479	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	317	3	1	4	3.7	O=C(Nc1nnc(-c2ccccc2F)s1)c1ccccc1F	nan
	CHEMBL1300733	19479	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	317	3	1	4	3.7	O=C(Nc1nnc(-c2ccccc2F)s1)c1ccccc1F	nan
	3815083	19518	26	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	269	1	1	5	2.5	N#Cc1cnn2c(N)c(-c3ccc(Cl)cc3)cnc12	nan
	CHEMBL1301028	19518	26	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	269	1	1	5	2.5	N#Cc1cnn2c(N)c(-c3ccc(Cl)cc3)cnc12	nan
	2219338	19671	9	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	6	2	3	5.0	O=C(Nc1cccc(C(F)(F)F)c1)c1cccnc1NCCc1ccccc1	nan
	CHEMBL1302293	19671	9	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	6	2	3	5.0	O=C(Nc1cccc(C(F)(F)F)c1)c1cccnc1NCCc1ccccc1	nan
	1217579	19677	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	2	0	6	4.5	N#Cc1ccc(-c2nc3cc(C#N)c(C#N)cc3nc2-c2ccccc2)cc1C#N	nan
	CHEMBL1302356	19677	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	2	0	6	4.5	N#Cc1ccc(-c2nc3cc(C#N)c(C#N)cc3nc2-c2ccccc2)cc1C#N	nan
	1244329	19751	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	4	1	7	3.6	COC(=O)c1c(-c2cccnc2)csc1NC(=O)c1ccc2c(c1)OCO2	nan
	CHEMBL1302889	19751	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	4	1	7	3.6	COC(=O)c1c(-c2cccnc2)csc1NC(=O)c1ccc2c(c1)OCO2	nan
	2740109	19888	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	2	0	5	3.5	N#Cc1c(N2CCOCC2)nsc1-c1ccc(C(F)(F)F)cc1	nan
	CHEMBL1303994	19888	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	2	0	5	3.5	N#Cc1c(N2CCOCC2)nsc1-c1ccc(C(F)(F)F)cc1	nan
	1462693	20158	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	8	2	7	2.3	COc1ccc(CNC(=O)CSc2nnc(NC(=O)C3CC3)s2)cc1	nan
	CHEMBL1306151	20158	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	8	2	7	2.3	COc1ccc(CNC(=O)CSc2nnc(NC(=O)C3CC3)s2)cc1	nan
	2158311	20160	13	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	4	1	5	5.1	O=C(CSc1ncnc2c1oc1ccccc12)Nc1ccccc1C(F)(F)F	nan
	CHEMBL1306166	20160	13	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	4	1	5	5.1	O=C(CSc1ncnc2c1oc1ccccc12)Nc1ccccc1C(F)(F)F	nan
	940263	20195	37	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	175	0	1	2	2.8	Cc1cc(S)c2ccccc2n1	nan
	CHEMBL1306515	20195	37	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	175	0	1	2	2.8	Cc1cc(S)c2ccccc2n1	nan
	3678328	20492	5	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	463	4	1	5	4.0	O=C(COC(=O)c1cccc(Br)c1)Nc1cccc2c1C(=O)c1ccccc1C2=O	nan
	CHEMBL1308878	20492	5	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	463	4	1	5	4.0	O=C(COC(=O)c1cccc(Br)c1)Nc1cccc2c1C(=O)c1ccccc1C2=O	nan
	3942275	20629	11	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	497	5	1	7	4.6	CC1CN(S(=O)(=O)c2ccc(C(=O)Nc3nc(-c4cc5ccccc5o4)cs3)cc2)CC(C)O1	nan
	CHEMBL1310132	20629	11	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	497	5	1	7	4.6	CC1CN(S(=O)(=O)c2ccc(C(=O)Nc3nc(-c4cc5ccccc5o4)cs3)cc2)CC(C)O1	nan
	2744150	21084	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	5	1	7	4.3	Cc1nc(-c2nnc(SCC(=O)Nc3cc(Cl)cc(Cl)c3)n2C)cs1	nan
	CHEMBL1313563	21084	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	5	1	7	4.3	Cc1nc(-c2nnc(SCC(=O)Nc3cc(Cl)cc(Cl)c3)n2C)cs1	nan
	2997549	21155	9	None	-7	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	465	5	1	8	2.9	Cc1ccc(S(=O)(=O)c2c(N)n(CCN3CCOCC3)c3nc4ccccc4nc23)cc1C	nan
	CHEMBL1314156	21155	9	None	-7	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	465	5	1	8	2.9	Cc1ccc(S(=O)(=O)c2c(N)n(CCN3CCOCC3)c3nc4ccccc4nc23)cc1C	nan
	16009918	21166	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	464	5	1	7	1.5	Cc1ccc(Cl)cc1NC(=O)CN(C)S(=O)(=O)c1ccc2c(c1)n(C)c(=O)c(=O)n2C	nan
	CHEMBL1314250	21166	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	464	5	1	7	1.5	Cc1ccc(Cl)cc1NC(=O)CN(C)S(=O)(=O)c1ccc2c(c1)n(C)c(=O)c(=O)n2C	nan
	135458483	21180	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	4	2	5	1.7	Cc1ccn2c(=O)c(C(=O)NCCc3ccccc3)c(O)nc2c1	nan
	CHEMBL1314355	21180	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	4	2	5	1.7	Cc1ccn2c(=O)c(C(=O)NCCc3ccccc3)c(O)nc2c1	nan
	16024181	21202	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	3	0	4	3.9	Cc1cccc(N2C(=O)CS(=O)(=O)C23C(=O)N(Cc2c(F)cccc2Cl)c2ccccc23)c1	nan
	CHEMBL1314689	21202	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	3	0	4	3.9	Cc1cccc(N2C(=O)CS(=O)(=O)C23C(=O)N(Cc2c(F)cccc2Cl)c2ccccc23)c1	nan
	4913767	21213	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	5	0	7	3.2	COC(=O)Cc1c(C)c2ccc3c(c2oc1=O)CN(Cc1ccccc1OC)CO3	nan
	CHEMBL1314916	21213	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	5	0	7	3.2	COC(=O)Cc1c(C)c2ccc3c(c2oc1=O)CN(Cc1ccccc1OC)CO3	nan
	16027662	21224	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	423	5	1	7	3.5	O=C(Nc1cccc(C(=O)OCc2cc(=O)n3ccsc3n2)c1)c1ccc(F)cc1	nan
	CHEMBL1315065	21224	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	423	5	1	7	3.5	O=C(Nc1cccc(C(=O)OCc2cc(=O)n3ccsc3n2)c1)c1ccc(F)cc1	nan
	16021060	21257	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	4	1	6	3.7	COc1ccc(NC(=O)c2cn3c4c(ccc(Cl)c4c2=O)OC(C)C3)cc1OC	nan
	CHEMBL1315440	21257	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	4	1	6	3.7	COc1ccc(NC(=O)c2cn3c4c(ccc(Cl)c4c2=O)OC(C)C3)cc1OC	nan
	4524401	21269	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	8	1	8	4.0	COC(=O)c1ccccc1NC(=O)CSc1nc2ccsc2c(=O)n1CCC(C)C	nan
	CHEMBL1315570	21269	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	8	1	8	4.0	COC(=O)c1ccccc1NC(=O)CSc1nc2ccsc2c(=O)n1CCC(C)C	nan
	16020822	21271	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	7	1	5	6.0	O=C(NC1CCCCC1)c1ccc(Cn2c(SCc3ccc(F)cc3)nc3cccnc32)cc1	nan
	CHEMBL1315619	21271	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	7	1	5	6.0	O=C(NC1CCCCC1)c1ccc(Cn2c(SCc3ccc(F)cc3)nc3cccnc32)cc1	nan
	16016226	21287	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	5	1	5	5.0	CC(=O)c1cccc(NC(=O)c2nc(-c3ccccc3)n(-c3cccc(Cl)c3)n2)c1	nan
	CHEMBL1315816	21287	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	5	1	5	5.0	CC(=O)c1cccc(NC(=O)c2nc(-c3ccccc3)n(-c3cccc(Cl)c3)n2)c1	nan
	16009840	21290	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	5	2	4	5.2	COc1ccccc1NC(=O)c1oc2ccccc2c1NC(=O)C1CCCCC1	nan
	CHEMBL1315829	21290	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	5	2	4	5.2	COc1ccccc1NC(=O)c1oc2ccccc2c1NC(=O)C1CCCCC1	nan
	16025104	21308	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	5	1	5	4.4	CC(=O)c1cccc(NC(=O)c2cnn(-c3cccc(C)c3)c2-n2cccc2)c1	nan
	CHEMBL1316030	21308	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	5	1	5	4.4	CC(=O)c1cccc(NC(=O)c2cnn(-c3cccc(C)c3)c2-n2cccc2)c1	nan
	1083262	21316	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	5	0	5	4.4	CCOC(=O)CSc1nc(-c2ccc(F)cc2)cc(C(F)(F)F)c1C#N	nan
	CHEMBL1316119	21316	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	5	0	5	4.4	CCOC(=O)CSc1nc(-c2ccc(F)cc2)cc(C(F)(F)F)c1C#N	nan
	20940443	21335	3	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	5	1	3	4.5	CCCNC(=O)c1cc(-c2ccccc2)c(N2CCCCC2)s1	nan
	CHEMBL1316420	21335	3	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	5	1	3	4.5	CCCNC(=O)c1cc(-c2ccccc2)c(N2CCCCC2)s1	nan
	16022216	21380	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	6	1	4	4.7	CC(=O)c1ccc(NC(=O)CC(c2cccs2)N2Cc3ccccc3C2=O)cc1	nan
	CHEMBL1317049	21380	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	6	1	4	4.7	CC(=O)c1ccc(NC(=O)CC(c2cccs2)N2Cc3ccccc3C2=O)cc1	nan
	16027421	21387	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	6	1	8	3.7	COc1cccc(C(=O)Nc2cccc(C(=O)OCc3cc(=O)n4c(C)csc4n3)c2)c1	nan
	CHEMBL1317129	21387	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	6	1	8	3.7	COc1cccc(C(=O)Nc2cccc(C(=O)OCc3cc(=O)n4c(C)csc4n3)c2)c1	nan
	2159322	21401	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	3	0	6	3.6	CCn1/c(=N/C(=O)c2ccc3c(c2)OCCO3)sc2c(C)ccc(OC)c21	nan
	CHEMBL1317343	21401	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	3	0	6	3.6	CCn1/c(=N/C(=O)c2ccc3c(c2)OCCO3)sc2c(C)ccc(OC)c21	nan
	16028188	21418	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	3	2	3	3.8	Cc1cccc(NC(=O)c2cc3c([nH]c2=O)CC(c2ccccc2)CC3=O)c1	nan
	CHEMBL1317555	21418	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	3	2	3	3.8	Cc1cccc(NC(=O)c2cc3c([nH]c2=O)CC(c2ccccc2)CC3=O)c1	nan
	16023037	21433	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	436	6	1	6	3.6	Cc1ccc(C(=O)Nc2nnc(S(=O)(=O)N(C)Cc3ccc(Cl)cc3)s2)cc1	nan
	CHEMBL1317727	21433	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	436	6	1	6	3.6	Cc1ccc(C(=O)Nc2nnc(S(=O)(=O)N(C)Cc3ccc(Cl)cc3)s2)cc1	nan
	2227086	21440	14	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	300	2	2	3	2.5	O=C(Nc1ccc2c(c1)C(=O)NC2=O)c1cccc(Cl)c1	nan
	CHEMBL1317881	21440	14	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	300	2	2	3	2.5	O=C(Nc1ccc2c(c1)C(=O)NC2=O)c1cccc(Cl)c1	nan
	16024891	21476	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	460	5	1	5	4.9	CSc1ccc(CNC(=O)C2CCN(c3nc4ccccc4nc3C(F)(F)F)CC2)cc1	nan
	CHEMBL1318327	21476	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	460	5	1	5	4.9	CSc1ccc(CNC(=O)C2CCN(c3nc4ccccc4nc3C(F)(F)F)CC2)cc1	nan
	16025877	21503	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	6	1	8	2.9	CC(C)Oc1ccc(CNC(=O)c2cnc3sc(N4CCCCC4)nn3c2=O)cc1	nan
	CHEMBL1318545	21503	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	6	1	8	2.9	CC(C)Oc1ccc(CNC(=O)c2cnc3sc(N4CCCCC4)nn3c2=O)cc1	nan
	16445400	21526	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	275	2	1	5	2.8	Cc1nonc1NC(=O)c1oc2ccc(F)cc2c1C	nan
	CHEMBL1318745	21526	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	275	2	1	5	2.8	Cc1nonc1NC(=O)c1oc2ccc(F)cc2c1C	nan
	16022946	21621	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	482	6	1	6	4.6	Cc1ccc(-n2nc3c(N4CCC(C(=O)NCCc5ccccc5C)CC4)nnc(C)c3c2C)cc1	nan
	CHEMBL1319510	21621	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	482	6	1	6	4.6	Cc1ccc(-n2nc3c(N4CCC(C(=O)NCCc5ccccc5C)CC4)nnc(C)c3c2C)cc1	nan
	16022818	21687	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	4	1	6	5.2	Cc1ccc(Cl)cc1NC(=O)C1CCN(c2nnc(C)c3c(C)n(-c4ccccc4)nc23)CC1	nan
	CHEMBL1320089	21687	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	4	1	6	5.2	Cc1ccc(Cl)cc1NC(=O)C1CCN(c2nnc(C)c3c(C)n(-c4ccccc4)nc23)CC1	nan
	4183241	21692	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	461	6	1	5	5.5	COc1ccc(-c2cc(C(F)(F)F)c(C#N)c(SCC(=O)Nc3ccc(F)cc3)n2)cc1	nan
	CHEMBL1320138	21692	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	461	6	1	5	5.5	COc1ccc(-c2cc(C(F)(F)F)c(C#N)c(SCC(=O)Nc3ccc(F)cc3)n2)cc1	nan
	3167480	21702	6	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	4	1	6	5.1	Cc1ccc2nc(SCC(=O)Nc3ccc4sc(C)nc4c3)c(C#N)cc2c1	nan
	CHEMBL1320193	21702	6	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	4	1	6	5.1	Cc1ccc2nc(SCC(=O)Nc3ccc4sc(C)nc4c3)c(C#N)cc2c1	nan
	16023651	21705	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	477	7	3	5	3.6	Cc1ccc(CNC(=O)c2ccc3c(c2)NC(=O)C(CS(=O)(=O)Cc2cccc(C)c2)N3)cc1	nan
	CHEMBL1320214	21705	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	477	7	3	5	3.6	Cc1ccc(CNC(=O)c2ccc3c(c2)NC(=O)C(CS(=O)(=O)Cc2cccc(C)c2)N3)cc1	nan
	16009865	21734	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	4	1	6	3.6	O=C(Cn1c(=O)n(-c2ccc(F)cc2)c(=O)c2sc3ccccc3c21)NC1CCCC1	nan
	CHEMBL1320479	21734	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	4	1	6	3.6	O=C(Cn1c(=O)n(-c2ccc(F)cc2)c(=O)c2sc3ccccc3c21)NC1CCCC1	nan
	3613580	21869	20	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	316	4	1	5	3.7	CNc1nc(-c2ccccc2)nc(-c2ccc(OC)cc2)c1C#N	nan
	CHEMBL1321693	21869	20	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	316	4	1	5	3.7	CNc1nc(-c2ccccc2)nc(-c2ccc(OC)cc2)c1C#N	nan
	16026062	22034	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	3	1	7	2.6	Cc1cccc(NC(=O)c2cnc3sc(N4CCCC4)nn3c2=O)c1C	nan
	CHEMBL1323207	22034	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	3	1	7	2.6	Cc1cccc(NC(=O)c2cnc3sc(N4CCCC4)nn3c2=O)c1C	nan
	720155	22064	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	344	4	2	2	4.8	Cc1cccc(NC(=O)c2cccc(C(=O)Nc3cccc(C)c3)c2)c1	nan
	CHEMBL1323476	22064	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	344	4	2	2	4.8	Cc1cccc(NC(=O)c2cccc(C(=O)Nc3cccc(C)c3)c2)c1	nan
	866639	22087	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	1	0	6	2.4	Cc1cccn2c(=O)c3cc(C(=O)N4COCC4(C)C)sc3nc12	nan
	CHEMBL1323660	22087	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	1	0	6	2.4	Cc1cccn2c(=O)c3cc(C(=O)N4COCC4(C)C)sc3nc12	nan
	7597258	22212	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	325	4	1	4	3.7	Cc1ccc(-c2nnc(NC(=O)Cc3ccc(F)cc3)o2)c(C)c1	nan
	CHEMBL1324652	22212	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	325	4	1	4	3.7	Cc1ccc(-c2nnc(NC(=O)Cc3ccc(F)cc3)o2)c(C)c1	nan
	20903561	22269	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	4	2	5	3.1	O=C(Nc1ccc(F)cc1)C1CCCN(S(=O)(=O)c2ccc3nc(O)ccc3c2)C1	nan
	CHEMBL1325113	22269	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	4	2	5	3.1	O=C(Nc1ccc(F)cc1)C1CCCN(S(=O)(=O)c2ccc3nc(O)ccc3c2)C1	nan
	1239703	22286	8	None	-7	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	5	1	7	3.0	CCc1nnc(NC(=O)CSc2nc3c(cc2C#N)CCCC3)s1	nan
	CHEMBL1325279	22286	8	None	-7	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	5	1	7	3.0	CCc1nnc(NC(=O)CSc2nc3c(cc2C#N)CCCC3)s1	nan
	4053254	22382	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	5	2	5	3.1	COc1ccc(NC(=O)CCn2c(=S)[nH]c3ccccc3c2=O)cc1	nan
	CHEMBL1326345	22382	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	5	2	5	3.1	COc1ccc(NC(=O)CCn2c(=S)[nH]c3ccccc3c2=O)cc1	nan
	2742890	22467	5	None	-7	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	3	2	2	4.3	COc1ccc2[nH]c(C(=O)Nc3ccc(F)cc3Br)cc2c1	nan
	CHEMBL1327081	22467	5	None	-7	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	3	2	2	4.3	COc1ccc2[nH]c(C(=O)Nc3ccc(F)cc3Br)cc2c1	nan
	16030465	22532	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	5	0	4	4.3	O=C(CSc1nc2ccccc2nc1Cc1ccccc1)N1CCCCC1	nan
	CHEMBL1327646	22532	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	5	0	4	4.3	O=C(CSc1nc2ccccc2nc1Cc1ccccc1)N1CCCCC1	nan
	2330460	22590	8	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	4	1	7	5.0	Cc1nn(-c2ccccc2Cl)c2sc(C(=O)Nc3nnc(C4CC4)s3)cc12	nan
	CHEMBL1328005	22590	8	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	4	1	7	5.0	Cc1nn(-c2ccccc2Cl)c2sc(C(=O)Nc3nnc(C4CC4)s3)cc12	nan
	1048410	23032	8	None	-2	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	6	2	4	5.6	COc1cc(NC(=O)c2ccc(-c3ccc(Br)cc3)o2)ccc1NC(=O)C(C)C	nan
	CHEMBL1331632	23032	8	None	-2	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	6	2	4	5.6	COc1cc(NC(=O)c2ccc(-c3ccc(Br)cc3)o2)ccc1NC(=O)C(C)C	nan
	1088560	23041	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	320	4	1	3	4.1	CC(=O)c1cn(CC(=O)Nc2ccc(C)c(C)c2)c2ccccc12	nan
	CHEMBL1331684	23041	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	320	4	1	3	4.1	CC(=O)c1cn(CC(=O)Nc2ccc(C)c(C)c2)c2ccccc12	nan
	16022830	23143	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	4	1	6	5.2	Cc1ccc(NC(=O)C2CCN(c3nnc(C)c4c(C)n(-c5ccccc5)nc34)CC2)c(Cl)c1	nan
	CHEMBL1332482	23143	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	4	1	6	5.2	Cc1ccc(NC(=O)C2CCN(c3nnc(C)c4c(C)n(-c5ccccc5)nc34)CC2)c(Cl)c1	nan
	4443607	23347	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	346	4	1	5	3.3	COc1cc2[nH]c(=S)n(Cc3ccc(F)cc3)c(=O)c2cc1OC	nan
	CHEMBL1334074	23347	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	346	4	1	5	3.3	COc1cc2[nH]c(=S)n(Cc3ccc(F)cc3)c(=O)c2cc1OC	nan
	3245441	23391	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	5	1	4	3.1	O=C(CCCN1C(=O)c2ccccc2C1=O)Nc1c2c(nc3c1CCC3)CCC2	nan
	CHEMBL1334367	23391	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	5	1	4	3.1	O=C(CCCN1C(=O)c2ccccc2C1=O)Nc1c2c(nc3c1CCC3)CCC2	nan
	16009378	23467	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	3	0	5	3.8	Cc1ccc(OCc2cc(=O)n3c4c(sc3n2)CCCC4)c(C)c1	nan
	CHEMBL1335076	23467	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	3	0	5	3.8	Cc1ccc(OCc2cc(=O)n3c4c(sc3n2)CCCC4)c(C)c1	nan
	135454500	23714	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	5	2	7	4.6	Cc1cc(-n2c(SCC(=O)Nc3ccc(F)c(F)c3)nc3nnc(C)c-3c2N)ccc1Cl	nan
	CHEMBL1337074	23714	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	5	2	7	4.6	Cc1cc(-n2c(SCC(=O)Nc3ccc(F)c(F)c3)nc3nnc(C)c-3c2N)ccc1Cl	nan
	16023881	23800	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	2	2	2	4.2	O=C(Nc1ccc(F)cc1F)c1cc2ccc3cccnc3c2[nH]1	nan
	CHEMBL1337846	23800	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	2	2	2	4.2	O=C(Nc1ccc(F)cc1F)c1cc2ccc3cccnc3c2[nH]1	nan
	3458131	23966	8	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	324	3	0	4	5.1	Cc1nc(SCc2ccc(F)cc2)c2oc3ccccc3c2n1	nan
	CHEMBL1339257	23966	8	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	324	3	0	4	5.1	Cc1nc(SCc2ccc(F)cc2)c2oc3ccccc3c2n1	nan
	3677224	23994	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	502	7	1	6	3.3	O=C(NCCc1ccccc1)c1cc(-c2ccncc2)nc2ccc(S(=O)(=O)N3CCOCC3)cc12	nan
	CHEMBL1339543	23994	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	502	7	1	6	3.3	O=C(NCCc1ccccc1)c1cc(-c2ccncc2)nc2ccc(S(=O)(=O)N3CCOCC3)cc12	nan
	4625935	24053	14	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	4	1	4	4.4	CC(=O)c1sc(NC(=O)c2ccc(F)cc2)nc1-c1ccccc1	nan
	CHEMBL1340080	24053	14	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	4	1	4	4.4	CC(=O)c1sc(NC(=O)c2ccc(F)cc2)nc1-c1ccccc1	nan
	1873236	24328	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	3	1	7	2.6	COC(=O)c1ccc2c(=O)n(Cc3ccc4c(c3)OCO4)c(=S)[nH]c2c1	nan
	CHEMBL1342433	24328	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	3	1	7	2.6	COC(=O)c1ccc2c(=O)n(Cc3ccc4c(c3)OCO4)c(=S)[nH]c2c1	nan
	1302080	24388	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	4	2	4	2.8	O=C(CCc1ccccc1)NC(=S)Nc1ccc2c(c1)C(=O)OC2	nan
	CHEMBL1342849	24388	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	4	2	4	2.8	O=C(CCc1ccccc1)NC(=S)Nc1ccc2c(c1)C(=O)OC2	nan
	3185654	24433	3	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	536	9	3	8	3.3	COc1ccccc1N(C(=O)c1snc(C(N)=O)c1N)C(C(=O)NC1CCCC1)c1ccc(N(C)C)cc1	nan
	CHEMBL1343261	24433	3	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	536	9	3	8	3.3	COc1ccccc1N(C(=O)c1snc(C(N)=O)c1N)C(C(=O)NC1CCCC1)c1ccc(N(C)C)cc1	nan
	1164441	24484	6	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	5	1	7	4.8	COc1ccc2nc(SCC(=O)Nc3ccc4sc(C)nc4c3)c(C#N)cc2c1	nan
	CHEMBL1343720	24484	6	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	5	1	7	4.8	COc1ccc2nc(SCC(=O)Nc3ccc4sc(C)nc4c3)c(C#N)cc2c1	nan
	653965	24509	4	None	-3	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	3	0	4	3.8	Cc1cc(C)c2nc(SCC(=O)N3CCCCC3)c(C#N)cc2c1	nan
	CHEMBL1343941	24509	4	None	-3	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	3	0	4	3.8	Cc1cc(C)c2nc(SCC(=O)N3CCCCC3)c(C#N)cc2c1	nan
	5068572	24975	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	358	5	1	6	3.1	COc1ccc(Cn2c(=S)[nH]c3cc(OC)c(OC)cc3c2=O)cc1	nan
	CHEMBL1347842	24975	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	358	5	1	6	3.1	COc1ccc(Cn2c(=S)[nH]c3cc(OC)c(OC)cc3c2=O)cc1	nan
	2992621	25020	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	4	1	4	3.0	COc1cccc2cc(C(=O)NCc3ccc(C)cc3)c(=O)oc12	nan
	CHEMBL1348238	25020	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	4	1	4	3.0	COc1cccc2cc(C(=O)NCc3ccc(C)cc3)c(=O)oc12	nan
	2785932	25096	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	275	0	0	5	1.4	Cn1c(=O)c2cc3ccc(Cl)cc3nc2n(C)c1=O	nan
	CHEMBL1348983	25096	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	275	0	0	5	1.4	Cn1c(=O)c2cc3ccc(Cl)cc3nc2n(C)c1=O	nan
	20929691	25121	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	6	1	6	3.0	Cc1ccc2c(=O)c(C(=O)c3ccc(F)cc3)cn(CC(=O)NCc3ccco3)c2n1	nan
	CHEMBL1349170	25121	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	6	1	6	3.0	Cc1ccc2c(=O)c(C(=O)c3ccc(F)cc3)cn(CC(=O)NCc3ccco3)c2n1	nan
	1261778	25353	11	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	3	1	3	5.6	Cc1cccc2c(C(=O)Nc3ccc(Br)cc3)cc(-c3ccccn3)nc12	nan
	CHEMBL1351124	25353	11	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	3	1	3	5.6	Cc1cccc2c(C(=O)Nc3ccc(Br)cc3)cc(-c3ccccn3)nc12	nan
	2309203	25356	7	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	464	7	2	4	4.3	O=C(NCCCCNC(=O)c1ccc(Br)s1)c1ccc(Br)s1	nan
	CHEMBL1351160	25356	7	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	464	7	2	4	4.3	O=C(NCCCCNC(=O)c1ccc(Br)s1)c1ccc(Br)s1	nan
	1945599	25489	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	5	2	6	3.7	COc1cc(C(=O)NC(=S)Nc2cccc3nc(C)ccc23)cc(OC)c1OC	nan
	CHEMBL1352289	25489	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	5	2	6	3.7	COc1cc(C(=O)NC(=S)Nc2cccc3nc(C)ccc23)cc(OC)c1OC	nan
	2345662	25598	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	307	5	1	6	2.8	COc1ccc(-c2nnc(NC(=O)C(C)C)s2)c(OC)c1	nan
	CHEMBL1353144	25598	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	307	5	1	6	2.8	COc1ccc(-c2nnc(NC(=O)C(C)C)s2)c(OC)c1	nan
	2588947	25634	5	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	5	2	5	3.2	COc1ccc2c(-c3ccccc3)cc(SCC(=O)NC(N)=O)nc2c1	nan
	CHEMBL1353338	25634	5	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	5	2	5	3.2	COc1ccc2c(-c3ccccc3)cc(SCC(=O)NC(N)=O)nc2c1	nan
	16024589	25767	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	463	6	1	5	4.0	Cc1ccc2c(=O)c(C(=O)c3ccc(F)cc3)cn(CC(=O)NCc3ccccc3Cl)c2n1	nan
	CHEMBL1354308	25767	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	463	6	1	5	4.0	Cc1ccc2c(=O)c(C(=O)c3ccc(F)cc3)cn(CC(=O)NCc3ccccc3Cl)c2n1	nan
	24981187	25775	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	494	7	0	7	2.0	CCOC(=O)C1CCN(C(=O)COC(=O)C2CCN(S(=O)(=O)c3ccc(C)c(C)c3)CC2)CC1	nan
	CHEMBL1354340	25775	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	494	7	0	7	2.0	CCOC(=O)C1CCN(C(=O)COC(=O)C2CCN(S(=O)(=O)c3ccc(C)c(C)c3)CC2)CC1	nan
	16015624	25805	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	9	1	6	5.8	Cc1ccccc1OCC(=O)Nc1ccc2nc(SCCOc3ccccc3)sc2c1	nan
	CHEMBL1354759	25805	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	9	1	6	5.8	Cc1ccccc1OCC(=O)Nc1ccc2nc(SCCOc3ccccc3)sc2c1	nan
	16022729	25863	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	5	1	8	2.5	Cc1noc(Cn2c(=O)c3ccccc3n(CC(=O)Nc3cc(Cl)ccc3C)c2=O)n1	nan
	CHEMBL1355436	25863	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	5	1	8	2.5	Cc1noc(Cn2c(=O)c3ccccc3n(CC(=O)Nc3cc(Cl)ccc3C)c2=O)n1	nan
	15989639	25866	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	8	1	7	3.4	COc1ccc(CCn2c(=O)c3ccccc3n(CC(=O)Nc3cccc(C)c3)c2=O)cc1OC	nan
	CHEMBL1355514	25866	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	8	1	7	3.4	COc1ccc(CCn2c(=O)c3ccccc3n(CC(=O)Nc3cccc(C)c3)c2=O)cc1OC	nan
	16023098	25871	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	2	1	5	4.1	Cc1nnc2c3ccccc3nc(Nc3ccc(F)cc3Cl)n12	nan
	CHEMBL1355617	25871	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	2	1	5	4.1	Cc1nnc2c3ccccc3nc(Nc3ccc(F)cc3Cl)n12	nan
	2150160	25872	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	6	1	6	4.2	COCCCNc1nc2c(-c3cccc(Br)c3)nnn2c2ccccc12	nan
	CHEMBL1355622	25872	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	6	1	6	4.2	COCCCNc1nc2c(-c3cccc(Br)c3)nnn2c2ccccc12	nan
	135546934	25877	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	3	3	7	4.3	Cc1cccc(NC(=O)c2sc3nc(-c4cc5ccc(O)cc5oc4=O)[nH]c(=O)c3c2C)c1	nan
	CHEMBL1355684	25877	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	3	3	7	4.3	Cc1cccc(NC(=O)c2sc3nc(-c4cc5ccc(O)cc5oc4=O)[nH]c(=O)c3c2C)c1	nan
	135419178	25898	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	396	5	2	5	4.8	CC(=O)Nc1ccc(/C=C/c2nc(-c3ccccc3O)n(-c3ccccc3)n2)cc1	nan
	CHEMBL1355898	25898	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	396	5	2	5	4.8	CC(=O)Nc1ccc(/C=C/c2nc(-c3ccccc3O)n(-c3ccccc3)n2)cc1	nan
	16017045	25943	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	4	0	6	4.8	CCC(C(=O)N1CCN(c2cccc(C)c2C)CC1)n1nc(C)c2sc3ccccc3c2c1=O	nan
	CHEMBL1356499	25943	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	4	0	6	4.8	CCC(C(=O)N1CCN(c2cccc(C)c2C)CC1)n1nc(C)c2sc3ccccc3c2c1=O	nan
	15990110	25945	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	5	0	5	5.3	Cc1ccc(C)c(N2CCN(C(c3ccccc3)c3nnc(-c4ccccc4)o3)CC2)c1	nan
	CHEMBL1356570	25945	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	5	0	5	5.3	Cc1ccc(C)c(N2CCN(C(c3ccccc3)c3nnc(-c4ccccc4)o3)CC2)c1	nan
	5886984	25950	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	4	0	4	6.8	COc1c(Cl)cc(Cl)cc1/C=C(\C#N)c1nc(-c2ccc(Cl)cc2)cs1	nan
	CHEMBL1356614	25950	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	4	0	4	6.8	COc1c(Cl)cc(Cl)cc1/C=C(\C#N)c1nc(-c2ccc(Cl)cc2)cs1	nan
	16018240	25972	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	6	1	5	5.2	Cc1c(C(=O)NCc2ccc(N(C)C)cc2)oc2c1-c1nn(Cc3cccc(Cl)c3)cc1CC2	nan
	CHEMBL1356884	25972	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	6	1	5	5.2	Cc1c(C(=O)NCc2ccc(N(C)C)cc2)oc2c1-c1nn(Cc3cccc(Cl)c3)cc1CC2	nan
	2219490	25982	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	5	1	4	5.1	O=C(Cn1cc(C(=O)c2ccco2)c2ccccc21)Nc1ccccc1C(F)(F)F	nan
	CHEMBL1357026	25982	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	5	1	4	5.1	O=C(Cn1cc(C(=O)c2ccco2)c2ccccc21)Nc1ccccc1C(F)(F)F	nan
	16007510	26007	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	440	7	1	4	5.6	CCOc1ccc(CNC(=O)CSc2c3c(nc4ccc(Cl)cc24)CCCC3)cc1	nan
	CHEMBL1357328	26007	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	440	7	1	4	5.6	CCOc1ccc(CNC(=O)CSc2c3c(nc4ccc(Cl)cc24)CCCC3)cc1	nan
	16010573	26008	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	410	8	1	7	2.6	CCOc1ccccc1NC(=O)Cn1c(=O)n(CCC(C)C)c(=O)c2cccnc21	nan
	CHEMBL1357333	26008	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	410	8	1	7	2.6	CCOc1ccccc1NC(=O)Cn1c(=O)n(CCC(C)C)c(=O)c2cccnc21	nan
	7533493	26014	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	7	1	6	4.1	CCOc1ccc(-c2nnc(SCC(=O)Nc3cc(F)ccc3F)o2)cc1	nan
	CHEMBL1357469	26014	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	7	1	6	4.1	CCOc1ccc(-c2nnc(SCC(=O)Nc3cc(F)ccc3F)o2)cc1	nan
	16030313	26038	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	5	1	5	4.1	Cc1ccccc1C(=O)Nc1ccc(OCc2cc(=O)n3cccc(C)c3n2)cc1	nan
	CHEMBL1357868	26038	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	5	1	5	4.1	Cc1ccccc1C(=O)Nc1ccc(OCc2cc(=O)n3cccc(C)c3n2)cc1	nan
	7244606	26041	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	410	4	0	7	2.9	C#CCn1/c(=N/C(=O)c2ccc3c(c2)OCCO3)sc2cc(OC)c(OC)cc21	nan
	CHEMBL1357945	26041	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	410	4	0	7	2.9	C#CCn1/c(=N/C(=O)c2ccc3c(c2)OCCO3)sc2cc(OC)c(OC)cc21	nan
	16018859	26045	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	5	1	5	4.1	O=C(CCCn1c(=O)c2cccn2c2cccnc21)Nc1ccccc1C(F)(F)F	nan
	CHEMBL1357984	26045	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	5	1	5	4.1	O=C(CCCn1c(=O)c2cccn2c2cccnc21)Nc1ccccc1C(F)(F)F	nan
	16009434	26049	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	7	1	7	3.4	O=C(COc1ccccc1)Nc1ccc(OCc2cc(=O)n3ccsc3n2)cc1	nan
	CHEMBL1358022	26049	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	7	1	7	3.4	O=C(COc1ccccc1)Nc1ccc(OCc2cc(=O)n3ccsc3n2)cc1	nan
	15987969	26125	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	492	7	1	4	4.1	CCC(=O)N1CCc2cc(Br)cc(S(=O)(=O)CCC(=O)Nc3cccc(CC)c3)c21	nan
	CHEMBL1358851	26125	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	492	7	1	4	4.1	CCC(=O)N1CCc2cc(Br)cc(S(=O)(=O)CCC(=O)Nc3cccc(CC)c3)c21	nan
	3799752	26126	8	None	-3	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	6	2	6	2.4	COc1ccc(OC)c(N/C=C2/C(=O)NC(=S)N(Cc3ccccc3)C2=O)c1	nan
	CHEMBL1358861	26126	8	None	-3	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	6	2	6	2.4	COc1ccc(OC)c(N/C=C2/C(=O)NC(=S)N(Cc3ccccc3)C2=O)c1	nan
	7210861	26203	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	5	2	5	3.6	CCn1c(SCC(=O)Nc2ccccc2)nc2c([nH]c3ccccc32)c1=O	nan
	CHEMBL1359450	26203	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	5	2	5	3.6	CCn1c(SCC(=O)Nc2ccccc2)nc2c([nH]c3ccccc32)c1=O	nan
	1818953	26362	16	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	488	6	0	6	5.7	C=C(C)Cn1c(SCC(=O)c2ccc(Br)cc2)nc2sc3c(c2c1=O)CCCC3	nan
	CHEMBL1360901	26362	16	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	488	6	0	6	5.7	C=C(C)Cn1c(SCC(=O)c2ccc(Br)cc2)nc2sc3c(c2c1=O)CCCC3	nan
	16022921	26424	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	498	7	1	7	4.7	CCOc1ccccc1CNC(=O)C1CCN(c2nnc(C)c3c(C)n(-c4ccc(C)cc4)nc23)CC1	nan
	CHEMBL1361507	26424	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	498	7	1	7	4.7	CCOc1ccccc1CNC(=O)C1CCN(c2nnc(C)c3c(C)n(-c4ccc(C)cc4)nc23)CC1	nan
	4329717	26437	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	3	2	3	4.2	CC(NC(=O)c1cc(O)nc2ccc(Br)cc12)c1ccccc1	nan
	CHEMBL1361599	26437	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	3	2	3	4.2	CC(NC(=O)c1cc(O)nc2ccc(Br)cc12)c1ccccc1	nan
	3475073	26475	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	4	1	2	5.4	Cc1cc2ccccc2n1CCNC(=O)c1cc(C(F)(F)F)cc(C(F)(F)F)c1	nan
	CHEMBL1361903	26475	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	4	1	2	5.4	Cc1cc2ccccc2n1CCNC(=O)c1cc(C(F)(F)F)cc(C(F)(F)F)c1	nan
	16022126	26504	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	441	5	1	5	4.5	COc1cc(OC)c(NC(=O)c2c(N3CCCC3=O)c3cc(C)ccc3n2C)cc1Cl	nan
	CHEMBL1362140	26504	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	441	5	1	5	4.5	COc1cc(OC)c(NC(=O)c2c(N3CCCC3=O)c3cc(C)ccc3n2C)cc1Cl	nan
	1984900	26529	8	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	531	8	1	7	5.0	CCOc1ccc(S(=O)(=O)[N-]c2nc3ccccc3nc2-[n+]2ccc(NC(=O)c3cccs3)cc2)cc1	nan
	CHEMBL1362375	26529	8	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	531	8	1	7	5.0	CCOc1ccc(S(=O)(=O)[N-]c2nc3ccccc3nc2-[n+]2ccc(NC(=O)c3cccs3)cc2)cc1	nan
	6471827	26560	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	5	1	9	2.4	Cc1nnc(NC(=O)C(C)Sc2nnc(-c3ccco3)n2C)s1	nan
	CHEMBL1362583	26560	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	5	1	9	2.4	Cc1nnc(NC(=O)C(C)Sc2nnc(-c3ccco3)n2C)s1	nan
	7693885	26573	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	308	4	1	4	3.9	COc1ccc(C(=O)Nc2cc(-c3ccc(C)cc3)no2)cc1	nan
	CHEMBL1362677	26573	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	308	4	1	4	3.9	COc1ccc(C(=O)Nc2cc(-c3ccc(C)cc3)no2)cc1	nan
	16019393	26584	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	6	1	8	4.0	CCCCNc1nc2c(S(=O)(=O)c3ccc(Cl)cc3)nnn2c2ccsc12	nan
	CHEMBL1362800	26584	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	6	1	8	4.0	CCCCNc1nc2c(S(=O)(=O)c3ccc(Cl)cc3)nnn2c2ccsc12	nan
	22334175	26602	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	548	10	2	10	2.8	COc1ccc(-n2nc(C(=O)NCC(=O)Nc3cc(OC)c(OC)c(OC)c3)c3ccccc3c2=O)cc1OC	nan
	CHEMBL1362992	26602	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	548	10	2	10	2.8	COc1ccc(-n2nc(C(=O)NCC(=O)Nc3cc(OC)c(OC)c(OC)c3)c3ccccc3c2=O)cc1OC	nan
	645413	26613	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	3	1	5	3.4	Cc1cc(C(F)F)n2nc(C(=O)Nc3ccccc3Br)nc2n1	nan
	CHEMBL1363101	26613	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	3	1	5	3.4	Cc1cc(C(F)F)n2nc(C(=O)Nc3ccccc3Br)nc2n1	nan
	16024545	26623	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	5	1	5	4.8	Cc1ccc(C)c(NC(=O)Cn2cc(C(=O)c3ccc(Cl)cc3)c(=O)c3ccc(C)nc32)c1	nan
	CHEMBL1363144	26623	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	5	1	5	4.8	Cc1ccc(C)c(NC(=O)Cn2cc(C(=O)c3ccc(Cl)cc3)c(=O)c3ccc(C)nc32)c1	nan
	4447999	26659	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	492	8	2	6	4.6	Cc1ccc(NC(=O)CSc2nc3ccccc3c(=O)n2CCC(=O)NC2CCCCC2)cc1C	nan
	CHEMBL1363483	26659	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	492	8	2	6	4.6	Cc1ccc(NC(=O)CSc2nc3ccccc3c(=O)n2CCC(=O)NC2CCCCC2)cc1C	nan
	16030946	26709	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	7	1	7	4.1	COc1ccc(NC(=O)CSc2ccc3nc(-c4ccccc4)cn3n2)cc1OC	nan
	CHEMBL1363950	26709	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	7	1	7	4.1	COc1ccc(NC(=O)CSc2ccc3nc(-c4ccccc4)cn3n2)cc1OC	nan
	1960168	26767	9	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	2	0	5	4.4	Cc1ccc(-c2nc3c(c(=O)c4ccccc4n3C)c(=O)n2-c2ccc(F)cc2)cc1	nan
	CHEMBL1364491	26767	9	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	2	0	5	4.4	Cc1ccc(-c2nc3c(c(=O)c4ccccc4n3C)c(=O)n2-c2ccc(F)cc2)cc1	nan
	1258567	26959	17	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	7	1	7	5.5	COc1ccc(-c2cc(-c3ccccc3)nc(SCC(=O)Nc3nccs3)c2C#N)cc1	nan
	CHEMBL1366086	26959	17	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	7	1	7	5.5	COc1ccc(-c2cc(-c3ccccc3)nc(SCC(=O)Nc3nccs3)c2C#N)cc1	nan
	5726342	26993	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	3	1	3	3.8	CN1C(=O)C(O)=C(C(=O)c2ccc(Br)cc2)C1c1ccc(F)cc1	nan
	CHEMBL1366379	26993	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	3	1	3	3.8	CN1C(=O)C(O)=C(C(=O)c2ccc(Br)cc2)C1c1ccc(F)cc1	nan
	16015810	27007	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	6	1	5	5.3	COc1ccc(OCC(=O)Nc2cccc(-c3nc4ccccc4s3)c2C)cc1	nan
	CHEMBL1366460	27007	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	6	1	5	5.3	COc1ccc(OCC(=O)Nc2cccc(-c3nc4ccccc4s3)c2C)cc1	nan
	5204153	27028	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	486	5	2	7	1.3	CCOC(=O)N1CCN(S(=O)(=O)c2ccc(C(=O)Nc3ccc4c(c3)C(=O)NC4=O)cc2)CC1	nan
	CHEMBL1366674	27028	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	486	5	2	7	1.3	CCOC(=O)N1CCN(S(=O)(=O)c2ccc(C(=O)Nc3ccc4c(c3)C(=O)NC4=O)cc2)CC1	nan
	16015685	27066	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	5	1	5	5.5	Cc1ccc(C(=O)Nc2ccc3nc(SCC(=O)N4CCc5ccccc54)sc3c2)cc1	nan
	CHEMBL1367053	27066	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	5	1	5	5.5	Cc1ccc(C(=O)Nc2ccc3nc(SCC(=O)N4CCc5ccccc54)sc3c2)cc1	nan
	561651	27179	21	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	288	3	0	3	4.6	c1ccc(C2=NN(c3ccccc3)C(c3ccco3)C2)cc1	nan
	CHEMBL1367925	27179	21	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	288	3	0	3	4.6	c1ccc(C2=NN(c3ccccc3)C(c3ccco3)C2)cc1	nan
	16022119	27408	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	489	6	0	8	3.9	COc1ccc2c(c1)c1c(c(=O)n(-c3ccc(OC)c(OC)c3)c(=O)n1Cc1ccc(F)cc1)n2C	nan
	CHEMBL1369667	27408	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	489	6	0	8	3.9	COc1ccc2c(c1)c1c(c(=O)n(-c3ccc(OC)c(OC)c3)c(=O)n1Cc1ccc(F)cc1)n2C	nan
	16024643	27438	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	8	1	5	3.9	CCc1ccc(C(=O)c2cn(CC(=O)NCCc3ccccc3)c3nc(C)ccc3c2=O)cc1	nan
	CHEMBL1369852	27438	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	8	1	5	3.9	CCc1ccc(C(=O)c2cn(CC(=O)NCCc3ccccc3)c3nc(C)ccc3c2=O)cc1	nan
	16018703	27482	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	4	0	6	3.4	Cc1ccc(Cl)cc1N1CCN(C(=O)CCn2c(=O)c3cccn3c3cccnc32)CC1	nan
	CHEMBL1370112	27482	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	4	0	6	3.4	Cc1ccc(Cl)cc1N1CCN(C(=O)CCn2c(=O)c3cccn3c3cccnc32)CC1	nan
	16017844	27559	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	6	1	6	1.6	COc1cccc(-n2ccn(CC(=O)NCc3ccc(C)cc3)c(=O)c2=O)c1	nan
	CHEMBL1370655	27559	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	6	1	6	1.6	COc1cccc(-n2ccn(CC(=O)NCc3ccc(C)cc3)c(=O)c2=O)c1	nan
	2053979	27574	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	3	0	5	4.0	CCN(C(=O)c1cc2c(=O)n3cccc(C)c3nc2s1)C1CCCCC1	nan
	CHEMBL1370734	27574	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	3	0	5	4.0	CCN(C(=O)c1cc2c(=O)n3cccc(C)c3nc2s1)C1CCCCC1	nan
	2999996	27601	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	3	0	9	2.9	O=C(OCc1cc(=O)n2c(n1)sc1ccccc12)c1ccc2c(=O)n3c(nc2c1)CCC3	nan
	CHEMBL1370976	27601	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	3	0	9	2.9	O=C(OCc1cc(=O)n2c(n1)sc1ccccc12)c1ccc2c(=O)n3c(nc2c1)CCC3	nan
	2212806	27655	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	5	2	4	5.1	Cc1cccc(NC(=O)c2cc(NC(=O)c3ccco3)ccc2N2CCCCC2)c1	nan
	CHEMBL1371405	27655	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	5	2	4	5.1	Cc1cccc(NC(=O)c2cc(NC(=O)c3ccco3)ccc2N2CCCCC2)c1	nan
	4069120	27673	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	5	1	5	4.7	COc1ccc(OC)c(NC(=O)c2oc(=O)c3ccccc3c2-c2ccccc2)c1	nan
	CHEMBL1371548	27673	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	5	1	5	4.7	COc1ccc(OC)c(NC(=O)c2oc(=O)c3ccccc3c2-c2ccccc2)c1	nan
	862401	27686	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	330	5	1	4	3.7	COc1ccc2nc(SCC(=O)NC3CCCC3)c(C)cc2c1	nan
	CHEMBL1371650	27686	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	330	5	1	4	3.7	COc1ccc2nc(SCC(=O)NC3CCCC3)c(C)cc2c1	nan
	941550	27690	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	315	4	1	6	3.4	COc1ccc2nc(O)c(COC(=O)c3cccs3)cc2c1	nan
	CHEMBL1371690	27690	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	315	4	1	6	3.4	COc1ccc2nc(O)c(COC(=O)c3cccs3)cc2c1	nan
	648869	27810	4	None	-3	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	5	0	5	3.9	CCOc1ccc2cc(C#N)c(SCC(=O)N3CCC(C)CC3)nc2c1	nan
	CHEMBL1372547	27810	4	None	-3	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	5	0	5	3.9	CCOc1ccc2cc(C#N)c(SCC(=O)N3CCC(C)CC3)nc2c1	nan
	664361	27857	12	None	-3	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	4	1	5	4.4	Cc1nc(SCC(=O)Nc2ccccc2)c2oc3ccccc3c2n1	nan
	CHEMBL1372818	27857	12	None	-3	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	4	1	5	4.4	Cc1nc(SCC(=O)Nc2ccccc2)c2oc3ccccc3c2n1	nan
	2404728	27985	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	4	2	5	2.4	O=C(COC(=O)c1ccc(Cl)cc1O)NC(=O)C1CCCCC1	nan
	CHEMBL1373640	27985	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	4	2	5	2.4	O=C(COC(=O)c1ccc(Cl)cc1O)NC(=O)C1CCCCC1	nan
	711468	28022	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	287	1	1	3	3.3	Cc1cc(-c2cccc(Br)c2)c(C#N)c(N)n1	nan
	CHEMBL1373906	28022	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	287	1	1	3	3.3	Cc1cc(-c2cccc(Br)c2)c(C#N)c(N)n1	nan
	660358	28064	18	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	6	1	8	4.8	CCOC(=O)c1sc(NC(=O)CSc2nc3c(cc2C#N)CCCCCC3)c(C#N)c1C	nan
	CHEMBL1374224	28064	18	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	6	1	8	4.8	CCOC(=O)c1sc(NC(=O)CSc2nc3c(cc2C#N)CCCCCC3)c(C#N)c1C	nan
	848636	28108	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	2	0	6	5.1	Cc1sc2ncnc(Sc3nc4ccccc4s3)c2c1C	nan
	CHEMBL1374559	28108	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	2	0	6	5.1	Cc1sc2ncnc(Sc3nc4ccccc4s3)c2c1C	nan
	22330687	28131	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	5	1	8	4.3	COc1ccc(C)cc1NC(=O)c1sc2ncnc(N3CCN(c4ccccn4)CC3)c2c1C	nan
	CHEMBL1374703	28131	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	5	1	8	4.3	COc1ccc(C)cc1NC(=O)c1sc2ncnc(N3CCN(c4ccccn4)CC3)c2c1C	nan
	16421351	28158	15	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	5	1	6	3.8	COc1ccc(-c2cc3ccc(O)c(CN4CCCC4)c3oc2=O)cc1OC	nan
	5513687	28158	15	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	5	1	6	3.8	COc1ccc(-c2cc3ccc(O)c(CN4CCCC4)c3oc2=O)cc1OC	nan
	CHEMBL1374848	28158	15	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	5	1	6	3.8	COc1ccc(-c2cc3ccc(O)c(CN4CCCC4)c3oc2=O)cc1OC	nan
	2113664	28285	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	5	0	8	4.2	CCc1cc2c(SCC(=O)C(C#N)=C3N(C)c4ccccc4N3C)ncnc2s1	nan
	CHEMBL1375768	28285	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	5	0	8	4.2	CCc1cc2c(SCC(=O)C(C#N)=C3N(C)c4ccccc4N3C)ncnc2s1	nan
	1049792	28336	21	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	5	0	5	5.0	COc1ccc(-c2cc(-c3ccc(OC)cc3)c(C#N)c(SC)n2)cc1	nan
	CHEMBL1376368	28336	21	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	5	0	5	5.0	COc1ccc(-c2cc(-c3ccc(OC)cc3)c(C#N)c(SC)n2)cc1	nan
	3141909	28341	8	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	239	2	0	4	3.0	Cc1cccc2cc(C#N)c(SCC#N)nc12	nan
	CHEMBL1376381	28341	8	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	239	2	0	4	3.0	Cc1cccc2cc(C#N)c(SCC#N)nc12	nan
	1086373	28394	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	7	1	6	3.6	COc1cccc(-c2ccc(C#N)c(SCC(=O)NCc3ccco3)n2)c1	nan
	CHEMBL1376846	28394	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	7	1	6	3.6	COc1cccc(-c2ccc(C#N)c(SCC(=O)NCc3ccco3)n2)c1	nan
	16024493	28483	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	6	1	5	3.3	Cc1ccc2c(=O)c(C(=O)c3ccccc3)cn(CC(=O)NCc3ccccc3)c2n1	nan
	CHEMBL1377756	28483	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	6	1	5	3.3	Cc1ccc2c(=O)c(C(=O)c3ccccc3)cn(CC(=O)NCc3ccccc3)c2n1	nan
	16018882	28489	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	495	9	1	5	4.2	CCOc1ccc(N(CC)S(=O)(=O)N2CCCC(C(=O)Nc3ccc(OC)c(Cl)c3)C2)cc1	nan
	CHEMBL1377806	28489	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	495	9	1	5	4.2	CCOc1ccc(N(CC)S(=O)(=O)N2CCCC(C(=O)Nc3ccc(OC)c(Cl)c3)C2)cc1	nan
	2426511	28556	3	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	240	0	0	4	2.7	Cc1cc(=O)n2c(sc3ccccc32)c1C#N	nan
	CHEMBL1378393	28556	3	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	240	0	0	4	2.7	Cc1cc(=O)n2c(sc3ccccc32)c1C#N	nan
	2060585	28571	61	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	224	1	1	2	1.4	O=C(c1ccccc1Cl)N1CCNCC1	nan
	CHEMBL1378602	28571	61	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	224	1	1	2	1.4	O=C(c1ccccc1Cl)N1CCNCC1	nan
	54680441	28645	17	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	294	3	3	4	2.6	O=C(NCc1ccccc1)c1c(O)nc2ccccc2c1O	nan
	CHEMBL1379243	28645	17	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	294	3	3	4	2.6	O=C(NCc1ccccc1)c1c(O)nc2ccccc2c1O	nan
	7502810	28703	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	5	1	6	3.9	Cc1cc(NC(=O)CSc2ccc(-c3ccc(Br)cc3)nn2)no1	nan
	CHEMBL1379696	28703	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	5	1	6	3.9	Cc1cc(NC(=O)CSc2ccc(-c3ccc(Br)cc3)nn2)no1	nan
	663350	28763	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	5	0	9	2.9	COc1cc(OC)c(-c2nn3c(-c4cccnc4)nnc3s2)cc1OC	nan
	CHEMBL1380292	28763	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	5	0	9	2.9	COc1cc(OC)c(-c2nn3c(-c4cccnc4)nnc3s2)cc1OC	nan
	551775	28857	13	None	-2	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	345	6	0	5	4.0	CCN(CC)C(=O)CSc1nc(C)cc(-c2cccs2)c1C#N	nan
	CHEMBL1380940	28857	13	None	-2	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	345	6	0	5	4.0	CCN(CC)C(=O)CSc1nc(C)cc(-c2cccs2)c1C#N	nan
	6470016	28993	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	4	2	2	3.4	CC1=C(C)CC(C(=O)NCc2cccc(Cl)c2)C(C(=O)O)C1	nan
	CHEMBL1382205	28993	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	4	2	2	3.4	CC1=C(C)CC(C(=O)NCc2cccc(Cl)c2)C(C(=O)O)C1	nan
	4908628	29002	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	356	4	1	4	3.4	Cc1ccc(S(=O)(=O)N(C)Cc2cc3cc(C)ccc3nc2O)cc1	nan
	CHEMBL1382276	29002	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	356	4	1	4	3.4	Cc1ccc(S(=O)(=O)N(C)Cc2cc3cc(C)ccc3nc2O)cc1	nan
	1450725	29005	3	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	3	0	7	1.8	N#Cc1cc2cc3c(cc2nc1SCC(=O)N1CCOCC1)OCO3	nan
	CHEMBL1382288	29005	3	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	3	0	7	1.8	N#Cc1cc2cc3c(cc2nc1SCC(=O)N1CCOCC1)OCO3	nan
	5155717	29162	5	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	4	2	5	2.1	NS(=O)(=O)c1ccc(CCn2c(=S)[nH]c3ccc(F)cc3c2=O)cc1	nan
	CHEMBL1383680	29162	5	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	4	2	5	2.1	NS(=O)(=O)c1ccc(CCn2c(=S)[nH]c3ccc(F)cc3c2=O)cc1	nan
	1271521	29356	11	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	4	1	5	4.9	O=C(Nc1ccc(-c2noc(-c3ccccc3F)n2)cc1)c1cccs1	nan
	CHEMBL1385411	29356	11	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	4	1	5	4.9	O=C(Nc1ccc(-c2noc(-c3ccccc3F)n2)cc1)c1cccs1	nan
	1604314	29494	12	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	4	0	6	3.6	CCOC(=O)C1=C(c2ccccc2)O/C(=C(/C(=O)OC)C(F)(F)F)S1	nan
	CHEMBL1386476	29494	12	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	4	0	6	3.6	CCOC(=O)C1=C(c2ccccc2)O/C(=C(/C(=O)OC)C(F)(F)F)S1	nan
	2815677	29510	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	260	3	0	6	1.5	CCOC(=O)c1cn2nc(N3CCCC3)ccc2n1	nan
	CHEMBL1386622	29510	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	260	3	0	6	1.5	CCOC(=O)c1cn2nc(N3CCCC3)ccc2n1	nan
	979520	29632	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	9	2	4	4.5	COc1cc(CNCc2ccccc2Cl)ccc1OCC(=O)NC1CCCCC1	nan
	CHEMBL1387627	29632	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	9	2	4	4.5	COc1cc(CNCc2ccccc2Cl)ccc1OCC(=O)NC1CCCCC1	nan
	855469	29668	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	4	1	6	3.4	Cc1cc(NC(=O)CSc2nc3c(C)cccc3cc2C#N)no1	nan
	CHEMBL1387916	29668	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	4	1	6	3.4	Cc1cc(NC(=O)CSc2nc3c(C)cccc3cc2C#N)no1	nan
	1026561	29679	11	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	7	2	3	4.5	CCOc1ccc(Br)cc1C(=O)Nc1ccc(C(=O)NCC(C)C)cc1	nan
	CHEMBL1388002	29679	11	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	7	2	3	4.5	CCOc1ccc(Br)cc1C(=O)Nc1ccc(C(=O)NCC(C)C)cc1	nan
	2372910	29724	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	274	2	0	5	3.3	c1ccc(-c2cc(-c3nnco3)c3ccccc3n2)nc1	nan
	CHEMBL1388328	29724	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	274	2	0	5	3.3	c1ccc(-c2cc(-c3nnco3)c3ccccc3n2)nc1	nan
	4909035	29964	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	4	0	5	4.0	Cc1cccc(-c2nc3c(c(SCC(=O)N4CCCC4)n2)COC(C)(C)C3)c1	nan
	CHEMBL1390262	29964	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	4	0	5	4.0	Cc1cccc(-c2nc3c(c(SCC(=O)N4CCCC4)n2)COC(C)(C)C3)c1	nan
	20969169	29991	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	4	1	7	4.1	COc1ccc(Cl)cc1NC(=O)c1sc2nc(C)nc(N3CCOCC3)c2c1C	nan
	CHEMBL1390480	29991	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	4	1	7	4.1	COc1ccc(Cl)cc1NC(=O)c1sc2nc(C)nc(N3CCOCC3)c2c1C	nan
	4688970	29998	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	3	1	6	4.2	Cc1nc(N2CCOCC2)c2c(C)c(C(=O)Nc3ccc(F)cc3Cl)sc2n1	nan
	CHEMBL1390558	29998	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	3	1	6	4.2	Cc1nc(N2CCOCC2)c2c(C)c(C(=O)Nc3ccc(F)cc3Cl)sc2n1	nan
	6621188	30002	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	363	6	2	4	2.3	CCc1ccc(NC(=O)CNC(=O)Cn2ccc3ccccc3c2=O)cc1	nan
	CHEMBL1390571	30002	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	363	6	2	4	2.3	CCc1ccc(NC(=O)CNC(=O)Cn2ccc3ccccc3c2=O)cc1	nan
	24687564	30139	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	441	6	2	7	4.0	CCOC(=O)c1c(NC(=O)COc2ccccc2C#N)sc2c1CC(C)(C)NC2(C)C	nan
	CHEMBL1391818	30139	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	441	6	2	7	4.0	CCOC(=O)c1c(NC(=O)COc2ccccc2C#N)sc2c1CC(C)(C)NC2(C)C	nan
	8030390	30236	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	4	1	5	3.1	Cc1c(C)c2ccc(OCC(=O)Nc3ccccn3)c(C)c2oc1=O	nan
	CHEMBL1392611	30236	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	4	1	5	3.1	Cc1c(C)c2ccc(OCC(=O)Nc3ccccn3)c(C)c2oc1=O	nan
	649622	30306	3	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	316	4	0	7	2.5	CCOC(=O)CSc1nc2cc3c(cc2cc1C#N)OCO3	nan
	CHEMBL1393221	30306	3	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	316	4	0	7	2.5	CCOC(=O)CSc1nc2cc3c(cc2cc1C#N)OCO3	nan
	16024685	30404	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	499	5	1	5	5.2	Cc1ccc2c(=O)c(C(=O)c3cccc(Cl)c3)cn(CC(=O)Nc3ccccc3C(F)(F)F)c2n1	nan
	CHEMBL1394039	30404	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	499	5	1	5	5.2	Cc1ccc2c(=O)c(C(=O)c3cccc(Cl)c3)cn(CC(=O)Nc3ccccc3C(F)(F)F)c2n1	nan
	3844740	30406	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	7	3	7	3.8	COc1ccc(C2C=C(c3ccc(Cl)cc3)Nc3nc(NC(=O)CCC(=O)O)nn32)cc1	nan
	CHEMBL1394052	30406	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	7	3	7	3.8	COc1ccc(C2C=C(c3ccc(Cl)cc3)Nc3nc(NC(=O)CCC(=O)O)nn32)cc1	nan
	16024945	30418	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	3	1	4	4.8	O=C(Nc1cccc(C(F)(F)F)c1)c1ccc2c(c1)nnn2C1CCCC1	nan
	CHEMBL1394171	30418	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	3	1	4	4.8	O=C(Nc1cccc(C(F)(F)F)c1)c1ccc2c(c1)nnn2C1CCCC1	nan
	2136700	30425	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	5	1	5	3.8	Cc1ccccc1NC(=O)Cn1cc(S(=O)(=O)c2ccccc2)c(=O)c2ccccc21	nan
	CHEMBL1394236	30425	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	5	1	5	3.8	Cc1ccccc1NC(=O)Cn1cc(S(=O)(=O)c2ccccc2)c(=O)c2ccccc21	nan
	16017140	30463	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	5	1	5	5.0	Cc1ccc(C)c(NC(=O)CCCn2nc(C)c3sc4ccccc4c3c2=O)c1	nan
	CHEMBL1394852	30463	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	5	1	5	5.0	Cc1ccc(C)c(NC(=O)CCCn2nc(C)c3sc4ccccc4c3c2=O)c1	nan
	16022416	30464	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	7	2	7	4.6	CCc1ccccc1Nc1nn2c(=O)c3ccc(C(=O)NCCc4ccccc4)cc3nc2s1	nan
	CHEMBL1394859	30464	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	7	2	7	4.6	CCc1ccccc1Nc1nn2c(=O)c3ccc(C(=O)NCCc4ccccc4)cc3nc2s1	nan
	16030605	30471	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	6	0	5	5.3	COc1ccccc1Cc1nc2ccccc2nc1SCC(=O)N1CCCc2ccccc21	nan
	CHEMBL1394911	30471	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	6	0	5	5.3	COc1ccccc1Cc1nc2ccccc2nc1SCC(=O)N1CCCc2ccccc21	nan
	16034772	30506	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	6	1	6	4.6	Cc1nn(CCCC(=O)Nc2cccc(C(F)(F)F)c2)c(=O)c2nn(-c3ccccc3)c(C)c12	nan
	CHEMBL1395185	30506	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	6	1	6	4.6	Cc1nn(CCCC(=O)Nc2cccc(C(F)(F)F)c2)c(=O)c2nn(-c3ccccc3)c(C)c12	nan
	2007143	30510	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	5	1	6	1.9	CCOC(=O)CNC(=O)c1ccc(-c2nn(C)c(=O)c3ccccc23)cc1	nan
	CHEMBL1395237	30510	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	5	1	6	1.9	CCOC(=O)CNC(=O)c1ccc(-c2nn(C)c(=O)c3ccccc23)cc1	nan
	16019606	30511	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	5	1	8	4.7	Cc1ccc(S(=O)(=O)c2nnn3c2nc(NCc2ccccc2Cl)c2sccc23)cc1	nan
	CHEMBL1395245	30511	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	5	1	8	4.7	Cc1ccc(S(=O)(=O)c2nnn3c2nc(NCc2ccccc2Cl)c2sccc23)cc1	nan
	16018799	30513	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	5	1	5	3.2	CCc1cccc(NC(=O)CCn2c(=O)c3cccn3c3cccnc32)c1	nan
	CHEMBL1395272	30513	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	5	1	5	3.2	CCc1cccc(NC(=O)CCn2c(=O)c3cccn3c3cccnc32)c1	nan
	15987986	30532	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	496	6	1	4	4.0	CCC(=O)N1CCc2cc(Br)cc(S(=O)(=O)CCC(=O)Nc3ccc(C)c(F)c3)c21	nan
	CHEMBL1395557	30532	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	496	6	1	4	4.0	CCC(=O)N1CCc2cc(Br)cc(S(=O)(=O)CCC(=O)Nc3ccc(C)c(F)c3)c21	nan
	16009626	30546	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	4	2	3	5.7	Cc1cc(C)cc(C(=O)Nc2c(C(=O)Nc3ccccc3F)oc3ccccc23)c1	nan
	CHEMBL1395778	30546	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	4	2	3	5.7	Cc1cc(C)cc(C(=O)Nc2c(C(=O)Nc3ccccc3F)oc3ccccc23)c1	nan
	16017553	30569	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	4	1	6	2.7	O=C(Nc1nnc(S(=O)(=O)N2CCCCC2)s1)c1ccccc1Br	nan
	CHEMBL1396131	30569	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	4	1	6	2.7	O=C(Nc1nnc(S(=O)(=O)N2CCCCC2)s1)c1ccccc1Br	nan
	16033012	30594	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	500	4	0	7	3.3	O=C(Cn1c(=O)n2nc(-c3cccc(F)c3)nc2c2ccccc21)N1CCN(c2ccccc2F)CC1	nan
	CHEMBL1396543	30594	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	500	4	0	7	3.3	O=C(Cn1c(=O)n2nc(-c3cccc(F)c3)nc2c2ccccc21)N1CCN(c2ccccc2F)CC1	nan
	15989006	30601	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	515	7	1	8	3.5	O=C(CCn1c(=O)c2sccc2n(Cc2ccc(F)cc2Cl)c1=O)NCc1ccc2c(c1)OCO2	nan
	CHEMBL1396634	30601	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	515	7	1	8	3.5	O=C(CCn1c(=O)c2sccc2n(Cc2ccc(F)cc2Cl)c1=O)NCc1ccc2c(c1)OCO2	nan
	16009460	30624	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	7	1	8	3.6	COc1ccc(C(=O)Nc2ccc(OCc3cc(=O)n4ccsc4n3)cc2)cc1OC	nan
	CHEMBL1396932	30624	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	7	1	8	3.6	COc1ccc(C(=O)Nc2ccc(OCc3cc(=O)n4ccsc4n3)cc2)cc1OC	nan
	3408184	30635	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	457	7	1	5	5.8	CCOc1ccc(-c2cc(C(F)(F)F)c(C#N)c(SCC(=O)Nc3ccccc3)n2)cc1	nan
	CHEMBL1397049	30635	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	457	7	1	5	5.8	CCOc1ccc(-c2cc(C(F)(F)F)c(C#N)c(SCC(=O)Nc3ccccc3)n2)cc1	nan
	4345038	30640	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	466	6	1	3	5.2	CN(Cc1ccccc1)S(=O)(=O)c1ccc(F)c(C(=O)Nc2cccc(Cl)c2Cl)c1	nan
	CHEMBL1397130	30640	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	466	6	1	3	5.2	CN(Cc1ccccc1)S(=O)(=O)c1ccc(F)c(C(=O)Nc2cccc(Cl)c2Cl)c1	nan
	16017005	30642	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	6	1	4	4.9	CCOc1ccc(NC(=O)C(=O)c2cc(C)n(-c3cc(C)cc(C)c3)c2C)cc1	nan
	CHEMBL1397170	30642	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	6	1	4	4.9	CCOc1ccc(NC(=O)C(=O)c2cc(C)n(-c3cc(C)cc(C)c3)c2C)cc1	nan
	16009843	30704	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	4	1	6	3.4	O=C(Cn1c(=O)n(-c2ccccc2)c(=O)c2sc3ccccc3c21)NC1CCCC1	nan
	CHEMBL1398005	30704	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	4	1	6	3.4	O=C(Cn1c(=O)n(-c2ccccc2)c(=O)c2sc3ccccc3c21)NC1CCCC1	nan
	15988021	30720	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	514	12	2	10	1.0	COCCNC(=O)CCn1c(=O)c2cc(OC)c(OC)cc2n(CC(=O)Nc2ccccc2OC)c1=O	nan
	CHEMBL1398191	30720	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	514	12	2	10	1.0	COCCNC(=O)CCn1c(=O)c2cc(OC)c(OC)cc2n(CC(=O)Nc2ccccc2OC)c1=O	nan
	2288826	30903	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	267	2	3	4	0.6	O=C1NC(=O)C(=CNc2cc(F)cc(F)c2)C(=O)N1	nan
	CHEMBL1400030	30903	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	267	2	3	4	0.6	O=C1NC(=O)C(=CNc2cc(F)cc(F)c2)C(=O)N1	nan
	16009302	30987	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	3	1	5	2.7	Cn1c2ccccc2c2cnn(CC(=O)Nc3ccccc3F)c(=O)c21	nan
	CHEMBL1400803	30987	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	3	1	5	2.7	Cn1c2ccccc2c2cnn(CC(=O)Nc3ccccc3F)c(=O)c21	nan
	16010052	31001	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	8	1	5	4.9	COc1ccc(CCNC(=O)Cn2c(-c3cccs3)cc3cc(F)ccc32)cc1OC	nan
	CHEMBL1400938	31001	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	8	1	5	4.9	COc1ccc(CCNC(=O)Cn2c(-c3cccs3)cc3cc(F)ccc32)cc1OC	nan
	16022925	31142	3	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	5	0	6	4.6	Cc1ccc(-n2nc3c(N4CCC(C(=O)N(C)Cc5ccccc5)CC4)nnc(C)c3c2C)cc1	nan
	CHEMBL1402121	31142	3	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	5	0	6	4.6	Cc1ccc(-n2nc3c(N4CCC(C(=O)N(C)Cc5ccccc5)CC4)nnc(C)c3c2C)cc1	nan
	3238641	31190	35	None	-354	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	258	5	1	3	3.0	COc1ccc(OCc2cccc(C(=O)O)c2)cc1	nan
	CHEMBL1402510	31190	35	None	-354	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	258	5	1	3	3.0	COc1ccc(OCc2cccc(C(=O)O)c2)cc1	nan
	24792811	31201	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	464	4	0	5	4.4	Cc1cccc(N2CCN(c3ccc4cc(S(=O)(=O)N5CCCCC5)ccc4n3)CC2C)c1	nan
	CHEMBL1402620	31201	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	464	4	0	5	4.4	Cc1cccc(N2CCN(c3ccc4cc(S(=O)(=O)N5CCCCC5)ccc4n3)CC2C)c1	nan
	13020032	31237	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	345	4	2	5	2.9	COc1ccc(C[C@H]2c3cc(O)c(OC)cc3CC[N+]2(C)[O-])cc1O	nan
	CHEMBL1402907	31237	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	345	4	2	5	2.9	COc1ccc(C[C@H]2c3cc(O)c(OC)cc3CC[N+]2(C)[O-])cc1O	nan
	3456065	31241	14	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	336	3	1	4	4.8	Oc1nnc(Cc2ccc(-c3ccc(Cl)cc3)o2)c2ccccc12	nan
	CHEMBL1402979	31241	14	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	336	3	1	4	4.8	Oc1nnc(Cc2ccc(-c3ccc(Cl)cc3)o2)c2ccccc12	nan
	807671	31278	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	248	2	2	4	2.7	Cc1nc(NC(=O)c2ccccc2O)sc1C	nan
	CHEMBL1403354	31278	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	248	2	2	4	2.7	Cc1nc(NC(=O)c2ccccc2O)sc1C	nan
	24979173	31318	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	8	1	6	3.2	COc1ccccc1NC(=O)COC(=O)c1ccccc1SCC(=O)N1CCCC1	nan
	CHEMBL1403792	31318	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	8	1	6	3.2	COc1ccccc1NC(=O)COC(=O)c1ccccc1SCC(=O)N1CCCC1	nan
	1300573	31328	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	4	1	4	4.7	Cc1cccc(NC(=O)Cn2nc(-c3ccc(Cl)cc3)c3ccccc3c2=O)c1	nan
	CHEMBL1403862	31328	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	4	1	4	4.7	Cc1cccc(NC(=O)Cn2nc(-c3ccc(Cl)cc3)c3ccccc3c2=O)c1	nan
	3176404	31378	15	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	306	5	2	3	3.9	Cc1cccc(CCNCc2cc3cccc(C)c3nc2O)c1	nan
	CHEMBL1404217	31378	15	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	306	5	2	3	3.9	Cc1cccc(CCNCc2cc3cccc(C)c3nc2O)c1	nan
	2941406	31435	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	1	2	5	4.2	Cc1c(C#N)c(N)nc2c3c(sc12)NC(=O)CC3c1ccc(Cl)cc1	nan
	CHEMBL1404915	31435	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	1	2	5	4.2	Cc1c(C#N)c(N)nc2c3c(sc12)NC(=O)CC3c1ccc(Cl)cc1	nan
	663707	31520	14	None	-2	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	310	3	0	4	4.8	Fc1ccc(CSc2ncnc3c2oc2ccccc23)cc1	nan
	CHEMBL1405769	31520	14	None	-2	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	310	3	0	4	4.8	Fc1ccc(CSc2ncnc3c2oc2ccccc23)cc1	nan
	3207570	31529	2	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	6	1	5	3.1	CCc1ccc2nc(SCC(=O)NCC3CCCO3)c(C#N)cc2c1	nan
	CHEMBL1405871	31529	2	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	6	1	5	3.1	CCc1ccc2nc(SCC(=O)NCC3CCCO3)c(C#N)cc2c1	nan
	2102520	31683	5	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	423	6	1	7	5.0	COc1cc(C(=O)Nc2nc3ccc(C)cc3s2)ccc1OCc1c(C)noc1C	nan
	CHEMBL1407262	31683	5	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	423	6	1	7	5.0	COc1cc(C(=O)Nc2nc3ccc(C)cc3s2)ccc1OCc1c(C)noc1C	nan
	672442	31768	15	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	2	1	5	3.3	N#Cc1c(N)nc(N2CCCC2)c(C#N)c1-c1ccc(Cl)cc1	nan
	CHEMBL1407760	31768	15	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	2	1	5	3.3	N#Cc1c(N)nc(N2CCCC2)c(C#N)c1-c1ccc(Cl)cc1	nan
	15989447	31779	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	479	8	1	5	4.1	O=C(CCCn1c(=O)c2ccccc2n(Cc2cccc(F)c2)c1=O)NCc1ccccc1Cl	nan
	CHEMBL1407901	31779	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	479	8	1	5	4.1	O=C(CCCn1c(=O)c2ccccc2n(Cc2cccc(F)c2)c1=O)NCc1ccccc1Cl	nan
	5524322	31815	16	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	307	4	1	5	4.5	CSc1nsc(/C=C/Nc2cccc(Cl)c2)c1C#N	nan
	CHEMBL1408147	31815	16	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	307	4	1	5	4.5	CSc1nsc(/C=C/Nc2cccc(Cl)c2)c1C#N	nan
	135454349	31899	16	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	346	3	2	6	2.6	CCc1ccc(N2CC(=O)C(c3nc(O)c4ccccc4n3)=C2N)cc1	nan
	CHEMBL1408793	31899	16	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	346	3	2	6	2.6	CCc1ccc(N2CC(=O)C(c3nc(O)c4ccccc4n3)=C2N)cc1	nan
	16012616	31949	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	4	0	10	3.5	Cc1cccn2c(=O)c3cc(C#N)c(=O)n(-c4nnc(SCc5ccccc5F)s4)c3nc12	nan
	CHEMBL1409190	31949	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	4	0	10	3.5	Cc1cccn2c(=O)c3cc(C#N)c(=O)n(-c4nnc(SCc5ccccc5F)s4)c3nc12	nan
	16026074	32006	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	465	4	1	4	4.1	CC1=C(c2ccc(C)c(C)c2)S(=O)(=O)N=C1N1CCC(C(=O)NCc2ccccc2C)CC1	nan
	CHEMBL1409660	32006	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	465	4	1	4	4.1	CC1=C(c2ccc(C)c(C)c2)S(=O)(=O)N=C1N1CCC(C(=O)NCc2ccccc2C)CC1	nan
	5294544	32015	15	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	261	1	1	4	2.4	CCn1c(=S)[nH]c2nc3c(cc2c1=O)CCCC3	nan
	CHEMBL1409738	32015	15	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	261	1	1	4	2.4	CCn1c(=S)[nH]c2nc3c(cc2c1=O)CCCC3	nan
	3208202	32057	7	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	5	3	7	3.3	CCc1cc2c(C)ccc(C)c2nc1SCC(=O)Nc1cnc(O)nc1O	nan
	CHEMBL1410014	32057	7	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	5	3	7	3.3	CCc1cc2c(C)ccc(C)c2nc1SCC(=O)Nc1cnc(O)nc1O	nan
	2136000	32066	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	7	1	7	4.0	CCOc1ccc(NC(=O)Cn2cc(C(=O)c3ccccc3)c(=O)c3cc4c(cc32)OCCO4)cc1	nan
	CHEMBL1410088	32066	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	7	1	7	4.0	CCOc1ccc(NC(=O)Cn2cc(C(=O)c3ccccc3)c(=O)c3cc4c(cc32)OCCO4)cc1	nan
	2056596	32180	7	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	4	2	5	2.6	CCn1ncc(Br)c1C(=O)Nc1sc2c(c1C(N)=O)CCC2	nan
	CHEMBL1411085	32180	7	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	4	2	5	2.6	CCn1ncc(Br)c1C(=O)Nc1sc2c(c1C(N)=O)CCC2	nan
	15988949	32194	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	550	11	2	7	4.5	Cc1ccc(NC(=O)Cn2c(=O)n(CCCCCC(=O)NCc3ccc(F)cc3)c(=O)c3sccc32)cc1C	nan
	CHEMBL1411183	32194	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	550	11	2	7	4.5	Cc1ccc(NC(=O)Cn2c(=O)n(CCCCCC(=O)NCc3ccc(F)cc3)c(=O)c3sccc32)cc1C	nan
	4390376	32223	3	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	5	1	6	3.7	COc1ccc(-c2csc(NC(=O)c3ccc(N4C(=O)CCC4=O)cc3)n2)cc1	nan
	CHEMBL1411409	32223	3	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	5	1	6	3.7	COc1ccc(-c2csc(NC(=O)c3ccc(N4C(=O)CCC4=O)cc3)n2)cc1	nan
	627327	32283	30	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	301	1	0	3	3.6	O=c1oc(-c2ccc(Br)cc2)nc2ccccc12	nan
	CHEMBL1411919	32283	30	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	301	1	0	3	3.6	O=c1oc(-c2ccc(Br)cc2)nc2ccccc12	nan
	16017002	32321	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	6	1	6	1.8	CCOc1ccc(CNC(=O)C(C)n2ncn3cccc3c2=O)cc1	nan
	CHEMBL1412238	32321	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	6	1	6	1.8	CCOc1ccc(CNC(=O)C(C)n2ncn3cccc3c2=O)cc1	nan
	16026072	32370	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	495	6	1	5	4.2	CCOc1ccccc1CNC(=O)C1CCN(C2=NS(=O)(=O)C(c3ccc(C)c(C)c3)=C2C)CC1	nan
	CHEMBL1412601	32370	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	495	6	1	5	4.2	CCOc1ccccc1CNC(=O)C1CCN(C2=NS(=O)(=O)C(c3ccc(C)c(C)c3)=C2C)CC1	nan
	646655	32381	3	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	5	1	5	2.8	Cc1ccc2nc(SCC(=O)NCC3CCCO3)c(C#N)cc2c1	nan
	CHEMBL1412670	32381	3	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	5	1	5	2.8	Cc1ccc2nc(SCC(=O)NCC3CCCO3)c(C#N)cc2c1	nan
	1246434	32385	13	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	3	1	5	4.7	O=C(Nc1nnc(C2CCCCC2)s1)c1ccc(Br)s1	nan
	CHEMBL1412704	32385	13	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	3	1	5	4.7	O=C(Nc1nnc(C2CCCCC2)s1)c1ccc(Br)s1	nan
	1952877	32405	14	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	400	5	2	5	2.0	Cc1cc(C)c2oc(C(=O)NCCc3ccc(S(N)(=O)=O)cc3)cc(=O)c2c1	nan
	CHEMBL1412873	32405	14	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	400	5	2	5	2.0	Cc1cc(C)c2oc(C(=O)NCCc3ccc(S(N)(=O)=O)cc3)cc(=O)c2c1	nan
	16017227	32429	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	3	0	6	2.2	Cc1nn(CC(=O)N2CCN(c3cccc(C(F)(F)F)c3)CC2)c(=O)c2cccn12	nan
	CHEMBL1413003	32429	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	3	0	6	2.2	Cc1nn(CC(=O)N2CCN(c3cccc(C(F)(F)F)c3)CC2)c(=O)c2cccn12	nan
	15996885	32436	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	510	8	1	8	3.7	COc1cccc(N2CCN(C(=O)CCCCCn3c(=S)[nH]c4cc5c(cc4c3=O)OCO5)CC2)c1	nan
	CHEMBL1413061	32436	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	510	8	1	8	3.7	COc1cccc(N2CCN(C(=O)CCCCCn3c(=S)[nH]c4cc5c(cc4c3=O)OCO5)CC2)c1	nan
	2314879	32484	2	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	307	3	1	6	3.3	CCCCn1c2nc3ccccc3nc2c2c(=N)oc(C)nc21	nan
	CHEMBL1413521	32484	2	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	307	3	1	6	3.3	CCCCn1c2nc3ccccc3nc2c2c(=N)oc(C)nc21	nan
	694926	32499	22	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	346	3	1	5	3.3	Cc1cccc(C(=O)Nc2nc3ccc(S(C)(=O)=O)cc3s2)c1	nan
	CHEMBL1413648	32499	22	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	346	3	1	5	3.3	Cc1cccc(C(=O)Nc2nc3ccc(S(C)(=O)=O)cc3s2)c1	nan
	16025383	32609	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	534	8	1	6	4.4	O=C(CSc1ncc2c(n1)-c1ccccc1N(Cc1ccc(F)cc1)S2(=O)=O)NCCc1ccccc1	nan
	CHEMBL1414539	32609	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	534	8	1	6	4.4	O=C(CSc1ncc2c(n1)-c1ccccc1N(Cc1ccc(F)cc1)S2(=O)=O)NCCc1ccccc1	nan
	16010143	32674	3	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	5	1	3	5.6	Cc1ccc(Cn2c(C(=O)NCc3ccccc3Cl)cc3sccc32)cc1	nan
	CHEMBL1415124	32674	3	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	5	1	3	5.6	Cc1ccc(Cn2c(C(=O)NCc3ccccc3Cl)cc3sccc32)cc1	nan
	663372	32676	14	None	-14	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	2	0	4	4.2	Cc1ccc(C2CC(=O)c3cnc(N4CC(C)CC(C)C4)nc3C2)cc1	nan
	CHEMBL1415139	32676	14	None	-14	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	2	0	4	4.2	Cc1ccc(C2CC(=O)c3cnc(N4CC(C)CC(C)C4)nc3C2)cc1	nan
	16029519	32687	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	494	5	0	6	2.9	CN(C)S(=O)(=O)c1ccc2c(c1)N(CC(=O)N1CCN(c3cccc(Cl)c3)CC1)CCS2	nan
	CHEMBL1415234	32687	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	494	5	0	6	2.9	CN(C)S(=O)(=O)c1ccc2c(c1)N(CC(=O)N1CCN(c3cccc(Cl)c3)CC1)CCS2	nan
	1088534	32721	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	336	6	1	4	3.9	CCOc1ccc(NC(=O)Cn2cc(C(C)=O)c3ccccc32)cc1	nan
	CHEMBL1415529	32721	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	336	6	1	4	3.9	CCOc1ccc(NC(=O)Cn2cc(C(C)=O)c3ccccc32)cc1	nan
	2701522	32744	9	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	309	6	1	6	2.8	CCSc1nnc(NC(=O)Cc2ccccc2OC)s1	nan
	CHEMBL1415759	32744	9	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	309	6	1	6	2.8	CCSc1nnc(NC(=O)Cc2ccccc2OC)s1	nan
	20880977	32848	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	508	9	1	8	2.5	O=C(CCc1nnc2n(Cc3ccc(Cl)cc3)c(=O)c3ccccc3n12)NCCCN1CCOCC1	nan
	CHEMBL1416665	32848	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	508	9	1	8	2.5	O=C(CCc1nnc2n(Cc3ccc(Cl)cc3)c(=O)c3ccccc3n12)NCCCN1CCOCC1	nan
	16025415	32865	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	530	6	1	6	5.5	Cc1ccc(C)c(NC(=O)CSc2ncc3c(n2)-c2ccccc2N(Cc2ccccc2C)S3(=O)=O)c1	nan
	CHEMBL1416823	32865	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	530	6	1	6	5.5	Cc1ccc(C)c(NC(=O)CSc2ncc3c(n2)-c2ccccc2N(Cc2ccccc2C)S3(=O)=O)c1	nan
	24792644	33001	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	2	0	4	3.8	CN(C)c1ccc(-c2ccc3c(=O)c4ccccc4n(C)c3c2)cn1	nan
	CHEMBL1417964	33001	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	2	0	4	3.8	CN(C)c1ccc(-c2ccc3c(=O)c4ccccc4n(C)c3c2)cn1	nan
	16030529	33016	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	7	0	4	5.8	CCN(C(=O)CSc1nc2ccccc2nc1Cc1ccc(F)cc1)c1cccc(C)c1	nan
	CHEMBL1418101	33016	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	7	0	4	5.8	CCN(C(=O)CSc1nc2ccccc2nc1Cc1ccc(F)cc1)c1cccc(C)c1	nan
	1936615	33079	11	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	5	1	7	4.5	CC1(C)Cc2nc3sc4c(SCC(=O)NCc5ccccc5)ncnc4c3cc2CO1	nan
	CHEMBL1418632	33079	11	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	5	1	7	4.5	CC1(C)Cc2nc3sc4c(SCC(=O)NCc5ccccc5)ncnc4c3cc2CO1	nan
	3574260	33152	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	5	2	6	3.1	O=C(CCn1c(=S)[nH]c2cc3c(cc2c1=O)OCO3)NCc1ccccc1Cl	nan
	CHEMBL1419267	33152	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	5	2	6	3.1	O=C(CCn1c(=S)[nH]c2cc3c(cc2c1=O)OCO3)NCc1ccccc1Cl	nan
	5069803	33617	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	4	0	4	2.2	CC(C)C(=O)N1CCN(CCN2C(=O)c3cccc4cccc(c34)C2=O)CC1	nan
	CHEMBL1423181	33617	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	4	0	4	2.2	CC(C)C(=O)N1CCN(CCN2C(=O)c3cccc4cccc(c34)C2=O)CC1	nan
	4298772	33677	14	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	278	3	1	4	2.8	Cc1ccc(NC(=O)c2ccc(-n3cccn3)nc2)cc1	nan
	CHEMBL1423637	33677	14	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	278	3	1	4	2.8	Cc1ccc(NC(=O)c2ccc(-n3cccn3)nc2)cc1	nan
	135521903	33740	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	7	2	7	4.7	Cc1ccc(-n2c(SCC(=O)NCCC3=CCCCC3)nc3nnc(C)c-3c2N)cc1Cl	nan
	CHEMBL1424164	33740	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	7	2	7	4.7	Cc1ccc(-n2c(SCC(=O)NCCC3=CCCCC3)nc3nnc(C)c-3c2N)cc1Cl	nan
	5009230	34018	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	320	3	1	3	4.6	O=c1c2ccc(Cl)cc2[nH]c(=S)n1CCC1=CCCCC1	nan
	CHEMBL1426475	34018	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	320	3	1	3	4.6	O=c1c2ccc(Cl)cc2[nH]c(=S)n1CCC1=CCCCC1	nan
	1004501	34034	13	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	471	8	1	6	5.8	COc1ccc(-c2cc(-c3cccs3)c(C#N)c(SCC(=O)NCc3ccccc3)n2)cc1	nan
	CHEMBL1426581	34034	13	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	471	8	1	6	5.8	COc1ccc(-c2cc(-c3cccs3)c(C#N)c(SCC(=O)NCc3ccccc3)n2)cc1	nan
	1398121	34057	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	309	2	1	4	5.1	Cc1nc(Nc2ccccc2)c2oc3ccc(Cl)cc3c2n1	nan
	CHEMBL1426816	34057	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	309	2	1	4	5.1	Cc1nc(Nc2ccccc2)c2oc3ccc(Cl)cc3c2n1	nan
	2916457	34116	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	277	2	0	4	2.1	O=C1c2nc3ccccn3c2C(=O)N1Cc1ccccc1	nan
	CHEMBL1427322	34116	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	277	2	0	4	2.1	O=C1c2nc3ccccn3c2C(=O)N1Cc1ccccc1	nan
	2785858	34356	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	241	0	0	5	0.8	Cn1c(=O)c2cc3ccccc3nc2n(C)c1=O	nan
	CHEMBL1429441	34356	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	241	0	0	5	0.8	Cn1c(=O)c2cc3ccccc3nc2n(C)c1=O	nan
	1474449	34604	14	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	310	2	1	5	3.8	Nc1c(-c2cccs2)cnc2c(-c3ccc(F)cc3)cnn12	nan
	CHEMBL1431364	34604	14	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	310	2	1	5	3.8	Nc1c(-c2cccs2)cnc2c(-c3ccc(F)cc3)cnn12	nan
	22548378	34609	3	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	4	1	6	2.0	CC(=O)c1ccc(N2CCN(S(=O)(=O)c3cc4c(cc3C)NC(=O)CO4)CC2)cc1	nan
	CHEMBL1431452	34609	3	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	4	1	6	2.0	CC(=O)c1ccc(N2CCN(S(=O)(=O)c3cc4c(cc3C)NC(=O)CO4)CC2)cc1	nan
	3239990	34665	7	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	3	0	7	3.1	CCOC(=O)N1CCN(C(=O)c2nn(-c3ccc(C)cc3)c(=O)c3c2c2ccccc2n3C)CC1	nan
	CHEMBL1431956	34665	7	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	3	0	7	3.1	CCOC(=O)N1CCN(C(=O)c2nn(-c3ccc(C)cc3)c(=O)c3c2c2ccccc2n3C)CC1	nan
	1480466	34684	23	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	4	1	5	4.6	CC(C)Nc1nc(-c2cccnc2)nc(-c2ccc(Cl)cc2)c1C#N	nan
	CHEMBL1432166	34684	23	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	4	1	5	4.6	CC(C)Nc1nc(-c2cccnc2)nc(-c2ccc(Cl)cc2)c1C#N	nan
	24792375	34705	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	6	1	6	2.5	COc1ccc2nc(SCC(=O)NCC3CCCO3)c(C#N)cc2c1	nan
	CHEMBL1432321	34705	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	6	1	6	2.5	COc1ccc2nc(SCC(=O)NCC3CCCO3)c(C#N)cc2c1	nan
	1049756	34835	14	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	5	2	5	4.3	COc1ccccc1NC(=O)c1c(NC(=O)c2ccco2)sc2c1CCC2	nan
	CHEMBL1433354	34835	14	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	5	2	5	4.3	COc1ccccc1NC(=O)c1c(NC(=O)c2ccco2)sc2c1CCC2	nan
	2227785	34847	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	7	1	7	5.3	COc1ccc(-c2nc3ccccc3s2)cc1NC(=O)c1cc(OC)c(OC)c(OC)c1	nan
	CHEMBL1433437	34847	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	7	1	7	5.3	COc1ccc(-c2nc3ccccc3s2)cc1NC(=O)c1cc(OC)c(OC)c(OC)c1	nan
	16027247	34859	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	5	1	5	4.9	COc1ccc2ncc3c(-c4ccc(C)c(C)c4)nn(CC(=O)NC4CCCC4)c3c2c1	nan
	CHEMBL1433603	34859	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	5	1	5	4.9	COc1ccc2ncc3c(-c4ccc(C)c(C)c4)nn(CC(=O)NC4CCCC4)c3c2c1	nan
	16024617	34880	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	489	7	1	6	4.8	CCc1ccc(C(=O)c2cn(CC(=O)Nc3ccc(OC)c(Cl)c3)c3nc(C)ccc3c2=O)cc1	nan
	CHEMBL1433920	34880	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	489	7	1	6	4.8	CCc1ccc(C(=O)c2cn(CC(=O)Nc3ccc(OC)c(Cl)c3)c3nc(C)ccc3c2=O)cc1	nan
	16019055	34899	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	436	6	1	5	4.0	Cc1ccccc1CCNC(=O)c1ccc(Cn2c(=O)c3cccn3c3cccnc32)cc1	nan
	CHEMBL1434234	34899	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	436	6	1	5	4.0	Cc1ccccc1CCNC(=O)c1ccc(Cn2c(=O)c3cccn3c3cccnc32)cc1	nan
	2135389	34902	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	460	7	1	6	4.0	COc1cccc(NC(=O)Cn2cc(C(=O)c3ccc(F)cc3)c(=O)c3cc(OC)ccc32)c1	nan
	CHEMBL1434264	34902	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	460	7	1	6	4.0	COc1cccc(NC(=O)Cn2cc(C(=O)c3ccc(F)cc3)c(=O)c3cc(OC)ccc32)c1	nan
	16026966	34908	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	6	0	9	3.1	O=C(COc1ccc(F)cc1)OCc1cc(=O)n2nc(-c3cccs3)sc2n1	nan
	CHEMBL1434365	34908	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	6	0	9	3.1	O=C(COc1ccc(F)cc1)OCc1cc(=O)n2nc(-c3cccs3)sc2n1	nan
	16021030	34919	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	6	1	3	5.9	CC(CNC(=O)Cn1c(-c2cccs2)cc2cc(Cl)ccc21)c1ccccc1	nan
	CHEMBL1434633	34919	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	6	1	3	5.9	CC(CNC(=O)Cn1c(-c2cccs2)cc2cc(Cl)ccc21)c1ccccc1	nan
	2134800	34953	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	9	1	7	4.1	COCCCn1c(SCC(=O)NCc2ccccc2)nc2c(sc3ccccc32)c1=O	nan
	CHEMBL1435016	34953	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	9	1	7	4.1	COCCCn1c(SCC(=O)NCc2ccccc2)nc2c(sc3ccccc32)c1=O	nan
	16022354	34980	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	7	1	6	4.9	Cc1ccc(Cn2c(SCC(=O)NCc3ccc(Cl)cc3)nc3ccsc3c2=O)cc1	nan
	CHEMBL1435272	34980	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	7	1	6	4.9	Cc1ccc(Cn2c(SCC(=O)NCc3ccc(Cl)cc3)nc3ccsc3c2=O)cc1	nan
	16022956	35020	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	488	6	1	6	4.7	Cc1nnc(N2CCC(C(=O)NCCc3ccccc3)CC2)c2nn(-c3ccc(Cl)cc3)c(C)c12	nan
	CHEMBL1435842	35020	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	488	6	1	6	4.7	Cc1nnc(N2CCC(C(=O)NCCc3ccccc3)CC2)c2nn(-c3ccc(Cl)cc3)c(C)c12	nan
	16015098	35021	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	5	1	4	4.5	Cc1nc(SCC(=O)Nc2ccccc2C)cc(-c2ccccc2)n1	nan
	CHEMBL1435853	35021	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	5	1	4	4.5	Cc1nc(SCC(=O)Nc2ccccc2C)cc(-c2ccccc2)n1	nan
	16024515	35025	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	475	6	1	6	4.5	COc1ccc(Cl)cc1NC(=O)Cn1cc(C(=O)c2ccc(C)cc2)c(=O)c2ccc(C)nc21	nan
	CHEMBL1435881	35025	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	475	6	1	6	4.5	COc1ccc(Cl)cc1NC(=O)Cn1cc(C(=O)c2ccc(C)cc2)c(=O)c2ccc(C)nc21	nan
	16025955	35034	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	4	1	8	1.6	O=C(NCc1ccccc1Cl)c1cnc2sc(N3CCOCC3)nn2c1=O	nan
	CHEMBL1436007	35034	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	4	1	8	1.6	O=C(NCc1ccccc1Cl)c1cnc2sc(N3CCOCC3)nn2c1=O	nan
	15988055	35056	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	366	2	1	8	3.4	Cc1cccc(C)c1Nc1nn2c(=O)c3cc4c(cc3nc2s1)OCO4	nan
	CHEMBL1436214	35056	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	366	2	1	8	3.4	Cc1cccc(C)c1Nc1nn2c(=O)c3cc4c(cc3nc2s1)OCO4	nan
	1166237	35067	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	491	8	1	7	5.4	CCOc1ccc(NC(=O)CCSc2nc(-c3ccc4c(c3)OCO4)cc(C(F)(F)F)n2)cc1	nan
	CHEMBL1436413	35067	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	491	8	1	7	5.4	CCOc1ccc(NC(=O)CCSc2nc(-c3ccc4c(c3)OCO4)cc(C(F)(F)F)n2)cc1	nan
	4076476	35085	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	5	1	4	5.1	COc1cccc(C(=O)Nc2c(C(=O)c3ccc(F)cc3)oc3ccccc23)c1	nan
	CHEMBL1436707	35085	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	5	1	4	5.1	COc1cccc(C(=O)Nc2c(C(=O)c3ccc(F)cc3)oc3ccccc23)c1	nan
	16012965	35092	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	6	1	3	5.3	CCCCN(Cc1cc2cc(C)ccc2nc1O)C(=O)c1cccc(Cl)c1	nan
	CHEMBL1436801	35092	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	6	1	3	5.3	CCCCN(Cc1cc2cc(C)ccc2nc1O)C(=O)c1cccc(Cl)c1	nan
	16031323	35097	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	494	8	1	8	3.7	COc1cc(-c2cc3n(C)c(C)c(CCC(=O)Nc4ccc(F)cc4)c(=O)n3n2)cc(OC)c1OC	nan
	CHEMBL1436894	35097	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	494	8	1	8	3.7	COc1cc(-c2cc3n(C)c(C)c(CCC(=O)Nc4ccc(F)cc4)c(=O)n3n2)cc(OC)c1OC	nan
	3533132	35174	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	5	1	5	3.3	COc1ccc(S(=O)(=O)N2CCCCC2)cc1NC(=O)c1cncc(Br)c1	nan
	CHEMBL1437784	35174	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	5	1	5	3.3	COc1ccc(S(=O)(=O)N2CCCCC2)cc1NC(=O)c1cncc(Br)c1	nan
	4650106	35216	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	480	5	2	5	4.2	O=C(NCc1cccnc1)c1ccc(Cn2c(=S)[nH]c3ccc(Br)cc3c2=O)cc1	nan
	CHEMBL1438098	35216	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	480	5	2	5	4.2	O=C(NCc1cccnc1)c1ccc(Cn2c(=S)[nH]c3ccc(Br)cc3c2=O)cc1	nan
	959085	35302	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	288	3	1	4	3.5	CC(=O)c1sc(NC(=O)c2ccc(C)c(C)c2)nc1C	nan
	CHEMBL1438925	35302	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	288	3	1	4	3.5	CC(=O)c1sc(NC(=O)c2ccc(C)c(C)c2)nc1C	nan
	16026319	35323	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	5	1	5	4.5	CCc1ccc(-n2nc(C)c3c(C)cc(=O)n(CC(=O)Nc4ccc(C)c(F)c4)c32)cc1	nan
	CHEMBL1439096	35323	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	5	1	5	4.5	CCc1ccc(-n2nc(C)c3c(C)cc(=O)n(CC(=O)Nc4ccc(C)c(F)c4)c32)cc1	nan
	16015553	35325	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	423	6	2	6	5.2	Cc1ccc(NC(=O)CSc2nc3ccc(NC(=O)c4ccco4)cc3s2)cc1	nan
	CHEMBL1439122	35325	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	423	6	2	6	5.2	Cc1ccc(NC(=O)CSc2nc3ccc(NC(=O)c4ccco4)cc3s2)cc1	nan
	15988982	35446	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	524	8	2	7	3.8	Cc1cccc(C)c1NC(=O)Cn1c(=O)n(CCC(=O)NCc2ccccc2Cl)c(=O)c2sccc21	nan
	CHEMBL1440158	35446	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	524	8	2	7	3.8	Cc1cccc(C)c1NC(=O)Cn1c(=O)n(CCC(=O)NCc2ccccc2Cl)c(=O)c2sccc21	nan
	2137007	35685	9	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	6	1	8	2.8	COCCNc1nc2c(S(=O)(=O)c3cc(C)ccc3C)nnn2c2ccccc12	nan
	CHEMBL1442335	35685	9	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	6	1	8	2.8	COCCNc1nc2c(S(=O)(=O)c3cc(C)ccc3C)nnn2c2ccccc12	nan
	3156591	35703	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	6	1	7	3.0	CCCNS(=O)(=O)c1cc(-c2nnc3c4ccccc4c(C)nn23)ccc1OC	nan
	CHEMBL1442508	35703	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	6	1	7	3.0	CCCNS(=O)(=O)c1cc(-c2nnc3c4ccccc4c(C)nn23)ccc1OC	nan
	16009539	35743	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	7	1	7	3.8	Cc1csc2nc(COc3ccc(NC(=O)COc4ccccc4F)cc3)cc(=O)n12	nan
	CHEMBL1442799	35743	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	7	1	7	3.8	Cc1csc2nc(COc3ccc(NC(=O)COc4ccccc4F)cc3)cc(=O)n12	nan
	1119348	35761	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	3	0	6	4.2	COc1cccc2cc(-c3nnc(-c4ccc(Cl)cc4)o3)c(=O)oc12	nan
	CHEMBL1443005	35761	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	3	0	6	4.2	COc1cccc2cc(-c3nnc(-c4ccc(Cl)cc4)o3)c(=O)oc12	nan
	3456574	35941	8	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	5	2	5	1.8	COCCn1c(=S)[nH]c2cc(C(=O)NC(C)C)ccc2c1=O	nan
	CHEMBL1444789	35941	8	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	5	2	5	1.8	COCCn1c(=S)[nH]c2cc(C(=O)NC(C)C)ccc2c1=O	nan
	15987577	35957	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	4	1	5	4.3	Cc1cc(Cl)ccc1OCC(=O)Nc1c(Cl)ccc2nsnc12	nan
	CHEMBL1444928	35957	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	4	1	5	4.3	Cc1cc(Cl)ccc1OCC(=O)Nc1c(Cl)ccc2nsnc12	nan
	1529015	35959	15	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	5	1	6	5.3	CCOC(=O)c1c(-c2ccc(C)s2)csc1NC(=O)c1cccs1	nan
	CHEMBL1444931	35959	15	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	5	1	6	5.3	CCOC(=O)c1c(-c2ccc(C)s2)csc1NC(=O)c1cccs1	nan
	3238506	35992	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	5	1	7	3.0	CCOC(=O)N1CCN(S(=O)(=O)c2ccc(C(=O)Nc3nc4ccccc4s3)cc2)CC1	nan
	CHEMBL1445199	35992	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	5	1	7	3.0	CCOC(=O)N1CCN(S(=O)(=O)c2ccc(C(=O)Nc3nc4ccccc4s3)cc2)CC1	nan
	629629	36009	11	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	4	1	3	5.4	CC(=O)Nc1ccc(-c2cc(-c3ccccc3)nc(-c3ccccc3)n2)cc1	nan
	CHEMBL1445350	36009	11	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	4	1	3	5.4	CC(=O)Nc1ccc(-c2cc(-c3ccccc3)nc(-c3ccccc3)n2)cc1	nan
	16008367	36036	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	6	1	6	4.6	COc1cc(OC)c(NC(=O)CSc2cc(=O)n(C)c3ccc(Cl)cc23)cc1Cl	nan
	CHEMBL1445604	36036	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	6	1	6	4.6	COc1cc(OC)c(NC(=O)CSc2cc(=O)n(C)c3ccc(Cl)cc23)cc1Cl	nan
	16031877	36063	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	5	0	7	4.0	CCOC(=O)C1CCCN(Cc2cn3c(-c4ccc(Br)cc4)nnc3s2)C1	nan
	CHEMBL1445888	36063	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	5	0	7	4.0	CCOC(=O)C1CCCN(Cc2cn3c(-c4ccc(Br)cc4)nnc3s2)C1	nan
	3116123	36083	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	5	2	7	2.1	COc1ccccc1NC(=O)CSc1nc(N)c(C#N)cc1C#N	nan
	CHEMBL1446094	36083	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	5	2	7	2.1	COc1ccccc1NC(=O)CSc1nc(N)c(C#N)cc1C#N	nan
	3462774	36119	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	8	2	5	3.6	CCOCCCn1c(=S)[nH]c2cc(C(=O)NCc3ccc(F)cc3)ccc2c1=O	nan
	CHEMBL1446438	36119	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	8	2	5	3.6	CCOCCCn1c(=S)[nH]c2cc(C(=O)NCc3ccc(F)cc3)ccc2c1=O	nan
	1478332	36348	21	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	297	2	0	5	3.1	CCOC(=O)c1cc2c(=O)c3cc(C)ccc3oc2nc1C	nan
	CHEMBL1448380	36348	21	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	297	2	0	5	3.1	CCOC(=O)c1cc2c(=O)c3cc(C)ccc3oc2nc1C	nan
	15990626	36375	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	4	0	4	6.1	CCOc1ccc2ncc3c(-c4ccc(C)cc4)nn(-c4cccc(F)c4)c3c2c1	nan
	CHEMBL1448570	36375	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	4	0	4	6.1	CCOc1ccc2ncc3c(-c4ccc(C)cc4)nn(-c4cccc(F)c4)c3c2c1	nan
	16007612	36411	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	495	7	1	5	3.8	Cc1ccc(CCNC(=O)c2cn(C)c3ccc(S(=O)(=O)N(C)C4CCCCC4)cc3c2=O)cc1	nan
	CHEMBL1448823	36411	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	495	7	1	5	3.8	Cc1ccc(CCNC(=O)c2cn(C)c3ccc(S(=O)(=O)N(C)C4CCCCC4)cc3c2=O)cc1	nan
	2201274	36453	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	331	5	1	6	3.5	COc1cccc(-c2nnc(NC(=O)Cc3cccs3)s2)c1	nan
	CHEMBL1449110	36453	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	331	5	1	6	3.5	COc1cccc(-c2nnc(NC(=O)Cc3cccs3)s2)c1	nan
	16017301	36626	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	7	1	7	3.2	CC(C)CN(c1ccccc1)S(=O)(=O)c1nnc(NC(=O)c2ccco2)s1	nan
	CHEMBL1450497	36626	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	7	1	7	3.2	CC(C)CN(c1ccccc1)S(=O)(=O)c1nnc(NC(=O)c2ccco2)s1	nan
	3646626	36643	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	485	9	1	7	5.3	CC(C)OCCCn1c(SCC(=O)Nc2ccc(F)cc2)nc2c(sc3ccccc32)c1=O	nan
	CHEMBL1450646	36643	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	485	9	1	7	5.3	CC(C)OCCCn1c(SCC(=O)Nc2ccc(F)cc2)nc2c(sc3ccccc32)c1=O	nan
	1389502	36693	9	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	361	2	1	3	4.0	O=C(Nc1cc(Cl)cc(Cl)c1)c1coc(=O)c(Br)c1	nan
	CHEMBL1451156	36693	9	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	361	2	1	3	4.0	O=C(Nc1cc(Cl)cc(Cl)c1)c1coc(=O)c(Br)c1	nan
	653554	36751	10	None	-1	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	6	1	7	4.1	Cc1sc2nc(SCC(=O)NCc3ccco3)n(-c3ccccc3)c(=O)c2c1C	nan
	CHEMBL1451583	36751	10	None	-1	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	6	1	7	4.1	Cc1sc2nc(SCC(=O)NCc3ccco3)n(-c3ccccc3)c(=O)c2c1C	nan
	135476823	36755	1	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	4	1	7	2.7	Cc1cccc(-n2c(SCC(=O)N3CCCC3)nc3nnc(C)c-3c2N)c1	nan
	CHEMBL1451599	36755	1	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	4	1	7	2.7	Cc1cccc(-n2c(SCC(=O)N3CCCC3)nc3nnc(C)c-3c2N)c1	nan
	2029273	36842	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	5	0	6	5.2	COc1cccc(-c2ccc(-c3noc(-c4ccccc4Br)n3)c(OC)n2)c1	nan
	CHEMBL1452203	36842	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	5	0	6	5.2	COc1cccc(-c2ccc(-c3noc(-c4ccccc4Br)n3)c(OC)n2)c1	nan
	5058847	36853	9	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	6	1	6	3.0	COc1cc(NC(=O)Cn2c(C)cc3ccccc3c2=O)cc(OC)c1OC	nan
	CHEMBL1452293	36853	9	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	6	1	6	3.0	COc1cc(NC(=O)Cn2c(C)cc3ccccc3c2=O)cc(OC)c1OC	nan
	16027444	36883	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	460	6	1	8	3.9	Cc1cccc(C(=O)Nc2ccc(C(=O)OCc3cc(=O)n4nc(C5CC5)sc4n3)cc2)c1	nan
	CHEMBL1452550	36883	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	460	6	1	8	3.9	Cc1cccc(C(=O)Nc2ccc(C(=O)OCc3cc(=O)n4nc(C5CC5)sc4n3)cc2)c1	nan
	4256434	37046	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	5	1	6	5.1	Cc1ccc(-c2nc(NC(=O)CSc3cc(C)c4ccccc4n3)ns2)cc1	nan
	CHEMBL1453902	37046	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	5	1	6	5.1	Cc1ccc(-c2nc(NC(=O)CSc3cc(C)c4ccccc4n3)ns2)cc1	nan
	16008459	37052	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	6	0	4	4.8	CCOc1ccc2c(c1)c(=O)c(C(=O)c1ccccc1)cn2Cc1ccccc1F	nan
	CHEMBL1453936	37052	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	6	0	4	4.8	CCOc1ccc2c(c1)c(=O)c(C(=O)c1ccccc1)cn2Cc1ccccc1F	nan
	991456	37077	2	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	6	2	4	4.1	COc1ccc(C(=O)Nc2ccc(Cl)cc2C(=O)NCc2ccco2)cc1	nan
	CHEMBL1454096	37077	2	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	6	2	4	4.1	COc1ccc(C(=O)Nc2ccc(Cl)cc2C(=O)NCc2ccco2)cc1	nan
	808336	37145	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	258	1	0	6	1.8	Cc1ccc(-c2nn3c(=O)c(C)nnc3s2)cc1	nan
	CHEMBL1454681	37145	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	258	1	0	6	1.8	Cc1ccc(-c2nn3c(=O)c(C)nnc3s2)cc1	nan
	16017701	37148	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	7	1	7	3.9	CCC(Sc1nc2nccnc2c(=O)n1Cc1ccc(C)cc1)C(=O)NC1CCCCC1	nan
	CHEMBL1454690	37148	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	7	1	7	3.9	CCC(Sc1nc2nccnc2c(=O)n1Cc1ccc(C)cc1)C(=O)NC1CCCCC1	nan
	15988663	37168	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	6	1	5	3.9	COc1ccc(OC)c(-c2cc(C(=O)NCc3ccc(Cl)cc3)no2)c1	nan
	CHEMBL1454826	37168	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	6	1	5	3.9	COc1ccc(OC)c(-c2cc(C(=O)NCc3ccc(Cl)cc3)no2)c1	nan
	599450	37264	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	2	1	3	3.6	O=C(Nc1ccc2c(c1)C(=O)OC2)c1ccc(C(F)(F)F)cc1	nan
	CHEMBL1455771	37264	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	2	1	3	3.6	O=C(Nc1ccc2c(c1)C(=O)OC2)c1ccc(C(F)(F)F)cc1	nan
	3981165	37296	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	6	1	5	2.5	CCOc1ncccc1C(=O)Nc1ccc(S(=O)(=O)N2CCCC2)cc1	nan
	CHEMBL1456046	37296	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	6	1	5	2.5	CCOc1ncccc1C(=O)Nc1ccc(S(=O)(=O)N2CCCC2)cc1	nan
	15989547	37311	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	461	8	1	5	3.6	O=C(CCn1c(=O)c2ccccc2n(Cc2cccc(Cl)c2)c1=O)NCCc1ccccc1	nan
	CHEMBL1456174	37311	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	461	8	1	5	3.6	O=C(CCn1c(=O)c2ccccc2n(Cc2cccc(Cl)c2)c1=O)NCCc1ccccc1	nan
	16027694	37346	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	7	1	8	3.4	Cc1ccccc1OCC(=O)Nc1ccccc1C(=O)OCc1cc(=O)n2ccsc2n1	nan
	CHEMBL1456495	37346	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	7	1	8	3.4	Cc1ccccc1OCC(=O)Nc1ccccc1C(=O)OCc1cc(=O)n2ccsc2n1	nan
	3242698	37376	12	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	5	2	7	4.2	Cc1ccccc1NC(=O)CSc1nc(N)c(C#N)c(-c2cccs2)c1C#N	nan
	CHEMBL1456820	37376	12	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	5	2	7	4.2	Cc1ccccc1NC(=O)CSc1nc(N)c(C#N)c(-c2cccs2)c1C#N	nan
	16024703	37429	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	5	1	5	4.0	Cc1ccc2c(=O)c(C(=O)c3cccc(Cl)c3)cn(CC(=O)NC3CCCCC3)c2n1	nan
	CHEMBL1457278	37429	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	5	1	5	4.0	Cc1ccc2c(=O)c(C(=O)c3cccc(Cl)c3)cn(CC(=O)NC3CCCCC3)c2n1	nan
	7066852	37439	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	3	2	3	5.8	Cc1ccc2nc(-c3c[nH]c4ccccc34)c(Nc3ccccc3C)n2c1	nan
	CHEMBL1457410	37439	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	3	2	3	5.8	Cc1ccc2nc(-c3c[nH]c4ccccc34)c(Nc3ccccc3C)n2c1	nan
	16030759	37455	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	4	0	6	4.4	O=C(c1ccc2c(c1)OCCO2)N(Cc1cccnc1)c1nc2ccc(F)cc2s1	nan
	CHEMBL1457518	37455	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	4	0	6	4.4	O=C(c1ccc2c(c1)OCCO2)N(Cc1cccnc1)c1nc2ccc(F)cc2s1	nan
	3347951	37461	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	4	1	6	2.5	CNC(=O)C(Sc1nc(C)nc2c1oc1ccccc12)C(C)=O	nan
	CHEMBL1457585	37461	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	4	1	6	2.5	CNC(=O)C(Sc1nc(C)nc2c1oc1ccccc12)C(C)=O	nan
	654954	37578	5	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	5	1	5	3.4	Cc1ccc2nc(SCC(=O)NCc3ccco3)c(C#N)cc2c1	nan
	CHEMBL1458514	37578	5	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	5	1	5	3.4	Cc1ccc2nc(SCC(=O)NCc3ccco3)c(C#N)cc2c1	nan
	861942	37635	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	344	5	0	6	3.7	COc1ccc(OC)c(-c2csc(N(C)C(=O)c3ccco3)n2)c1	nan
	CHEMBL1458992	37635	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	344	5	0	6	3.7	COc1ccc(OC)c(-c2csc(N(C)C(=O)c3ccco3)n2)c1	nan
	2570053	37915	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	316	5	0	7	1.8	Cc1ccnc2nc(C(=O)OCCOc3ccc(F)cc3)nn12	nan
	CHEMBL1461384	37915	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	316	5	0	7	1.8	Cc1ccnc2nc(C(=O)OCCOc3ccc(F)cc3)nn12	nan
	2109478	37941	2	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	322	4	1	5	3.9	Cc1cc(NC(=O)COc2ccc3oc4ccccc4c3c2)no1	nan
	CHEMBL1461645	37941	2	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	322	4	1	5	3.9	Cc1cc(NC(=O)COc2ccc3oc4ccccc4c3c2)no1	nan
	3243431	37949	7	None	-11	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	6	2	4	5.6	CCOc1ccc(C(=O)Nc2ccc(NC(=O)c3ccco3)c(Cl)c2)cc1Br	nan
	CHEMBL1461732	37949	7	None	-11	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	6	2	4	5.6	CCOc1ccc(C(=O)Nc2ccc(NC(=O)c3ccco3)c(Cl)c2)cc1Br	nan
	24789924	38040	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	510	8	1	8	3.7	COc1ccc(N2CCN(C(=O)CCCCCn3c(=S)[nH]c4cc5c(cc4c3=O)OCO5)CC2)cc1	nan
	CHEMBL1462423	38040	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	510	8	1	8	3.7	COc1ccc(N2CCN(C(=O)CCCCCn3c(=S)[nH]c4cc5c(cc4c3=O)OCO5)CC2)cc1	nan
	651585	38067	4	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	302	3	0	7	2.1	COC(=O)CSc1nc2cc3c(cc2cc1C#N)OCO3	nan
	CHEMBL1462713	38067	4	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	302	3	0	7	2.1	COC(=O)CSc1nc2cc3c(cc2cc1C#N)OCO3	nan
	2134888	38072	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	467	9	1	9	2.4	COc1ccc(C=O)cc1Cn1c(=O)n(CCC(=O)NCc2ccco2)c(=O)c2sccc21	nan
	CHEMBL1462748	38072	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	467	9	1	9	2.4	COc1ccc(C=O)cc1Cn1c(=O)n(CCC(=O)NCc2ccco2)c(=O)c2sccc21	nan
	658551	38367	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	304	6	1	7	2.0	CCCOC(=O)CSc1nc(N)c(C#N)c(CC)c1C#N	nan
	CHEMBL1465062	38367	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	304	6	1	7	2.0	CCCOC(=O)CSc1nc(N)c(C#N)c(CC)c1C#N	nan
	2571531	38392	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	7	0	10	3.3	CCCCn1c(SCc2cc(=O)n3ccsc3n2)nc2cc(C(=O)OC)ccc2c1=O	nan
	CHEMBL1465204	38392	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	7	0	10	3.3	CCCCn1c(SCc2cc(=O)n3ccsc3n2)nc2cc(C(=O)OC)ccc2c1=O	nan
	2207742	38394	8	None	-11	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	4	2	6	3.8	CCc1c(C)sc(N=C(S)Nc2nc(C)cc(C)n2)c1C(=O)OC	nan
	CHEMBL1465216	38394	8	None	-11	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	4	2	6	3.8	CCc1c(C)sc(N=C(S)Nc2nc(C)cc(C)n2)c1C(=O)OC	nan
	1299194	38576	11	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	8	1	8	3.9	CCOC(=O)c1ccc(NC(=O)CSc2nnc(-c3cccs3)n2CC)cc1	nan
	CHEMBL1466656	38576	11	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	8	1	8	3.9	CCOC(=O)c1ccc(NC(=O)CSc2nnc(-c3cccs3)n2CC)cc1	nan
	7502637	38630	9	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	7	1	8	3.3	COc1ccc(-c2ccc(SCC(=O)Nc3nccs3)nn2)cc1OC	nan
	CHEMBL1467089	38630	9	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	7	1	8	3.3	COc1ccc(-c2ccc(SCC(=O)Nc3nccs3)nn2)cc1OC	nan
	1086372	38646	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	8	1	5	4.7	COc1cccc(-c2ccc(C#N)c(SCC(=O)NCCc3cccc(Cl)c3)n2)c1	nan
	CHEMBL1467241	38646	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	8	1	5	4.7	COc1cccc(-c2ccc(C#N)c(SCC(=O)NCCc3cccc(Cl)c3)n2)c1	nan
	865458	38657	7	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	230	2	0	4	2.8	COc1ccc2nc(SC)c(C#N)cc2c1	nan
	CHEMBL1467309	38657	7	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	230	2	0	4	2.8	COc1ccc2nc(SC)c(C#N)cc2c1	nan
	20886167	38951	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	361	5	1	5	2.6	COc1cccc(CNC(=O)Cn2c(=O)c3cccn3c3ccccc32)c1	nan
	CHEMBL1469817	38951	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	361	5	1	5	2.6	COc1cccc(CNC(=O)Cn2c(=O)c3cccn3c3ccccc32)c1	nan
	2045894	38961	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	3	0	5	4.9	Cc1ccc(-c2nc(=S)c3c(n2Cc2cccnc2)CC(C)(C)OC3)cc1	nan
	CHEMBL1469903	38961	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	3	0	5	4.9	Cc1ccc(-c2nc(=S)c3c(n2Cc2cccnc2)CC(C)(C)OC3)cc1	nan
	1035368	39082	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	5	1	7	4.2	COc1ccc2nc(NC(=O)CSc3nc4ccccc4o3)sc2c1	nan
	CHEMBL1470920	39082	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	5	1	7	4.2	COc1ccc2nc(NC(=O)CSc3nc4ccccc4o3)sc2c1	nan
	16009198	39260	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	7	1	7	4.2	CCc1ccc(C(=O)c2cn(CC(=O)Nc3ccc(OC)cc3)c3cc4c(cc3c2=O)OCO4)cc1	nan
	CHEMBL1472528	39260	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	7	1	7	4.2	CCc1ccc(C(=O)c2cn(CC(=O)Nc3ccc(OC)cc3)c3cc4c(cc3c2=O)OCO4)cc1	nan
	15988292	39272	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	586	8	3	6	6.3	COCCCNC(=O)c1sc2nc(C)c(C(=O)Nc3ccc(Cl)cc3)c(-c3ccc(Br)cc3)c2c1N	nan
	CHEMBL1472621	39272	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	586	8	3	6	6.3	COCCCNC(=O)c1sc2nc(C)c(C(=O)Nc3ccc(Cl)cc3)c(-c3ccc(Br)cc3)c2c1N	nan
	16027199	39293	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	457	6	1	6	3.7	CC(C)NC(=O)C1CCC(Cn2c(=O)c3sccc3n(Cc3ccc(F)cc3)c2=O)CC1	nan
	CHEMBL1472919	39293	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	457	6	1	6	3.7	CC(C)NC(=O)C1CCC(Cn2c(=O)c3sccc3n(Cc3ccc(F)cc3)c2=O)CC1	nan
	15988974	39297	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	546	12	2	7	4.6	CCc1ccccc1NC(=O)Cn1c(=O)n(CCCCCC(=O)NCc2ccc(C)cc2)c(=O)c2sccc21	nan
	CHEMBL1472973	39297	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	546	12	2	7	4.6	CCc1ccccc1NC(=O)Cn1c(=O)n(CCCCCC(=O)NCc2ccc(C)cc2)c(=O)c2sccc21	nan
	9505887	39310	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	2	0	6	2.3	N#Cc1ccc(OC(=O)C2CCN(C3=NS(=O)(=O)c4ccccc43)CC2)cc1	nan
	CHEMBL1473154	39310	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	2	0	6	2.3	N#Cc1ccc(OC(=O)C2CCN(C3=NS(=O)(=O)c4ccccc43)CC2)cc1	nan
	16021070	39314	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	4	1	6	3.7	COc1ccc(OC)c(NC(=O)c2cn3c4c(ccc(Cl)c4c2=O)OC(C)C3)c1	nan
	CHEMBL1473236	39314	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	4	1	6	3.7	COc1ccc(OC)c(NC(=O)c2cn3c4c(ccc(Cl)c4c2=O)OC(C)C3)c1	nan
	7786274	39322	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	4	2	5	3.0	O=C(COC(=O)c1cc(Br)ccc1O)Nc1cccnc1Cl	nan
	CHEMBL1473370	39322	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	4	2	5	3.0	O=C(COC(=O)c1cc(Br)ccc1O)Nc1cccnc1Cl	nan
	16017273	39337	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	318	3	1	5	1.7	Cc1nn(CC(=O)Nc2cc(F)ccc2F)c(=O)c2cccn12	nan
	CHEMBL1473495	39337	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	318	3	1	5	1.7	Cc1nn(CC(=O)Nc2cc(F)ccc2F)c(=O)c2cccn12	nan
	15990603	39373	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	4	0	5	6.2	CCOC(=O)c1ccc2ncc3c(-c4ccccc4)nn(-c4ccc(F)c(Cl)c4)c3c2c1	nan
	CHEMBL1474033	39373	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	4	0	5	6.2	CCOC(=O)c1ccc2ncc3c(-c4ccccc4)nn(-c4ccc(F)c(Cl)c4)c3c2c1	nan
	16015614	39393	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	7	1	5	5.1	CC(C)C(=O)Nc1ccc2nc(SCCOc3ccccc3)sc2c1	nan
	CHEMBL1474414	39393	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	7	1	5	5.1	CC(C)C(=O)Nc1ccc2nc(SCCOc3ccccc3)sc2c1	nan
	16012115	39401	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	7	1	6	3.7	COc1cccc(CNC(=O)Cn2ncc3c4ccccc4n(Cc4ccccc4)c3c2=O)c1	nan
	CHEMBL1474469	39401	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	7	1	6	3.7	COc1cccc(CNC(=O)Cn2ncc3c4ccccc4n(Cc4ccccc4)c3c2=O)c1	nan
	15987618	39420	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	3	0	4	5.7	CCN(C(=O)c1cc2c(=O)oc3ccccc3c2s1)c1cccc(C(F)(F)F)c1	nan
	CHEMBL1474699	39420	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	3	0	4	5.7	CCN(C(=O)c1cc2c(=O)oc3ccccc3c2s1)c1cccc(C(F)(F)F)c1	nan
	16016392	39421	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	3	1	4	4.9	CC(C)NC(=O)N1[C@H](c2cccs2)[C@@H](C)C(=O)[C@@H](C)[C@@H]1c1cccs1	nan
	CHEMBL1474706	39421	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	3	1	4	4.9	CC(C)NC(=O)N1[C@H](c2cccs2)[C@@H](C)C(=O)[C@@H](C)[C@@H]1c1cccs1	nan
	15989047	39453	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	502	8	1	9	3.0	N#Cc1ccccc1Cn1c(=O)n(CCCC(=O)NCc2ccc3c(c2)OCO3)c(=O)c2sccc21	nan
	CHEMBL1475184	39453	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	502	8	1	9	3.0	N#Cc1ccccc1Cn1c(=O)n(CCCC(=O)NCc2ccc3c(c2)OCO3)c(=O)c2sccc21	nan
	1300955	39479	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	5	1	6	4.1	COc1ccc(CNc2ncnc3c2cnn3-c2ccc(Cl)cc2)cc1	nan
	CHEMBL1475511	39479	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	5	1	6	4.1	COc1ccc(CNc2ncnc3c2cnn3-c2ccc(Cl)cc2)cc1	nan
	16021946	39511	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	471	4	0	6	4.8	Cc1ccc2c(c1)c1c(c(=O)n(-c3ccccc3C)c(=O)n1CC(=O)c1ccc(Cl)cc1)n2C	nan
	CHEMBL1475915	39511	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	471	4	0	6	4.8	Cc1ccc2c(c1)c1c(c(=O)n(-c3ccccc3C)c(=O)n1CC(=O)c1ccc(Cl)cc1)n2C	nan
	16009716	39547	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	4	1	6	4.1	O=C(Cn1c(=O)n(-c2ccccc2Cl)c(=O)c2sc3ccccc3c21)NC1CCCC1	nan
	CHEMBL1476522	39547	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	4	1	6	4.1	O=C(Cn1c(=O)n(-c2ccccc2Cl)c(=O)c2sc3ccccc3c21)NC1CCCC1	nan
	2387574	39635	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	366	5	1	6	4.0	CCS(=O)(=O)c1ccc2oc(Nc3cc(Cl)ccc3OC)nc2c1	nan
	CHEMBL1477466	39635	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	366	5	1	6	4.0	CCS(=O)(=O)c1ccc2oc(Nc3cc(Cl)ccc3OC)nc2c1	nan
	651813	39636	7	None	-7	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	6	1	6	4.1	CCc1nc(SCC(=O)NCc2ccco2)c2c3c(sc2n1)CCCC3	nan
	CHEMBL1477471	39636	7	None	-7	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	6	1	6	4.1	CCc1nc(SCC(=O)NCc2ccco2)c2c3c(sc2n1)CCCC3	nan
	135542325	39673	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	5	2	7	4.0	Cc1nnc2nc(SCC(=O)NC3CCCCC3)n(-c3ccc(Br)cc3)c(N)c1-2	nan
	CHEMBL1477773	39673	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	5	2	7	4.0	Cc1nnc2nc(SCC(=O)NC3CCCCC3)n(-c3ccc(Br)cc3)c(N)c1-2	nan
	4154279	39690	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	4	1	5	5.5	Cc1c(Cl)cccc1NC(=O)CSc1ncnc2c1sc1ccccc12	nan
	CHEMBL1477945	39690	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	4	1	5	5.5	Cc1c(Cl)cccc1NC(=O)CSc1ncnc2c1sc1ccccc12	nan
	647217	39738	1	None	1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	9	1	8	3.5	CCS(=O)(=O)Nc1ccc(-c2nnc(SCC(=O)c3cccc(OC)c3)o2)cc1	nan
	CHEMBL1478450	39738	1	None	1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	9	1	8	3.5	CCS(=O)(=O)Nc1ccc(-c2nnc(SCC(=O)c3cccc(OC)c3)o2)cc1	nan
	356316	39847	11	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	300	2	0	4	2.9	Cc1ccc(S(=O)(=O)c2cc3ccccc3oc2=O)cc1	nan
	CHEMBL1479392	39847	11	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	300	2	0	4	2.9	Cc1ccc(S(=O)(=O)c2cc3ccccc3oc2=O)cc1	nan
	16009796	39985	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	4	0	6	4.4	COc1ccc(-n2c(=O)c3sc4ccccc4c3n(Cc3ccccc3)c2=O)cc1	nan
	CHEMBL1480505	39985	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	4	0	6	4.4	COc1ccc(-n2c(=O)c3sc4ccccc4c3n(Cc3ccccc3)c2=O)cc1	nan
	16024583	40013	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	5	1	7	3.5	Cc1ccc2c(=O)c(C(=O)c3ccc(F)cc3)cn(CC(=O)Nc3ccc4c(c3)OCCO4)c2n1	nan
	CHEMBL1480766	40013	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	5	1	7	3.5	Cc1ccc2c(=O)c(C(=O)c3ccc(F)cc3)cn(CC(=O)Nc3ccc4c(c3)OCCO4)c2n1	nan
	3273049	40105	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	533	7	1	7	4.4	CCOC(=O)c1c(NC(=O)c2ccc(S(=O)(=O)N3CCC(C)CC3)cc2)sc2c1CCN(C(C)C)C2	nan
	CHEMBL1481475	40105	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	533	7	1	7	4.4	CCOC(=O)c1c(NC(=O)c2ccc(S(=O)(=O)N3CCC(C)CC3)cc2)sc2c1CCN(C(C)C)C2	nan
	3662250	40132	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	5	1	7	2.9	COc1ccc(-c2cc(C(=O)Nc3cc(C)on3)no2)cc1OC	nan
	CHEMBL1481783	40132	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	5	1	7	2.9	COc1ccc(-c2cc(C(=O)Nc3cc(C)on3)no2)cc1OC	nan
	5763301	40209	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	296	2	0	3	3.8	Cn1c(/C=C/c2ccc(Cl)cc2)nc2ccccc2c1=O	nan
	CHEMBL1482443	40209	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	296	2	0	3	3.8	Cn1c(/C=C/c2ccc(Cl)cc2)nc2ccccc2c1=O	nan
	16030274	40277	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	5	2	3	4.4	Cc1cccc2c(=O)cc(CSCC(=O)Nc3ccc(Cl)cc3)[nH]c12	nan
	CHEMBL1483081	40277	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	5	2	3	4.4	Cc1cccc2c(=O)cc(CSCC(=O)Nc3ccc(Cl)cc3)[nH]c12	nan
	135419126	40321	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	2	1	3	6.5	Oc1ccc(Cl)cc1C1=Nc2ccccc2N=C(c2cccc(Br)c2)C1	nan
	CHEMBL1483478	40321	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	2	1	3	6.5	Oc1ccc(Cl)cc1C1=Nc2ccccc2N=C(c2cccc(Br)c2)C1	nan
	16010346	40336	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	491	5	0	7	5.0	Cc1ccc(S(=O)(=O)c2nnn3c2nc(N(C)Cc2ccccc2)c2cc(Cl)ccc23)cc1C	nan
	CHEMBL1483574	40336	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	491	5	0	7	5.0	Cc1ccc(S(=O)(=O)c2nnn3c2nc(N(C)Cc2ccccc2)c2cc(Cl)ccc23)cc1C	nan
	1482113	40529	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	5	2	5	3.7	COCc1cc(O)nc2cc(NC(=O)c3cccc(OC)c3)c(C)cc12	nan
	CHEMBL1485213	40529	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	5	2	5	3.7	COCc1cc(O)nc2cc(NC(=O)c3cccc(OC)c3)c(C)cc12	nan
	848452	40565	11	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	4	1	4	2.9	COC(=O)c1ccc2ccn(CC(=O)NC3CCCCC3)c2c1	nan
	CHEMBL1485568	40565	11	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	4	1	4	2.9	COC(=O)c1ccc2ccn(CC(=O)NC3CCCCC3)c2c1	nan
	6491858	40686	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	361	5	2	7	3.4	COc1cccc(NC(=O)CSc2nc(O)c3c(C)csc3n2)c1	nan
	CHEMBL1486601	40686	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	361	5	2	7	3.4	COc1cccc(NC(=O)CSc2nc(O)c3c(C)csc3n2)c1	nan
	12005495	40721	3	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	400	6	2	4	4.0	Cc1cccc(C)c1NC(=O)C(NS(=O)(=O)c1cccs1)c1ccccc1	nan
	CHEMBL1486971	40721	3	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	400	6	2	4	4.0	Cc1cccc(C)c1NC(=O)C(NS(=O)(=O)c1cccs1)c1ccccc1	nan
	2007999	40792	8	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	358	4	1	6	3.4	CC(C)c1nc2sc3c(SCC(N)=O)ncnc3c2c2c1CCC2	nan
	CHEMBL1487512	40792	8	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	358	4	1	6	3.4	CC(C)c1nc2sc3c(SCC(N)=O)ncnc3c2c2c1CCC2	nan
	1604294	40819	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	7	0	4	5.9	Cc1ccc(OCCCCn2c(-c3ccc(Cl)cc3)nc3ccccc3c2=O)cc1	nan
	CHEMBL1487726	40819	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	7	0	4	5.9	Cc1ccc(OCCCCn2c(-c3ccc(Cl)cc3)nc3ccccc3c2=O)cc1	nan
	3847044	40985	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	5	0	8	4.1	COC(=O)CSc1nc2sc3c(c2c(=O)n1-c1ccc(C)cc1)CC(C(C)C)OC3	nan
	CHEMBL1488882	40985	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	5	0	8	4.1	COC(=O)CSc1nc2sc3c(c2c(=O)n1-c1ccc(C)cc1)CC(C(C)C)OC3	nan
	3531068	41054	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	512	5	1	8	4.5	COC(=O)c1ccc(C(=O)OC)c(NC(=O)c2cc3nc(-c4ccc(C)cc4)cc(C(F)(F)F)n3n2)c1	nan
	CHEMBL1489426	41054	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	512	5	1	8	4.5	COC(=O)c1ccc(C(=O)OC)c(NC(=O)c2cc3nc(-c4ccc(C)cc4)cc(C(F)(F)F)n3n2)c1	nan
	3149408	41140	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	6	6	8	-1.2	Cc1ccc(C2=NNC(C(O)C(O)C(O)C(O)CO)S2)cc1	nan
	CHEMBL1490120	41140	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	6	6	8	-1.2	Cc1ccc(C2=NNC(C(O)C(O)C(O)C(O)CO)S2)cc1	nan
	15996835	41208	9	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	6	2	6	3.9	COc1cc2nc(S)nc(NCCc3ccc(C)cc3)c2cc1OC	nan
	CHEMBL1490579	41208	9	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	6	2	6	3.9	COc1cc2nc(S)nc(NCCc3ccc(C)cc3)c2cc1OC	nan
	5216415	41246	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	3	0	5	5.2	COc1cccc2cc(-c3nc(-c4ccc(Cl)cc4)cs3)c(=O)oc12	nan
	CHEMBL1490839	41246	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	3	0	5	5.2	COc1cccc2cc(-c3nc(-c4ccc(Cl)cc4)cs3)c(=O)oc12	nan
	16022523	41305	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	442	3	0	7	2.3	Cn1cnc2c(=O)oc3ccc(S(=O)(=O)N4CCN(c5ccccc5F)CC4)cc3c21	nan
	CHEMBL1491216	41305	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	442	3	0	7	2.3	Cn1cnc2c(=O)oc3ccc(S(=O)(=O)N4CCN(c5ccccc5F)CC4)cc3c21	nan
	16034710	41531	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	6	1	5	3.9	Cc1ccc2c(=O)c(C(=O)c3cccc(Cl)c3)cn(CC(=O)NCc3ccccc3)c2n1	nan
	CHEMBL1492881	41531	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	6	1	5	3.9	Cc1ccc2c(=O)c(C(=O)c3cccc(Cl)c3)cn(CC(=O)NCc3ccccc3)c2n1	nan
	1319924	41559	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	495	9	0	6	4.8	CCCS(=O)(=O)c1c(S(=O)(=O)CCC)c2cc(CC)ccn2c1C(=O)c1ccc(Cl)cc1	nan
	CHEMBL1493213	41559	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	495	9	0	6	4.8	CCCS(=O)(=O)c1c(S(=O)(=O)CCC)c2cc(CC)ccn2c1C(=O)c1ccc(Cl)cc1	nan
	16423380	41575	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	410	5	1	7	2.9	COc1ccc(-c2cc3ccc(O)c(CN4CCN(C)CC4)c3oc2=O)cc1OC	nan
	7205024	41575	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	410	5	1	7	2.9	COc1ccc(-c2cc3ccc(O)c(CN4CCN(C)CC4)c3oc2=O)cc1OC	nan
	CHEMBL1493339	41575	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	410	5	1	7	2.9	COc1ccc(-c2cc3ccc(O)c(CN4CCN(C)CC4)c3oc2=O)cc1OC	nan
	6823777	41601	7	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	526	8	3	6	3.3	Cc1ccc(-n2c([S-])c(C(=O)Nc3ccc(OC(F)F)cc3)[n+]3ccc(C(=O)NCCO)cc23)cc1C	nan
	CHEMBL1493546	41601	7	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	526	8	3	6	3.3	Cc1ccc(-n2c([S-])c(C(=O)Nc3ccc(OC(F)F)cc3)[n+]3ccc(C(=O)NCCO)cc23)cc1C	nan
	1091748	41605	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	4	2	5	3.5	O=C(Nc1ccccc1C(=O)Nc1ccc2c(c1)OCO2)c1ccco1	nan
	CHEMBL1493592	41605	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	4	2	5	3.5	O=C(Nc1ccccc1C(=O)Nc1ccc2c(c1)OCO2)c1ccco1	nan
	4885142	41993	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	3	0	4	4.4	CC(=O)c1ccc(N2CCN(c3ccnc4cc(Cl)ccc34)CC2)cc1	nan
	CHEMBL1497325	41993	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	3	0	4	4.4	CC(=O)c1ccc(N2CCN(c3ccnc4cc(Cl)ccc34)CC2)cc1	nan
	665746	42048	12	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	358	3	0	5	3.5	O=C1c2oc3ccccc3c(=O)c2C(c2cccnc2)N1Cc1ccco1	nan
	CHEMBL1497863	42048	12	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	358	3	0	5	3.5	O=C1c2oc3ccccc3c(=O)c2C(c2cccnc2)N1Cc1ccco1	nan
	1478337	42077	13	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	2	1	4	5.2	Cc1ccc2oc3nc(C)c(C(=O)Nc4cccc(C(F)(F)F)c4)cc3c(=O)c2c1	nan
	CHEMBL1498149	42077	13	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	2	1	4	5.2	Cc1ccc2oc3nc(C)c(C(=O)Nc4cccc(C(F)(F)F)c4)cc3c(=O)c2c1	nan
	1877175	42166	9	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	320	5	1	6	2.9	CCOc1ccc(C(=O)Nc2nc(C)c(C(=O)OC)s2)cc1	nan
	CHEMBL1498972	42166	9	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	320	5	1	6	2.9	CCOc1ccc(C(=O)Nc2nc(C)c(C(=O)OC)s2)cc1	nan
	663555	42413	9	None	-1	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	293	3	1	4	3.6	Cc1cccc(C(=O)OCc2cc3ccccc3nc2O)c1	nan
	CHEMBL1501108	42413	9	None	-1	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	293	3	1	4	3.6	Cc1cccc(C(=O)OCc2cc3ccccc3nc2O)c1	nan
	1482342	42593	22	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	263	2	1	7	2.2	CSc1nc2ncc(-c3ccsc3)c(N)n2n1	nan
	CHEMBL1502638	42593	22	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	263	2	1	7	2.2	CSc1nc2ncc(-c3ccsc3)c(N)n2n1	nan
	6624089	42868	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	5	1	4	3.3	O=C(Cn1c(=O)c2cccn2c2ccccc21)NCCc1ccc(Cl)cc1	nan
	CHEMBL1505154	42868	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	5	1	4	3.3	O=C(Cn1c(=O)c2cccn2c2ccccc21)NCCc1ccc(Cl)cc1	nan
	1488509	42896	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	240	3	1	4	1.9	O=C(Nc1ccnc(-c2ccncc2)n1)C1CC1	nan
	CHEMBL1505422	42896	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	240	3	1	4	1.9	O=C(Nc1ccnc(-c2ccncc2)n1)C1CC1	nan
	8484069	43076	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	7	2	8	3.3	CC(=O)c1ccc(NC(=O)CSc2nnc(NC(=O)c3ccco3)s2)cc1	nan
	CHEMBL1506911	43076	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	7	2	8	3.3	CC(=O)c1ccc(NC(=O)CSc2nnc(NC(=O)c3ccco3)s2)cc1	nan
	2880344	43121	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	6	2	6	4.7	COc1ccc(CC(=O)Nc2ccc(-c3nc4cc(C)ccc4o3)c(O)c2)cc1OC	nan
	CHEMBL1507312	43121	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	6	2	6	4.7	COc1ccc(CC(=O)Nc2ccc(-c3nc4cc(C)ccc4o3)c(O)c2)cc1OC	nan
	1440345	43210	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	273	3	1	3	3.2	Cc1cc2cc3c(cc2nc1SCC(=O)O)CCC3	nan
	CHEMBL1508003	43210	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	273	3	1	3	3.2	Cc1cc2cc3c(cc2nc1SCC(=O)O)CCC3	nan
	4435004	43398	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	297	4	1	3	3.8	CCCn1c(NC(=O)c2ccc(F)cc2)nc2ccccc21	nan
	CHEMBL1509719	43398	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	297	4	1	3	3.8	CCCn1c(NC(=O)c2ccc(F)cc2)nc2ccccc21	nan
	2676980	43420	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	336	3	1	6	2.6	O=C(Cn1cnc2ccccc2c1=O)Nc1nc2ccccc2s1	nan
	CHEMBL1509918	43420	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	336	3	1	6	2.6	O=C(Cn1cnc2ccccc2c1=O)Nc1nc2ccccc2s1	nan
	2402709	43470	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	7	2	7	3.0	NS(=O)(=O)c1ccc(NC(=O)COC(=O)c2cn(-c3ccccc3)nc2-c2ccccc2)cc1	nan
	CHEMBL1510422	43470	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	7	2	7	3.0	NS(=O)(=O)c1ccc(NC(=O)COC(=O)c2cn(-c3ccccc3)nc2-c2ccccc2)cc1	nan
	16024491	43676	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	5	1	7	3.3	Cc1ccc2c(=O)c(C(=O)c3ccccc3)cn(CC(=O)Nc3ccc4c(c3)OCCO4)c2n1	nan
	CHEMBL1512438	43676	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	5	1	7	3.3	Cc1ccc2c(=O)c(C(=O)c3ccccc3)cn(CC(=O)Nc3ccc4c(c3)OCCO4)c2n1	nan
	7184798	43684	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	7	1	7	3.5	CC(C)Cn1c(=O)c2sccc2n2c(CCCC(=O)NC3CCCCC3)nnc12	nan
	CHEMBL1512523	43684	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	7	1	7	3.5	CC(C)Cn1c(=O)c2sccc2n2c(CCCC(=O)NC3CCCCC3)nnc12	nan
	16025847	43702	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	4	1	7	2.4	Cc1cccc(CNC(=O)c2cnc3sc(N4CCCCC4)nn3c2=O)c1	nan
	CHEMBL1512717	43702	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	4	1	7	2.4	Cc1cccc(CNC(=O)c2cnc3sc(N4CCCCC4)nn3c2=O)c1	nan
	16026525	43703	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	5	1	5	4.6	CCc1ccccc1NC(=O)C(C)n1c(=O)cc(C)c2c(C)nn(-c3ccccc3)c21	nan
	CHEMBL1512723	43703	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	5	1	5	4.6	CCc1ccccc1NC(=O)C(C)n1c(=O)cc(C)c2c(C)nn(-c3ccccc3)c21	nan
	16026338	43705	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	4	1	5	4.7	Cc1ccc(-n2nc(C)c3c(C)cc(=O)n(CC(=O)Nc4cc(Cl)ccc4C)c32)cc1	nan
	CHEMBL1512750	43705	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	4	1	5	4.7	Cc1ccc(-n2nc(C)c3c(C)cc(=O)n(CC(=O)Nc4cc(Cl)ccc4C)c32)cc1	nan
	7066893	43725	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	351	4	2	6	4.8	COc1cc(-c2nc3sccn3c2Nc2cccc(C)c2)ccc1O	nan
	CHEMBL1513064	43725	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	351	4	2	6	4.8	COc1cc(-c2nc3sccn3c2Nc2cccc(C)c2)ccc1O	nan
	16025357	43735	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	544	6	1	6	5.8	Cc1ccc(CN2c3ccccc3-c3nc(SCC(=O)Nc4c(C)cc(C)cc4C)ncc3S2(=O)=O)cc1	nan
	CHEMBL1513190	43735	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	544	6	1	6	5.8	Cc1ccc(CN2c3ccccc3-c3nc(SCC(=O)Nc4c(C)cc(C)cc4C)ncc3S2(=O)=O)cc1	nan
	16010879	43763	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	7	1	7	4.9	COc1cc2nc(NCCc3cccc(C)c3)n3nc(-c4ccccc4)nc3c2cc1OC	nan
	CHEMBL1513631	43763	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	7	1	7	4.9	COc1cc2nc(NCCc3cccc(C)c3)n3nc(-c4ccccc4)nc3c2cc1OC	nan
	2947326	43790	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	6	2	6	3.9	CCOC(=O)c1ccc(NC(=O)CSc2nc3c(C)c(Br)cnc3[nH]2)cc1	nan
	CHEMBL1514184	43790	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	6	2	6	3.9	CCOC(=O)c1ccc(NC(=O)CSc2nc3c(C)c(Br)cnc3[nH]2)cc1	nan
	15988389	43827	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	6	2	3	5.3	O=C(NCCc1ccccc1)c1cc(-c2ccccc2)nc2n[nH]c(-c3ccccc3)c12	nan
	CHEMBL1514741	43827	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	6	2	3	5.3	O=C(NCCc1ccccc1)c1cc(-c2ccccc2)nc2n[nH]c(-c3ccccc3)c12	nan
	16027439	43861	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	5	1	7	4.3	Cc1csc2nc(COC(=O)c3cccc(NC(=O)c4cccc(Cl)c4)c3)cc(=O)n12	nan
	CHEMBL1515224	43861	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	5	1	7	4.3	Cc1csc2nc(COC(=O)c3cccc(NC(=O)c4cccc(Cl)c4)c3)cc(=O)n12	nan
	3324743	43865	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	7	1	4	5.2	CCc1ccc(OCC(=O)Nc2c(C(=O)c3ccccc3)oc3ccccc23)cc1	nan
	CHEMBL1515282	43865	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	7	1	4	5.2	CCc1ccc(OCC(=O)Nc2c(C(=O)c3ccccc3)oc3ccccc23)cc1	nan
	1035668	43910	19	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	5	1	5	5.7	Cc1cccc(NC(=O)CSc2nc(-c3cccs3)cc(C(F)(F)F)c2C#N)c1	nan
	CHEMBL1515955	43910	19	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	5	1	5	5.7	Cc1cccc(NC(=O)CSc2nc(-c3cccs3)cc(C(F)(F)F)c2C#N)c1	nan
	16009680	43928	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	4	0	4	4.6	Cc1ccc(S(=O)(=O)c2cn(Cc3ccc(F)cc3)c3cc(F)c(F)cc3c2=O)cc1	nan
	CHEMBL1516142	43928	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	4	0	4	4.6	Cc1ccc(S(=O)(=O)c2cn(Cc3ccc(F)cc3)c3cc(F)c(F)cc3c2=O)cc1	nan
	1516716	43951	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	3	3	5	3.7	Nc1c(C(=O)Nc2ccc(C(=O)O)cc2)sc2nc3c(cc12)CCCC3	nan
	CHEMBL1516550	43951	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	3	3	5	3.7	Nc1c(C(=O)Nc2ccc(C(=O)O)cc2)sc2nc3c(cc12)CCCC3	nan
	15989644	43953	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	531	5	1	5	4.1	Cc1ccc(NC(=O)Cn2cc(S(=O)(=O)N3CCC(C)CC3)c3ccccc3c2=O)c(Br)c1	nan
	CHEMBL1516553	43953	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	531	5	1	5	4.1	Cc1ccc(NC(=O)Cn2cc(S(=O)(=O)N3CCC(C)CC3)c3ccccc3c2=O)c(Br)c1	nan
	16027696	43990	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	7	1	8	3.4	Cc1cccc(OCC(=O)Nc2ccccc2C(=O)OCc2cc(=O)n3ccsc3n2)c1	nan
	CHEMBL1516896	43990	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	7	1	8	3.4	Cc1cccc(OCC(=O)Nc2ccccc2C(=O)OCc2cc(=O)n3ccsc3n2)c1	nan
	16009847	44048	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	4	0	6	5.1	O=c1c2sc3ccccc3c2n(Cc2cccc(C(F)(F)F)c2)c(=O)n1Cc1ccco1	nan
	CHEMBL1517455	44048	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	4	0	6	5.1	O=c1c2sc3ccccc3c2n(Cc2cccc(C(F)(F)F)c2)c(=O)n1Cc1ccco1	nan
	16010572	44050	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	426	7	1	8	4.0	COc1ccc(OC)c(CCNc2nc3ccccc3c3nc(-c4cccnc4)nn23)c1	nan
	CHEMBL1517540	44050	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	426	7	1	8	4.0	COc1ccc(OC)c(CCNc2nc3ccccc3c3nc(-c4cccnc4)nn23)c1	nan
	1073734	44058	18	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	3	1	5	3.6	Cc1ccc(C(=O)Nc2nc3ccc(S(C)(=O)=O)cc3s2)cc1C	nan
	CHEMBL1517640	44058	18	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	3	1	5	3.6	Cc1ccc(C(=O)Nc2nc3ccc(S(C)(=O)=O)cc3s2)cc1C	nan
	15990463	44129	3	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	543	8	2	6	4.6	Cc1cccc(NC(=O)CSC2=Nc3ccccc3C3=NC(CCC(=O)NCc4ccc(F)cc4)C(=O)N23)c1	nan
	CHEMBL1518319	44129	3	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	543	8	2	6	4.6	Cc1cccc(NC(=O)CSC2=Nc3ccccc3C3=NC(CCC(=O)NCc4ccc(F)cc4)C(=O)N23)c1	nan
	890719	44181	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	289	4	2	4	0.9	CCN1C(=O)/C(=C\NCc2ccccc2)C(=O)NC1=S	nan
	CHEMBL1518771	44181	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	289	4	2	4	0.9	CCN1C(=O)/C(=C\NCc2ccccc2)C(=O)NC1=S	nan
	4457184	44202	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	358	2	2	7	2.2	N#Cc1c(N2CCCCC2)nc(N)c2c(N)nc3c(c12)CC(CCl)O3	nan
	CHEMBL1518944	44202	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	358	2	2	7	2.2	N#Cc1c(N2CCCCC2)nc(N)c2c(N)nc3c(c12)CC(CCl)O3	nan
	16013971	44232	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	4	0	7	3.7	Cc1nnc(N2CCN(c3ccc(Cl)cc3)CC2)c2c1nnn2Cc1ccc(F)cc1	nan
	CHEMBL1519203	44232	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	4	0	7	3.7	Cc1nnc(N2CCN(c3ccc(Cl)cc3)CC2)c2c1nnn2Cc1ccc(F)cc1	nan
	1557528	44252	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	8	0	5	5.1	Cc1ccc(OCCOCCn2c(-c3ccc(Cl)cc3)nc3ccccc3c2=O)cc1	nan
	CHEMBL1519353	44252	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	8	0	5	5.1	Cc1ccc(OCCOCCn2c(-c3ccc(Cl)cc3)nc3ccccc3c2=O)cc1	nan
	2158290	44286	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	552	9	0	9	3.8	CCOC(=O)c1cc2c(=O)n3ccccc3nc2n(CCCOC)/c1=N/C(=O)C(C)(C)Oc1ccc(Cl)cc1	nan
	CHEMBL1519687	44286	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	552	9	0	9	3.8	CCOC(=O)c1cc2c(=O)n3ccccc3nc2n(CCCOC)/c1=N/C(=O)C(C)(C)Oc1ccc(Cl)cc1	nan
	4379652	44426	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	447	6	1	10	1.1	Cn1c(=O)c2c(SCC(=O)NCC3CCCO3)nc(-c3cccs3)nc2n(C)c1=O	nan
	CHEMBL1520875	44426	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	447	6	1	10	1.1	Cn1c(=O)c2c(SCC(=O)NCC3CCCO3)nc(-c3cccs3)nc2n(C)c1=O	nan
	5925852	44472	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	493	5	1	10	3.2	COC(=O)c1ccc(C2C(C(=O)c3ccc4c(c3)OCCO4)=C(O)C(=O)N2c2nnc(C)s2)cc1	nan
	CHEMBL1521267	44472	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	493	5	1	10	3.2	COC(=O)c1ccc(C2C(C(=O)c3ccc4c(c3)OCCO4)=C(O)C(=O)N2c2nnc(C)s2)cc1	nan
	16018871	44507	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	7	1	6	2.8	COc1ccc(CNC(=O)CCCn2c(=O)c3cccn3c3cccnc32)cc1	nan
	CHEMBL1521570	44507	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	7	1	6	2.8	COc1ccc(CNC(=O)CCCn2c(=O)c3cccn3c3cccnc32)cc1	nan
	17252948	44608	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	336	3	1	5	3.9	Cc1ccc(NC(=O)c2cc(-c3ccc4c(c3)OCO4)on2)cc1C	nan
	CHEMBL1522534	44608	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	336	3	1	5	3.9	Cc1ccc(NC(=O)c2cc(-c3ccc4c(c3)OCO4)on2)cc1C	nan
	16009486	44645	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	481	8	1	9	3.9	COc1cc(C(=O)Nc2ccccc2OCc2cc(=O)n3c(C)csc3n2)cc(OC)c1OC	nan
	CHEMBL1522858	44645	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	481	8	1	9	3.9	COc1cc(C(=O)Nc2ccccc2OCc2cc(=O)n3c(C)csc3n2)cc(OC)c1OC	nan
	932437	44675	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	336	2	0	4	4.9	Cc1ccc(-c2nnc3c4ccccc4c(-c4ccccc4)nn23)cc1	nan
	CHEMBL1523117	44675	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	336	2	0	4	4.9	Cc1ccc(-c2nnc3c4ccccc4c(-c4ccccc4)nn23)cc1	nan
	2084813	44723	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	288	3	2	2	3.5	CC(=O)c1c(C)[nH]c(C(=O)Nc2cc(F)ccc2C)c1C	nan
	CHEMBL1523555	44723	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	288	3	2	2	3.5	CC(=O)c1c(C)[nH]c(C(=O)Nc2cc(F)ccc2C)c1C	nan
	663733	44766	12	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	4	1	8	3.1	Cc1nc2c(sc3nc4c(cc32)COC(C)(C)C4)c(=O)n1CC(=O)NCc1ccco1	nan
	CHEMBL1523984	44766	12	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	4	1	8	3.1	Cc1nc2c(sc3nc4c(cc32)COC(C)(C)C4)c(=O)n1CC(=O)NCc1ccco1	nan
	16027443	44870	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	5	1	7	4.3	Cc1csc2nc(COC(=O)c3ccccc3NC(=O)c3ccccc3Cl)cc(=O)n12	nan
	CHEMBL1525043	44870	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	5	1	7	4.3	Cc1csc2nc(COC(=O)c3ccccc3NC(=O)c3ccccc3Cl)cc(=O)n12	nan
	1299413	44961	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	6	1	5	3.1	C=CCn1c(SCC(=O)NC2CCCCC2)nc2ccccc2c1=O	nan
	CHEMBL1525864	44961	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	6	1	5	3.1	C=CCn1c(SCC(=O)NC2CCCCC2)nc2ccccc2c1=O	nan
	4174172	45120	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	499	7	0	6	4.9	COc1cc2c(cc1OC)C(COc1ccc3c(C)cc(=O)oc3c1)N(C(=O)Cc1ccccc1)CC2	nan
	CHEMBL1527205	45120	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	499	7	0	6	4.9	COc1cc2c(cc1OC)C(COc1ccc3c(C)cc(=O)oc3c1)N(C(=O)Cc1ccccc1)CC2	nan
	757005	45399	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	313	8	2	5	2.7	CCCc1cc(C(=O)OC)c(NC(=O)CCCC(=O)O)s1	nan
	CHEMBL1529664	45399	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	313	8	2	5	2.7	CCCc1cc(C(=O)OC)c(NC(=O)CCCC(=O)O)s1	nan
	4067774	45502	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	7	1	4	6.0	CCCOc1ccc(C(=O)Nc2c(C(=O)c3ccc(C)cc3)oc3ccccc23)cc1	nan
	CHEMBL1530590	45502	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	7	1	4	6.0	CCCOc1ccc(C(=O)Nc2c(C(=O)c3ccc(C)cc3)oc3ccccc23)cc1	nan
	3420293	45639	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	504	4	1	7	2.9	Cc1ccc(NC(=O)c2sc3ncn(CC(=O)N4CCOCC4)c(=O)c3c2C)c(Br)c1	nan
	CHEMBL1531811	45639	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	504	4	1	7	2.9	Cc1ccc(NC(=O)c2sc3ncn(CC(=O)N4CCOCC4)c(=O)c3c2C)c(Br)c1	nan
	821799	45665	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	295	1	0	5	2.1	CSc1nc2ccc(Br)cn2c(=O)c1C#N	nan
	CHEMBL1532047	45665	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	295	1	0	5	2.1	CSc1nc2ccc(Br)cn2c(=O)c1C#N	nan
	1475615	45694	15	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	5	1	6	5.0	O=C(Nc1cc2c(=O)n(-c3ccc(Oc4ccccc4)cc3)ccc2oc1=O)c1ccccc1	nan
	CHEMBL1532311	45694	15	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	5	1	6	5.0	O=C(Nc1cc2c(=O)n(-c3ccc(Oc4ccccc4)cc3)ccc2oc1=O)c1ccccc1	nan
	15989915	45738	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	6	1	5	4.6	COc1ccc(C2CC(=O)c3c([nH]c(C(=O)OCc4ccccc4)c3C)C2)cc1OC	nan
	CHEMBL1532686	45738	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	6	1	5	4.6	COc1ccc(C2CC(=O)c3c([nH]c(C(=O)OCc4ccccc4)c3C)C2)cc1OC	nan
	656128	45767	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	302	5	0	6	2.8	CCOc1ccc2cc(C#N)c(SCC(=O)OC)nc2c1	nan
	CHEMBL1532931	45767	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	302	5	0	6	2.8	CCOc1ccc2cc(C#N)c(SCC(=O)OC)nc2c1	nan
	3137936	45895	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	346	4	2	5	3.4	COC(=O)c1c(NC(C)=O)sc(C(=O)Nc2ccccc2C)c1C	nan
	CHEMBL1534032	45895	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	346	4	2	5	3.4	COC(=O)c1c(NC(C)=O)sc(C(=O)Nc2ccccc2C)c1C	nan
	16011802	45944	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	4	1	6	3.4	COc1ccc(C(=O)Nc2ccc3nc4n(c(=O)c3c2)CCCCC4)cc1OC	nan
	CHEMBL1534572	45944	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	4	1	6	3.4	COc1ccc(C(=O)Nc2ccc3nc4n(c(=O)c3c2)CCCCC4)cc1OC	nan
	3410008	45964	9	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	6	2	5	2.8	CCOc1ccc(N/C=C2/C(=O)NC(=S)N(Cc3ccccc3)C2=O)cc1	nan
	CHEMBL1534800	45964	9	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	6	2	5	2.8	CCOc1ccc(N/C=C2/C(=O)NC(=S)N(Cc3ccccc3)C2=O)cc1	nan
	5949916	46006	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	361	4	1	4	4.0	Cc1[nH]c2nc(SCC(=O)c3ccccc3)nc-2cc1Br	nan
	CHEMBL1535293	46006	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	361	4	1	4	4.0	Cc1[nH]c2nc(SCC(=O)c3ccccc3)nc-2cc1Br	nan
	2820834	46017	5	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	6	1	7	5.6	CSc1sc(-c2nnc(SCC(=O)Nc3ccc(Cl)cc3)n2C)c2c1C=CCC2	nan
	CHEMBL1535400	46017	5	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	6	1	7	5.6	CSc1sc(-c2nnc(SCC(=O)Nc3ccc(Cl)cc3)n2C)c2c1C=CCC2	nan
	16019886	46083	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	5	1	5	3.2	Cc1cccc(NC(=O)CN2C(=O)CSc3ccc(S(=O)(=O)N4CCCC4)cc32)c1C	nan
	CHEMBL1536151	46083	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	5	1	5	3.2	Cc1cccc(NC(=O)CN2C(=O)CSc3ccc(S(=O)(=O)N4CCCC4)cc32)c1C	nan
	891752	46143	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	319	3	1	4	3.6	COc1cc(Cl)c(C)cc1NC(=O)c1ccc2c(c1)OCO2	nan
	CHEMBL1536712	46143	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	319	3	1	4	3.6	COc1cc(Cl)c(C)cc1NC(=O)c1ccc2c(c1)OCO2	nan
	664078	46436	1	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	4	1	4	3.3	COc1cccc(OCc2nc3cc(Br)c[nH]c-3n2)c1	nan
	CHEMBL1539150	46436	1	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	4	1	4	3.3	COc1cccc(OCc2nc3cc(Br)c[nH]c-3n2)c1	nan
	841141	46786	10	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	318	4	2	5	2.2	COC(=O)c1c(NC(=O)c2ccccc2)sc(C(N)=O)c1C	nan
	CHEMBL1542119	46786	10	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	318	4	2	5	2.2	COC(=O)c1c(NC(=O)c2ccccc2)sc(C(N)=O)c1C	nan
	664933	46948	10	None	-2	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	4	1	5	4.6	Cc1nc(SCC(=O)Nc2ccc(F)cc2)c2oc3ccccc3c2n1	nan
	CHEMBL1543543	46948	10	None	-2	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	4	1	5	4.6	Cc1nc(SCC(=O)Nc2ccc(F)cc2)c2oc3ccccc3c2n1	nan
	3240821	47020	8	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	498	7	1	8	2.9	O=C(CCCCCn1c(=S)[nH]c2cc3c(cc2c1=O)OCO3)N1CCN(C(=O)c2ccco2)CC1	nan
	CHEMBL1544051	47020	8	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	498	7	1	8	2.9	O=C(CCCCCn1c(=S)[nH]c2cc3c(cc2c1=O)OCO3)N1CCN(C(=O)c2ccco2)CC1	nan
	1861702	47077	8	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	5	1	8	2.7	CC(C)OC(=O)CSc1nc(N)c(C#N)c(-c2ccco2)c1C#N	nan
	CHEMBL1544436	47077	8	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	5	1	8	2.7	CC(C)OC(=O)CSc1nc(N)c(C#N)c(-c2ccco2)c1C#N	nan
	3164596	47206	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	309	4	1	4	2.7	COc1ccc2cc(C(=O)NCc3ccccc3)c(=O)oc2c1	nan
	CHEMBL1545409	47206	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	309	4	1	4	2.7	COc1ccc2cc(C(=O)NCc3ccccc3)c(=O)oc2c1	nan
	4340721	47260	7	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	293	3	1	4	4.0	COc1ccc2cc(C#N)c(Nc3cccc(F)c3)nc2c1	nan
	CHEMBL1545865	47260	7	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	293	3	1	4	4.0	COc1ccc2cc(C#N)c(Nc3cccc(F)c3)nc2c1	nan
	2106365	47263	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	305	2	1	5	4.1	Oc1nc(-c2cccnc2)nc2sc(-c3ccccc3)cc12	nan
	CHEMBL1545901	47263	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	305	2	1	5	4.1	Oc1nc(-c2cccnc2)nc2sc(-c3ccccc3)cc12	nan
	902245	47410	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	305	3	1	3	4.9	CCc1cc2cc(C(=O)Nc3ccc(F)cc3)sc2s1	nan
	CHEMBL1547204	47410	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	305	3	1	3	4.9	CCc1cc2cc(C(=O)Nc3ccc(F)cc3)sc2s1	nan
	1088622	47440	13	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	4	1	9	1.2	CCOc1ccc(-c2c(C#N)c(N)nc3c2c(=O)n(C)c(=O)n3C)cc1OC	nan
	CHEMBL1547487	47440	13	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	4	1	9	1.2	CCOc1ccc(-c2c(C#N)c(N)nc3c2c(=O)n(C)c(=O)n3C)cc1OC	nan
	2801256	47579	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	231	1	1	5	2.4	Cc1nc(-c2cc(C#N)c(O)nc2C)cs1	nan
	CHEMBL1548830	47579	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	231	1	1	5	2.4	Cc1nc(-c2cc(C#N)c(O)nc2C)cs1	nan
	4601866	47690	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	552	10	3	6	3.4	NS(=O)(=O)c1ccc(CCNC(=O)CCCCCn2c(=S)[nH]c3ccc(Br)cc3c2=O)cc1	nan
	CHEMBL1549770	47690	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	552	10	3	6	3.4	NS(=O)(=O)c1ccc(CCNC(=O)CCCCCn2c(=S)[nH]c3ccc(Br)cc3c2=O)cc1	nan
	2731089	47738	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	9	2	7	2.6	COc1ccc(CCNC(=S)NC(=O)c2cc(OC)c(OC)c(OC)c2)cc1OC	nan
	CHEMBL1550121	47738	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	9	2	7	2.6	COc1ccc(CCNC(=S)NC(=O)c2cc(OC)c(OC)c(OC)c2)cc1OC	nan
	5122884	47770	4	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	348	4	1	5	2.8	COc1ccc2cc(CCN3C(=O)c4ccccc4C3=O)c(O)nc2c1	nan
	CHEMBL1550382	47770	4	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	348	4	1	5	2.8	COc1ccc2cc(CCN3C(=O)c4ccccc4C3=O)c(O)nc2c1	nan
	1490541	47776	14	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	283	3	1	3	4.2	Cc1ccccc1CNc1ncnc2cc(Cl)ccc12	nan
	CHEMBL1550435	47776	14	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	283	3	1	3	4.2	Cc1ccccc1CNc1ncnc2cc(Cl)ccc12	nan
	15944825	47838	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	464	5	1	5	4.2	Cc1ccc(NC(=O)Cn2cc(S(=O)(=O)c3ccc(C)cc3)c(=O)c3cc(F)ccc32)cc1	nan
	CHEMBL1550942	47838	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	464	5	1	5	4.2	Cc1ccc(NC(=O)Cn2cc(S(=O)(=O)c3ccc(C)cc3)c(=O)c3cc(F)ccc32)cc1	nan
	15988480	47856	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	373	4	1	6	2.4	COC(=O)c1cc(Cl)ccc1NC(=O)Cn1c(C)cc(C)c(C#N)c1=O	nan
	CHEMBL1551156	47856	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	373	4	1	6	2.4	COC(=O)c1cc(Cl)ccc1NC(=O)Cn1c(C)cc(C)c(C#N)c1=O	nan
	16025269	47859	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	5	2	5	4.7	COC(=O)c1c(SCC(=O)Nc2ccccc2C(F)(F)F)[nH]c2ccc(Cl)cc2c1=O	nan
	CHEMBL1551199	47859	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	5	2	5	4.7	COC(=O)c1c(SCC(=O)Nc2ccccc2C(F)(F)F)[nH]c2ccc(Cl)cc2c1=O	nan
	16009432	47874	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	5	1	6	3.9	Cc1cccc(C(=O)Nc2ccc(OCc3cc(=O)n4ccsc4n3)cc2)c1	nan
	CHEMBL1551357	47874	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	5	1	6	3.9	Cc1cccc(C(=O)Nc2ccc(OCc3cc(=O)n4ccsc4n3)cc2)c1	nan
	3151519	47877	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	447	8	3	8	1.4	Cc1cccn2c(=O)c3cc(C(=O)NCc4ccccc4)c(=N)n(CCOCCO)c3nc12	nan
	CHEMBL1551451	47877	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	447	8	3	8	1.4	Cc1cccn2c(=O)c3cc(C(=O)NCc4ccccc4)c(=N)n(CCOCCO)c3nc12	nan
	16007408	47883	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	2	2	3	3.7	Cc1ccc(NC(=O)c2cc3c(=O)[nH]c4ccccc4c3n2C)cc1F	nan
	CHEMBL1551538	47883	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	2	2	3	3.7	Cc1ccc(NC(=O)c2cc3c(=O)[nH]c4ccccc4c3n2C)cc1F	nan
	16021062	47893	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	3	1	6	3.5	COC(=O)c1ccccc1NC(=O)c1cn2c3c(ccc(Cl)c3c1=O)OC(C)C2	nan
	CHEMBL1551793	47893	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	3	1	6	3.5	COC(=O)c1ccccc1NC(=O)c1cn2c3c(ccc(Cl)c3c1=O)OC(C)C2	nan
	1189625	47900	17	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	7	1	5	5.3	CCOc1ccc(C(=O)Nc2c(C(=O)c3ccc(OC)cc3)oc3ccccc23)cc1	nan
	CHEMBL1551857	47900	17	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	7	1	5	5.3	CCOc1ccc(C(=O)Nc2c(C(=O)c3ccc(OC)cc3)oc3ccccc23)cc1	nan
	16008906	47907	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	4	1	5	3.0	COc1cccc(CNC(=O)c2cc3c(=O)n(C)c4ccccc4c3n2C)c1	nan
	CHEMBL1551951	47907	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	4	1	5	3.0	COc1cccc(CNC(=O)c2cc3c(=O)n(C)c4ccccc4c3n2C)c1	nan
	16011042	47917	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	2	2	3	4.8	O=C(Nc1ccc(F)cc1)c1ccc2c(c1)NC(=O)c1ccccc1S2	nan
	CHEMBL1552027	47917	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	2	2	3	4.8	O=C(Nc1ccc(F)cc1)c1ccc2c(c1)NC(=O)c1ccccc1S2	nan
	4412264	47918	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	7	0	8	4.5	CCOC(=O)CSc1nc2c(sc3cccc(F)c32)c(=O)n1Cc1ccc(OC)cc1	nan
	CHEMBL1552040	47918	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	7	0	8	4.5	CCOC(=O)CSc1nc2c(sc3cccc(F)c32)c(=O)n1Cc1ccc(OC)cc1	nan
	1187153	47920	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	6	1	6	3.5	CCOC(=O)c1cnc2c(Cl)c(Cl)ccc2c1NCCN1CCOCC1	nan
	CHEMBL1552062	47920	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	6	1	6	3.5	CCOC(=O)c1cnc2c(Cl)c(Cl)ccc2c1NCCN1CCOCC1	nan
	16027700	47942	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	463	7	1	8	3.7	Cc1ccc(OCC(=O)Nc2ccccc2C(=O)OCc2cc(=O)n3ccsc3n2)cc1C	nan
	CHEMBL1552279	47942	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	463	7	1	8	3.7	Cc1ccc(OCC(=O)Nc2ccccc2C(=O)OCc2cc(=O)n3ccsc3n2)cc1C	nan
	16032167	47960	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	6	2	8	3.5	Cn1c(SCC(=O)Nc2nc3ccccc3s2)ncc(C(=O)Nc2ccc(F)cc2)c1=O	nan
	CHEMBL1552642	47960	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	6	2	8	3.5	Cn1c(SCC(=O)Nc2nc3ccccc3s2)ncc(C(=O)Nc2ccc(F)cc2)c1=O	nan
	16024489	47978	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	5	1	5	4.5	Cc1ccc2c(=O)c(C(=O)c3ccccc3)cn(CC(=O)Nc3ccc(C)c(Cl)c3)c2n1	nan
	CHEMBL1552935	47978	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	5	1	5	4.5	Cc1ccc2c(=O)c(C(=O)c3ccccc3)cn(CC(=O)Nc3ccc(C)c(Cl)c3)c2n1	nan
	16030793	47979	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	7	1	5	5.2	COc1ccccc1-c1cc(NC(=O)COc2ccccc2Cl)n(-c2ccccc2)n1	nan
	CHEMBL1552946	47979	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	7	1	5	5.2	COc1ccccc1-c1cc(NC(=O)COc2ccccc2Cl)n(-c2ccccc2)n1	nan
	16020265	47986	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	6	2	6	2.5	Cc1ccc(-n2c(=O)c3ccc(C(=O)NCc4ccccc4Cl)cc3n(CC(N)=O)c2=O)cc1	nan
	CHEMBL1552986	47986	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	6	2	6	2.5	Cc1ccc(-n2c(=O)c3ccc(C(=O)NCc4ccccc4Cl)cc3n(CC(N)=O)c2=O)cc1	nan
	16024860	48007	3	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	4	1	4	3.9	O=S(=O)(c1ccc2nc(Nc3ccc(F)cc3)ccc2c1)N1CCCC1	nan
	CHEMBL1553226	48007	3	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	4	1	4	3.9	O=S(=O)(c1ccc2nc(Nc3ccc(F)cc3)ccc2c1)N1CCCC1	nan
	16014611	48016	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	4	1	5	3.1	CSc1ccc(NC(=O)C2CCN(c3ncccn3)CC2)cc1	nan
	CHEMBL1553334	48016	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	4	1	5	3.1	CSc1ccc(NC(=O)C2CCN(c3ncccn3)CC2)cc1	nan
	16018242	48032	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	477	6	1	6	5.5	COc1ccc(NC(=O)c2oc3c(c2C)-c2nn(Cc4ccccc4Cl)cc2CC3)cc1OC	nan
	CHEMBL1553551	48032	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	477	6	1	6	5.5	COc1ccc(NC(=O)c2oc3c(c2C)-c2nn(Cc4ccccc4Cl)cc2CC3)cc1OC	nan
	16020219	48035	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	2	1	4	4.2	Cn1c(=O)c2cc(C(=O)NC3CCCCCC3)sc2c2ccccc21	nan
	CHEMBL1553584	48035	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	2	1	4	4.2	Cn1c(=O)c2cc(C(=O)NC3CCCCCC3)sc2c2ccccc21	nan
	3158758	48037	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	4	1	6	4.2	COc1cc(OC)c(C2Nc3c(C)cccc3-c3cc(C)nn32)cc1OC	nan
	CHEMBL1553632	48037	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	4	1	6	4.2	COc1cc(OC)c(C2Nc3c(C)cccc3-c3cc(C)nn32)cc1OC	nan
	15989000	48040	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	481	7	1	8	2.8	O=C(CCn1c(=O)c2sccc2n(Cc2ccccc2F)c1=O)NCc1ccc2c(c1)OCO2	nan
	CHEMBL1553743	48040	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	481	7	1	8	2.8	O=C(CCn1c(=O)c2sccc2n(Cc2ccccc2F)c1=O)NCc1ccc2c(c1)OCO2	nan
	2580267	48047	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	4	1	5	2.9	Cc1cc(C)cc(NC(=O)COC(=O)c2ccc3c(c2)OCCO3)c1	nan
	CHEMBL1553826	48047	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	4	1	5	2.9	Cc1cc(C)cc(NC(=O)COC(=O)c2ccc3c(c2)OCCO3)c1	nan
	16033854	48051	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	3	1	8	3.1	COC(=O)c1ccc2c(=O)n3nc(Nc4ccc(F)cc4F)sc3nc2c1	nan
	CHEMBL1553893	48051	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	3	1	8	3.1	COC(=O)c1ccc2c(=O)n3nc(Nc4ccc(F)cc4F)sc3nc2c1	nan
	16030113	48066	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	5	1	6	3.5	Cc1cccc(CNC(=O)Cn2nc(C)c3nn(-c4ccc(Cl)cc4)c(C)c3c2=O)c1	nan
	CHEMBL1554129	48066	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	5	1	6	3.5	Cc1cccc(CNC(=O)Cn2nc(C)c3nn(-c4ccc(Cl)cc4)c(C)c3c2=O)c1	nan
	4361698	48085	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	540	5	0	8	3.8	CCOC(=O)c1cc2c(=O)n3ccccc3nc2n(CC2CCCO2)/c1=N\C(=O)c1cccc(C(F)(F)F)c1	nan
	CHEMBL1554379	48085	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	540	5	0	8	3.8	CCOC(=O)c1cc2c(=O)n3ccccc3nc2n(CC2CCCO2)/c1=N\C(=O)c1cccc(C(F)(F)F)c1	nan
	16282512	48087	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	442	6	1	5	3.2	Cc1ccc(NC(=O)CN(C)C(=O)COc2ncnc3ccc(Br)cc23)cc1	nan
	CHEMBL1554437	48087	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	442	6	1	5	3.2	Cc1ccc(NC(=O)CN(C)C(=O)COc2ncnc3ccc(Br)cc23)cc1	nan
	16009851	48090	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	489	6	1	7	4.2	COc1cccc(NC(=O)Cn2c(=O)n(Cc3ccc(F)cc3)c(=O)c3sc4ccccc4c32)c1	nan
	CHEMBL1554474	48090	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	489	6	1	7	4.2	COc1cccc(NC(=O)Cn2c(=O)n(Cc3ccc(F)cc3)c(=O)c3sc4ccccc4c32)c1	nan
	16011879	48091	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	295	4	1	2	4.1	Cc1ccc(CNC(=O)Cc2csc3ccccc23)cc1	nan
	CHEMBL1554476	48091	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	295	4	1	2	4.1	Cc1ccc(CNC(=O)Cc2csc3ccccc23)cc1	nan
	15988910	48094	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	5	0	10	2.6	COc1cc(OC)cc(-n2c(=O)c3sccc3n(Cc3cc(=O)n4c(C)cccc4n3)c2=O)c1	nan
	CHEMBL1554524	48094	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	5	0	10	2.6	COc1cc(OC)cc(-n2c(=O)c3sccc3n(Cc3cc(=O)n4c(C)cccc4n3)c2=O)c1	nan
	16009798	48095	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	361	3	1	5	4.8	Fc1cccc(-c2nnn3c2nc(NC2CCCCC2)c2ccccc23)c1	nan
	CHEMBL1554525	48095	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	361	3	1	5	4.8	Fc1cccc(-c2nnn3c2nc(NC2CCCCC2)c2ccccc23)c1	nan
	16019045	48096	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	482	8	1	7	4.0	CCOc1cc(CNC(=O)c2ccc(Cn3c(=O)c4cccn4c4cccnc43)cc2)ccc1OC	nan
	CHEMBL1554576	48096	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	482	8	1	7	4.0	CCOc1cc(CNC(=O)c2ccc(Cn3c(=O)c4cccn4c4cccnc43)cc2)ccc1OC	nan
	16010240	48110	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	332	3	1	3	5.3	CC(C)c1ccc(NC(=O)c2cc3sc(Cl)cc3n2C)cc1	nan
	CHEMBL1554758	48110	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	332	3	1	3	5.3	CC(C)c1ccc(NC(=O)c2cc3sc(Cl)cc3n2C)cc1	nan
	16016717	48141	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	4	2	3	6.0	CCc1ccccc1NC(=O)Nc1ccc2c(c1)N(CC)C(=O)c1ccccc1S2	nan
	CHEMBL1555228	48141	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	4	2	3	6.0	CCc1ccccc1NC(=O)Nc1ccc2c(c1)N(CC)C(=O)c1ccccc1S2	nan
	15999699	48143	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	5	1	5	3.7	CCCCNC(=O)c1nn(-c2ccc(C)cc2)c(=O)c2c1c1ccccc1n2C	nan
	CHEMBL1555241	48143	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	5	1	5	3.7	CCCCNC(=O)c1nn(-c2ccc(C)cc2)c(=O)c2c1c1ccccc1n2C	nan
	16024527	48223	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	6	1	6	4.2	COc1ccc(C(=O)c2cn(CC(=O)Nc3cc(C)ccc3C)c3nc(C)ccc3c2=O)cc1	nan
	CHEMBL1556147	48223	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	6	1	6	4.2	COc1ccc(C(=O)c2cn(CC(=O)Nc3cc(C)ccc3C)c3nc(C)ccc3c2=O)cc1	nan
	884827	48224	16	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	298	4	1	5	3.8	CCOc1ccc(Nc2nc3ccccc3c(=O)s2)cc1	nan
	CHEMBL1556149	48224	16	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	298	4	1	5	3.8	CCOc1ccc(Nc2nc3ccccc3c(=O)s2)cc1	nan
	1299811	48245	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	3	0	8	3.4	COC(=O)CSc1ncnc2c1sc1nc3c(cc12)COC(C)(C)C3	nan
	CHEMBL1556306	48245	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	3	0	8	3.4	COC(=O)CSc1ncnc2c1sc1nc3c(cc12)COC(C)(C)C3	nan
	1297627	48275	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	373	3	1	3	4.1	CC(=O)c1ccc(NC(=S)N2CCN(c3cccc(Cl)c3)CC2)cc1	nan
	CHEMBL1556657	48275	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	373	3	1	3	4.1	CC(=O)c1ccc(NC(=S)N2CCN(c3cccc(Cl)c3)CC2)cc1	nan
	1262055	48277	7	None	-2	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	6	1	6	5.3	CCn1c(SCC(=O)Nc2cccc(F)c2)nnc1-c1cc2cc(Br)ccc2o1	nan
	CHEMBL1556666	48277	7	None	-2	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	6	1	6	5.3	CCn1c(SCC(=O)Nc2cccc(F)c2)nnc1-c1cc2cc(Br)ccc2o1	nan
	2769090	48437	23	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	320	3	0	5	2.8	CC(=O)c1cc(C#N)c(N2CCN(c3ccccc3)CC2)nc1C	nan
	CHEMBL1558006	48437	23	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	320	3	0	5	2.8	CC(=O)c1cc(C#N)c(N2CCN(c3ccccc3)CC2)nc1C	nan
	16015862	48608	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	5	1	4	5.7	Cc1ccc(SCC(=O)Nc2ccc3oc(-c4ccc(F)cc4)nc3c2)cc1	nan
	CHEMBL1559463	48608	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	5	1	4	5.7	Cc1ccc(SCC(=O)Nc2ccc3oc(-c4ccc(F)cc4)nc3c2)cc1	nan
	3208119	48634	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	5	1	5	4.4	CCc1cc2ccc(C)c(C)c2nc1SCC(=O)Nc1cc(C)on1	nan
	CHEMBL1559714	48634	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	5	1	5	4.4	CCc1cc2ccc(C)c(C)c2nc1SCC(=O)Nc1cc(C)on1	nan
	16286863	48807	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	5	2	6	2.7	CC(OC(=O)c1cc(Br)ccc1O)C(=O)NCc1ccc2c(c1)OCO2	nan
	CHEMBL1561413	48807	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	5	2	6	2.7	CC(OC(=O)c1cc(Br)ccc1O)C(=O)NCc1ccc2c(c1)OCO2	nan
	24686491	48965	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	5	1	5	3.2	COc1ccc(S(=O)(=O)N2CCCCCC2)cc1C(=O)Nc1ccc(C)cn1	nan
	CHEMBL1562813	48965	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	5	1	5	3.2	COc1ccc(S(=O)(=O)N2CCCCCC2)cc1C(=O)Nc1ccc(C)cn1	nan
	135884418	48981	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	366	4	1	7	3.9	COc1cc2ccccc2cc1C(=O)OCc1nc(O)c2sccc2n1	nan
	CHEMBL1562918	48981	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	366	4	1	7	3.9	COc1cc2ccccc2cc1C(=O)OCc1nc(O)c2sccc2n1	nan
	664089	49031	8	None	-3	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	4	1	5	4.6	Cc1nc(SCC(=O)Nc2cccc(F)c2)c2oc3ccccc3c2n1	nan
	CHEMBL1563407	49031	8	None	-3	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	4	1	5	4.6	Cc1nc(SCC(=O)Nc2cccc(F)c2)c2oc3ccccc3c2n1	nan
	16008603	49032	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	410	6	1	7	1.5	COc1ccc(CNC(=O)CCc2c(C)nc3c(c2C)c(=O)n(C)c(=O)n3C)cc1	nan
	CHEMBL1563417	49032	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	410	6	1	7	1.5	COc1ccc(CNC(=O)CCc2c(C)nc3c(c2C)c(=O)n(C)c(=O)n3C)cc1	nan
	16025580	49080	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	488	4	1	6	4.6	Cc1cc(C)c(NC(=O)CSc2ncc3c(n2)-c2cc(Cl)ccc2N(C)S3(=O)=O)c(C)c1	nan
	CHEMBL1563792	49080	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	488	4	1	6	4.6	Cc1cc(C)c(NC(=O)CSc2ncc3c(n2)-c2cc(Cl)ccc2N(C)S3(=O)=O)c(C)c1	nan
	654285	49197	1	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	283	1	0	6	1.7	N#Cc1cc2cc3c(cc2nc1N1CCOCC1)OCO3	nan
	CHEMBL1564877	49197	1	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	283	1	0	6	1.7	N#Cc1cc2cc3c(cc2nc1N1CCOCC1)OCO3	nan
	4282255	49298	11	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	293	4	1	6	2.6	COc1cc([N+](=O)[O-])cc2sc(NC(=O)C3CC3)nc12	nan
	CHEMBL1565614	49298	11	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	293	4	1	6	2.6	COc1cc([N+](=O)[O-])cc2sc(NC(=O)C3CC3)nc12	nan
	151922	49568	57	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	276	12	1	1	5.2	O=C(O)CCCCCCCCCCCc1ccccc1	nan
	CHEMBL1567811	49568	57	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	276	12	1	1	5.2	O=C(O)CCCCCCCCCCCc1ccccc1	nan
	4289114	49691	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	6	1	4	6.0	Cc1ccc(C(=O)c2oc3ccccc3c2NC(=O)C(C)Oc2ccccc2Cl)cc1	nan
	CHEMBL1568822	49691	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	6	1	4	6.0	Cc1ccc(C(=O)c2oc3ccccc3c2NC(=O)C(C)Oc2ccccc2Cl)cc1	nan
	650090	49722	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	6	0	9	2.7	Cn1c(=O)c2c(nc(SCC(=O)c3cccs3)n2Cc2ccc(F)cc2)n(C)c1=O	nan
	CHEMBL1569069	49722	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	6	0	9	2.7	Cn1c(=O)c2c(nc(SCC(=O)c3cccs3)n2Cc2ccc(F)cc2)n(C)c1=O	nan
	1336265	49860	7	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	3	2	6	2.5	COC(=O)c1sc(NC(=S)NC(=O)c2ccccc2F)nc1C	nan
	CHEMBL1570262	49860	7	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	3	2	6	2.5	COC(=O)c1sc(NC(=S)NC(=O)c2ccccc2F)nc1C	nan
	1834757	49901	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	5	0	5	6.7	CCN(CC)c1ccc2cc(-c3nc(-c4ccc(Cl)cc4Cl)cs3)c(=O)oc2c1	nan
	CHEMBL1570631	49901	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	5	0	5	6.7	CCN(CC)c1ccc2cc(-c3nc(-c4ccc(Cl)cc4Cl)cs3)c(=O)oc2c1	nan
	661116	49979	8	None	-1	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	5	1	8	3.2	COc1ccc(-n2ncc3c(NCc4ccc5c(c4)OCO5)ncnc32)cc1	nan
	CHEMBL1571331	49979	8	None	-1	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	5	1	8	3.2	COc1ccc(-n2ncc3c(NCc4ccc5c(c4)OCO5)ncnc32)cc1	nan
	3228933	50038	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	6	1	8	3.5	CCc1nc(SCC(=O)Nc2c(C)nn(C)c2C)c2cnn(-c3ccccc3)c2n1	nan
	CHEMBL1571990	50038	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	6	1	8	3.5	CCc1nc(SCC(=O)Nc2c(C)nn(C)c2C)c2cnn(-c3ccccc3)c2n1	nan
	998563	50048	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	358	3	1	3	5.8	Cc1ccc(NC(=O)c2cc(-c3cccs3)nc3ccccc23)c(C)c1	nan
	CHEMBL1572046	50048	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	358	3	1	3	5.8	Cc1ccc(NC(=O)c2cc(-c3cccs3)nc3ccccc23)c(C)c1	nan
	5038692	50086	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	4	1	6	1.9	O=C(O)C1Cc2ccccc2CN1C(=O)CSc1nnc2ccccn12	nan
	CHEMBL1572334	50086	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	4	1	6	1.9	O=C(O)C1Cc2ccccc2CN1C(=O)CSc1nnc2ccccn12	nan
	16020271	50360	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	539	7	1	6	5.1	COc1ccc(-n2c(=O)c3ccc(C(=O)NCc4ccc(C)cc4)cc3n(Cc3cccc(Cl)c3)c2=O)cc1	nan
	CHEMBL1575057	50360	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	539	7	1	6	5.1	COc1ccc(-n2c(=O)c3ccc(C(=O)NCc4ccc(C)cc4)cc3n(Cc3cccc(Cl)c3)c2=O)cc1	nan
	1637692	50371	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	7	1	5	4.1	CC(=O)c1sc(NC(=O)CCCOc2ccc(Cl)cc2)nc1C	nan
	CHEMBL1575283	50371	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	7	1	5	4.1	CC(=O)c1sc(NC(=O)CCCOc2ccc(Cl)cc2)nc1C	nan
	2446441	50640	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	348	3	2	2	4.2	CC(=O)c1c(C)[nH]c(C(=O)Nc2ccc(C)cc2Br)c1C	nan
	CHEMBL1577640	50640	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	348	3	2	2	4.2	CC(=O)c1c(C)[nH]c(C(=O)Nc2ccc(C)cc2Br)c1C	nan
	2868371	50665	12	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	6	2	7	2.5	CCOc1ccccc1NC(=O)CSc1nc(N)c(C#N)cc1C#N	nan
	CHEMBL1577894	50665	12	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	6	2	7	2.5	CCOc1ccccc1NC(=O)CSc1nc(N)c(C#N)cc1C#N	nan
	7207360	50669	9	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	7	1	7	3.4	CCOC(=O)c1ccc(NC(=O)CSc2ccc(-c3ccncc3)nn2)cc1	nan
	CHEMBL1577921	50669	9	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	7	1	7	3.4	CCOC(=O)c1ccc(NC(=O)CSc2ccc(-c3ccncc3)nn2)cc1	nan
	24891931	50749	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	498	8	2	7	0.7	NS(=O)(=O)c1ccc(CCNC(=O)C(=O)c2cn(CC(=O)N3CCOCC3)c3ccccc23)cc1	nan
	CHEMBL1578510	50749	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	498	8	2	7	0.7	NS(=O)(=O)c1ccc(CCNC(=O)C(=O)c2cn(CC(=O)N3CCOCC3)c3ccccc23)cc1	nan
	712274	50787	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	3	3	5	2.2	NC(=O)c1ccc2nc(NC(=O)c3ccc(N)cc3)sc2c1	nan
	CHEMBL1578798	50787	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	3	3	5	2.2	NC(=O)c1ccc2nc(NC(=O)c3ccc(N)cc3)sc2c1	nan
	7416477	50937	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	348	4	1	4	3.5	Cc1cccc(C(=O)OCC(=O)c2cccc(Br)c2)c1O	nan
	CHEMBL1580196	50937	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	348	4	1	4	3.5	Cc1cccc(C(=O)OCC(=O)c2cccc(Br)c2)c1O	nan
	16193583	50966	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	496	10	1	8	3.3	CCCCNC(=O)CSc1nc2ccc(N3CCOCC3)cc2c(=O)n1Cc1ccc(OC)cc1	nan
	CHEMBL1580449	50966	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	496	10	1	8	3.3	CCCCNC(=O)CSc1nc2ccc(N3CCOCC3)cc2c(=O)n1Cc1ccc(OC)cc1	nan
	135421577	51010	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	311	3	2	3	2.0	C=CCN1C(=O)/C(=C/c2cc3ccccc3[nH]2)C(=O)NC1=S	nan
	CHEMBL1580833	51010	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	311	3	2	3	2.0	C=CCN1C(=O)/C(=C/c2cc3ccccc3[nH]2)C(=O)NC1=S	nan
	652265	51065	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	5	1	5	4.1	O=C(Nc1ccc(Oc2ccccc2)cc1)C1CCN(c2ncccn2)CC1	nan
	CHEMBL1581276	51065	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	5	1	5	4.1	O=C(Nc1ccc(Oc2ccccc2)cc1)C1CCN(c2ncccn2)CC1	nan
	4455225	51154	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	9	2	5	3.5	CCOCCCn1c(=S)[nH]c2cc(C(=O)NCCc3ccccc3)ccc2c1=O	nan
	CHEMBL1582016	51154	2	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	9	2	5	3.5	CCOCCCn1c(=S)[nH]c2cc(C(=O)NCCc3ccccc3)ccc2c1=O	nan
	135693216	51404	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	5	2	5	2.9	Cc1cccc(CCNC(=O)Cn2ncc3c4ccccc4nc-3c2O)c1	nan
	CHEMBL1584056	51404	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	5	2	5	2.9	Cc1cccc(CCNC(=O)Cn2ncc3c4ccccc4nc-3c2O)c1	nan
	3662539	51427	7	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	1	4	7	3.1	N#Cc1c(N)nc2c3c(sc(=N)c2c1N)NC(=O)CC3c1c(F)cccc1Cl	nan
	CHEMBL1584309	51427	7	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	1	4	7	3.1	N#Cc1c(N)nc2c3c(sc(=N)c2c1N)NC(=O)CC3c1c(F)cccc1Cl	nan
	24819718	51559	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	1	1	2	4.0	O=C(c1cc2ccccc2cc1O)N1CCCC(C(F)(F)F)C1	nan
	CHEMBL1585344	51559	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	1	1	2	4.0	O=C(c1cc2ccccc2cc1O)N1CCCC(C(F)(F)F)C1	nan
	2112635	51712	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	4	2	6	2.9	Cc1nc(NCc2ccc(S(N)(=O)=O)cc2)c2c(C)c(C)sc2n1	nan
	CHEMBL1586644	51712	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	4	2	6	2.9	Cc1nc(NCc2ccc(S(N)(=O)=O)cc2)c2c(C)c(C)sc2n1	nan
	135441025	51726	13	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	319	3	2	4	3.7	CCCn1c(=O)c(-c2nc3ccccc3[nH]2)c(O)c2ccccc21	nan
	CHEMBL1586724	51726	13	None	-3	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	319	3	2	4	3.7	CCCn1c(=O)c(-c2nc3ccccc3[nH]2)c(O)c2ccccc21	nan
	2158327	51767	10	None	-17	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	5	1	5	3.9	O=C(CSc1ncnc2c1oc1ccccc12)NCc1ccc(F)cc1	nan
	CHEMBL1587044	51767	10	None	-17	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	5	1	5	3.9	O=C(CSc1ncnc2c1oc1ccccc12)NCc1ccc(F)cc1	nan
	20876043	51938	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	446	6	1	8	0.5	COc1cccc(NC(=O)CN(C)S(=O)(=O)c2ccc3c(c2)n(C)c(=O)c(=O)n3C)c1	nan
	CHEMBL1588535	51938	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	446	6	1	8	0.5	COc1cccc(NC(=O)CN(C)S(=O)(=O)c2ccc3c(c2)n(C)c(=O)c(=O)n3C)c1	nan
	16016041	52089	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	358	4	1	4	4.5	COc1ccc(CC(=O)Nc2nc3c(s2)CC(C(C)(C)C)CC3)cc1	nan
	CHEMBL1589883	52089	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	358	4	1	4	4.5	COc1ccc(CC(=O)Nc2nc3c(s2)CC(C(C)(C)C)CC3)cc1	nan
	4671465	52114	14	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	6	2	4	3.3	NC(=O)c1ccc(NC(=O)c2ccc(COc3ccc(F)cc3)o2)cc1	nan
	CHEMBL1590137	52114	14	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	6	2	4	3.3	NC(=O)c1ccc(NC(=O)c2ccc(COc3ccc(F)cc3)o2)cc1	nan
	16009149	52144	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	410	5	1	3	5.5	Cc1ccc(CNC(=O)CSc2c3c(nc4cc(Cl)ccc24)CCCC3)cc1	nan
	CHEMBL1590589	52144	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	410	5	1	3	5.5	Cc1ccc(CNC(=O)CSc2c3c(nc4cc(Cl)ccc24)CCCC3)cc1	nan
	16026741	52152	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	6	0	8	2.8	O=C(COc1ccc(Cl)cc1)OCc1cc(=O)n2nc(C3CC3)sc2n1	nan
	CHEMBL1590675	52152	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	6	0	8	2.8	O=C(COc1ccc(Cl)cc1)OCc1cc(=O)n2nc(C3CC3)sc2n1	nan
	16025957	52158	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	4	1	8	1.6	O=C(NCc1ccc(Cl)cc1)c1cnc2sc(N3CCOCC3)nn2c1=O	nan
	CHEMBL1590760	52158	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	4	1	8	1.6	O=C(NCc1ccc(Cl)cc1)c1cnc2sc(N3CCOCC3)nn2c1=O	nan
	16033877	52159	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	5	2	8	4.0	O=C(NCc1cccs1)c1ccc2c(=O)n3nc(Nc4ccccc4)sc3nc2c1	nan
	CHEMBL1590761	52159	8	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	5	2	8	4.0	O=C(NCc1cccs1)c1ccc2c(=O)n3nc(Nc4ccccc4)sc3nc2c1	nan
	18567961	52176	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	9	2	6	3.3	COc1ccc(C(=O)Nc2nc(CC(=O)NCCc3ccccc3OC)cs2)cc1	nan
	CHEMBL1590928	52176	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	9	2	6	3.3	COc1ccc(C(=O)Nc2nc(CC(=O)NCCc3ccccc3OC)cs2)cc1	nan
	16021437	52203	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	6	2	4	6.6	Cc1cc(Nc2cccc(Cl)c2)nc2ccc(NC(=O)COc3ccc(Cl)cc3)cc12	nan
	CHEMBL1591314	52203	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	6	2	4	6.6	Cc1cc(Nc2cccc(Cl)c2)nc2ccc(NC(=O)COc3ccc(Cl)cc3)cc12	nan
	16030267	52215	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	5	0	4	4.6	Cc1ccc(Cc2nc3ccccc3nc2SCC(=O)N2CCCCC2)cc1	nan
	CHEMBL1591398	52215	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	5	0	4	4.6	Cc1ccc(Cc2nc3ccccc3nc2SCC(=O)N2CCCCC2)cc1	nan
	15988978	52216	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	475	5	1	7	3.9	COc1ccc(NC(=O)Cn2c(=O)n(-c3cccc(C(F)(F)F)c3)c(=O)c3sccc32)cc1	nan
	CHEMBL1591409	52216	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	475	5	1	7	3.9	COc1ccc(NC(=O)Cn2c(=O)n(-c3cccc(C(F)(F)F)c3)c(=O)c3sccc32)cc1	nan
	4905426	52219	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	294	4	1	2	3.4	COc1ccc2cc(C(=O)N(C)Cc3ccccc3)[nH]c2c1	nan
	CHEMBL1591442	52219	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	294	4	1	2	3.4	COc1ccc2cc(C(=O)N(C)Cc3ccccc3)[nH]c2c1	nan
	15989516	52260	3	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	538	9	2	6	4.0	O=C(Cn1c(=O)n(CC2CCC(C(=O)NCCc3ccccc3)CC2)c(=O)c2ccccc21)Nc1ccccc1	nan
	CHEMBL1592027	52260	3	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	538	9	2	6	4.0	O=C(Cn1c(=O)n(CC2CCC(C(=O)NCCc3ccccc3)CC2)c(=O)c2ccccc21)Nc1ccccc1	nan
	15991260	52280	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	4	2	7	1.4	CCn1c(=N)c(C(=O)NCC2CCCO2)cc2c(=O)n3cc(C)ccc3nc21	nan
	CHEMBL1592271	52280	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	4	2	7	1.4	CCn1c(=N)c(C(=O)NCC2CCCO2)cc2c(=O)n3cc(C)ccc3nc21	nan
	16027708	52303	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	461	5	1	7	4.7	CC(C)(C)c1ccc(C(=O)Nc2ccccc2C(=O)OCc2cc(=O)n3ccsc3n2)cc1	nan
	CHEMBL1592618	52303	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	461	5	1	7	4.7	CC(C)(C)c1ccc(C(=O)Nc2ccccc2C(=O)OCc2cc(=O)n3ccsc3n2)cc1	nan
	16027669	52304	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	493	5	1	7	4.9	O=C(Nc1ccccc1C(=O)OCc1cc(=O)n2c3c(sc2n1)CCCC3)c1cccc(Cl)c1	nan
	CHEMBL1592645	52304	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	493	5	1	7	4.9	O=C(Nc1ccccc1C(=O)OCc1cc(=O)n2c3c(sc2n1)CCCC3)c1cccc(Cl)c1	nan
	16024581	52315	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	6	1	5	3.7	Cc1ccc(CNC(=O)Cn2cc(C(=O)c3ccc(F)cc3)c(=O)c3ccc(C)nc32)cc1	nan
	CHEMBL1592799	52315	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	6	1	5	3.7	Cc1ccc(CNC(=O)Cn2cc(C(=O)c3ccc(F)cc3)c(=O)c3ccc(C)nc32)cc1	nan
	16020979	52346	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	8	1	7	4.5	COc1cc(NC(=O)Cn2c(SCc3ccc(F)cc3)nc3cccnc32)cc(OC)c1	nan
	CHEMBL1593212	52346	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	8	1	7	4.5	COc1cc(NC(=O)Cn2c(SCc3ccc(F)cc3)nc3cccnc32)cc(OC)c1	nan
	16012982	52360	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	4	1	3	5.7	Cc1cccc(N(Cc2cc3ccccc3nc2O)C(=O)c2cccc(Cl)c2)c1	nan
	CHEMBL1593385	52360	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	4	1	3	5.7	Cc1cccc(N(Cc2cc3ccccc3nc2O)C(=O)c2cccc(Cl)c2)c1	nan
	5143379	52361	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	6	2	3	5.0	CC(=O)Nc1cc(C(=O)NCc2ccc(F)cc2)ccc1Sc1ccc(F)cc1	nan
	CHEMBL1593424	52361	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	6	2	3	5.0	CC(=O)Nc1cc(C(=O)NCc2ccc(F)cc2)ccc1Sc1ccc(F)cc1	nan
	16322180	52377	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	356	4	1	5	3.7	Cc1nc(SC(C)C(=O)NC2(C#N)CCCCC2)c(C#N)c(C)c1C	nan
	CHEMBL1593705	52377	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	356	4	1	5	3.7	Cc1nc(SC(C)C(=O)NC2(C#N)CCCCC2)c(C#N)c(C)c1C	nan
	16024549	52383	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	475	7	1	6	4.6	CCOc1ccccc1NC(=O)Cn1cc(C(=O)c2ccc(Cl)cc2)c(=O)c2ccc(C)nc21	nan
	CHEMBL1593798	52383	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	475	7	1	6	4.6	CCOc1ccccc1NC(=O)Cn1cc(C(=O)c2ccc(Cl)cc2)c(=O)c2ccc(C)nc21	nan
	16019841	52387	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	457	8	1	7	4.1	CC(C)Cn1c(=O)c2sccc2n2c(CCCC(=O)NCc3ccccc3Cl)nnc12	nan
	CHEMBL1593835	52387	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	457	8	1	7	4.1	CC(C)Cn1c(=O)c2sccc2n2c(CCCC(=O)NCc3ccccc3Cl)nnc12	nan
	16026849	52394	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	6	1	5	3.8	COc1ccc(Cn2ccc3nc(C)c(C(=O)NCc4ccc(F)cc4)cc3c2=O)cc1	nan
	CHEMBL1593965	52394	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	6	1	5	3.8	COc1ccc(Cn2ccc3nc(C)c(C(=O)NCc4ccc(F)cc4)cc3c2=O)cc1	nan
	16024916	52400	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	6	1	5	4.9	CSc1ccc(CCNC(=O)C2CCN(c3nc4ccccc4nc3C(F)(F)F)CC2)cc1	nan
	CHEMBL1594028	52400	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	6	1	5	4.9	CSc1ccc(CCNC(=O)C2CCN(c3nc4ccccc4nc3C(F)(F)F)CC2)cc1	nan
	16024610	52410	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	6	1	5	4.8	CCc1ccc(C(=O)c2cn(CC(=O)Nc3cccc(C)c3C)c3nc(C)ccc3c2=O)cc1	nan
	CHEMBL1594130	52410	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	6	1	5	4.8	CCc1ccc(C(=O)c2cn(CC(=O)Nc3cccc(C)c3C)c3nc(C)ccc3c2=O)cc1	nan
	2140504	52556	20	None	-3	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	344	4	1	6	3.4	N#Cc1cc2c(nc1SCC(=O)Nc1nccs1)CCCCC2	nan
	CHEMBL1595336	52556	20	None	-3	3	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	344	4	1	6	3.4	N#Cc1cc2c(nc1SCC(=O)Nc1nccs1)CCCCC2	nan
	16024587	52639	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	6	1	5	3.4	Cc1ccc2c(=O)c(C(=O)c3ccc(F)cc3)cn(CC(=O)NCc3ccccc3)c2n1	nan
	CHEMBL1596100	52639	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	6	1	5	3.4	Cc1ccc2c(=O)c(C(=O)c3ccc(F)cc3)cn(CC(=O)NCc3ccccc3)c2n1	nan
	865538	52677	7	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	273	3	1	3	4.0	Cc1ccc2nc(NCc3ccccc3)c(C#N)cc2c1	nan
	CHEMBL1596421	52677	7	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	273	3	1	3	4.0	Cc1ccc2nc(NCc3ccccc3)c(C#N)cc2c1	nan
	16008803	52688	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	4	1	4	5.8	CCOc1ccccc1NC(=O)c1cc2c(Cl)nc3ccccc3c2s1	nan
	CHEMBL1596557	52688	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	4	1	4	5.8	CCOc1ccccc1NC(=O)c1cc2c(Cl)nc3ccccc3c2s1	nan
	1191858	52696	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	6	0	6	3.8	COc1ccc(-c2cc(=O)c3cc(OCC(=O)OC(C)C)ccc3o2)cc1	nan
	CHEMBL1596612	52696	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	6	0	6	3.8	COc1ccc(-c2cc(=O)c3cc(OCC(=O)OC(C)C)ccc3o2)cc1	nan
	16011437	52700	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	508	10	1	6	5.8	COc1ccc(Cn2c(SCc3ccc(C(=O)NCCc4ccccc4)cc3)nc3cccnc32)cc1	nan
	CHEMBL1596645	52700	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	508	10	1	6	5.8	COc1ccc(Cn2c(SCc3ccc(C(=O)NCCc4ccccc4)cc3)nc3cccnc32)cc1	nan
	2110721	52719	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	310	3	2	2	3.5	CC(=O)c1c(C)[nH]c(C(=O)Nc2ccc(F)c(F)c2F)c1C	nan
	CHEMBL1596828	52719	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	310	3	2	2	3.5	CC(=O)c1c(C)[nH]c(C(=O)Nc2ccc(F)c(F)c2F)c1C	nan
	15991384	52755	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	4	1	4	6.2	COc1c(C)cccc1C(=O)Nc1ccc(-c2nc3ccccc3s2)c(Cl)c1	nan
	CHEMBL1597164	52755	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	4	1	4	6.2	COc1c(C)cccc1C(=O)Nc1ccc(-c2nc3ccccc3s2)c(Cl)c1	nan
	9397360	52932	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	4	1	8	3.6	CCc1nnc(NC(=O)C2CCN(c3ncnc4sc(C)c(C)c34)CC2)s1	nan
	CHEMBL1598832	52932	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	4	1	8	3.6	CCc1nnc(NC(=O)C2CCN(c3ncnc4sc(C)c(C)c34)CC2)s1	nan
	1873710	52954	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	5	0	5	5.3	CCOc1nc(-c2ccc(C)cc2)ccc1-c1noc(-c2ccccc2F)n1	nan
	CHEMBL1599008	52954	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	5	0	5	5.3	CCOc1nc(-c2ccc(C)cc2)ccc1-c1noc(-c2ccccc2F)n1	nan
	16016553	52974	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	5	1	5	4.1	Cc1cc(C)cc(OCC(=O)Nc2nonc2-c2ccc(Br)cc2)c1	nan
	CHEMBL1599164	52974	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	5	1	5	4.1	Cc1cc(C)cc(OCC(=O)Nc2nonc2-c2ccc(Br)cc2)c1	nan
	16027417	52994	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	483	7	1	8	4.1	Cc1csc2nc(COC(=O)c3cccc(NC(=O)COc4ccccc4Cl)c3)cc(=O)n12	nan
	CHEMBL1599306	52994	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	483	7	1	8	4.1	Cc1csc2nc(COC(=O)c3cccc(NC(=O)COc4ccccc4Cl)c3)cc(=O)n12	nan
	5059359	53062	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	2	0	6	4.4	Cn1c(=O)c2c(-c3ccccc3)n3c4ccccc4nc(-c4ccccc4)c3c2n(C)c1=O	nan
	CHEMBL1599921	53062	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	2	0	6	4.4	Cn1c(=O)c2c(-c3ccccc3)n3c4ccccc4nc(-c4ccccc4)c3c2n(C)c1=O	nan
	16019821	53143	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	6	2	6	3.4	CCOc1ccc(NC(=O)C2CCCN(S(=O)(=O)c3ccc4nc(O)ccc4c3)C2)cc1	nan
	CHEMBL1600701	53143	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	6	2	6	3.4	CCOc1ccc(NC(=O)C2CCCN(S(=O)(=O)c3ccc4nc(O)ccc4c3)C2)cc1	nan
	16021830	53271	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	4	1	4	4.4	CSc1ncc(C(=O)Nc2ccc(F)cc2F)c(-c2ccccc2)n1	nan
	CHEMBL1602038	53271	1	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	4	1	4	4.4	CSc1ncc(C(=O)Nc2ccc(F)cc2F)c(-c2ccccc2)n1	nan
	4197620	53292	15	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	335	3	1	6	2.7	COc1ccc(Cl)cc1NC(=O)c1cnc2sccn2c1=O	nan
	CHEMBL1602236	53292	15	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	335	3	1	6	2.7	COc1ccc(Cl)cc1NC(=O)c1cnc2sccn2c1=O	nan
	16026568	53326	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	4	1	5	4.8	Cc1cc(C)c(NC(=O)C(C)n2c(=O)cc(-c3ccccc3)c3c(C)nn(C)c32)c(C)c1	nan
	CHEMBL1602546	53326	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	4	1	5	4.8	Cc1cc(C)c(NC(=O)C(C)n2c(=O)cc(-c3ccccc3)c3c(C)nn(C)c32)c(C)c1	nan
	1482197	53357	21	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	319	5	0	4	4.0	COc1ccc(C(=O)c2ccc(-c3ccc(OC)cc3)nc2)cc1	nan
	CHEMBL1602835	53357	21	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	319	5	0	4	4.0	COc1ccc(C(=O)c2ccc(-c3ccc(OC)cc3)nc2)cc1	nan
	16023008	53371	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	488	6	1	7	4.1	COc1ccc(-n2nc3c(N4CCC(C(=O)NCc5cccc(F)c5)CC4)nnc(C)c3c2C)cc1	nan
	CHEMBL1602958	53371	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	488	6	1	7	4.1	COc1ccc(-n2nc3c(N4CCC(C(=O)NCc5cccc(F)c5)CC4)nnc(C)c3c2C)cc1	nan
	4077604	53437	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	4	2	5	3.1	O=C(NCC1CCCO1)c1ccc2c(=O)n(-c3ccc(F)cc3)c(=S)[nH]c2c1	nan
	CHEMBL1603522	53437	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	4	2	5	3.1	O=C(NCC1CCCO1)c1ccc2c(=O)n(-c3ccc(F)cc3)c(=S)[nH]c2c1	nan
	16008430	53513	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	503	6	0	6	5.0	COc1ccc(N2CCN(C(=O)CCc3c(C)nc4cc(-c5ccc(Cl)cc5)nn4c3C)CC2)cc1	nan
	CHEMBL1604039	53513	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	503	6	0	6	5.0	COc1ccc(N2CCN(C(=O)CCc3c(C)nc4cc(-c5ccc(Cl)cc5)nn4c3C)CC2)cc1	nan
	2319103	53523	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	556	7	2	6	4.7	CC(=O)Nc1ccc(S(=O)(=O)[N-]c2nc3ccccc3nc2-[n+]2ccc(NC(=O)c3ccc(F)cc3)cc2)cc1	nan
	CHEMBL1604161	53523	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	556	7	2	6	4.7	CC(=O)Nc1ccc(S(=O)(=O)[N-]c2nc3ccccc3nc2-[n+]2ccc(NC(=O)c3ccc(F)cc3)cc2)cc1	nan
	1105833	53582	7	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	2	0	2	5.2	N#Cc1c(-c2cccc(F)c2)cc(-c2ccccc2)nc1Br	nan
	CHEMBL1604724	53582	7	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	2	0	2	5.2	N#Cc1c(-c2cccc(F)c2)cc(-c2ccccc2)nc1Br	nan
	13283806	53695	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	2	0	3	4.2	O=S1(=O)c2ccccc2N(Cc2ccccc2)c2ccccc21	nan
	CHEMBL1605626	53695	0	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	2	0	3	4.2	O=S1(=O)c2ccccc2N(Cc2ccccc2)c2ccccc21	nan
	606829	53776	16	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	301	2	1	2	5.1	Cc1ccc(NC(=O)c2sc3ccccc3c2Cl)cc1	nan
	CHEMBL1606319	53776	16	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	301	2	1	2	5.1	Cc1ccc(NC(=O)c2sc3ccccc3c2Cl)cc1	nan
	2877673	53816	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	6	0	4	4.3	CCCC(=O)N1CCN(c2ccc(C(=O)c3ccc(OC)c(Br)c3)cc2F)CC1	nan
	CHEMBL1606636	53816	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	6	0	4	4.3	CCCC(=O)N1CCN(c2ccc(C(=O)c3ccc(OC)c(Br)c3)cc2F)CC1	nan
	16025505	53880	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	454	5	1	6	4.1	CC(C)c1ccc(NC(=O)CSc2ncc3c(n2)-c2ccccc2N(C)S3(=O)=O)cc1	nan
	CHEMBL1607091	53880	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	454	5	1	6	4.1	CC(C)c1ccc(NC(=O)CSc2ncc3c(n2)-c2ccccc2N(C)S3(=O)=O)cc1	nan
	16019209	53894	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	483	6	1	7	4.2	COc1ccc(Cn2c(=O)c3oc4ccccc4c3n(CC(=O)Nc3c(C)cccc3C)c2=O)cc1	nan
	CHEMBL1607174	53894	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	483	6	1	7	4.2	COc1ccc(Cn2c(=O)c3oc4ccccc4c3n(CC(=O)Nc3c(C)cccc3C)c2=O)cc1	nan
	1166591	53993	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	7	1	5	5.4	COc1ccc(-c2cc(C(F)(F)F)nc(SCCC(=O)Nc3ccccc3F)n2)cc1	nan
	CHEMBL1608012	53993	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	7	1	5	5.4	COc1ccc(-c2cc(C(F)(F)F)nc(SCCC(=O)Nc3ccccc3F)n2)cc1	nan
	939124	54215	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	298	3	1	6	3.6	CC(=O)c1c(C)nc(Nc2nc3ccccc3s2)nc1C	nan
	CHEMBL1609840	54215	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	298	3	1	6	3.6	CC(=O)c1c(C)nc(Nc2nc3ccccc3s2)nc1C	nan
	15989162	54245	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	542	10	2	7	3.8	COc1ccccc1CNC(=O)CCCn1c(=O)c2ccccc2n(CC(=O)Nc2c(C)cc(C)cc2C)c1=O	nan
	CHEMBL1610075	54245	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	542	10	2	7	3.8	COc1ccccc1CNC(=O)CCCn1c(=O)c2ccccc2n(CC(=O)Nc2c(C)cc(C)cc2C)c1=O	nan
	2542807	54282	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	4	1	4	4.2	Cc1cc(C)c(NC(=O)CSc2nc(C)cc(C)c2C#N)c(C)c1	nan
	CHEMBL1610420	54282	13	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	4	1	4	4.2	Cc1cc(C)c(NC(=O)CSc2nc(C)cc(C)c2C#N)c(C)c1	nan
	1192919	54411	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	5	1	4	5.1	COc1ccc(C(=O)c2oc3ccccc3c2NC(=O)c2ccc(F)cc2)cc1	nan
	CHEMBL1611527	54411	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	5	1	4	5.1	COc1ccc(C(=O)c2oc3ccccc3c2NC(=O)c2ccc(F)cc2)cc1	nan
	16024853	54532	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	5	1	4	4.2	O=C(NCCc1ccccc1)C1CCN(c2nc3ccccc3nc2C(F)(F)F)CC1	nan
	CHEMBL1612612	54532	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	5	1	4	4.2	O=C(NCCc1ccccc1)C1CCN(c2nc3ccccc3nc2C(F)(F)F)CC1	nan
	24789826	54780	0	None	-56	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	7	1	4	5.8	CCN(CC)c1ccc(-c2sc(Nc3ccccc3)n[n+]2-c2ccc(F)cc2)cc1	nan
	CHEMBL1307717	54780	0	None	-56	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	7	1	4	5.8	CCN(CC)c1ccc(-c2sc(Nc3ccccc3)n[n+]2-c2ccc(F)cc2)cc1	nan
	CHEMBL1616626	54780	0	None	-56	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	7	1	4	5.8	CCN(CC)c1ccc(-c2sc(Nc3ccccc3)n[n+]2-c2ccc(F)cc2)cc1	nan
	135448704	54973	33	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	281	1	4	4	1.4	N=C(N)Nc1nc(O)c2cc(Br)ccc2n1	nan
	CHEMBL1319156	54973	33	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	281	1	4	4	1.4	N=C(N)Nc1nc(O)c2cc(Br)ccc2n1	nan
	CHEMBL1618027	54973	33	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	281	1	4	4	1.4	N=C(N)Nc1nc(O)c2cc(Br)ccc2n1	nan
	3773369	55428	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	4	1	5	2.9	COc1ccc(CCn2c(S)nc3ccccc3c2=O)cc1	nan
	CHEMBL1483432	55428	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	4	1	5	2.9	COc1ccc(CCn2c(S)nc3ccccc3c2=O)cc1	nan
	CHEMBL1622111	55428	12	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	4	1	5	2.9	COc1ccc(CCn2c(S)nc3ccccc3c2=O)cc1	nan
	6886091	107374	7	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	426	3	1	6	3.2	Cn1c(=O)n(C)c2cc(/C=N/NC(=O)c3cc4cc(Br)ccc4o3)ccc21	nan
	CHEMBL3192586	107374	7	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	426	3	1	6	3.2	Cn1c(=O)n(C)c2cc(/C=N/NC(=O)c3cc4cc(Br)ccc4o3)ccc21	nan
	3221539	107433	4	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	8	0	6	3.2	CCOc1ccc2nc3c(cc2c1)CN(CCOC)/C(=N\CCOC)S3	nan
	CHEMBL3193316	107433	4	None	-2	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	8	0	6	3.2	CCOc1ccc2nc3c(cc2c1)CN(CCOC)/C(=N\CCOC)S3	nan
	9615796	107762	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	3	1	5	2.3	Cn1c(=O)n(C)c2cc(/C=N/NC(=O)c3ccc(Cl)cc3)ccc21	nan
	CHEMBL3197069	107762	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	3	1	5	2.3	Cn1c(=O)n(C)c2cc(/C=N/NC(=O)c3ccc(Cl)cc3)ccc21	nan
	24892226	107852	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	478	8	0	9	2.2	COC(=O)Cn1/c(=N\C(=O)CCS(=O)(=O)c2ccccc2)sc2c(OC)ccc(OC)c21	nan
	CHEMBL3197975	107852	9	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	478	8	0	9	2.2	COC(=O)Cn1/c(=N\C(=O)CCS(=O)(=O)c2ccccc2)sc2c(OC)ccc(OC)c21	nan
	6341421	107904	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	291	3	1	3	3.6	CCCn1c(C)cs/c1=N\C(=S)Nc1ccccc1	nan
	CHEMBL3198424	107904	6	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	291	3	1	3	3.6	CCCn1c(C)cs/c1=N\C(=S)Nc1ccccc1	nan
	6065517	108316	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	253	5	2	4	1.1	CC(C)NC(=O)CC(=O)N/N=C/c1cccs1	nan
	CHEMBL3209441	108316	4	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	253	5	2	4	1.1	CC(C)NC(=O)CC(=O)N/N=C/c1cccs1	nan
	135485035	108466	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	3	1	5	3.9	COc1ccc(Cl)cc1/N=C/c1c(O)oc2ccccc2c1=O	nan
	CHEMBL3211560	108466	10	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	3	1	5	3.9	COc1ccc(Cl)cc1/N=C/c1c(O)oc2ccccc2c1=O	nan
	17584634	108669	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	4	0	5	2.7	COc1ccc(C(=O)/N=C2\SC3CS(=O)(=O)CC3N2Cc2ccc(F)cc2)cc1	nan
	CHEMBL3214247	108669	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	4	0	5	2.7	COc1ccc(C(=O)/N=C2\SC3CS(=O)(=O)CC3N2Cc2ccc(F)cc2)cc1	nan
	6869045	112101	4	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	301	7	2	5	1.8	NCCCCCC(=O)N/N=C/c1coc2ccccc2c1=O	nan
	CHEMBL3194304	112101	4	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	301	7	2	5	1.8	NCCCCCC(=O)N/N=C/c1coc2ccccc2c1=O	nan
	CHEMBL3301898	112101	4	None	-1	2	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	301	7	2	5	1.8	NCCCCCC(=O)N/N=C/c1coc2ccccc2c1=O	nan
	658981	116563	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	255	2	1	5	2.7	CCOC(=O)c1c(N)sc(=S)c2c1CCC2	nan
	CHEMBL3392035	116563	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	255	2	1	5	2.7	CCOC(=O)c1c(N)sc(=S)c2c1CCC2	nan
	2241546	119905	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	295	3	1	4	3.8	Cc1ccc(C(=O)Nc2nc(-c3ccccc3)ns2)cc1	nan
	CHEMBL353651	119905	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	295	3	1	4	3.8	Cc1ccc(C(=O)Nc2nc(-c3ccccc3)ns2)cc1	nan
	878295	172642	29	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	255	1	1	1	3.8	O=c1cc(-c2ccccc2)c2cc(Cl)ccc2[nH]1	nan
	CHEMBL452292	172642	29	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	255	1	1	1	3.8	O=c1cc(-c2ccccc2)c2cc(Cl)ccc2[nH]1	nan
	16010872	197393	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	7	1	7	4.4	COc1cc2nc(NCCC(C)C)n3nc(-c4ccccc4)nc3c2cc1OC	nan
	CHEMBL587492	197393	7	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	7	1	7	4.4	COc1cc2nc(NCCC(C)C)n3nc(-c4ccccc4)nc3c2cc1OC	nan
	16017892	197451	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	4	1	6	3.4	CCOc1ccc(NC(=O)c2sc3nc4n(c(=O)c3c2C)CCC4)cc1	nan
	CHEMBL589232	197451	5	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	4	1	6	3.4	CCOc1ccc(NC(=O)c2sc3nc4n(c(=O)c3c2C)CCC4)cc1	nan
	1370186	197998	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	358	5	1	4	4.8	Cc1ccccc1OCC(=O)Nc1ccc(-c2nc3ccccc3o2)cc1	nan
	CHEMBL593119	197998	11	None	-	1	Human	4.5	pPotency	=	4.5	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	358	5	1	4	4.8	Cc1ccccc1OCC(=O)Nc1ccc(-c2nc3ccccc3o2)cc1	nan
	372	58	96	None	-107	5	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	301	2	4	9	-1.3	OC[C@H]1O[C@H]([C@@H]([C@@H]1O)O)n1cnc2c1nc(Cl)nc2N	nan
	8974	58	96	None	-107	5	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	301	2	4	9	-1.3	OC[C@H]1O[C@H]([C@@H]([C@@H]1O)O)n1cnc2c1nc(Cl)nc2N	nan
	CHEMBL285819	58	96	None	-107	5	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	301	2	4	9	-1.3	OC[C@H]1O[C@H]([C@@H]([C@@H]1O)O)n1cnc2c1nc(Cl)nc2N	nan
	16019683	23875	0	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	6	1	7	2.6	Cc1ccc(CNC(=O)CCCc2nnc3n(C)c(=O)c4sccc4n23)cc1	nan
	CHEMBL1338399	23875	0	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	6	1	7	2.6	Cc1ccc(CNC(=O)CCCc2nnc3n(C)c(=O)c4sccc4n23)cc1	nan
	3486944	24797	8	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	2	0	4	2.5	Cc1cc(C=C2C(=O)N(C)C(=O)N(C)C2=O)c(C)n1-c1ccccc1	nan
	CHEMBL1346519	24797	8	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	2	0	4	2.5	Cc1cc(C=C2C(=O)N(C)C(=O)N(C)C2=O)c(C)n1-c1ccccc1	nan
	665622	29939	7	None	3	2	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	5	1	11	2.8	CC1(C)Cc2c(sc3c2c2ncnn2c2nnc(SCC(=O)NCc4ccco4)n32)CO1	nan
	CHEMBL1390005	29939	7	None	3	2	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	5	1	11	2.8	CC1(C)Cc2c(sc3c2c2ncnn2c2nnc(SCC(=O)NCc4ccco4)n32)CO1	nan
	16019552	34965	11	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	5	1	8	4.1	Cc1ccc(CNc2nc3c(S(=O)(=O)c4ccccc4)nnn3c3ccsc23)cc1	nan
	CHEMBL1435107	34965	11	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	5	1	8	4.1	Cc1ccc(CNc2nc3c(S(=O)(=O)c4ccccc4)nnn3c3ccsc23)cc1	nan
	665286	35352	9	None	3	2	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	483	6	1	11	3.2	CCC1(C)Cc2c(sc3c2c2ncnn2c2nnc(SCC(=O)NCc4ccco4)n32)CO1	nan
	CHEMBL1439367	35352	9	None	3	2	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	483	6	1	11	3.2	CCC1(C)Cc2c(sc3c2c2ncnn2c2nnc(SCC(=O)NCc4ccco4)n32)CO1	nan
	2054021	35576	15	None	1	2	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	4	1	7	3.6	O=C(CSc1ncnc2c1oc1ccccc12)Nc1nccs1	nan
	CHEMBL1441380	35576	15	None	1	2	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	4	1	7	3.6	O=C(CSc1ncnc2c1oc1ccccc12)Nc1nccs1	nan
	1395606	35614	9	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	5	1	5	4.7	CCOc1ccc(-n2nc3ccc(NC(=O)c4ccc(C)cc4C)cc3n2)cc1	nan
	CHEMBL1441729	35614	9	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	5	1	5	4.7	CCOc1ccc(-n2nc3ccc(NC(=O)c4ccc(C)cc4C)cc3n2)cc1	nan
	997264	38632	5	None	1	2	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	5	2	5	2.9	Cc1ccc2cc(C#N)c(SCC(=O)NNC(=O)Cc3ccccc3)nc2c1	nan
	CHEMBL1467097	38632	5	None	1	2	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	5	2	5	2.9	Cc1ccc2cc(C#N)c(SCC(=O)NNC(=O)Cc3ccccc3)nc2c1	nan
	1552186	39292	17	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	530	5	1	4	6.8	Cc1ccc2nc(-c3ccc(NC(=O)COc4ccc(Br)cc4Br)cc3)sc2c1	nan
	CHEMBL1472916	39292	17	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	530	5	1	4	6.8	Cc1ccc2nc(-c3ccc(NC(=O)COc4ccc(Br)cc4Br)cc3)sc2c1	nan
	16009715	41706	11	None	1	2	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	4	1	5	4.7	Fc1ccc(-c2nnn3c2nc(NCc2ccccc2)c2ccccc23)cc1	nan
	CHEMBL1494680	41706	11	None	1	2	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	4	1	5	4.7	Fc1ccc(-c2nnn3c2nc(NCc2ccccc2)c2ccccc23)cc1	nan
	16018178	47987	5	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	5	1	4	5.5	Cc1ccc(CNC(=O)c2oc3c(c2C)-c2nn(Cc4ccc(Cl)cc4)cc2CC3)cc1	nan
	CHEMBL1552994	47987	5	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	5	1	4	5.5	Cc1ccc(CNC(=O)c2oc3c(c2C)-c2nn(Cc4ccc(Cl)cc4)cc2CC3)cc1	nan
	15991072	52142	5	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	3	1	4	6.3	O=C(Nc1ccc2oc(-c3ccc(Br)cc3)nc2c1)c1cc2ccccc2o1	nan
	CHEMBL1590554	52142	5	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	3	1	4	6.3	O=C(Nc1ccc2oc(-c3ccc(Br)cc3)nc2c1)c1cc2ccccc2o1	nan
	2988582	52330	14	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	363	3	1	4	5.1	Cc1cc(-c2nc3ncccc3o2)ccc1NC(=O)c1ccc(Cl)cc1	nan
	CHEMBL1592961	52330	14	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	363	3	1	4	5.1	Cc1cc(-c2nc3ncccc3o2)ccc1NC(=O)c1ccc(Cl)cc1	nan
	15988483	52393	5	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	400	4	2	4	3.7	CC(=O)c1ccc(NC(=O)c2cc3c([nH]c2=O)CC(c2ccccc2)CC3=O)cc1	nan
	CHEMBL1593961	52393	5	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	400	4	2	4	3.7	CC(=O)c1ccc(NC(=O)c2cc3c([nH]c2=O)CC(c2ccccc2)CC3=O)cc1	nan
	1367050	53700	12	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	7	1	6	3.8	CCOc1ccc(-n2nc3ccc(NC(=O)COc4ccccc4)cc3n2)cc1	nan
	CHEMBL1605697	53700	12	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	7	1	6	3.8	CCOc1ccc(-n2nc3ccc(NC(=O)COc4ccccc4)cc3n2)cc1	nan
	4429605	71350	12	None	-1	2	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	6	0	7	3.1	CCOC(=O)c1s/c(=N\C(=O)c2ccc(S(=O)(=O)N(C)c3ccccc3)cc2)n(C)c1C	nan
	CHEMBL1964939	71350	12	None	-1	2	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	6	0	7	3.1	CCOC(=O)c1s/c(=N\C(=O)c2ccc(S(=O)(=O)N(C)c3ccccc3)cc2)n(C)c1C	nan
	16010338	5800	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	472	7	2	8	2.9	CCc1ccc(S(=O)(=O)c2nnn3c2nc(NCCNC(C)=O)c2cc(Cl)ccc23)cc1	nan
	CHEMBL1079456	5800	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	472	7	2	8	2.9	CCc1ccc(S(=O)(=O)c2nnn3c2nc(NCCNC(C)=O)c2cc(Cl)ccc23)cc1	nan
	135446757	7970	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	326	2	1	2	3.9	O=c1[nH]c(/C=C/c2ccc(Br)cc2)nc2ccccc12	nan
	CHEMBL1091028	7970	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	326	2	1	2	3.9	O=c1[nH]c(/C=C/c2ccc(Br)cc2)nc2ccccc12	nan
	250997	10390	3	None	-12	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	398	7	2	10	3.5	COc1cc(SSc2cc(OC)cc([N+](=O)[O-])c2N)c(N)c([N+](=O)[O-])c1	nan
	CHEMBL116548	10390	3	None	-12	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	398	7	2	10	3.5	COc1cc(SSc2cc(OC)cc([N+](=O)[O-])c2N)c(N)c([N+](=O)[O-])c1	nan
	16019609	10512	10	None	-223	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	5	1	8	4.7	Cc1ccc(S(=O)(=O)c2nnn3c2nc(NC(C)c2ccccc2)c2sccc23)cc1	nan
	CHEMBL1170098	10512	10	None	-223	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	5	1	8	4.7	Cc1ccc(S(=O)(=O)c2nnn3c2nc(NC(C)c2ccccc2)c2sccc23)cc1	nan
	16019288	10591	7	None	-234	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	4	1	8	4.2	O=S(=O)(c1cccc(Cl)c1)c1nnn2c1nc(NC1CCCC1)c1sccc12	nan
	CHEMBL1170696	10591	7	None	-234	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	4	1	8	4.2	O=S(=O)(c1cccc(Cl)c1)c1nnn2c1nc(NC1CCCC1)c1sccc12	nan
	16019546	10610	6	None	-676	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	5	1	8	3.8	O=S(=O)(c1ccccc1)c1nnn2c1nc(NCc1ccccc1)c1sccc12	nan
	CHEMBL1170891	10610	6	None	-676	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	5	1	8	3.8	O=S(=O)(c1ccccc1)c1nnn2c1nc(NCc1ccccc1)c1sccc12	nan
	16019576	10796	6	None	-1995	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	5	1	9	3.8	O=S(=O)(c1ccccc1)c1nnn2c1nc(NCc1cccs1)c1sccc12	nan
	CHEMBL1172726	10796	6	None	-1995	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	5	1	9	3.8	O=S(=O)(c1ccccc1)c1nnn2c1nc(NCc1cccs1)c1sccc12	nan
	7246142	10821	9	None	-85	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	4	1	8	3.6	CC(C)Nc1nc2c(S(=O)(=O)c3cccc(Cl)c3)nnn2c2ccsc12	nan
	CHEMBL1172934	10821	9	None	-85	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	4	1	8	3.6	CC(C)Nc1nc2c(S(=O)(=O)c3cccc(Cl)c3)nnn2c2ccsc12	nan
	747391	15489	17	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	5	1	6	3.8	CCOC(=O)c1sc(NC(=O)c2ccco2)nc1-c1ccccc1	nan
	CHEMBL1222145	15489	17	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	5	1	6	3.8	CCOC(=O)c1sc(NC(=O)c2ccco2)nc1-c1ccccc1	nan
	5309696	19358	1	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	5	1	6	2.8	CCn1c(=O)cc(OCC(=O)Nc2nc(C)cs2)c2ccccc21	nan
	CHEMBL1299766	19358	1	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	5	1	6	2.8	CCn1c(=O)cc(OCC(=O)Nc2nc(C)cs2)c2ccccc21	nan
	1716419	19433	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	6	1	5	4.7	CCCCNC(=O)c1nn2c(C(F)(F)F)cc(-c3ccc(OC)cc3)nc2c1Br	nan
	CHEMBL1300444	19433	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	6	1	5	4.7	CCCCNC(=O)c1nn2c(C(F)(F)F)cc(-c3ccc(OC)cc3)nc2c1Br	nan
	135468422	19459	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	498	7	2	9	4.4	COc1ccc(NC(=O)CSc2nc3nnc(C)c-3c(N)n2-c2ccc(Cl)c(C)c2)cc1OC	nan
	CHEMBL1300619	19459	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	498	7	2	9	4.4	COc1ccc(NC(=O)CSc2nc3nnc(C)c-3c(N)n2-c2ccc(Cl)c(C)c2)cc1OC	nan
	5112617	19611	6	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	325	4	3	4	2.2	CC(C)CC(=O)NC(=S)Nc1sc2c(c1C(N)=O)CCC2	nan
	CHEMBL1301780	19611	6	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	325	4	3	4	2.2	CC(C)CC(=O)NC(=S)Nc1sc2c(c1C(N)=O)CCC2	nan
	1440349	19646	4	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	4	1	3	5.4	Cc1cc2cc3c(cc2nc1SCC(=O)Nc1c(C)cccc1C)CCC3	nan
	CHEMBL1302141	19646	4	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	4	1	3	5.4	Cc1cc2cc3c(cc2nc1SCC(=O)Nc1c(C)cccc1C)CCC3	nan
	648939	19648	4	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	5	1	5	3.1	Cc1cc(C)c2cc(C#N)c(SCC(=O)NCC3CCCO3)nc2c1	nan
	CHEMBL1302172	19648	4	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	5	1	5	3.1	Cc1cc(C)c2cc(C#N)c(SCC(=O)NCC3CCCO3)nc2c1	nan
	3221134	19690	4	None	-5	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	6	1	6	4.0	COCCN(Cc1cc2cc(C)ccc2n2nnnc12)C(S)=Nc1ccccc1C	nan
	CHEMBL1302436	19690	4	None	-5	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	6	1	6	4.0	COCCN(Cc1cc2cc(C)ccc2n2nnnc12)C(S)=Nc1ccccc1C	nan
	1864418	19692	8	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	5	1	6	3.5	CC(C)Cc1nc2sc3c(SCC(N)=O)ncnc3c2c2c1CCC2	nan
	CHEMBL1302453	19692	8	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	5	1	6	3.5	CC(C)Cc1nc2sc3c(SCC(N)=O)ncnc3c2c2c1CCC2	nan
	22334119	19709	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	490	8	2	7	2.6	COc1ccc(-n2nc(C(=O)NCC(=O)NCc3ccc(F)cc3)c3ccccc3c2=O)cc1OC	nan
	CHEMBL1302552	19709	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	490	8	2	7	2.6	COc1ccc(-n2nc(C(=O)NCC(=O)NCc3ccc(F)cc3)c3ccccc3c2=O)cc1OC	nan
	1173246	19873	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	5	2	6	4.2	Cc1ccc(C)c2c1cc(C)c1nnc(SCC(=O)Nc3cccc(C(=O)O)c3)n12	nan
	CHEMBL1303849	19873	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	5	2	6	4.2	Cc1ccc(C)c2c1cc(C)c1nnc(SCC(=O)Nc3cccc(C(=O)O)c3)n12	nan
	135455179	19992	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	297	3	1	4	3.0	Cc1cccc(NC2=NC(=O)C(Cc3ccccc3)S2)n1	nan
	135480855	19992	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	297	3	1	4	3.0	Cc1cccc(NC2=NC(=O)C(Cc3ccccc3)S2)n1	nan
	135554164	19992	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	297	3	1	4	3.0	Cc1cccc(NC2=NC(=O)C(Cc3ccccc3)S2)n1	nan
	CHEMBL1304888	19992	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	297	3	1	4	3.0	Cc1cccc(NC2=NC(=O)C(Cc3ccccc3)S2)n1	nan
	16188302	20073	6	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	3	1	4	5.4	CCN(C(=O)c1cc2c(O)nc3ccc(C)cc3c2s1)c1cccc(C)c1	nan
	CHEMBL1305636	20073	6	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	3	1	4	5.4	CCN(C(=O)c1cc2c(O)nc3ccc(C)cc3c2s1)c1cccc(C)c1	nan
	3612019	20131	11	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	306	2	2	4	2.5	O=C(Nc1ccc2c(c1)C(=O)NC2=O)c1ccc(Cl)s1	nan
	CHEMBL1305985	20131	11	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	306	2	2	4	2.5	O=C(Nc1ccc2c(c1)C(=O)NC2=O)c1ccc(Cl)s1	nan
	4243407	20293	9	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	510	5	1	7	4.8	CC1(C)Cc2nc3sc4c(=O)n(CC(=O)NC(c5ccccc5)c5ccccc5)cnc4c3cc2CO1	nan
	CHEMBL1307313	20293	9	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	510	5	1	7	4.8	CC1(C)Cc2nc3sc4c(=O)n(CC(=O)NC(c5ccccc5)c5ccccc5)cnc4c3cc2CO1	nan
	664182	20338	9	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	6	1	7	4.9	CC(C)c1nc2sc3c(SCC(=O)NCc4ccco4)ncnc3c2c2c1CCC2	nan
	CHEMBL1307669	20338	9	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	6	1	7	4.9	CC(C)c1nc2sc3c(SCC(=O)NCc4ccco4)ncnc3c2c2c1CCC2	nan
	2823681	20449	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	2	2	1	4.9	Cc1cc(C)c2[nH]c(C(=O)Nc3ccc(F)cc3Br)cc2c1	nan
	CHEMBL1308537	20449	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	2	2	1	4.9	Cc1cc(C)c2[nH]c(C(=O)Nc3ccc(F)cc3Br)cc2c1	nan
	135443911	20463	17	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	363	4	1	6	3.5	COc1ccc(N2CC(=O)C(c3nc(-c4ccccc4)cs3)=C2N)cc1	nan
	CHEMBL1308652	20463	17	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	363	4	1	6	3.5	COc1ccc(N2CC(=O)C(c3nc(-c4ccccc4)cs3)=C2N)cc1	nan
	7206305	20536	3	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	5	1	8	2.9	Cc1cc(NC(=O)CSc2ccc(-c3ccc4c(c3)OCO4)nn2)no1	nan
	CHEMBL1309267	20536	3	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	5	1	8	2.9	Cc1cc(NC(=O)CSc2ccc(-c3ccc4c(c3)OCO4)nn2)no1	nan
	546665	20662	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	325	2	1	5	3.0	CC(C)(C)S(=O)(=O)c1cnc(-c2ccc(Cl)cc2)nc1N	nan
	CHEMBL1310343	20662	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	325	2	1	5	3.0	CC(C)(C)S(=O)(=O)c1cnc(-c2ccc(Cl)cc2)nc1N	nan
	54693834	20747	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	356	3	2	5	2.9	CC1CCc2cc(F)cc3c(O)c(C(=O)NCc4ccco4)c(=O)n1c23	nan
	CHEMBL1311072	20747	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	356	3	2	5	2.9	CC1CCc2cc(F)cc3c(O)c(C(=O)NCc4ccco4)c(=O)n1c23	nan
	16746300	20770	0	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	618	8	0	8	6.1	COc1cc(OC)c2c(-c3ccccc3)cc(=O)oc2c1C(CC(=O)N1CCN(c2ccccc2)CC1)c1ccc2c(c1)OCO2	nan
	CHEMBL1311273	20770	0	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	618	8	0	8	6.1	COc1cc(OC)c2c(-c3ccccc3)cc(=O)oc2c1C(CC(=O)N1CCN(c2ccccc2)CC1)c1ccc2c(c1)OCO2	nan
	3413238	20772	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	3	2	7	2.8	NS(=O)(=O)c1ccc2nc(NC(=O)c3ccc4ncsc4c3)sc2c1	nan
	CHEMBL1311288	20772	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	3	2	7	2.8	NS(=O)(=O)c1ccc2nc(NC(=O)c3ccc4ncsc4c3)sc2c1	nan
	245201	20786	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	214	3	1	7	0.9	CNc1nc(SC)n(C)c(=O)c1N=O	nan
	CHEMBL1311401	20786	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	214	3	1	7	0.9	CNc1nc(SC)n(C)c(=O)c1N=O	nan
	16194626	20835	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	7	1	6	2.6	COc1ccc(N2CCN(C(c3cccs3)C(C)NS(C)(=O)=O)CC2)cc1	nan
	CHEMBL1311746	20835	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	7	1	6	2.6	COc1ccc(N2CCN(C(c3cccs3)C(C)NS(C)(=O)=O)CC2)cc1	nan
	3586870	20946	14	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	252	3	0	4	3.4	COc1ccc(Oc2cnc3ccccc3n2)cc1	nan
	CHEMBL1312526	20946	14	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	252	3	0	4	3.4	COc1ccc(Oc2cnc3ccccc3n2)cc1	nan
	645988	20975	9	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	5	1	5	4.3	O=C(CSc1nc2c(c(C(F)(F)F)n1)CCc1ccccc1-2)NCc1ccco1	nan
	CHEMBL1312719	20975	9	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	5	1	5	4.3	O=C(CSc1nc2c(c(C(F)(F)F)n1)CCc1ccccc1-2)NCc1ccco1	nan
	660699	21049	11	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	7	2	7	3.6	N#Cc1c(N)nc(SCC(=O)NCCc2ccccc2)c(C#N)c1-c1cccs1	nan
	CHEMBL1313254	21049	11	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	7	2	7	3.6	N#Cc1c(N)nc(SCC(=O)NCCc2ccccc2)c(C#N)c1-c1cccs1	nan
	6619041	21051	7	None	-6	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	502	9	2	8	3.2	CCOc1ccc(NC(=O)CNC(=O)c2nn(-c3ccc(OC)c(OC)c3)c(=O)c3ccccc23)cc1	nan
	CHEMBL1313270	21051	7	None	-6	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	502	9	2	8	3.2	CCOc1ccc(NC(=O)CNC(=O)c2nn(-c3ccc(OC)c(OC)c3)c(=O)c3ccccc23)cc1	nan
	2731590	21091	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	1	1	5	2.8	O=c1c2ccccc2[nH]c(=S)n1-c1ccc2c(c1)OCCO2	nan
	CHEMBL1313595	21091	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	1	1	5	2.8	O=c1c2ccccc2[nH]c(=S)n1-c1ccc2c(c1)OCCO2	nan
	11957277	21108	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	7	0	8	3.9	O=[N+]([O-])C(/C=C(\Cl)[N+](=O)[O-])=C1N(Cc2ccc(Cl)nc2)CCN1Cc1ccc(Cl)nc1	nan
	CHEMBL1313693	21108	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	7	0	8	3.9	O=[N+]([O-])C(/C=C(\Cl)[N+](=O)[O-])=C1N(Cc2ccc(Cl)nc2)CCN1Cc1ccc(Cl)nc1	nan
	16012576	21168	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	6	1	7	4.1	COc1cc(NC(=O)CCc2c(C)nc3c4c(C)cc(C)nc4nn3c2C)cc(OC)c1	nan
	CHEMBL1314269	21168	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	6	1	7	4.1	COc1cc(NC(=O)CCc2c(C)nc3c4c(C)cc(C)nc4nn3c2C)cc(OC)c1	nan
	16020367	21174	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	6	1	8	4.4	COC(=O)c1ccccc1NC(=O)c1cc2c(-c3ccc(OC)c(OC)c3)nn(C)c2s1	nan
	CHEMBL1314309	21174	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	6	1	8	4.4	COC(=O)c1ccccc1NC(=O)c1cc2c(-c3ccc(OC)c(OC)c3)nn(C)c2s1	nan
	16009631	21177	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	461	6	1	7	4.5	COc1ccc(C(=O)Nc2cccc(OCc3cc(=O)n4c5c(sc4n3)CCCC5)c2)cc1	nan
	CHEMBL1314331	21177	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	461	6	1	7	4.5	COc1ccc(C(=O)Nc2cccc(OCc3cc(=O)n4c5c(sc4n3)CCCC5)c2)cc1	nan
	16008545	21178	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	5	0	6	4.3	COc1ccc(C(=O)c2cn(Cc3cccc(C)c3)c3cc4c(cc3c2=O)OCO4)cc1	nan
	CHEMBL1314337	21178	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	5	0	6	4.3	COc1ccc(C(=O)c2cn(Cc3cccc(C)c3)c3cc4c(cc3c2=O)OCO4)cc1	nan
	16018962	21183	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	5	1	5	3.6	O=C(NCc1ccccc1)c1ccc(Cn2c(=O)c3cccn3c3cccnc32)cc1	nan
	CHEMBL1314402	21183	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	5	1	5	3.6	O=C(NCc1ccccc1)c1ccc(Cn2c(=O)c3cccn3c3cccnc32)cc1	nan
	16026094	21194	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	4	1	7	3.1	CC(C)c1ccc(NC(=O)c2cnc3sc(N4CCCC4)nn3c2=O)cc1	nan
	CHEMBL1314533	21194	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	4	1	7	3.1	CC(C)c1ccc(NC(=O)c2cnc3sc(N4CCCC4)nn3c2=O)cc1	nan
	2152595	21208	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	4	0	7	2.9	COC(=O)c1ccc2c(c1)s/c(=N/C(=O)c1ccc(S(=O)(=O)N3CCCCC3)cc1)n2C	nan
	CHEMBL1314815	21208	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	4	0	7	2.9	COC(=O)c1ccc2c(c1)s/c(=N/C(=O)c1ccc(S(=O)(=O)N3CCCCC3)cc1)n2C	nan
	135437061	21209	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	6	3	6	3.9	Cc1ccc(-n2c(SCC(=O)NCc3ccccc3)nc3[nH]nc(C)c3c2=N)cc1Cl	nan
	CHEMBL1314816	21209	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	6	3	6	3.9	Cc1ccc(-n2c(SCC(=O)NCc3ccccc3)nc3[nH]nc(C)c3c2=N)cc1Cl	nan
	16019424	21214	3	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	4	0	8	4.5	CC1CCCN(c2nc3c(S(=O)(=O)c4ccc(C(C)C)cc4)nnn3c3ccsc23)C1	nan
	CHEMBL1314919	21214	3	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	4	0	8	4.5	CC1CCCN(c2nc3c(S(=O)(=O)c4ccc(C(C)C)cc4)nnn3c3ccsc23)C1	nan
	16010115	21218	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	4	1	5	2.8	Cc1ccc(CNC(=O)C2CCN(c3nc4ccccc4n(C)c3=O)CC2)cc1	nan
	CHEMBL1314966	21218	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	4	1	5	2.8	Cc1ccc(CNC(=O)C2CCN(c3nc4ccccc4n(C)c3=O)CC2)cc1	nan
	16020210	21223	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	576	8	2	8	4.0	CCc1ccc(NC(=O)Cn2c(=O)n(-c3ccccc3)c(=O)c3ccc(C(=O)NCc4ccc5c(c4)OCO5)cc32)cc1	nan
	CHEMBL1315042	21223	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	576	8	2	8	4.0	CCc1ccc(NC(=O)Cn2c(=O)n(-c3ccccc3)c(=O)c3ccc(C(=O)NCc4ccc5c(c4)OCO5)cc32)cc1	nan
	16021834	21235	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	4	1	4	4.7	CSc1ncc(C(=O)Nc2c(C)cccc2C)c(-c2ccccc2)n1	nan
	CHEMBL1315205	21235	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	4	1	4	4.7	CSc1ncc(C(=O)Nc2c(C)cccc2C)c(-c2ccccc2)n1	nan
	3516704	21238	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	467	10	1	7	4.4	CCOCCCn1c(SCC(=O)NCc2ccccc2)nc2c(sc3ccccc32)c1=O	nan
	CHEMBL1315294	21238	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	467	10	1	7	4.4	CCOCCCn1c(SCC(=O)NCc2ccccc2)nc2c(sc3ccccc32)c1=O	nan
	16009766	21254	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	440	6	2	5	6.1	CCOc1ccc(NC(=O)c2oc3ccccc3c2NC(=O)c2cc3ccccc3o2)cc1	nan
	CHEMBL1315409	21254	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	440	6	2	5	6.1	CCOc1ccc(NC(=O)c2oc3ccccc3c2NC(=O)c2cc3ccccc3o2)cc1	nan
	16018863	21261	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	5	1	5	3.8	O=C(CCCn1c(=O)c2cccn2c2cccnc21)Nc1ccccc1Br	nan
	CHEMBL1315473	21261	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	5	1	5	3.8	O=C(CCCn1c(=O)c2cccn2c2cccnc21)Nc1ccccc1Br	nan
	16026940	21279	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	6	0	9	3.3	Cc1cccc(OCC(=O)OCc2cc(=O)n3nc(-c4cccs4)sc3n2)c1	nan
	CHEMBL1315714	21279	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	6	0	9	3.3	Cc1cccc(OCC(=O)OCc2cc(=O)n3nc(-c4cccs4)sc3n2)c1	nan
	2808363	21301	21	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	286	3	1	5	2.7	COC(=O)c1sccc1NC(=O)c1ccc(C#N)cc1	nan
	CHEMBL1315955	21301	21	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	286	3	1	5	2.7	COC(=O)c1sccc1NC(=O)c1ccc(C#N)cc1	nan
	16019191	21315	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	6	1	2	5.2	O=C(CCc1cn(Cc2ccc(F)cc2)c2ccccc12)NC1CCCCC1	nan
	CHEMBL1316117	21315	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	6	1	2	5.2	O=C(CCc1cn(Cc2ccc(F)cc2)c2ccccc12)NC1CCCCC1	nan
	16031991	21320	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	7	1	8	4.1	CCOC(=O)c1ccc(NC(=O)CSc2ccc(-c3sc(C)nc3C)nn2)cc1	nan
	CHEMBL1316148	21320	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	7	1	8	4.1	CCOC(=O)c1ccc(NC(=O)CSc2ccc(-c3sc(C)nc3C)nn2)cc1	nan
	2135282	21321	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	500	8	1	8	4.0	CCOc1ccc(NC(=O)Cn2cc(C(=O)c3ccc(OC)cc3)c(=O)c3cc4c(cc32)OCO4)cc1	nan
	CHEMBL1316149	21321	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	500	8	1	8	4.0	CCOc1ccc(NC(=O)Cn2cc(C(=O)c3ccc(OC)cc3)c(=O)c3cc4c(cc32)OCO4)cc1	nan
	16008335	21326	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	498	6	2	6	4.4	O=C(Nc1ccc(C(F)(F)F)cc1)C1CCC(CNS(=O)(=O)c2cccc3nsnc23)CC1	nan
	CHEMBL1316232	21326	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	498	6	2	6	4.4	O=C(Nc1ccc(C(F)(F)F)cc1)C1CCC(CNS(=O)(=O)c2cccc3nsnc23)CC1	nan
	16034305	21338	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	480	7	1	5	4.5	CC(C)CCNC(=O)c1cc(-c2cccnc2)nc2ccc(S(=O)(=O)N3CCC(C)CC3)cc12	nan
	CHEMBL1316467	21338	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	480	7	1	5	4.5	CC(C)CCNC(=O)c1cc(-c2cccnc2)nc2ccc(S(=O)(=O)N3CCC(C)CC3)cc12	nan
	3162808	21342	15	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	4	0	6	4.8	COc1ccc(C2CC(=O)c3cnc4c(-c5ccc(F)cc5)c(C)nn4c3C2)cc1OC	nan
	CHEMBL1316500	21342	15	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	4	0	6	4.8	COc1ccc(C2CC(=O)c3cnc4c(-c5ccc(F)cc5)c(C)nn4c3C2)cc1OC	nan
	3674872	21343	14	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	6	1	8	3.0	CCn1c(SCC(=O)Nc2ccccc2C(=O)OC)nc2ccsc2c1=O	nan
	CHEMBL1316511	21343	14	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	6	1	8	3.0	CCn1c(SCC(=O)Nc2ccccc2C(=O)OC)nc2ccsc2c1=O	nan
	7223037	21390	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	6	2	4	4.3	CCc1ccccc1NC(=O)C(=O)NCCc1sc(-c2cccc(C)c2)nc1C	nan
	CHEMBL1317197	21390	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	6	2	4	4.3	CCc1ccccc1NC(=O)C(=O)NCCc1sc(-c2cccc(C)c2)nc1C	nan
	16026110	21400	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	5	1	5	4.2	CC1=C(c2ccc(C(C)C)cc2)S(=O)(=O)N=C1N1CCC(C(=O)NCc2ccc(C)o2)CC1	nan
	CHEMBL1317332	21400	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	5	1	5	4.2	CC1=C(c2ccc(C(C)C)cc2)S(=O)(=O)N=C1N1CCC(C(=O)NCc2ccc(C)o2)CC1	nan
	7205418	21414	15	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	4	1	5	4.4	Cc1ccc(-n2ncc3c(NCc4ccccc4)ncnc32)cc1Cl	nan
	CHEMBL1317524	21414	15	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	4	1	5	4.4	Cc1ccc(-n2ncc3c(NCc4ccccc4)ncnc32)cc1Cl	nan
	16008313	21427	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	478	6	2	6	4.4	Cc1ccc(NC(=O)C2CCC(CNS(=O)(=O)c3cccc4nsnc34)CC2)c(Cl)c1	nan
	CHEMBL1317641	21427	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	478	6	2	6	4.4	Cc1ccc(NC(=O)C2CCC(CNS(=O)(=O)c3cccc4nsnc34)CC2)c(Cl)c1	nan
	16026429	21431	0	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	3	1	7	1.2	Cc1cc2c(cc1NS(=O)(=O)c1cccc(C#N)c1)n(C)c(=O)c(=O)n2C	nan
	CHEMBL1317692	21431	0	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	3	1	7	1.2	Cc1cc2c(cc1NS(=O)(=O)c1cccc(C#N)c1)n(C)c(=O)c(=O)n2C	nan
	15989759	21443	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	307	3	1	5	3.3	Cc1ccc2nc(NCc3ccc(F)cc3)c3nncn3c2c1	nan
	CHEMBL1317896	21443	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	307	3	1	5	3.3	Cc1ccc2nc(NCc3ccc(F)cc3)c3nncn3c2c1	nan
	16016705	21460	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	330	5	1	4	2.6	O=C(CCC(=O)N1CCOc2ccccc21)NCc1cccs1	nan
	CHEMBL1318069	21460	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	330	5	1	4	2.6	O=C(CCC(=O)N1CCOc2ccccc21)NCc1cccs1	nan
	15988587	21467	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	507	6	1	6	4.5	O=C(Cn1c(=O)n(Cc2ccc(F)cc2)c(=O)c2sc3ccccc3c21)NCc1ccccc1Cl	nan
	CHEMBL1318209	21467	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	507	6	1	6	4.5	O=C(Cn1c(=O)n(Cc2ccc(F)cc2)c(=O)c2sc3ccccc3c21)NCc1ccccc1Cl	nan
	7245933	21471	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	6	0	6	3.4	CCOc1ccc(S(=O)(=O)c2cc3cccc(OCC)c3oc2=O)cc1	nan
	CHEMBL1318269	21471	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	6	0	6	3.4	CCOc1ccc(S(=O)(=O)c2cc3cccc(OCC)c3oc2=O)cc1	nan
	1164100	21509	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	5	0	6	3.4	COc1cccc(-c2nnc(SCC(=O)N3CCc4ccccc43)o2)c1	nan
	CHEMBL1318572	21509	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	5	0	6	3.4	COc1cccc(-c2nnc(SCC(=O)N3CCc4ccccc43)o2)c1	nan
	4077176	21519	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	5	1	3	5.6	CCC(C)NC(=O)c1cc(Sc2cccc(Cl)c2)nc2ccccc12	nan
	CHEMBL1318673	21519	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	5	1	3	5.6	CCC(C)NC(=O)c1cc(Sc2cccc(Cl)c2)nc2ccccc12	nan
	4055959	21544	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	4	1	5	3.6	Cc1ccc(NC(=O)c2oc3ccc(S(=O)(=O)N4CCOCC4)cc3c2C)c(C)c1	nan
	CHEMBL1318877	21544	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	4	1	5	3.6	Cc1ccc(NC(=O)c2oc3ccc(S(=O)(=O)N4CCOCC4)cc3c2C)c(C)c1	nan
	16022946	21621	1	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	482	6	1	6	4.6	Cc1ccc(-n2nc3c(N4CCC(C(=O)NCCc5ccccc5C)CC4)nnc(C)c3c2C)cc1	nan
	CHEMBL1319510	21621	1	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	482	6	1	6	4.6	Cc1ccc(-n2nc3c(N4CCC(C(=O)NCCc5ccccc5C)CC4)nnc(C)c3c2C)cc1	nan
	2967498	21683	21	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	300	5	1	5	3.6	O=C(Nc1nccs1)c1ccc(COc2ccccc2)o1	nan
	CHEMBL1320036	21683	21	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	300	5	1	5	3.6	O=C(Nc1nccs1)c1ccc(COc2ccccc2)o1	nan
	5139336	21697	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	5	1	5	4.4	Cc1cccc2sc(NC(=O)c3ccc(OCC4CCCO4)cc3)nc12	nan
	CHEMBL1320175	21697	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	5	1	5	4.4	Cc1cccc2sc(NC(=O)c3ccc(OCC4CCCO4)cc3)nc12	nan
	16030546	21704	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	6	1	6	3.5	COc1ccccc1C(=O)Nc1cccc(OCc2cc(=O)n3ccccc3n2)c1	nan
	CHEMBL1320207	21704	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	6	1	6	3.5	COc1ccccc1C(=O)Nc1cccc(OCc2cc(=O)n3ccccc3n2)c1	nan
	16030772	21749	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	6	1	9	1.8	Cn1c(=O)c2c(SCC(=O)NCc3ccco3)nc(-c3ccccc3F)nc2n(C)c1=O	nan
	CHEMBL1320595	21749	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	6	1	9	1.8	Cn1c(=O)c2c(SCC(=O)NCc3ccco3)nc(-c3ccccc3F)nc2n(C)c1=O	nan
	16016685	21759	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	4	2	3	4.3	CCCCNC(=O)Nc1ccc2c(c1)N(C)C(=O)c1ccccc1S2	nan
	CHEMBL1320647	21759	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	4	2	3	4.3	CCCCNC(=O)Nc1ccc2c(c1)N(C)C(=O)c1ccccc1S2	nan
	16033946	21765	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	5	1	7	4.4	CCOC(=O)c1ccc(Nc2ncnc3c2cnn3-c2cccc(Cl)c2)cc1	nan
	CHEMBL1320676	21765	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	5	1	7	4.4	CCOC(=O)c1ccc(Nc2ncnc3c2cnn3-c2cccc(Cl)c2)cc1	nan
	944701	21771	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	299	4	1	6	2.9	COc1ccc2nc(O)c(COC(=O)c3ccco3)cc2c1	nan
	CHEMBL1320788	21771	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	299	4	1	6	2.9	COc1ccc2nc(O)c(COC(=O)c3ccco3)cc2c1	nan
	5135847	21803	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	5	2	4	3.8	CCOC(=O)c1cc2c(nc1N=C(S)NCc1ccccc1)CCCC2	nan
	CHEMBL1321064	21803	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	5	2	4	3.8	CCOC(=O)c1cc2c(nc1N=C(S)NCc1ccccc1)CCCC2	nan
	3634798	21806	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	7	0	7	4.5	CCOC(=O)CSc1nc2c(sc3ccccc32)c(=O)n1CCc1ccccc1	nan
	CHEMBL1321100	21806	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	7	0	7	4.5	CCOC(=O)CSc1nc2c(sc3ccccc32)c(=O)n1CCc1ccccc1	nan
	6473515	21822	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	6	2	5	3.1	COc1ccc(S(=O)(=O)Nc2ccccn2)cc1C(=O)Nc1ccccc1	nan
	CHEMBL1321208	21822	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	6	2	5	3.1	COc1ccc(S(=O)(=O)Nc2ccccn2)cc1C(=O)Nc1ccccc1	nan
	16026080	21857	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	4	1	7	2.6	CCc1ccccc1NC(=O)c1cnc2sc(N3CCCC3)nn2c1=O	nan
	CHEMBL1321609	21857	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	4	1	7	2.6	CCc1ccccc1NC(=O)c1cnc2sc(N3CCCC3)nn2c1=O	nan
	661514	21862	9	None	-2	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	4	0	8	2.7	COc1ccc(-c2nnc3sc(CN4C(=O)c5ccccc5C4=O)nn23)cc1	nan
	CHEMBL1321633	21862	9	None	-2	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	4	0	8	2.7	COc1ccc(-c2nnc3sc(CN4C(=O)c5ccccc5C4=O)nn23)cc1	nan
	963196	21900	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	346	5	1	3	4.5	Cc1ccc(NC(=O)Cn2cc(C(=O)C3CC3)c3ccccc32)c(C)c1	nan
	CHEMBL1321920	21900	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	346	5	1	3	4.5	Cc1ccc(NC(=O)Cn2cc(C(=O)C3CC3)c3ccccc32)c(C)c1	nan
	1034156	21903	15	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	4	2	4	2.9	Cc1cc2oc(C(=O)NCc3ccc(S(N)(=O)=O)cc3)c(C)c2cc1C	nan
	CHEMBL1321976	21903	15	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	4	2	4	2.9	Cc1cc2oc(C(=O)NCc3ccc(S(N)(=O)=O)cc3)c(C)c2cc1C	nan
	16026098	21904	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	4	1	5	3.7	CC1=C(c2ccc(C)c(C)c2)S(=O)(=O)N=C1N1CCC(C(=O)NCc2ccc(C)o2)CC1	nan
	CHEMBL1321983	21904	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	4	1	5	3.7	CC1=C(c2ccc(C)c(C)c2)S(=O)(=O)N=C1N1CCC(C(=O)NCc2ccc(C)o2)CC1	nan
	1480476	21957	23	None	-12	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	4	1	5	4.6	CC(C)Nc1nc(-c2ccncc2)nc(-c2ccc(Cl)cc2)c1C#N	nan
	CHEMBL1322430	21957	23	None	-12	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	4	1	5	4.6	CC(C)Nc1nc(-c2ccncc2)nc(-c2ccc(Cl)cc2)c1C#N	nan
	16021832	22075	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	4	1	4	4.7	CSc1ncc(C(=O)Nc2cccc(C)c2C)c(-c2ccccc2)n1	nan
	CHEMBL1323559	22075	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	4	1	4	4.7	CSc1ncc(C(=O)Nc2cccc(C)c2C)c(-c2ccccc2)n1	nan
	4868391	22122	30	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	300	3	1	3	4.5	Sc1ncc(-c2ccc(Cl)cc2)n1Cc1ccccc1	nan
	CHEMBL1323909	22122	30	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	300	3	1	3	4.5	Sc1ncc(-c2ccc(Cl)cc2)n1Cc1ccccc1	nan
	7284118	22126	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	9	1	5	3.2	CCOc1ccc(CCNC(=O)Cn2ccc3ccccc3c2=O)cc1OCC	nan
	CHEMBL1323924	22126	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	9	1	5	3.2	CCOc1ccc(CCNC(=O)Cn2ccc3ccccc3c2=O)cc1OCC	nan
	2135896	22144	4	None	-158	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	7	2	7	2.4	COc1ccc(OC)c(NC(=O)c2nnn(CCc3ccccc3)c2N)c1	nan
	CHEMBL1324085	22144	4	None	-158	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	7	2	7	2.4	COc1ccc(OC)c(NC(=O)c2nnn(CCc3ccccc3)c2N)c1	nan
	3422137	22149	15	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	502	8	0	9	2.0	COCCn1c(CN2CCN(C(c3ccccc3)c3ccccc3)CC2)nc2c1c(=O)n(C)c(=O)n2C	nan
	CHEMBL1324117	22149	15	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	502	8	0	9	2.0	COCCn1c(CN2CCN(C(c3ccccc3)c3ccccc3)CC2)nc2c1c(=O)n(C)c(=O)n2C	nan
	16015664	22199	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	486	7	1	6	6.6	CCOc1ccc(C(=O)c2oc3ccccc3c2NC(=O)c2cc(-c3ccc(Cl)cc3)on2)cc1	nan
	CHEMBL1324545	22199	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	486	7	1	6	6.6	CCOc1ccc(C(=O)c2oc3ccccc3c2NC(=O)c2cc(-c3ccc(Cl)cc3)on2)cc1	nan
	5299986	22242	18	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	4	1	5	5.1	N#Cc1cc2c(nc1SCC(=O)Nc1ccc(Cl)c(C(F)(F)F)c1)C1CCN2CC1	nan
	CHEMBL1324899	22242	18	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	4	1	5	5.1	N#Cc1cc2c(nc1SCC(=O)Nc1ccc(Cl)c(C(F)(F)F)c1)C1CCN2CC1	nan
	2967360	22263	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	5	1	4	5.3	Cc1ccc(N(Cc2cc3ccc(C)cc3nc2O)S(=O)(=O)c2ccccc2)c(C)c1	nan
	CHEMBL1325059	22263	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	5	1	4	5.3	Cc1ccc(N(Cc2cc3ccc(C)cc3nc2O)S(=O)(=O)c2ccccc2)c(C)c1	nan
	4013085	22281	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	304	4	2	7	2.7	CCOC(=O)c1ccc(NC2Nc3cc(C)nn3S2)cc1	nan
	CHEMBL1325232	22281	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	304	4	2	7	2.7	CCOC(=O)c1ccc(NC2Nc3cc(C)nn3S2)cc1	nan
	4877095	22299	5	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	4	1	6	4.1	CCOC(=O)c1sc(NC(=O)c2cc3c(s2)CCC(C)C3)nc1C	nan
	CHEMBL1325413	22299	5	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	4	1	6	4.1	CCOC(=O)c1sc(NC(=O)c2cc3c(s2)CCC(C)C3)nc1C	nan
	16012280	22309	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	5	1	7	1.7	Cc1cccc(C)c1NC(=O)CCS(=O)(=O)c1ccc2c(c1)n(C)c(=O)c(=O)n2C	nan
	CHEMBL1325535	22309	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	5	1	7	1.7	Cc1cccc(C)c1NC(=O)CCS(=O)(=O)c1ccc2c(c1)n(C)c(=O)c(=O)n2C	nan
	16011188	22322	3	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	4	1	5	4.4	COC(=O)c1cc2oc3ccccc3c2n1CC(=O)Nc1ccc(C)cc1C	nan
	CHEMBL1325716	22322	3	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	4	1	5	4.4	COC(=O)c1cc2oc3ccccc3c2n1CC(=O)Nc1ccc(C)cc1C	nan
	709602	22330	4	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	335	3	2	5	3.6	Cc1c(NC(=O)c2nc[nH]n2)cccc1-c1nc2ccccc2s1	nan
	CHEMBL1325780	22330	4	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	335	3	2	5	3.6	Cc1c(NC(=O)c2nc[nH]n2)cccc1-c1nc2ccccc2s1	nan
	3619431	22393	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	6	0	4	5.7	O=C(c1cccs1)c1cn(CCOc2ccc(Cl)cc2)c2ccccc12	nan
	CHEMBL1326440	22393	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	6	0	4	5.7	O=C(c1cccs1)c1cn(CCOc2ccc(Cl)cc2)c2ccccc12	nan
	663870	22400	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	293	3	1	4	3.6	Cc1ccc(C(=O)OCc2cc3ccccc3nc2O)cc1	nan
	CHEMBL1326511	22400	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	293	3	1	4	3.6	Cc1ccc(C(=O)OCc2cc3ccccc3nc2O)cc1	nan
	16018929	22410	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	11	1	7	3.6	CCOc1ccc(CCNC(=O)CCCn2c(=O)c3cccn3c3cccnc32)cc1OCC	nan
	CHEMBL1326604	22410	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	11	1	7	3.6	CCOc1ccc(CCNC(=O)CCCn2c(=O)c3cccn3c3cccnc32)cc1OCC	nan
	17583882	22419	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	7	1	5	3.5	CCCCc1cc(=O)oc2cc(OCC(=O)Nc3ccccn3)ccc12	nan
	CHEMBL1326654	22419	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	7	1	5	3.5	CCCCc1cc(=O)oc2cc(OCC(=O)Nc3ccccn3)ccc12	nan
	1477181	22462	17	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	332	5	1	6	3.7	CC(=O)c1cc(C#N)c(NCc2cc(-c3ccccc3)no2)nc1C	nan
	CHEMBL1327040	22462	17	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	332	5	1	6	3.7	CC(=O)c1cc(C#N)c(NCc2cc(-c3ccccc3)no2)nc1C	nan
	16034758	22470	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	345	4	2	6	2.6	COc1ccc(NC(=O)c2sc3nc[nH]c(=O)c3c2C)cc1OC	nan
	CHEMBL1327116	22470	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	345	4	2	6	2.6	COc1ccc(NC(=O)c2sc3nc[nH]c(=O)c3c2C)cc1OC	nan
	16008896	22478	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	4	1	5	3.0	COc1ccc(CNC(=O)c2cc3c(=O)n(C)c4ccccc4c3n2C)cc1	nan
	CHEMBL1327173	22478	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	4	1	5	3.0	COc1ccc(CNC(=O)c2cc3c(=O)n(C)c4ccccc4c3n2C)cc1	nan
	4227789	22509	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	467	6	0	5	5.5	CCN(CC)C(=O)C1CCCN(c2ncnc3c2c(-c2ccccc2)cn3-c2cccc(C)c2)C1	nan
	CHEMBL1327499	22509	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	467	6	0	5	5.5	CCN(CC)C(=O)C1CCCN(c2ncnc3c2c(-c2ccccc2)cn3-c2cccc(C)c2)C1	nan
	16032611	22613	1	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	4	2	3	2.9	O=C(NC1CC(=O)N(c2ccc(Cl)cc2)C1)C(=O)c1c[nH]c2ccccc12	nan
	CHEMBL1328167	22613	1	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	4	2	3	2.9	O=C(NC1CC(=O)N(c2ccc(Cl)cc2)C1)C(=O)c1c[nH]c2ccccc12	nan
	1426216	22683	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	490	6	2	8	4.1	Cc1cc(=O)n2c(C(=O)Nc3ccc(C(=O)OC(C)C)cc3)c(C(=O)Nc3ccccc3)sc2n1	nan
	CHEMBL1328860	22683	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	490	6	2	8	4.1	Cc1cc(=O)n2c(C(=O)Nc3ccc(C(=O)OC(C)C)cc3)c(C(=O)Nc3ccccc3)sc2n1	nan
	857007	22684	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	5	1	4	4.2	Cc1cc2cc(C)c(SCC(=O)NCc3ccco3)nc2cc1C	nan
	CHEMBL1328861	22684	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	5	1	4	4.2	Cc1cc2cc(C)c(SCC(=O)NCc3ccco3)nc2cc1C	nan
	16015065	22697	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	7	1	6	5.3	CC(=O)c1cccc(NC(=O)c2sc(-n3nc(C)c(CCC(C)C)c3C)nc2C)c1	nan
	CHEMBL1328989	22697	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	7	1	6	5.3	CC(=O)c1cccc(NC(=O)c2sc(-n3nc(C)c(CCC(C)C)c3C)nc2C)c1	nan
	7294635	22724	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	4	2	4	4.7	Nc1c(C(=O)Nc2ccccc2Cl)c2ccccn2c1C(=O)c1ccccc1	nan
	CHEMBL1329216	22724	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	4	2	4	4.7	Nc1c(C(=O)Nc2ccccc2Cl)c2ccccn2c1C(=O)c1ccccc1	nan
	2986428	22755	10	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	4	1	8	4.0	CC(C)CNc1ncnc2c1sc1nc(N3CCOCC3)c3c(c12)CC(C)(C)OC3	nan
	CHEMBL1329460	22755	10	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	4	1	8	4.0	CC(C)CNc1ncnc2c1sc1nc(N3CCOCC3)c3c(c12)CC(C)(C)OC3	nan
	7422802	22759	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	4	1	5	2.8	Cc1ccc(Cn2cccc(C(=O)Nc3cc(C)on3)c2=O)cc1	nan
	CHEMBL1329510	22759	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	4	1	5	2.8	Cc1ccc(Cn2cccc(C(=O)Nc3cc(C)on3)c2=O)cc1	nan
	7889414	22805	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	6	1	10	1.5	CCCn1c(N)c(C(=O)CSc2ncnc3sccc23)c(=O)n(C)c1=O	nan
	CHEMBL1329885	22805	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	6	1	10	1.5	CCCn1c(N)c(C(=O)CSc2ncnc3sccc23)c(=O)n(C)c1=O	nan
	1038210	22815	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	6	0	8	2.7	CCOC(=O)CCSc1nc(N2CCOCC2)c2c(c1C#N)CC(C)(C)OC2	nan
	CHEMBL1329993	22815	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	6	0	8	2.7	CCOC(=O)CCSc1nc(N2CCOCC2)c2c(c1C#N)CC(C)(C)OC2	nan
	16009180	22862	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	7	1	7	4.2	CCc1ccc(C(=O)c2cn(CC(=O)Nc3ccc4c(c3)OCO4)c3ccc(OC)cc3c2=O)cc1	nan
	CHEMBL1330381	22862	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	7	1	7	4.2	CCc1ccc(C(=O)c2cn(CC(=O)Nc3ccc4c(c3)OCO4)c3ccc(OC)cc3c2=O)cc1	nan
	1510063	22876	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	4	1	4	3.4	CCC(=O)c1cc2c(cc1NC(=O)c1ccccc1F)OCCO2	nan
	CHEMBL1330472	22876	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	4	1	4	3.4	CCC(=O)c1cc2c(cc1NC(=O)c1ccccc1F)OCCO2	nan
	16019798	22911	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	471	6	2	6	2.6	COc1ccc(NC(=O)C2CCCN(S(=O)(=O)c3ccc4[nH]c(=O)ccc4c3)C2)cc1OC	nan
	CHEMBL1330797	22911	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	471	6	2	6	2.6	COc1ccc(NC(=O)C2CCCN(S(=O)(=O)c3ccc4[nH]c(=O)ccc4c3)C2)cc1OC	nan
	1078194	22960	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	7	2	5	3.5	Cc1ccc(OCC(=O)Nc2ccc(S(=O)(=O)Nc3ccccn3)cc2)cc1C	nan
	CHEMBL1331082	22960	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	7	2	5	3.5	Cc1ccc(OCC(=O)Nc2ccc(S(=O)(=O)Nc3ccccn3)cc2)cc1C	nan
	1367422	22962	13	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	3	2	6	3.6	O=C(NC(=S)Nc1cccc(-c2nc3ncccc3o2)c1)c1ccco1	nan
	CHEMBL1331090	22962	13	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	3	2	6	3.6	O=C(NC(=S)Nc1cccc(-c2nc3ncccc3o2)c1)c1ccco1	nan
	15990786	22984	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	496	13	2	5	6.4	CCCCN(CCCNC(=O)c1cc(Nc2ccc(OC)cc2)nc2ccccc12)Cc1ccccc1	nan
	CHEMBL1331246	22984	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	496	13	2	5	6.4	CCCCN(CCCNC(=O)c1cc(Nc2ccc(OC)cc2)nc2ccccc12)Cc1ccccc1	nan
	1426224	22992	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	5	2	6	4.1	CCc1ccc(NC(=O)c2c(C(=O)Nc3ccccc3)sc3nc(C)cc(=O)n23)cc1	nan
	CHEMBL1331302	22992	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	5	2	6	4.1	CCc1ccc(NC(=O)c2c(C(=O)Nc3ccccc3)sc3nc(C)cc(=O)n23)cc1	nan
	16009858	23021	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	9	2	6	5.7	CCOc1ccc(C(=O)Nc2c(C(=O)Nc3ccccc3OC)oc3ccccc23)cc1OCC	nan
	CHEMBL1331538	23021	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	9	2	6	5.7	CCOc1ccc(C(=O)Nc2c(C(=O)Nc3ccccc3OC)oc3ccccc23)cc1OCC	nan
	965763	23054	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	4	1	4	3.8	Cc1cc(OCC(=O)Nc2ccc3oc(=O)ccc3c2)ccc1Cl	nan
	CHEMBL1331830	23054	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	4	1	4	3.8	Cc1cc(OCC(=O)Nc2ccc3oc(=O)ccc3c2)ccc1Cl	nan
	4216258	23090	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	457	8	3	6	6.0	CCOc1ccccc1Nc1sc(C(=O)c2ccccc2)c(N)c1C(=O)Nc1ccccc1	nan
	CHEMBL1332095	23090	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	457	8	3	6	6.0	CCOc1ccccc1Nc1sc(C(=O)c2ccccc2)c(N)c1C(=O)Nc1ccccc1	nan
	2670204	23101	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	7	0	9	1.7	COc1ccc(C(=O)COC(=O)c2ccc(-n3cnnn3)cc2)c(OC)c1	nan
	CHEMBL1332216	23101	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	7	0	9	1.7	COc1ccc(C(=O)COC(=O)c2ccc(-n3cnnn3)cc2)c(OC)c1	nan
	2151601	23120	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	5	1	6	5.5	Cc1ccc(-n2c(SCC(=O)Nc3cccc(C)c3)nc3c(oc4ccccc43)c2=O)cc1	nan
	CHEMBL1332323	23120	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	5	1	6	5.5	Cc1ccc(-n2c(SCC(=O)Nc3cccc(C)c3)nc3c(oc4ccccc43)c2=O)cc1	nan
	16012517	23124	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	464	6	2	5	6.3	CCOc1ccc(-c2cc(NC(=O)Nc3ccccc3C(F)(F)F)c(C(=O)OC)s2)cc1	nan
	CHEMBL1332340	23124	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	464	6	2	5	6.3	CCOc1ccc(-c2cc(NC(=O)Nc3ccccc3C(F)(F)F)c(C(=O)OC)s2)cc1	nan
	2243529	23125	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	279	1	0	3	3.7	O=C(c1cccs1)N1C(=O)c2cccc3cccc1c23	nan
	CHEMBL1332342	23125	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	279	1	0	3	3.7	O=C(c1cccs1)N1C(=O)c2cccc3cccc1c23	nan
	867009	23242	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	320	4	2	3	3.7	COc1ccc(Cl)cc1NC(=O)c1[nH]c(C)c(C(C)=O)c1C	nan
	CHEMBL1333261	23242	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	320	4	2	3	3.7	COc1ccc(Cl)cc1NC(=O)c1[nH]c(C)c(C(C)=O)c1C	nan
	677173	23269	14	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	278	4	2	4	3.5	CCCc1nnc(N=C(S)Nc2ccccc2)s1	nan
	CHEMBL1333504	23269	14	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	278	4	2	4	3.5	CCCc1nnc(N=C(S)Nc2ccccc2)s1	nan
	3623159	23303	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	7	1	4	5.3	CCOc1ccc(Sc2cc(C(=O)NC(C)CC)c3ccccc3n2)cc1	nan
	CHEMBL1333744	23303	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	7	1	4	5.3	CCOc1ccc(Sc2cc(C(=O)NC(C)CC)c3ccccc3n2)cc1	nan
	16008956	23341	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	436	7	1	6	4.2	CCn1c(=O)c2cc(C(=O)NCCc3ccc(OC)c(OC)c3)sc2c2ccccc21	nan
	CHEMBL1334014	23341	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	436	7	1	6	4.2	CCn1c(=O)c2cc(C(=O)NCCc3ccc(OC)c(OC)c3)sc2c2ccccc21	nan
	2196864	23386	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	7	1	7	4.2	CCn1c(Cc2ccccc2)nnc1SCC(=O)Nc1nc2ccccc2s1	nan
	CHEMBL1334332	23386	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	7	1	7	4.2	CCn1c(Cc2ccccc2)nnc1SCC(=O)Nc1nc2ccccc2s1	nan
	3622707	23459	8	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	324	3	0	4	5.1	Cc1nc(SCc2cccc(F)c2)c2oc3ccccc3c2n1	nan
	CHEMBL1335007	23459	8	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	324	3	0	4	5.1	Cc1nc(SCc2cccc(F)c2)c2oc3ccccc3c2n1	nan
	16008370	23485	0	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	5	1	4	3.7	Cn1c(=O)cc(SCC(=O)NCc2ccc(F)cc2)c2cc(Cl)ccc21	nan
	CHEMBL1335160	23485	0	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	5	1	4	3.7	Cn1c(=O)cc(SCC(=O)NCc2ccc(F)cc2)c2cc(Cl)ccc21	nan
	16020489	23524	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	5	0	5	3.7	CCN(CC)c1cc2c(cc1F)c(=O)c(S(=O)(=O)c1cccc(C)c1)cn2C	nan
	CHEMBL1335441	23524	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	5	0	5	3.7	CCN(CC)c1cc2c(cc1F)c(=O)c(S(=O)(=O)c1cccc(C)c1)cn2C	nan
	16012518	23528	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	7	1	5	5.3	CCOc1ccccc1NC(=O)CCc1c(C)nc2c(c(C)nn2-c2ccccc2)c1C	nan
	CHEMBL1335479	23528	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	7	1	5	5.3	CCOc1ccccc1NC(=O)CCc1c(C)nc2c(c(C)nn2-c2ccccc2)c1C	nan
	16018933	23535	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	9	1	7	2.8	COc1ccc(OC)c(CCNC(=O)CCCn2c(=O)c3cccn3c3cccnc32)c1	nan
	CHEMBL1335514	23535	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	9	1	7	2.8	COc1ccc(OC)c(CCNC(=O)CCCn2c(=O)c3cccn3c3cccnc32)c1	nan
	16022436	23546	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	489	6	2	7	5.2	CCc1ccccc1Nc1nn2c(=O)c3ccc(C(=O)NCc4ccccc4Cl)cc3nc2s1	nan
	CHEMBL1335596	23546	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	489	6	2	7	5.2	CCc1ccccc1Nc1nn2c(=O)c3ccc(C(=O)NCc4ccccc4Cl)cc3nc2s1	nan
	3221114	23586	4	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	398	6	1	6	3.3	COCCN=C(S)N(Cc1cc2cc(C)ccc2n2nnnc12)C1CCCC1	nan
	CHEMBL1335947	23586	4	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	398	6	1	6	3.3	COCCN=C(S)N(Cc1cc2cc(C)ccc2n2nnnc12)C1CCCC1	nan
	16015039	23603	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	6	1	7	5.4	CCc1ccccc1NC(=O)c1sc(-n2nc(C)c(Cc3ccc4c(c3)OCO4)c2C)nc1C	nan
	CHEMBL1336092	23603	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	6	1	7	5.4	CCc1ccccc1NC(=O)c1sc(-n2nc(C)c(Cc3ccc4c(c3)OCO4)c2C)nc1C	nan
	2138945	23627	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	4	1	5	3.5	O=C(Nc1nc2ccc(S(=O)(=O)N3CCCC3)cc2s1)c1ccc(F)cc1	nan
	CHEMBL1336262	23627	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	4	1	5	3.5	O=C(Nc1nc2ccc(S(=O)(=O)N3CCCC3)cc2s1)c1ccc(F)cc1	nan
	6220215	23684	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	320	1	2	3	3.2	CC1=CC2=NC(=O)/C(=C\c3c(C)[nH]c4ccc(C)cc34)C(=N)N2O1	nan
	CHEMBL1336784	23684	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	320	1	2	3	3.2	CC1=CC2=NC(=O)/C(=C\c3c(C)[nH]c4ccc(C)cc34)C(=N)N2O1	nan
	16026936	23721	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	6	0	9	3.0	O=C(COc1ccccc1)OCc1cc(=O)n2nc(-c3cccs3)sc2n1	nan
	CHEMBL1337126	23721	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	6	0	9	3.0	O=C(COc1ccccc1)OCc1cc(=O)n2nc(-c3cccs3)sc2n1	nan
	1486592	23773	15	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	286	4	1	7	1.7	COc1ccc(Nc2nc(N(C)C)oc(=O)c2C#N)cc1	nan
	CHEMBL1337568	23773	15	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	286	4	1	7	1.7	COc1ccc(Nc2nc(N(C)C)oc(=O)c2C#N)cc1	nan
	1485789	23794	21	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	295	3	0	2	4.3	O=C(c1ccc(F)cc1)c1ccc(-c2ccc(F)cc2)nc1	nan
	CHEMBL1337770	23794	21	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	295	3	0	2	4.3	O=C(c1ccc(F)cc1)c1ccc(-c2ccc(F)cc2)nc1	nan
	16033861	23828	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	461	6	2	8	4.6	CCc1ccccc1Nc1nn2c(=O)c3ccc(C(=O)NCc4cccs4)cc3nc2s1	nan
	CHEMBL1338096	23828	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	461	6	2	8	4.6	CCc1ccccc1Nc1nn2c(=O)c3ccc(C(=O)NCc4cccs4)cc3nc2s1	nan
	1265732	23880	14	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	5	1	4	5.4	O=C(Cn1c(S)nc(-c2ccccc2)c1-c1ccccc1)c1ccccc1	nan
	CHEMBL1338427	23880	14	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	5	1	4	5.4	O=C(Cn1c(S)nc(-c2ccccc2)c1-c1ccccc1)c1ccccc1	nan
	16026086	23937	0	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	3	1	7	2.3	Cc1ccccc1NC(=O)c1cnc2sc(N3CCCC3)nn2c1=O	nan
	CHEMBL1339014	23937	0	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	3	1	7	2.3	Cc1ccccc1NC(=O)c1cnc2sc(N3CCCC3)nn2c1=O	nan
	15944700	24146	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	4	2	5	4.4	O=C(Nc1cc(Cl)cc(Cl)c1)c1ccc(Cn2c(=O)[nH]c3ccsc3c2=O)cc1	nan
	CHEMBL1340950	24146	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	4	2	5	4.4	O=C(Nc1cc(Cl)cc(Cl)c1)c1ccc(Cn2c(=O)[nH]c3ccsc3c2=O)cc1	nan
	5069163	24161	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	7	2	7	2.9	COc1ccc(CNC(=O)CCCn2c(=S)[nH]c3cc4c(cc3c2=O)OCO4)cc1	nan
	CHEMBL1341068	24161	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	7	2	7	2.9	COc1ccc(CNC(=O)CCCn2c(=S)[nH]c3cc4c(cc3c2=O)OCO4)cc1	nan
	855559	24284	2	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	5	0	6	3.5	CCN(C(=O)c1ccco1)c1nnc(-c2ccc(OC)cc2)s1	nan
	CHEMBL1342076	24284	2	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	5	0	6	3.5	CCN(C(=O)c1ccco1)c1nnc(-c2ccc(OC)cc2)s1	nan
	3149126	24298	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	454	10	2	7	3.5	CCOCCCn1c(SCC(=O)Nc2ccc(NC(C)=O)cc2)nc2ccccc2c1=O	nan
	CHEMBL1342207	24298	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	454	10	2	7	3.5	CCOCCCn1c(SCC(=O)Nc2ccc(NC(C)=O)cc2)nc2ccccc2c1=O	nan
	1086862	24317	16	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	7	1	7	3.4	COc1ccc(C(=O)Nc2nnc(Cc3ccc(OC)c(OC)c3)s2)cc1	nan
	CHEMBL1342348	24317	16	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	7	1	7	3.4	COc1ccc(C(=O)Nc2nnc(Cc3ccc(OC)c(OC)c3)s2)cc1	nan
	5443591	24356	7	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	8	1	6	3.8	CCOC(=O)/C(C#N)=C\c1ccc(OCC(=O)Nc2ccc(C)cc2C)c(OC)c1	nan
	CHEMBL1342661	24356	7	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	8	1	6	3.8	CCOC(=O)/C(C#N)=C\c1ccc(OCC(=O)Nc2ccc(C)cc2C)c(OC)c1	nan
	665611	24393	9	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	2	1	6	3.9	Cc1cc(-c2nnc3sc(-c4ccc(Cl)cc4Cl)nn23)[nH]n1	nan
	CHEMBL1342889	24393	9	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	2	1	6	3.9	Cc1cc(-c2nnc3sc(-c4ccc(Cl)cc4Cl)nn23)[nH]n1	nan
	5063932	24451	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	4	2	5	3.6	O=C(NCc1ccco1)c1ccc2c(=O)n(-c3ccccc3)c(=S)[nH]c2c1	nan
	CHEMBL1343363	24451	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	4	2	5	3.6	O=C(NCc1ccco1)c1ccc2c(=O)n(-c3ccccc3)c(=S)[nH]c2c1	nan
	2452051	24600	4	None	-2	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	5	1	8	4.6	N#Cc1ccc(CSc2nnc(NC(=O)c3ccc4ncsc4c3)s2)cc1	nan
	CHEMBL1344739	24600	4	None	-2	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	5	1	8	4.6	N#Cc1ccc(CSc2nnc(NC(=O)c3ccc4ncsc4c3)s2)cc1	nan
	2335388	24688	1	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	2	1	5	3.0	Cc1ccnc(NC(=O)c2ccc3c(c2)S(=O)(=O)c2ccccc2C3=O)c1	nan
	CHEMBL1345474	24688	1	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	2	1	5	3.0	Cc1ccnc(NC(=O)c2ccc3c(c2)S(=O)(=O)c2ccccc2C3=O)c1	nan
	666154	24689	9	None	-3	3	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	345	2	1	6	4.2	Cc1ccc(-n2nc(C)c3c(-c4cccs4)c(C#N)c(N)nc32)cc1	nan
	CHEMBL1345487	24689	9	None	-3	3	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	345	2	1	6	4.2	Cc1ccc(-n2nc(C)c3c(-c4cccs4)c(C#N)c(N)nc32)cc1	nan
	2040126	24694	12	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	461	7	2	6	2.6	Cc1ccc(/C=C2\SC(=S)N(CCC(=O)NNS(=O)(=O)c3ccccc3)C2=O)cc1	nan
	CHEMBL1345551	24694	12	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	461	7	2	6	2.6	Cc1ccc(/C=C2\SC(=S)N(CCC(=O)NNS(=O)(=O)c3ccccc3)C2=O)cc1	nan
	3185713	24767	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	550	10	3	8	3.1	CCc1ccccc1N(C(=O)c1snc(C(N)=O)c1N)C(C(=O)NCC1CCCO1)c1ccc(N(C)C)cc1	nan
	CHEMBL1346198	24767	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	550	10	3	8	3.1	CCc1ccccc1N(C(=O)c1snc(C(N)=O)c1N)C(C(=O)NCC1CCCO1)c1ccc(N(C)C)cc1	nan
	1409877	24829	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	4	1	5	2.8	Cc1cccc(NC(=O)COC(=O)c2ccc3c(c2)OCO3)c1C	nan
	CHEMBL1346710	24829	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	4	1	5	2.8	Cc1cccc(NC(=O)COC(=O)c2ccc3c(c2)OCO3)c1C	nan
	3846689	24847	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	317	3	0	6	2.4	COCc1nc2oc3ccc(F)cc3c(=O)c2cc1C(=O)OC	nan
	CHEMBL1346831	24847	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	317	3	0	6	2.4	COCc1nc2oc3ccc(F)cc3c(=O)c2cc1C(=O)OC	nan
	2813569	24896	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	356	4	0	6	3.3	O=C(COc1ncnc2cc(Cl)ccc12)c1ccc2c(c1)OCCO2	nan
	CHEMBL1347186	24896	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	356	4	0	6	3.3	O=C(COc1ncnc2cc(Cl)ccc12)c1ccc2c(c1)OCCO2	nan
	2426514	24957	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	267	1	0	5	2.6	Cc1cc(=O)n2nc(-c3ccccc3)sc2c1C#N	nan
	CHEMBL1347674	24957	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	267	1	0	5	2.6	Cc1cc(=O)n2nc(-c3ccccc3)sc2c1C#N	nan
	2950848	25030	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	347	6	1	5	3.2	COCc1cc(C)nc(SCC(=O)NC2CCCCC2C)c1C#N	nan
	CHEMBL1348333	25030	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	347	6	1	5	3.2	COCc1cc(C)nc(SCC(=O)NC2CCCCC2C)c1C#N	nan
	664720	25075	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	4	1	7	5.4	CC(C)c1nc2sc3c(NCc4ccco4)ncnc3c2c2c1COC(C)(C)C2	nan
	CHEMBL1348840	25075	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	4	1	7	5.4	CC(C)c1nc2sc3c(NCc4ccco4)ncnc3c2c2c1COC(C)(C)C2	nan
	780682	25180	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	291	4	1	3	3.8	C=CCn1c(NC(=O)c2ccc(C)cc2)nc2ccccc21	nan
	CHEMBL1349635	25180	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	291	4	1	3	3.8	C=CCn1c(NC(=O)c2ccc(C)cc2)nc2ccccc21	nan
	7157934	25291	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	4	2	5	1.6	O=C(Nc1ccc2c(c1)C(=O)NC2=O)c1ccc(S(=O)(=O)N2CCCC2)cc1	nan
	CHEMBL1350603	25291	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	4	2	5	1.6	O=C(Nc1ccc2c(c1)C(=O)NC2=O)c1ccc(S(=O)(=O)N2CCCC2)cc1	nan
	16194401	25392	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	396	3	2	6	2.8	CCOC(=O)N1CCC(NC(=O)c2cc3c(O)nc4ccccc4c3n2C)CC1	nan
	CHEMBL1351462	25392	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	396	3	2	6	2.8	CCOC(=O)N1CCC(NC(=O)c2cc3c(O)nc4ccccc4c3n2C)CC1	nan
	1433829	25524	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	313	5	1	5	2.5	COc1ccc2nc(SCC(=O)NC3CC3)c(C#N)cc2c1	nan
	CHEMBL1352517	25524	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	313	5	1	5	2.5	COc1ccc2nc(SCC(=O)NC3CC3)c(C#N)cc2c1	nan
	5112429	25557	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	5	2	7	1.9	N#CCC(=O)NNc1c([N+](=O)[O-])cc(C(F)(F)F)cc1[N+](=O)[O-]	nan
	CHEMBL1352781	25557	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	5	2	7	1.9	N#CCC(=O)NNc1c([N+](=O)[O-])cc(C(F)(F)F)cc1[N+](=O)[O-]	nan
	4850085	25588	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	7	2	8	2.8	CCOC(=O)c1sc2nc(C)nc(NCCc3ccc(S(N)(=O)=O)cc3)c2c1C	nan
	CHEMBL1353043	25588	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	7	2	8	2.8	CCOC(=O)c1sc2nc(C)nc(NCCc3ccc(S(N)(=O)=O)cc3)c2c1C	nan
	3350830	25730	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	4	2	4	4.7	Cc1cc(C)c(NC(=O)CSc2nc3cc(Br)c[nH]c-3n2)c(Cl)c1	nan
	CHEMBL1354025	25730	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	4	2	4	4.7	Cc1cc(C)c(NC(=O)CSc2nc3cc(Br)c[nH]c-3n2)c(Cl)c1	nan
	16017542	25773	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	446	7	1	7	3.6	CCN(c1ccc(C)cc1C)S(=O)(=O)c1nnc(NC(=O)c2ccccc2OC)s1	nan
	CHEMBL1354338	25773	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	446	7	1	7	3.6	CCN(c1ccc(C)cc1C)S(=O)(=O)c1nnc(NC(=O)c2ccccc2OC)s1	nan
	3415736	25787	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	471	7	2	6	2.3	COc1ccc(CNC(=O)c2cc(=O)[nH]c3ccc(S(=O)(=O)N4CCCC4)cc23)c(OC)c1	nan
	CHEMBL1354486	25787	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	471	7	2	6	2.3	COc1ccc(CNC(=O)c2cc(=O)[nH]c3ccc(S(=O)(=O)N4CCCC4)cc23)c(OC)c1	nan
	16008465	25794	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	5	1	4	4.5	Cc1nc2cc(-c3cccc(F)c3)nn2c(C)c1CCC(=O)NC1CCCCC1	nan
	CHEMBL1354574	25794	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	5	1	4	4.5	Cc1nc2cc(-c3cccc(F)c3)nn2c(C)c1CCC(=O)NC1CCCCC1	nan
	16008364	25795	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	4	1	4	5.0	Cc1ccc(NC(=O)CSc2cc(=O)n(C)c3ccc(Cl)cc23)c(Br)c1	nan
	CHEMBL1354597	25795	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	4	1	4	5.0	Cc1ccc(NC(=O)CSc2cc(=O)n(C)c3ccc(Cl)cc23)c(Br)c1	nan
	16034362	25797	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	546	9	1	9	2.1	CSCCC(NS(=O)(=O)c1ccc2c(c1)oc(=O)n2C)C(=O)N1CCN(c2ccc(C(C)=O)cc2)CC1	nan
	CHEMBL1354617	25797	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	546	9	1	9	2.1	CSCCC(NS(=O)(=O)c1ccc2c(c1)oc(=O)n2C)C(=O)N1CCN(c2ccc(C(C)=O)cc2)CC1	nan
	16029590	25802	0	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	5	1	3	5.8	O=C(Nc1ccc(Br)cc1F)c1ccc2nc(CCc3ccccc3)oc2c1	nan
	CHEMBL1354702	25802	0	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	5	1	3	5.8	O=C(Nc1ccc(Br)cc1F)c1ccc2nc(CCc3ccccc3)oc2c1	nan
	16024765	25807	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	3	1	4	3.8	O=C(Cn1c(=O)c(C(F)(F)F)nc2ccccc21)Nc1cccc(Br)c1	nan
	CHEMBL1354803	25807	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	3	1	4	3.8	O=C(Cn1c(=O)c(C(F)(F)F)nc2ccccc21)Nc1cccc(Br)c1	nan
	16026345	25813	0	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	4	1	5	2.6	Cc1ccc(-n2nc(C)c3c(C)cc(=O)n(CC(=O)NC(C)C)c32)cc1	nan
	CHEMBL1354863	25813	0	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	4	1	5	2.6	Cc1ccc(-n2nc(C)c3c(C)cc(=O)n(CC(=O)NC(C)C)c32)cc1	nan
	7872437	25815	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	410	5	3	6	3.8	CC(=O)Nc1ccc(NC(=O)CCc2nc(O)c3c4c(sc3n2)CCCC4)cc1	nan
	CHEMBL1354869	25815	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	410	5	3	6	3.8	CC(=O)Nc1ccc(NC(=O)CCc2nc(O)c3c4c(sc3n2)CCCC4)cc1	nan
	2135022	25825	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	7	1	7	4.3	CCOc1ccc(NC(=O)Cn2cc(C(=O)c3ccc(C)cc3)c(=O)c3cc4c(cc32)OCO4)cc1	nan
	CHEMBL1354981	25825	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	7	1	7	4.3	CCOc1ccc(NC(=O)Cn2cc(C(=O)c3ccc(C)cc3)c(=O)c3cc4c(cc32)OCO4)cc1	nan
	135416424	25828	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	3	2	6	4.8	Cc1ccc2oc(-c3cc(NC(=O)c4ccc5c(c4)OCCO5)cc(C)c3O)nc2c1	nan
	CHEMBL1355004	25828	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	3	2	6	4.8	Cc1ccc2oc(-c3cc(NC(=O)c4ccc5c(c4)OCCO5)cc(C)c3O)nc2c1	nan
	16019041	25847	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	8	1	6	3.2	CC(C)OCCCNC(=O)c1ccc(Cn2c(=O)c3cccn3c3cccnc32)cc1	nan
	CHEMBL1355237	25847	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	8	1	6	3.2	CC(C)OCCCNC(=O)c1ccc(Cn2c(=O)c3cccn3c3cccnc32)cc1	nan
	135437043	25857	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	8	3	7	3.3	CCOc1ccc(-n2c(SCC(=O)NCc3ccccc3)nc3[nH]nc(C)c3c2=N)cc1	nan
	CHEMBL1355309	25857	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	8	3	7	3.3	CCOc1ccc(-n2c(SCC(=O)NCc3ccccc3)nc3[nH]nc(C)c3c2=N)cc1	nan
	16011751	25862	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	6	2	7	3.3	CCOC(=O)c1ccc(NC(=O)CC(=O)Nc2ccc3nc4n(c(=O)c3c2)CCCCC4)cc1	nan
	CHEMBL1355424	25862	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	6	2	7	3.3	CCOC(=O)c1ccc(NC(=O)CC(=O)Nc2ccc3nc4n(c(=O)c3c2)CCCCC4)cc1	nan
	16027630	25865	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	7	1	8	3.4	Cc1ccccc1OCC(=O)Nc1ccc(C(=O)OCc2cc(=O)n3ccsc3n2)cc1	nan
	CHEMBL1355500	25865	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	7	1	8	3.4	Cc1ccccc1OCC(=O)Nc1ccc(C(=O)OCc2cc(=O)n3ccsc3n2)cc1	nan
	16025481	25870	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	6	1	7	3.4	CCOc1ccc(NC(=O)CSc2ncc3c(n2)-c2ccccc2N(C)S3(=O)=O)cc1	nan
	CHEMBL1355611	25870	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	6	1	7	3.4	CCOc1ccc(NC(=O)CSc2ncc3c(n2)-c2ccccc2N(C)S3(=O)=O)cc1	nan
	16020103	25878	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	482	7	1	7	4.2	CCOc1ccc(CNC(=O)c2nn(-c3ccc(OC)cc3)c(=O)c3c2c2ccccc2n3C)cc1	nan
	CHEMBL1355692	25878	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	482	7	1	7	4.2	CCOc1ccc(CNC(=O)c2nn(-c3ccc(OC)cc3)c(=O)c3c2c2ccccc2n3C)cc1	nan
	16026942	25884	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	6	0	9	3.3	Cc1ccc(OCC(=O)OCc2cc(=O)n3nc(-c4cccs4)sc3n2)cc1	nan
	CHEMBL1355764	25884	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	6	0	9	3.3	Cc1ccc(OCC(=O)OCc2cc(=O)n3nc(-c4cccs4)sc3n2)cc1	nan
	16011703	25888	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	6	1	7	3.6	COc1ccc(CCNc2nc3ccc(Cl)cc3n3cnnc23)cc1OC	nan
	CHEMBL1355798	25888	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	6	1	7	3.6	COc1ccc(CCNc2nc3ccc(Cl)cc3n3cnnc23)cc1OC	nan
	16026082	25889	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	4	1	7	2.6	CCc1ccc(NC(=O)c2cnc3sc(N4CCCC4)nn3c2=O)cc1	nan
	CHEMBL1355799	25889	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	4	1	7	2.6	CCc1ccc(NC(=O)c2cnc3sc(N4CCCC4)nn3c2=O)cc1	nan
	16027128	25916	0	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	3	0	4	4.6	Cc1cc(=O)n(Cc2cccc(Br)c2)c2c1c(C)nn2-c1ccccc1	nan
	CHEMBL1356158	25916	0	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	3	0	4	4.6	Cc1cc(=O)n(Cc2cccc(Br)c2)c2c1c(C)nn2-c1ccccc1	nan
	16020942	25924	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	5	1	3	5.4	CC(NC(=O)Cn1c(-c2cccs2)cc2cc(F)ccc21)c1ccccc1	nan
	CHEMBL1356228	25924	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	5	1	3	5.4	CC(NC(=O)Cn1c(-c2cccs2)cc2cc(F)ccc21)c1ccccc1	nan
	2869380	25941	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	4	2	3	5.9	O=C(Nc1sc2c(c1C(=O)Nc1ccccc1Cl)CCCC2)c1ccccc1F	nan
	CHEMBL1356452	25941	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	4	2	3	5.9	O=C(Nc1sc2c(c1C(=O)Nc1ccccc1Cl)CCCC2)c1ccccc1F	nan
	4802695	25947	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	5	3	5	2.2	O=C(COC(=O)c1cc(Cl)ccc1O)NC(=O)NCc1ccccc1	nan
	CHEMBL1356574	25947	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	5	3	5	2.2	O=C(COC(=O)c1cc(Cl)ccc1O)NC(=O)NCc1ccccc1	nan
	16015066	25954	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	5	1	4	4.8	Cc1nc(SCC(=O)Nc2ccccc2Cl)cc(-c2ccccc2)n1	nan
	CHEMBL1356682	25954	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	5	1	4	4.8	Cc1nc(SCC(=O)Nc2ccccc2Cl)cc(-c2ccccc2)n1	nan
	16018801	25968	0	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	7	2	7	1.0	NS(=O)(=O)c1ccc(CCNC(=O)CCn2c(=O)c3cccn3c3cccnc32)cc1	nan
	CHEMBL1356848	25968	0	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	7	2	7	1.0	NS(=O)(=O)c1ccc(CCNC(=O)CCn2c(=O)c3cccn3c3cccnc32)cc1	nan
	24687225	25973	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	504	8	0	8	3.1	COc1cccc(COC(=O)c2cc(S(=O)(=O)N3CCCCC3)ccc2N2CCOCC2)c1OC	nan
	CHEMBL1356898	25973	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	504	8	0	8	3.1	COc1cccc(COC(=O)c2cc(S(=O)(=O)N3CCCCC3)ccc2N2CCOCC2)c1OC	nan
	16015534	25978	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	6	1	6	4.3	CCOC(=O)CSc1nc2ccc(NC(=O)c3ccc(F)cc3)cc2s1	nan
	CHEMBL1357001	25978	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	6	1	6	4.3	CCOC(=O)CSc1nc2ccc(NC(=O)c3ccc(F)cc3)cc2s1	nan
	15989556	25979	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	465	8	1	9	2.5	COc1ccc(NC(=O)Cn2c(=O)n(Cc3ccco3)c(=O)c3cc(OC)c(OC)cc32)cc1	nan
	CHEMBL1357013	25979	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	465	8	1	9	2.5	COc1ccc(NC(=O)Cn2c(=O)n(Cc3ccco3)c(=O)c3cc(OC)c(OC)cc32)cc1	nan
	16025511	25993	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	454	5	1	6	4.0	CCN1c2ccccc2-c2nc(SCC(=O)Nc3cccc(C)c3C)ncc2S1(=O)=O	nan
	CHEMBL1357149	25993	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	454	5	1	6	4.0	CCN1c2ccccc2-c2nc(SCC(=O)Nc3cccc(C)c3C)ncc2S1(=O)=O	nan
	20903553	26011	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	441	5	2	6	3.0	COc1ccc(NC(=O)C2CCCN(S(=O)(=O)c3ccc4nc(O)ccc4c3)C2)cc1	nan
	CHEMBL1357354	26011	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	441	5	2	6	3.0	COc1ccc(NC(=O)C2CCCN(S(=O)(=O)c3ccc4nc(O)ccc4c3)C2)cc1	nan
	16031127	26022	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	6	2	5	5.2	CSc1ccc(CNC(=O)c2ccccc2NC(=O)c2nsc3ccccc23)cc1	nan
	CHEMBL1357550	26022	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	6	2	5	5.2	CSc1ccc(CNC(=O)c2ccccc2NC(=O)c2nsc3ccccc23)cc1	nan
	1146087	26026	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	7	1	5	4.7	COc1ccc(-c2cc(C(F)(F)F)nc(SCC(=O)NCc3ccc(F)cc3)n2)cc1	nan
	CHEMBL1357694	26026	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	7	1	5	4.7	COc1ccc(-c2cc(C(F)(F)F)nc(SCC(=O)NCc3ccc(F)cc3)n2)cc1	nan
	16027571	26047	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	6	1	9	2.9	CS(=O)(=O)Nc1ccccc1C(=O)OCc1cc(=O)n2nc(C3CCCCC3)sc2n1	nan
	CHEMBL1358013	26047	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	6	1	9	2.9	CS(=O)(=O)Nc1ccccc1C(=O)OCc1cc(=O)n2nc(C3CCCCC3)sc2n1	nan
	16027432	26057	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	426	5	1	9	3.1	Cc1nn2c(=O)cc(COC(=O)c3ccccc3NC(=O)c3cccs3)nc2s1	nan
	CHEMBL1358125	26057	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	426	5	1	9	3.1	Cc1nn2c(=O)cc(COC(=O)c3ccccc3NC(=O)c3cccs3)nc2s1	nan
	16012175	26061	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	7	1	5	4.7	Cc1ccccc1Cn1c2ccccc2c2cnn(CC(=O)NCCc3ccc(Cl)cc3)c(=O)c21	nan
	CHEMBL1358188	26061	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	7	1	5	4.7	Cc1ccccc1Cn1c2ccccc2c2cnn(CC(=O)NCCc3ccc(Cl)cc3)c(=O)c21	nan
	16011822	26066	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	6	1	7	4.2	CCOc1ccc(NC(=O)C2CCN(c3nnc(-n4c(C)ccc4C)s3)CC2)cc1	nan
	CHEMBL1358209	26066	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	6	1	7	4.2	CCOc1ccc(NC(=O)C2CCN(c3nnc(-n4c(C)ccc4C)s3)CC2)cc1	nan
	16015787	26067	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	6	1	6	6.0	COc1ccc(-c2cc(C(=O)Nc3c(C(=O)c4ccc(C)c(F)c4)oc4ccccc34)no2)cc1	nan
	CHEMBL1358232	26067	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	6	1	6	6.0	COc1ccc(-c2cc(C(=O)Nc3c(C(=O)c4ccc(C)c(F)c4)oc4ccccc34)no2)cc1	nan
	16009454	26102	3	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	7	1	7	3.7	CC(Oc1ccccc1)C(=O)Nc1ccc(OCc2cc(=O)n3ccsc3n2)cc1	nan
	CHEMBL1358685	26102	3	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	7	1	7	3.7	CC(Oc1ccccc1)C(=O)Nc1ccc(OCc2cc(=O)n3ccsc3n2)cc1	nan
	16022826	26124	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	6	1	7	4.7	CCOc1ccc(NC(=O)C2CCN(c3nnc(C)c4c(C)n(-c5ccccc5)nc34)CC2)cc1	nan
	CHEMBL1358850	26124	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	6	1	7	4.7	CCOc1ccc(NC(=O)C2CCN(c3nnc(C)c4c(C)n(-c5ccccc5)nc34)CC2)cc1	nan
	654435	26146	14	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	4	1	6	4.2	O=C(CSc1nc2ccccc2o1)Nc1nc2ccccc2s1	nan
	CHEMBL1359027	26146	14	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	4	1	6	4.2	O=C(CSc1nc2ccccc2o1)Nc1nc2ccccc2s1	nan
	16009817	26153	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	4	1	7	5.0	Brc1cccc(-c2nnn3c2nc(NCc2ccc4c(c2)OCO4)c2ccccc23)c1	nan
	CHEMBL1359062	26153	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	4	1	7	5.0	Brc1cccc(-c2nnn3c2nc(NCc2ccc4c(c2)OCO4)c2ccccc23)c1	nan
	16009648	26225	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	5	0	5	4.3	COc1ccc(Cn2cc(S(=O)(=O)c3ccc(C)cc3)c(=O)c3cc(F)ccc32)cc1	nan
	CHEMBL1359678	26225	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	5	0	5	4.3	COc1ccc(Cn2cc(S(=O)(=O)c3ccc(C)cc3)c(=O)c3cc(F)ccc32)cc1	nan
	16020569	26261	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	5	0	5	4.3	CCCn1cc(S(=O)(=O)c2ccc(C)cc2)c(=O)c2cc(F)c(N3CCCC3)cc21	nan
	CHEMBL1360010	26261	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	5	0	5	4.3	CCCn1cc(S(=O)(=O)c2ccc(C)cc2)c(=O)c2cc(F)c(N3CCCC3)cc21	nan
	135546909	26273	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	464	7	2	6	3.7	COc1ccc(CN2CCc3nc(SCC(=O)Nc4cc(C)cc(C)c4)[nH]c(=O)c3C2)cc1	nan
	CHEMBL1360113	26273	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	464	7	2	6	3.7	COc1ccc(CN2CCc3nc(SCC(=O)Nc4cc(C)cc(C)c4)[nH]c(=O)c3C2)cc1	nan
	3185716	26297	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	564	10	3	8	3.7	CC(C)c1ccc(N(C(=O)c2snc(C(N)=O)c2N)C(C(=O)NCC2CCCO2)c2ccc(N(C)C)cc2)cc1	nan
	CHEMBL1360292	26297	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	564	10	3	8	3.7	CC(C)c1ccc(N(C(=O)c2snc(C(N)=O)c2N)C(C(=O)NCC2CCCO2)c2ccc(N(C)C)cc2)cc1	nan
	2819025	26316	13	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	235	1	1	5	1.9	N#Cc1cnc2cc(-c3ccccc3)nn2c1N	nan
	CHEMBL1360465	26316	13	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	235	1	1	5	1.9	N#Cc1cnc2cc(-c3ccccc3)nn2c1N	nan
	2141195	26337	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	6	1	5	4.7	CCc1ccc2c(c1)c(=O)c(S(=O)(=O)c1ccccc1)cn2CC(=O)Nc1cc(C)ccc1C	nan
	CHEMBL1360707	26337	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	6	1	5	4.7	CCc1ccc2c(c1)c(=O)c(S(=O)(=O)c1ccccc1)cn2CC(=O)Nc1cc(C)ccc1C	nan
	135436940	26339	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	5	1	7	5.0	Oc1cc(-c2ccc(F)cc2)nc(SCc2nc(-c3cccc(Cl)c3)no2)n1	nan
	CHEMBL1360713	26339	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	5	1	7	5.0	Oc1cc(-c2ccc(F)cc2)nc(SCc2nc(-c3cccc(Cl)c3)no2)n1	nan
	16009483	26358	3	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	9	1	7	1.4	CCCCN(C)CCNC(=O)C1CCCN(S(=O)(=O)c2ccc3c(c2)oc(=O)n3C)C1	nan
	CHEMBL1360843	26358	3	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	9	1	7	1.4	CCCCN(C)CCNC(=O)C1CCCN(S(=O)(=O)c2ccc3c(c2)oc(=O)n3C)C1	nan
	2135565	26409	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	502	7	1	7	4.2	CCOc1ccc(C(=O)c2cn(CC(=O)Nc3ccc4c(c3)OCCO4)c3ccc(F)cc3c2=O)cc1	nan
	CHEMBL1361368	26409	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	502	7	1	7	4.2	CCOc1ccc(C(=O)c2cn(CC(=O)Nc3ccc4c(c3)OCCO4)c3ccc(F)cc3c2=O)cc1	nan
	7598414	26471	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	4	1	5	2.8	Cc1cccc(Cn2cccc(C(=O)Nc3cc(C)on3)c2=O)c1	nan
	CHEMBL1361891	26471	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	4	1	5	2.8	Cc1cccc(Cn2cccc(C(=O)Nc3cc(C)on3)c2=O)c1	nan
	1071174	26473	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	8	1	7	3.8	CCOc1ccc(-n2c(SCC(=O)NCc3ccco3)nc3ccccc3c2=O)cc1	nan
	CHEMBL1361894	26473	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	8	1	7	3.8	CCOc1ccc(-n2c(SCC(=O)NCc3ccco3)nc3ccccc3c2=O)cc1	nan
	857565	26538	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	4	1	5	4.2	Cc1cc(NC(=O)CSc2nc3c(C)c(C)ccc3cc2C)no1	nan
	CHEMBL1362451	26538	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	4	1	5	4.2	Cc1cc(NC(=O)CSc2nc3c(C)c(C)ccc3cc2C)no1	nan
	790083	26636	50	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	330	3	0	4	4.2	COc1ccccc1-c1nc(-c2ccc(Br)cc2)no1	nan
	CHEMBL1363291	26636	50	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	330	3	0	4	4.2	COc1ccccc1-c1nc(-c2ccc(Br)cc2)no1	nan
	2137970	26695	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	482	6	1	6	4.1	COc1ccc(S(=O)(=O)c2cn(CC(=O)Nc3ccccc3)c3ccc(Cl)cc3c2=O)cc1	nan
	CHEMBL1363852	26695	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	482	6	1	6	4.1	COc1ccc(S(=O)(=O)c2cn(CC(=O)Nc3ccccc3)c3ccc(Cl)cc3c2=O)cc1	nan
	22522543	26744	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	331	3	1	4	3.2	Cc1ccc(NC(=O)Cn2c(=O)c3cccn3c3ccccc32)cc1	nan
	CHEMBL1364334	26744	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	331	3	1	4	3.2	Cc1ccc(NC(=O)Cn2c(=O)c3cccn3c3ccccc32)cc1	nan
	1581690	26785	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	10	2	6	4.6	CCCCCOc1ccc(C(=O)Nc2ccc(S(=O)(=O)Nc3cc(C)on3)cc2)cc1	nan
	CHEMBL1364631	26785	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	10	2	6	4.6	CCCCCOc1ccc(C(=O)Nc2ccc(S(=O)(=O)Nc3cc(C)on3)cc2)cc1	nan
	1759638	26813	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	513	5	1	5	5.3	Cc1c(CCC(=O)N2CCC(C(=O)O)(c3ccccc3)CC2)c(=O)oc2cc3oc4c(c3cc12)CCCC4	nan
	CHEMBL1364853	26813	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	513	5	1	5	5.3	Cc1c(CCC(=O)N2CCC(C(=O)O)(c3ccccc3)CC2)c(=O)oc2cc3oc4c(c3cc12)CCCC4	nan
	2137118	26914	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	494	6	1	6	4.2	COc1ccc2c(c1)c(=O)c(S(=O)(=O)c1ccc(F)cc1)cn2CC(=O)Nc1ccc(C)cc1C	nan
	CHEMBL1365673	26914	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	494	6	1	6	4.2	COc1ccc2c(c1)c(=O)c(S(=O)(=O)c1ccc(F)cc1)cn2CC(=O)Nc1ccc(C)cc1C	nan
	16008395	26940	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	7	1	6	3.7	CCn1c(=O)cc(OCC(=O)Nc2cc(Cl)c(OC)cc2OC)c2ccccc21	nan
	CHEMBL1365942	26940	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	7	1	6	3.7	CCn1c(=O)cc(OCC(=O)Nc2cc(Cl)c(OC)cc2OC)c2ccccc21	nan
	2155747	26949	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	7	1	8	3.2	CCOc1ccc(-c2nnc(SCC(=O)Nc3cc(C)on3)o2)cc1	nan
	CHEMBL1366006	26949	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	7	1	8	3.2	CCOc1ccc(-c2nnc(SCC(=O)Nc3cc(C)on3)o2)cc1	nan
	16012964	26951	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	5	1	3	5.0	CCCN(Cc1cc2cc(C)ccc2nc1O)C(=O)c1cccc(Cl)c1	nan
	CHEMBL1366015	26951	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	5	1	3	5.0	CCCN(Cc1cc2cc(C)ccc2nc1O)C(=O)c1cccc(Cl)c1	nan
	2474394	27003	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	363	3	1	4	3.5	CCCn1c(=O)[nH]c(=O)c2c(C(F)(F)F)cc(-c3ccc(C)cc3)nc21	nan
	CHEMBL1366444	27003	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	363	3	1	4	3.5	CCCn1c(=O)[nH]c(=O)c2c(C(F)(F)F)cc(-c3ccc(C)cc3)nc21	nan
	17757029	27035	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	7	0	8	4.6	CCOC(=O)COc1ccc([N+](=O)[O-])cc1-c1ccnc2cc(-c3ccc(Cl)cc3)nn12	nan
	CHEMBL1366773	27035	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	7	0	8	4.6	CCOC(=O)COc1ccc([N+](=O)[O-])cc1-c1ccnc2cc(-c3ccc(Cl)cc3)nn12	nan
	5087310	27187	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	5	1	7	2.8	COc1cc2c(cc1OC)n(CC(=O)NC1CCCCCC1)n1c(C)cc(=O)nc21	nan
	CHEMBL1367963	27187	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	412	5	1	7	2.8	COc1cc2c(cc1OC)n(CC(=O)NC1CCCCCC1)n1c(C)cc(=O)nc21	nan
	4825943	27196	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	4	1	7	2.8	CC(Sc1nc2ccccc2c(=O)n1C)C(=O)Nc1ccc2c(c1)OCCO2	nan
	CHEMBL1368013	27196	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	4	1	7	2.8	CC(Sc1nc2ccccc2c(=O)n1C)C(=O)Nc1ccc2c(c1)OCCO2	nan
	16022825	27216	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	463	5	1	10	1.9	Cc1ccc(C)c(NC(=O)Cn2c(=O)n(Cc3nc(C)no3)c(=O)c3cc4c(cc32)OCO4)c1	nan
	CHEMBL1368194	27216	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	463	5	1	10	1.9	Cc1ccc(C)c(NC(=O)Cn2c(=O)n(Cc3nc(C)no3)c(=O)c3cc4c(cc32)OCO4)c1	nan
	709853	27259	17	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	5	1	5	2.7	COc1ccc(CNC(=O)c2cc3cccc(OC)c3oc2=O)cc1	nan
	CHEMBL1368522	27259	17	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	5	1	5	2.7	COc1ccc(CNC(=O)c2cc3cccc(OC)c3oc2=O)cc1	nan
	16019023	27279	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	8	1	6	2.9	CCOCCCNC(=O)c1ccc(Cn2c(=O)c3cccn3c3cccnc32)cc1	nan
	CHEMBL1368698	27279	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	8	1	6	2.9	CCOCCCNC(=O)c1ccc(Cn2c(=O)c3cccn3c3cccnc32)cc1	nan
	1898787	27294	18	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	4	1	8	1.9	COC(=O)CSc1nc(N)c(C#N)c(-c2ccco2)c1C#N	nan
	CHEMBL1368847	27294	18	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	4	1	8	1.9	COC(=O)CSc1nc(N)c(C#N)c(-c2ccco2)c1C#N	nan
	16746213	27308	0	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	542	11	3	5	4.4	NC(=O)CC(NC(=O)Cc1ccc(Br)cc1)c1ccc(NCCc2ccccc2F)c([N+](=O)[O-])c1	nan
	CHEMBL1368944	27308	0	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	542	11	3	5	4.4	NC(=O)CC(NC(=O)Cc1ccc(Br)cc1)c1ccc(NCCc2ccccc2F)c([N+](=O)[O-])c1	nan
	15989069	27310	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	528	12	1	9	2.7	CCN(CC)C(=O)Cn1c(=O)n(CCCCCC(=O)NCc2ccc3c(c2)OCO3)c(=O)c2sccc21	nan
	CHEMBL1368950	27310	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	528	12	1	9	2.7	CCN(CC)C(=O)Cn1c(=O)n(CCCCCC(=O)NCc2ccc3c(c2)OCO3)c(=O)c2sccc21	nan
	3417357	27350	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	495	4	0	6	4.9	Cc1cc(C)c(Cn2c(=O)n(-c3ccccc3Cl)c(=O)c3c(C)c(C(=O)N(C)C)sc32)c(C)c1	nan
	CHEMBL1369202	27350	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	495	4	0	6	4.9	Cc1cc(C)c(Cn2c(=O)n(-c3ccccc3Cl)c(=O)c3c(C)c(C(=O)N(C)C)sc32)c(C)c1	nan
	4454678	27378	12	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	5	1	7	4.4	Cc1cc(OCC(=O)Nc2cc(-c3nn4c(C)nnc4s3)ccc2C)ccc1Cl	nan
	CHEMBL1369422	27378	12	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	5	1	7	4.4	Cc1cc(OCC(=O)Nc2cc(-c3nn4c(C)nnc4s3)ccc2C)ccc1Cl	nan
	16034378	27456	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	325	7	1	4	3.5	COc1ccc(C(=O)CCC(=O)Nc2cccc(C(C)=O)c2)cc1	nan
	CHEMBL1369934	27456	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	325	7	1	4	3.5	COc1ccc(C(=O)CCC(=O)Nc2cccc(C(C)=O)c2)cc1	nan
	16746462	27477	0	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	400	8	1	6	3.3	COc1cc(O)c(C(CCN2CCOCC2)c2ccc(N(C)C)cc2)c(OC)c1	nan
	CHEMBL1370067	27477	0	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	400	8	1	6	3.3	COc1cc(O)c(C(CCN2CCOCC2)c2ccc(N(C)C)cc2)c(OC)c1	nan
	3236293	27479	9	None	-3	3	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	7	1	8	3.3	CCCCn1c(SCC(=O)Nc2cc(C)on2)nc2ccsc2c1=O	nan
	CHEMBL1370078	27479	9	None	-3	3	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	7	1	8	3.3	CCCCn1c(SCC(=O)Nc2cc(C)on2)nc2ccsc2c1=O	nan
	5310561	27531	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	5	2	7	2.8	CCOc1ccccc1-c1nc(C(N)=O)c2nc(O)n(-c3ccc(F)cc3)c2n1	nan
	CHEMBL1370473	27531	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	5	2	7	2.8	CCOc1ccccc1-c1nc(C(N)=O)c2nc(O)n(-c3ccc(F)cc3)c2n1	nan
	667326	27544	11	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	7	1	5	3.5	CCOCCCNc1ncc2c(n1)CC(c1ccc(C)cc1)CC2=O	nan
	CHEMBL1370544	27544	11	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	7	1	5	3.5	CCOCCCNc1ncc2c(n1)CC(c1ccc(C)cc1)CC2=O	nan
	135546918	27557	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	6	2	6	3.6	CCCN1CCc2nc(SCC(=O)Nc3ccc(C)c(Cl)c3)nc(O)c2C1	nan
	CHEMBL1370635	27557	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	6	2	6	3.6	CCCN1CCc2nc(SCC(=O)Nc3ccc(C)c(Cl)c3)nc(O)c2C1	nan
	3628612	27588	16	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	7	1	5	4.4	CCc1nc(SCC(=O)NCCc2ccccc2)c2oc3ccccc3c2n1	nan
	CHEMBL1370855	27588	16	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	7	1	5	4.4	CCc1nc(SCC(=O)NCCc2ccccc2)c2oc3ccccc3c2n1	nan
	1348188	27734	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	4	1	3	5.6	Cc1cccc(-c2nc3cc(NC(=O)Cc4ccc(Cl)cc4)ccc3o2)c1	nan
	CHEMBL1372034	27734	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	4	1	3	5.6	Cc1cccc(-c2nc3cc(NC(=O)Cc4ccc(Cl)cc4)ccc3o2)c1	nan
	1854798	27759	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	1	0	5	3.6	Cn1c(=O)nc2n(-c3ccc(Br)cc3)c3cccc(Cl)c3cc-2c1=O	nan
	CHEMBL1372184	27759	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	1	0	5	3.6	Cn1c(=O)nc2n(-c3ccc(Br)cc3)c3cccc(Cl)c3cc-2c1=O	nan
	16019423	27829	1	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	6	1	9	5.0	CC(C)c1ccc(S(=O)(=O)c2nnn3c2nc(NCc2cccs2)c2sccc23)cc1	nan
	CHEMBL1372659	27829	1	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	6	1	9	5.0	CC(C)c1ccc(S(=O)(=O)c2nnn3c2nc(NCc2cccs2)c2sccc23)cc1	nan
	16031591	27889	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	5	0	6	3.4	CC(=O)c1ccc(N2CCN(S(=O)(=O)c3ccc(-c4coc(C)n4)cc3)CC2)cc1	nan
	CHEMBL1373010	27889	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	5	0	6	3.4	CC(=O)c1ccc(N2CCN(S(=O)(=O)c3ccc(-c4coc(C)n4)cc3)CC2)cc1	nan
	2684697	27963	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	3	1	5	3.7	COc1ccc(C)cc1NC(=O)c1ccc2c(=O)n3c(nc2c1)CCCCC3	nan
	CHEMBL1373515	27963	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	3	1	5	3.7	COc1ccc(C)cc1NC(=O)c1ccc2c(=O)n3c(nc2c1)CCCCC3	nan
	652717	27979	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	7	2	5	5.1	CCN1CCCC1CN(Cc1cc2cc(C)cc(C)c2nc1O)C(=O)Nc1ccccc1OC	nan
	CHEMBL1373605	27979	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	7	2	5	5.1	CCN1CCCC1CN(Cc1cc2cc(C)cc(C)c2nc1O)C(=O)Nc1ccccc1OC	nan
	16015413	27990	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	8	1	6	6.2	COc1cc(C)ccc1OCCSc1nc2ccc(NC(=O)c3ccc(F)cc3)cc2s1	nan
	CHEMBL1373657	27990	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	8	1	6	6.2	COc1cc(C)ccc1OCCSc1nc2ccc(NC(=O)c3ccc(F)cc3)cc2s1	nan
	16033161	28026	3	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	497	8	2	5	4.6	O=C(Nc1ccc(N2CCN(CCOc3ccc(Cl)cc3)CC2)c(C(=O)O)c1)c1ccc(F)cc1	nan
	CHEMBL1373926	28026	3	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	497	8	2	5	4.6	O=C(Nc1ccc(N2CCN(CCOc3ccc(Cl)cc3)CC2)c(C(=O)O)c1)c1ccc(F)cc1	nan
	16030696	28032	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	489	6	1	9	2.9	CC(=O)c1ccc(NC(=O)CSc2nc(-c3ccccc3C)nc3c2c(=O)n(C)c(=O)n3C)cc1	nan
	CHEMBL1374004	28032	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	489	6	1	9	2.9	CC(=O)c1ccc(NC(=O)CSc2nc(-c3ccccc3C)nc3c2c(=O)n(C)c(=O)n3C)cc1	nan
	15997814	28077	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	361	5	2	6	4.2	COc1cc2nc(S)nc(NCc3cccc(Cl)c3)c2cc1OC	nan
	CHEMBL1374312	28077	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	361	5	2	6	4.2	COc1cc2nc(S)nc(NCc3cccc(Cl)c3)c2cc1OC	nan
	4521283	28084	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	525	4	1	5	4.7	O=C(CN1C(=O)c2ccccc2Sc2ccc(C(=O)N3CCOCC3)cc21)Nc1ccc(Cl)cc1F	nan
	CHEMBL1374381	28084	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	525	4	1	5	4.7	O=C(CN1C(=O)c2ccccc2Sc2ccc(C(=O)N3CCOCC3)cc21)Nc1ccc(Cl)cc1F	nan
	3734127	28122	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	5	2	4	4.0	CCc1ccc(NC(=O)CSc2nc3cc(Br)c[nH]c-3n2)cc1	nan
	CHEMBL1374637	28122	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	5	2	4	4.0	CCc1ccc(NC(=O)CSc2nc3cc(Br)c[nH]c-3n2)cc1	nan
	669593	28137	14	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	248	2	1	5	2.1	O=C(Nc1nccs1)c1ccc2c(c1)OCO2	nan
	CHEMBL1374723	28137	14	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	248	2	1	5	2.1	O=C(Nc1nccs1)c1ccc2c(c1)OCO2	nan
	656234	28178	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	4	1	7	3.3	O=c1c2ccccc2nc(CSc2[nH]cnc3ncnc2-3)n1-c1ccccc1	nan
	CHEMBL1375001	28178	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	4	1	7	3.3	O=c1c2ccccc2nc(CSc2[nH]cnc3ncnc2-3)n1-c1ccccc1	nan
	4074625	28192	14	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	305	3	3	6	0.3	COC(=O)c1ccccc1NC=C1C(=O)NC(=S)NC1=O	nan
	CHEMBL1375120	28192	14	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	305	3	3	6	0.3	COC(=O)c1ccccc1NC=C1C(=O)NC(=S)NC1=O	nan
	828451	28292	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	303	4	1	4	4.6	CCOc1ccc(Nc2nc3c(C)cccc3cc2C#N)cc1	nan
	CHEMBL1375831	28292	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	303	4	1	4	4.6	CCOc1ccc(Nc2nc3c(C)cccc3cc2C#N)cc1	nan
	7246250	28297	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	3	0	5	3.4	COc1cc(Br)cc2cc(S(=O)(=O)c3ccccc3)c(=O)oc12	nan
	CHEMBL1375897	28297	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	3	0	5	3.4	COc1cc(Br)cc2cc(S(=O)(=O)c3ccccc3)c(=O)oc12	nan
	16029523	28319	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	478	5	0	6	2.3	CN(C)S(=O)(=O)c1ccc2c(c1)N(CC(=O)N1CCN(c3ccc(F)cc3)CC1)CCS2	nan
	CHEMBL1376205	28319	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	478	5	0	6	2.3	CN(C)S(=O)(=O)c1ccc2c(c1)N(CC(=O)N1CCN(c3ccc(F)cc3)CC1)CCS2	nan
	4048244	28347	10	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	546	13	1	8	4.1	CCOC(=O)c1sc(-c2ccccc2)cc1NC(=O)c1ccc(S(=O)(=O)N(CCOC)CCOC)cc1	nan
	CHEMBL1376427	28347	10	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	546	13	1	8	4.1	CCOC(=O)c1sc(-c2ccccc2)cc1NC(=O)c1ccc(S(=O)(=O)N(CCOC)CCOC)cc1	nan
	1629947	28386	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	4	2	4	1.6	O=C1NC(=S)NC(=O)C1=Cc1ccc2c(c1)CCN2CCCCl	nan
	CHEMBL1376754	28386	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	4	2	4	1.6	O=C1NC(=S)NC(=O)C1=Cc1ccc2c(c1)CCN2CCCCl	nan
	1281315	28402	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	489	4	2	6	6.1	COc1ccc(-c2c3c(nc4sc(C(=O)Nc5ccccc5F)c(N)c24)CC(C)(C)CC3=O)cc1	nan
	CHEMBL1376941	28402	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	489	4	2	6	6.1	COc1ccc(-c2c3c(nc4sc(C(=O)Nc5ccccc5F)c(N)c24)CC(C)(C)CC3=O)cc1	nan
	3640458	28426	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	505	6	1	7	3.6	CCOC(=O)c1c(NC(=O)c2ccc(S(=O)(=O)N3CCC(C)CC3)cc2)sc2c1CCN(C)C2	nan
	CHEMBL1377235	28426	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	505	6	1	7	3.6	CCOC(=O)c1c(NC(=O)c2ccc(S(=O)(=O)N3CCC(C)CC3)cc2)sc2c1CCN(C)C2	nan
	4307577	28462	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	466	10	2	4	6.4	CC(C)c1ccc(Nc2cc(C(=O)NCCCN(C)Cc3ccccc3)c3ccccc3n2)cc1	nan
	CHEMBL1377592	28462	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	466	10	2	4	6.4	CC(C)c1ccc(Nc2cc(C(=O)NCCCN(C)Cc3ccccc3)c3ccccc3n2)cc1	nan
	16193746	28542	5	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	489	4	1	6	2.3	Cc1ccc(N2C(=O)C3C4C=CC(CN=C(S)N5CCN(c6ccccn6)CC5)(O4)C3C2=O)cc1	nan
	CHEMBL1378295	28542	5	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	489	4	1	6	2.3	Cc1ccc(N2C(=O)C3C4C=CC(CN=C(S)N5CCN(c6ccccn6)CC5)(O4)C3C2=O)cc1	nan
	2220966	28584	10	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	297	2	1	3	3.4	Cc1c(Cl)ccc2c(C(N)=O)cc(-c3ccccn3)nc12	nan
	CHEMBL1378741	28584	10	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	297	2	1	3	3.4	Cc1c(Cl)ccc2c(C(N)=O)cc(-c3ccccn3)nc12	nan
	7422753	28599	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	347	5	2	4	2.2	NC(=O)c1ccc(NC(=O)c2cccn(Cc3ccccc3)c2=O)cc1	nan
	CHEMBL1378862	28599	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	347	5	2	4	2.2	NC(=O)c1ccc(NC(=O)c2cccn(Cc3ccccc3)c2=O)cc1	nan
	2815317	28607	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	2	0	5	3.8	Cc1cc(C)c2c(n1)sc1c(=O)n(Cc3ccc(F)cc3)cnc12	nan
	CHEMBL1378935	28607	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	2	0	5	3.8	Cc1cc(C)c2c(n1)sc1c(=O)n(Cc3ccc(F)cc3)cnc12	nan
	16193948	28623	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	5	2	6	3.5	CCOC(=O)c1[nH]c2ccc(OC)cc2c1N=C(S)N1CCN(c2ccccn2)CC1	nan
	CHEMBL1379050	28623	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	5	2	6	3.5	CCOC(=O)c1[nH]c2ccc(OC)cc2c1N=C(S)N1CCN(c2ccccn2)CC1	nan
	24746968	28744	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	4	1	6	4.1	Cc1nc(Nc2ccccc2F)c2nnn(Cc3ccccc3Cl)c2n1	nan
	CHEMBL1380147	28744	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	4	1	6	4.1	Cc1nc(Nc2ccccc2F)c2nnn(Cc3ccccc3Cl)c2n1	nan
	725312	28767	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	4	1	6	3.0	CCn1cnc2sc(C(=O)Nc3ccccc3OC)c(C)c2c1=O	nan
	CHEMBL1380313	28767	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	4	1	6	3.0	CCn1cnc2sc(C(=O)Nc3ccccc3OC)c(C)c2c1=O	nan
	24792708	28800	3	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	8	2	7	3.3	COc1ccc(CNC(=O)CSc2nnc(NC(=O)c3ccccc3F)s2)cc1	nan
	CHEMBL1380537	28800	3	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	8	2	7	3.3	COc1ccc(CNC(=O)CSc2nnc(NC(=O)c3ccccc3F)s2)cc1	nan
	3604840	28830	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	4	1	5	3.7	COc1cccc(-c2cc(C(=O)Nc3cccnc3Cl)no2)c1	nan
	CHEMBL1380782	28830	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	4	1	5	3.7	COc1cccc(-c2cc(C(=O)Nc3cccnc3Cl)no2)c1	nan
	1980822	28983	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	361	5	2	4	3.9	COc1ccc(C(=O)Nc2ccccc2C(=O)Nc2cccc(C)n2)cc1	nan
	CHEMBL1382084	28983	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	361	5	2	4	3.9	COc1ccc(C(=O)Nc2ccccc2C(=O)Nc2cccc(C)n2)cc1	nan
	555289	29043	19	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	311	4	1	4	3.6	Cc1cc(C)c(C#N)c(SCC(=O)Nc2ccccc2C)n1	nan
	CHEMBL1382619	29043	19	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	311	4	1	4	3.6	Cc1cc(C)c(C#N)c(SCC(=O)Nc2ccccc2C)n1	nan
	9550495	29239	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	5	1	5	4.2	Cc1ccc(-c2nc3ncccc3o2)cc1NC(=O)COc1ccccc1	nan
	CHEMBL1384380	29239	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	5	1	5	4.2	Cc1ccc(-c2nc3ncccc3o2)cc1NC(=O)COc1ccccc1	nan
	7161160	29256	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	5	1	7	0.3	CCOc1ccccc1NS(=O)(=O)c1cn(C)c(=O)n(C)c1=O	nan
	CHEMBL1384530	29256	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	5	1	7	0.3	CCOc1ccccc1NS(=O)(=O)c1cn(C)c(=O)n(C)c1=O	nan
	4271811	29311	17	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	336	6	0	5	3.2	CCCc1nc2ccccc2c(=O)n1CC(=O)c1ccc(OC)cc1	nan
	CHEMBL1384958	29311	17	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	336	6	0	5	3.2	CCCc1nc2ccccc2c(=O)n1CC(=O)c1ccc(OC)cc1	nan
	2123263	29320	7	None	-5	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	495	7	2	9	3.5	CCCn1c(N)c(-c2nc(C3CCCC3)c(C(=O)c3ccc(NC(C)=O)cc3)s2)c(=O)n(C)c1=O	nan
	CHEMBL1385062	29320	7	None	-5	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	495	7	2	9	3.5	CCCn1c(N)c(-c2nc(C3CCCC3)c(C(=O)c3ccc(NC(C)=O)cc3)s2)c(=O)n(C)c1=O	nan
	3243476	29366	10	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	322	1	1	4	3.4	CC(=O)Nc1nc2c(c3c1c(=O)oc1ccccc13)CC(C)CC2	nan
	CHEMBL1385469	29366	10	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	322	1	1	4	3.4	CC(=O)Nc1nc2c(c3c1c(=O)oc1ccccc13)CC(C)CC2	nan
	645034	29418	4	None	-6	3	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	295	1	0	5	2.9	N#Cc1cc2cc3c(cc2nc1N1CCCCC1)OCCO3	nan
	CHEMBL1385946	29418	4	None	-6	3	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	295	1	0	5	2.9	N#Cc1cc2cc3c(cc2nc1N1CCCCC1)OCCO3	nan
	1233014	29439	9	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	290	4	1	6	2.4	Cc1ccc(C#N)c(SCC(=O)Nc2nccs2)n1	nan
	CHEMBL1386142	29439	9	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	290	4	1	6	2.4	Cc1ccc(C#N)c(SCC(=O)Nc2nccs2)n1	nan
	818106	29467	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	302	3	0	4	4.0	COc1ccc(-c2nc3c4ccccc4ccn3c2C=O)cc1	nan
	CHEMBL1386316	29467	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	302	3	0	4	4.0	COc1ccc(-c2nc3c4ccccc4ccn3c2C=O)cc1	nan
	2803005	29470	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	326	2	1	2	3.8	NC(=O)c1cc(-c2ccccc2)nc2ccc(Br)cc12	nan
	CHEMBL1386328	29470	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	326	2	1	2	3.8	NC(=O)c1cc(-c2ccccc2)nc2ccc(Br)cc12	nan
	743778	29504	12	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	243	1	1	3	3.2	Cc1cc(-c2ccc(Cl)cc2)c(C#N)c(N)n1	nan
	CHEMBL1386595	29504	12	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	243	1	1	3	3.2	Cc1cc(-c2ccc(Cl)cc2)c(C#N)c(N)n1	nan
	1078300	29508	9	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	5	1	6	4.4	COc1ccccc1NC(=O)c1sc2ncn(Cc3cccc(C)c3)c(=O)c2c1C	nan
	CHEMBL1386617	29508	9	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	5	1	6	4.4	COc1ccccc1NC(=O)c1sc2ncn(Cc3cccc(C)c3)c(=O)c2c1C	nan
	2197659	29560	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	5	1	5	2.6	COc1ccc2c(c1)c(=O)oc1cc(OCC(=O)NC3CC3)ccc12	nan
	CHEMBL1387003	29560	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	5	1	5	2.6	COc1ccc2c(c1)c(=O)oc1cc(OCC(=O)NC3CC3)ccc12	nan
	2368754	29582	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	306	2	0	4	2.1	CCN1C(=O)C(=C2C=C(C)OC(C)=C2)C(=O)N(CC)C1=S	nan
	CHEMBL1387204	29582	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	306	2	0	4	2.1	CCN1C(=O)C(=C2C=C(C)OC(C)=C2)C(=O)N(CC)C1=S	nan
	1590813	29627	18	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	3	1	1	5.9	O=C(Nc1ccc(Cl)cc1Cl)c1ccc(-c2ccccc2)cc1	nan
	CHEMBL1387594	29627	18	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	3	1	1	5.9	O=C(Nc1ccc(Cl)cc1Cl)c1ccc(-c2ccccc2)cc1	nan
	16194196	29640	0	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	7	1	8	2.6	CCOC(=O)N1CCN(C(=O)CCCCCn2c(=S)[nH]c3cc4c(cc3c2=O)OCO4)CC1	nan
	CHEMBL1387679	29640	0	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	7	1	8	2.6	CCOC(=O)N1CCN(C(=O)CCCCCn2c(=S)[nH]c3cc4c(cc3c2=O)OCO4)CC1	nan
	3961803	29662	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	4	1	8	-0.6	Cn1nc(C(=O)OCC(=O)NC2CCS(=O)(=O)C2)c2ccccc2c1=O	nan
	CHEMBL1387823	29662	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	4	1	8	-0.6	Cn1nc(C(=O)OCC(=O)NC2CCS(=O)(=O)C2)c2ccccc2c1=O	nan
	649021	29711	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	472	5	1	9	3.8	Cc1cccc2cc(C(c3nnnn3Cc3ccc4c(c3)OCO4)N3CCC(C)CC3)c(O)nc12	nan
	CHEMBL1388237	29711	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	472	5	1	9	3.8	Cc1cccc2cc(C(c3nnnn3Cc3ccc4c(c3)OCO4)N3CCC(C)CC3)c(O)nc12	nan
	2565451	29728	7	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	6	1	7	2.1	CCOC(=O)c1sc(NC(=O)c2ccc(S(=O)(=O)N(C)C)cc2)nc1C	nan
	CHEMBL1388388	29728	7	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	6	1	7	2.1	CCOC(=O)c1sc(NC(=O)c2ccc(S(=O)(=O)N(C)C)cc2)nc1C	nan
	20874214	29755	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	410	6	1	8	3.7	CC(C)c1nn2c(=O)cc(COc3cccc(NC(=O)c4ccco4)c3)nc2s1	nan
	CHEMBL1388517	29755	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	410	6	1	8	3.7	CC(C)c1nn2c(=O)cc(COc3cccc(NC(=O)c4ccco4)c3)nc2s1	nan
	736044	29814	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	320	3	2	5	1.3	NS(=O)(=O)c1ccc(NC(=O)c2ccc3c(c2)OCO3)cc1	nan
	CHEMBL1389015	29814	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	320	3	2	5	1.3	NS(=O)(=O)c1ccc(NC(=O)c2ccc3c(c2)OCO3)cc1	nan
	3581200	29883	4	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	6	1	5	4.9	O=C(Nc1nc(-c2ccc(F)c(F)c2)cs1)c1ccc(OCC2CCCO2)cc1	nan
	CHEMBL1389543	29883	4	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	6	1	5	4.9	O=C(Nc1nc(-c2ccc(F)c(F)c2)cs1)c1ccc(OCC2CCCO2)cc1	nan
	2815149	29999	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	299	1	0	4	3.3	Cn1c2ccccc2n2c(=O)cc(-c3ccccc3)c(C#N)c12	nan
	CHEMBL1390567	29999	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	299	1	0	4	3.3	Cn1c2ccccc2n2c(=O)cc(-c3ccccc3)c(C#N)c12	nan
	1480454	30145	17	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	301	3	0	5	3.1	CN(C)c1nc(-c2cccnc2)nc(-c2ccccc2)c1C#N	nan
	CHEMBL1391874	30145	17	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	301	3	0	5	3.1	CN(C)c1nc(-c2cccnc2)nc(-c2ccccc2)c1C#N	nan
	3151961	30155	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	291	3	1	6	2.6	CC(C)c1nnc(NC(=O)c2ccc3c(c2)OCO3)s1	nan
	CHEMBL1391972	30155	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	291	3	1	6	2.6	CC(C)c1nnc(NC(=O)c2ccc3c(c2)OCO3)s1	nan
	2818919	30295	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	351	2	0	5	5.2	FC(F)(F)c1cc(-c2cccs2)nc2cc(-c3cccs3)nn12	nan
	CHEMBL1393159	30295	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	351	2	0	5	5.2	FC(F)(F)c1cc(-c2cccs2)nc2cc(-c3cccs3)nn12	nan
	3597887	30302	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	486	8	1	7	4.2	Cc1ccc(-c2nc(S(=O)(=O)c3ccc(C)cc3)c(SCC(=O)NCC3CCCO3)o2)cc1	nan
	CHEMBL1393192	30302	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	486	8	1	7	4.2	Cc1ccc(-c2nc(S(=O)(=O)c3ccc(C)cc3)c(SCC(=O)NCC3CCCO3)o2)cc1	nan
	6498520	30352	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	6	1	6	2.9	CN=C(S)N(Cc1cc2cc(C)ccc2n2nnnc12)CC(C)(C)CN(C)C	nan
	CHEMBL1393589	30352	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	6	1	6	2.9	CN=C(S)N(Cc1cc2cc(C)ccc2n2nnnc12)CC(C)(C)CN(C)C	nan
	938851	30385	11	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	299	3	1	5	3.7	Cc1ccc2nc(O)c(COC(=O)c3cccs3)cc2c1	nan
	CHEMBL1393863	30385	11	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	299	3	1	5	3.7	Cc1ccc2nc(O)c(COC(=O)c3cccs3)cc2c1	nan
	2810066	30395	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	4	1	6	2.9	COc1cc2nc(NC(=O)c3ccccc3)sc(=O)c2cc1OC	nan
	CHEMBL1393944	30395	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	4	1	6	2.9	COc1cc2nc(NC(=O)c3ccccc3)sc(=O)c2cc1OC	nan
	16010814	30407	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	441	3	0	7	4.3	Clc1cccc(N2CCN(c3nc4ccccc4c4nc(-c5cccnc5)nn34)CC2)c1	nan
	CHEMBL1394069	30407	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	441	3	0	7	4.3	Clc1cccc(N2CCN(c3nc4ccccc4c4nc(-c5cccnc5)nn34)CC2)c1	nan
	16018745	30421	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	7	2	3	5.9	Cc1ccc(Cn2c(C(=O)O)c(CNCc3ccccc3Cl)c3ccc(C)cc32)cc1	nan
	CHEMBL1394183	30421	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	7	2	3	5.9	Cc1ccc(Cn2c(C(=O)O)c(CNCc3ccccc3Cl)c3ccc(C)cc32)cc1	nan
	16030321	30422	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	6	1	6	3.8	COc1ccccc1C(=O)Nc1ccc(OCc2cc(=O)n3cccc(C)c3n2)cc1	nan
	CHEMBL1394221	30422	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	6	1	6	3.8	COc1ccccc1C(=O)Nc1ccc(OCc2cc(=O)n3cccc(C)c3n2)cc1	nan
	16019476	30424	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	6	1	9	4.4	CCc1ccc(S(=O)(=O)c2nnn3c2nc(NCc2cccs2)c2sccc23)cc1	nan
	CHEMBL1394231	30424	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	6	1	9	4.4	CCc1ccc(S(=O)(=O)c2nnn3c2nc(NCc2cccs2)c2sccc23)cc1	nan
	16012300	30429	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	293	3	1	2	5.0	Cc1ccc(NC(=O)c2ccc(-c3ccccc3)s2)cc1	nan
	CHEMBL1394287	30429	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	293	3	1	2	5.0	Cc1ccc(NC(=O)c2ccc(-c3ccccc3)s2)cc1	nan
	16015419	30460	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	464	8	1	6	6.3	COc1cc(C)ccc1OCCSc1nc2ccc(NC(=O)c3ccc(C)cc3)cc2s1	nan
	CHEMBL1394800	30460	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	464	8	1	6	6.3	COc1cc(C)ccc1OCCSc1nc2ccc(NC(=O)c3ccc(C)cc3)cc2s1	nan
	5297365	30469	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	4	1	5	4.4	N#Cc1cc2c(nc1SCC(=O)Nc1cccc(C(F)(F)F)c1)C1CCN2CC1	nan
	CHEMBL1394905	30469	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	4	1	5	4.4	N#Cc1cc2c(nc1SCC(=O)Nc1cccc(C(F)(F)F)c1)C1CCN2CC1	nan
	1308289	30470	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	479	6	0	6	4.2	CCS(=O)(=O)c1c(S(=O)(=O)CC)c2cc(C(C)(C)C)ccn2c1C(=O)c1ccc(F)cc1	nan
	CHEMBL1394907	30470	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	479	6	0	6	4.2	CCS(=O)(=O)c1c(S(=O)(=O)CC)c2cc(C(C)(C)C)ccn2c1C(=O)c1ccc(F)cc1	nan
	7338094	30484	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	398	4	1	5	5.2	Cc1ccn2c(Nc3ccccc3C)c(-c3ccc(N4CCOCC4)cc3)nc2c1	nan
	CHEMBL1395018	30484	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	398	4	1	5	5.2	Cc1ccn2c(Nc3ccccc3C)c(-c3ccc(N4CCOCC4)cc3)nc2c1	nan
	1598875	30486	16	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	5	2	7	3.4	COC(=O)c1ccccc1NC(=O)CSc1nc2sc3c(c2c(=O)[nH]1)CCCC3	nan
	CHEMBL1395042	30486	16	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	5	2	7	3.4	COC(=O)c1ccccc1NC(=O)CSc1nc2sc3c(c2c(=O)[nH]1)CCCC3	nan
	705204	30496	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	319	1	1	5	3.7	N#Cc1c(N)n(-c2cccc(Cl)c2)c2nc3ccccc3nc12	nan
	CHEMBL1395126	30496	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	319	1	1	5	3.7	N#Cc1c(N)n(-c2cccc(Cl)c2)c2nc3ccccc3nc12	nan
	16011870	30502	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	498	6	0	6	6.9	Cc1oc(-c2ccccc2F)nc1Cn1c(SCc2cccc(C(F)(F)F)c2)nc2ccncc21	nan
	CHEMBL1395173	30502	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	498	6	0	6	6.9	Cc1oc(-c2ccccc2F)nc1Cn1c(SCc2cccc(C(F)(F)F)c2)nc2ccncc21	nan
	16011750	30503	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	7	1	7	4.2	CCC(C(=O)NCc1cc(OC)ccc1OC)n1nc(C)c2sc3ccccc3c2c1=O	nan
	CHEMBL1395174	30503	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	7	1	7	4.2	CCC(C(=O)NCc1cc(OC)ccc1OC)n1nc(C)c2sc3ccccc3c2c1=O	nan
	7150993	30505	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	6	1	6	4.6	Cc1ccc2nc(NC(=O)CSc3nccn3Cc3ccccc3)sc2c1	nan
	CHEMBL1395184	30505	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	6	1	6	4.6	Cc1ccc2nc(NC(=O)CSc3nccn3Cc3ccccc3)sc2c1	nan
	16022376	30531	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	7	1	6	4.7	O=C(CSc1nc2ccsc2c(=O)n1Cc1ccc(F)cc1)NCc1ccc(Cl)cc1	nan
	CHEMBL1395536	30531	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	7	1	6	4.7	O=C(CSc1nc2ccsc2c(=O)n1Cc1ccc(F)cc1)NCc1ccc(Cl)cc1	nan
	16008365	30558	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	5	1	5	3.9	COc1cccc(NC(=O)CSc2cc(=O)n(C)c3ccc(Cl)cc23)c1	nan
	CHEMBL1395994	30558	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	5	1	5	3.9	COc1cccc(NC(=O)CSc2cc(=O)n(C)c3ccc(Cl)cc23)c1	nan
	16016520	30566	16	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	292	2	2	2	3.4	Cc1cccc(NC(=O)c2ccc3[nH]c(C)cc(=O)c3c2)c1	nan
	CHEMBL1396103	30566	16	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	292	2	2	2	3.4	Cc1cccc(NC(=O)c2ccc3[nH]c(C)cc(=O)c3c2)c1	nan
	16012961	30588	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	4	0	7	3.2	COc1ccc(Cc2nc3c4cnn(-c5cccc(F)c5)c4ncn3n2)cc1	nan
	CHEMBL1396439	30588	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	4	0	7	3.2	COc1ccc(Cc2nc3c4cnn(-c5cccc(F)c5)c4ncn3n2)cc1	nan
	16011203	30608	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	4	1	6	3.8	CCc1nn(CC(=O)Nc2c(C)cc(C)cc2C)c(=O)c2cc3sccc3n12	nan
	CHEMBL1396725	30608	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	4	1	6	3.8	CCc1nn(CC(=O)Nc2c(C)cc(C)cc2C)c(=O)c2cc3sccc3n12	nan
	5300039	30632	14	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	446	2	2	5	4.7	Nc1c(C(=O)Nc2ccc(Br)cc2F)sc2nc3c(cc12)N1CCC3CC1	nan
	CHEMBL1397016	30632	14	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	446	2	2	5	4.7	Nc1c(C(=O)Nc2ccc(Br)cc2F)sc2nc3c(cc12)N1CCC3CC1	nan
	16029565	30646	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	5	1	5	4.0	Cc1ccc(C)c(NC(=O)Cn2cc(C(=O)c3ccncc3)c(=O)c3cc(F)ccc32)c1	nan
	CHEMBL1397193	30646	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	5	1	5	4.0	Cc1ccc(C)c(NC(=O)Cn2cc(C(=O)c3ccncc3)c(=O)c3cc(F)ccc32)c1	nan
	9114471	30659	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	3	2	7	1.5	N#Cc1cc(C#N)c(SCC(=O)N2CC(=O)Nc3ccccc32)nc1N	nan
	CHEMBL1397378	30659	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	3	2	7	1.5	N#Cc1cc(C#N)c(SCC(=O)N2CC(=O)Nc3ccccc32)nc1N	nan
	16029539	30663	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	6	1	5	4.7	Cc1ccc2c(c1)c(=O)c(C(=O)c1ccncc1)cn2CC(=O)Nc1ccc(C(C)C)cc1	nan
	CHEMBL1397433	30663	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	6	1	5	4.7	Cc1ccc2c(c1)c(=O)c(C(=O)c1ccncc1)cn2CC(=O)Nc1ccc(C(C)C)cc1	nan
	16021836	30666	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	5	1	4	4.1	CSc1ncc(C(=O)NCc2ccc(C)cc2)c(-c2ccccc2)n1	nan
	CHEMBL1397498	30666	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	5	1	4	4.1	CSc1ncc(C(=O)NCc2ccc(C)cc2)c(-c2ccccc2)n1	nan
	16024513	30668	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	5	1	5	4.8	Cc1ccc(C(=O)c2cn(CC(=O)Nc3ccc(C)cc3Cl)c3nc(C)ccc3c2=O)cc1	nan
	CHEMBL1397525	30668	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	5	1	5	4.8	Cc1ccc(C(=O)c2cn(CC(=O)Nc3ccc(C)cc3Cl)c3nc(C)ccc3c2=O)cc1	nan
	4069971	30694	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	8	1	4	5.3	CCCCNC(=O)c1cc(Sc2ccc(OCC)cc2)nc2ccccc12	nan
	CHEMBL1397896	30694	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	8	1	4	5.3	CCCCNC(=O)c1cc(Sc2ccc(OCC)cc2)nc2ccccc12	nan
	402652	30712	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	2	1	6	3.7	O=c1c2ccccc2nc2sc(Nc3cccc(Cl)c3)nn12	nan
	CHEMBL1398128	30712	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	2	1	6	3.7	O=c1c2ccccc2nc2sc(Nc3cccc(Cl)c3)nn12	nan
	15988651	30713	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	4	1	4	3.8	O=C(Nc1cccc(C(F)(F)F)c1)C1CCN(S(=O)(=O)c2cccs2)CC1	nan
	CHEMBL1398130	30713	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	4	1	4	3.8	O=C(Nc1cccc(C(F)(F)F)c1)C1CCN(S(=O)(=O)c2cccs2)CC1	nan
	135455820	30724	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	2	1	5	4.6	Oc1ncnc2c1sc1nc(C(F)F)cc(-c3ccccc3)c12	nan
	CHEMBL1398293	30724	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	2	1	5	4.6	Oc1ncnc2c1sc1nc(C(F)F)cc(-c3ccccc3)c12	nan
	16019015	30735	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	6	1	5	3.5	CC(C)CCNC(=O)c1ccc(Cn2c(=O)c3cccn3c3cccnc32)cc1	nan
	CHEMBL1398441	30735	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	6	1	5	3.5	CC(C)CCNC(=O)c1ccc(Cn2c(=O)c3cccn3c3cccnc32)cc1	nan
	16032326	30752	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	5	1	6	5.9	CN1CCc2c(sc(NC(=O)CSc3ccc(F)cc3)c2-c2nc3ccccc3s2)C1	nan
	CHEMBL1398567	30752	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	5	1	6	5.9	CN1CCc2c(sc(NC(=O)CSc3ccc(F)cc3)c2-c2nc3ccccc3s2)C1	nan
	2105201	30780	8	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	521	8	1	9	4.9	CCOC(=O)c1c(NC(=O)CSc2nc3ccccc3c(=O)n2-c2ccccc2)sc(C(C)=O)c1C	nan
	CHEMBL1398840	30780	8	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	521	8	1	9	4.9	CCOC(=O)c1c(NC(=O)CSc2nc3ccccc3c(=O)n2-c2ccccc2)sc(C(C)=O)c1C	nan
	16021149	30825	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	7	1	5	5.8	O=C(NC1CCCCC1)c1ccc(Cn2c(SCc3ccccc3)nc3cccnc32)cc1	nan
	CHEMBL1399300	30825	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	7	1	5	5.8	O=C(NC1CCCCC1)c1ccc(Cn2c(SCc3ccccc3)nc3cccnc32)cc1	nan
	8351751	30853	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	7	0	8	2.1	CCOc1ccc(C(=O)COC(=O)c2ccc(-n3cnnn3)cc2)cc1	nan
	CHEMBL1399515	30853	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	7	0	8	2.1	CCOc1ccc(C(=O)COC(=O)c2ccc(-n3cnnn3)cc2)cc1	nan
	1386490	30867	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	6	0	5	4.8	COc1cccc(OCCn2c(-c3ccc(Cl)cc3)nc3ccccc3c2=O)c1	nan
	CHEMBL1399670	30867	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	6	0	5	4.8	COc1cccc(OCCn2c(-c3ccc(Cl)cc3)nc3ccccc3c2=O)c1	nan
	16007871	30878	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	490	5	1	4	5.2	O=C(NCc1ccco1)c1ccc2c(c1)N(Cc1ccc(Cl)cc1)C(=O)c1ccccc1[S+]2[O-]	nan
	CHEMBL1399777	30878	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	490	5	1	4	5.2	O=C(NCc1ccco1)c1ccc2c(c1)N(Cc1ccc(Cl)cc1)C(=O)c1ccccc1[S+]2[O-]	nan
	16011403	30880	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	500	8	1	5	6.0	O=C(NCc1ccc(F)cc1)c1ccc(Cn2c(SCc3ccc(F)cc3)nc3cccnc32)cc1	nan
	CHEMBL1399789	30880	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	500	8	1	5	6.0	O=C(NCc1ccc(F)cc1)c1ccc(Cn2c(SCc3ccc(F)cc3)nc3cccnc32)cc1	nan
	7293305	30883	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	7	1	5	3.6	COCCn1ccc2c(OCC(=O)Nc3c(C)cc(C)cc3C)cccc2c1=O	nan
	CHEMBL1399845	30883	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	7	1	5	3.6	COCCn1ccc2c(OCC(=O)Nc3c(C)cc(C)cc3C)cccc2c1=O	nan
	16030115	31020	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	5	1	6	4.4	CCc1cccc(C)c1NC(=O)Cn1nc(C)c2nn(-c3ccc(Cl)cc3)c(C)c2c1=O	nan
	CHEMBL1401110	31020	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	5	1	6	4.4	CCc1cccc(C)c1NC(=O)Cn1nc(C)c2nn(-c3ccc(Cl)cc3)c(C)c2c1=O	nan
	1163266	31034	9	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	249	1	1	5	2.2	Cc1ccc(-c2cc3ncc(C#N)c(N)n3n2)cc1	nan
	CHEMBL1401234	31034	9	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	249	1	1	5	2.2	Cc1ccc(-c2cc3ncc(C#N)c(N)n3n2)cc1	nan
	16024855	31056	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	3	1	4	5.1	Cc1cc(C)cc(NC(=O)C2CCN(c3nc4ccccc4nc3C(F)(F)F)CC2)c1	nan
	CHEMBL1401368	31056	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	3	1	4	5.1	Cc1cc(C)cc(NC(=O)C2CCN(c3nc4ccccc4nc3C(F)(F)F)CC2)c1	nan
	16011339	31162	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	6	2	5	5.2	CCOC(=O)c1ccccc1NC(=O)NC(C)c1c(-n2cccc2)sc(C)c1C	nan
	CHEMBL1402306	31162	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	6	2	5	5.2	CCOC(=O)c1ccccc1NC(=O)NC(C)c1c(-n2cccc2)sc(C)c1C	nan
	16019019	31172	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	6	1	5	3.7	O=C(NCCc1ccccc1)c1ccc(Cn2c(=O)c3cccn3c3cccnc32)cc1	nan
	CHEMBL1402402	31172	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	6	1	5	3.7	O=C(NCCc1ccccc1)c1ccc(Cn2c(=O)c3cccn3c3cccnc32)cc1	nan
	16011789	31246	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	344	3	0	5	3.6	Cc1ccc(-n2ncc3c(=O)n(Cc4ccccc4C)cnc32)cc1C	nan
	CHEMBL1403021	31246	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	344	3	0	5	3.6	Cc1ccc(-n2ncc3c(=O)n(Cc4ccccc4C)cnc32)cc1C	nan
	7096324	31263	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	330	3	2	3	2.5	NS(=O)(=O)c1ccc(NC(=O)c2ccc3c(c2)CCCC3)cc1	nan
	CHEMBL1403204	31263	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	330	3	2	3	2.5	NS(=O)(=O)c1ccc(NC(=O)c2ccc3c(c2)CCCC3)cc1	nan
	135437062	31288	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	6	3	6	3.5	CCC(C)NC(=O)CSc1nc2[nH]nc(C)c2c(=N)n1-c1ccc(C)c(Cl)c1	nan
	CHEMBL1403479	31288	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	6	3	6	3.5	CCC(C)NC(=O)CSc1nc2[nH]nc(C)c2c(=N)n1-c1ccc(C)c(Cl)c1	nan
	16026084	31349	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	3	1	7	2.1	O=C(Nc1cccc(F)c1)c1cnc2sc(N3CCCC3)nn2c1=O	nan
	CHEMBL1404065	31349	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	3	1	7	2.1	O=C(Nc1cccc(F)c1)c1cnc2sc(N3CCCC3)nn2c1=O	nan
	15999042	31385	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	4	1	6	2.8	O=C(Cn1c(=O)n(-c2ccc(F)cc2)c(=O)c2sccc21)NC1CCCCC1	nan
	CHEMBL1404291	31385	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	4	1	6	2.8	O=C(Cn1c(=O)n(-c2ccc(F)cc2)c(=O)c2sccc21)NC1CCCCC1	nan
	1617675	31427	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	3	0	5	6.2	Cc1cccc(-c2nc3c4c(-c5ccccc5)c(-c5ccccc5)oc4ncn3n2)c1	nan
	CHEMBL1404812	31427	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	3	0	5	6.2	Cc1cccc(-c2nc3c4c(-c5ccccc5)c(-c5ccccc5)oc4ncn3n2)c1	nan
	2390567	31461	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	4	2	6	2.9	N#Cc1ccsc1NC(=O)COC(=O)c1cc(Br)ccc1O	nan
	CHEMBL1405202	31461	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	4	2	6	2.9	N#Cc1ccsc1NC(=O)COC(=O)c1cc(Br)ccc1O	nan
	15988048	31521	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	538	10	2	9	2.1	COc1cc2c(=O)n(CCC(=O)NCC3CCCO3)c(=O)n(CC(=O)Nc3c(C)cccc3C)c2cc1OC	nan
	CHEMBL1405772	31521	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	538	10	2	9	2.1	COc1cc2c(=O)n(CCC(=O)NCC3CCCO3)c(=O)n(CC(=O)Nc3c(C)cccc3C)c2cc1OC	nan
	16024912	31525	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	442	5	1	4	4.5	Cc1ccccc1CCNC(=O)C1CCN(c2nc3ccccc3nc2C(F)(F)F)CC1	nan
	CHEMBL1405829	31525	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	442	5	1	4	4.5	Cc1ccccc1CCNC(=O)C1CCN(c2nc3ccccc3nc2C(F)(F)F)CC1	nan
	2991576	31726	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	3	1	6	2.6	CCCCc1nc2sc3c(=O)n(N)cnc3c2c2c1CCC2	nan
	CHEMBL1407541	31726	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	3	1	6	2.6	CCCCc1nc2sc3c(=O)n(N)cnc3c2c2c1CCC2	nan
	3583749	31763	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	477	5	1	7	3.0	COC(=O)c1c(NC(=O)c2ccc(S(=O)(=O)N3CCCCC3)cc2)sc2c1CCN(C)C2	nan
	CHEMBL1407736	31763	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	477	5	1	7	3.0	COC(=O)c1c(NC(=O)c2ccc(S(=O)(=O)N3CCCCC3)cc2)sc2c1CCN(C)C2	nan
	3245299	31773	8	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	5	2	7	2.7	CCOc1ccccc1-c1nc(C(N)=O)c2nc(O)n(-c3ccccc3)c2n1	nan
	CHEMBL1407835	31773	8	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	5	2	7	2.7	CCOc1ccccc1-c1nc(C(N)=O)c2nc(O)n(-c3ccccc3)c2n1	nan
	6485917	31822	14	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	9	1	8	2.6	COc1ccc(CNCCSc2nnnn2-c2ccccc2)c(OC)c1	nan
	CHEMBL1408179	31822	14	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	9	1	8	2.6	COc1ccc(CNCCSc2nnnn2-c2ccccc2)c(OC)c1	nan
	2265197	31831	17	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	334	4	2	2	4.3	O=C(Nc1ccccc1C(=O)Nc1ccccc1)c1ccccc1F	nan
	CHEMBL1408256	31831	17	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	334	4	2	2	4.3	O=C(Nc1ccccc1C(=O)Nc1ccccc1)c1ccccc1F	nan
	15989388	31916	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	510	7	1	6	3.3	CCc1ccc(NC(=O)Cn2c(=O)n(CCC(=O)N3CCc4ccccc4C3)c(=O)c3ccccc32)cc1	nan
	CHEMBL1408914	31916	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	510	7	1	6	3.3	CCc1ccc(NC(=O)Cn2c(=O)n(CCC(=O)N3CCc4ccccc4C3)c(=O)c3ccccc32)cc1	nan
	1082765	32005	14	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	8	1	6	2.9	COc1ccc(CCNC(=O)COc2ccc3c(C)cc(=O)oc3c2)cc1OC	nan
	CHEMBL1409638	32005	14	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	8	1	6	2.9	COc1ccc(CCNC(=O)COc2ccc3c(C)cc(=O)oc3c2)cc1OC	nan
	1913870	32032	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	7	2	6	3.1	O=C(/C=C\Nc1ccc(S(=O)(=O)Nc2ncccn2)cc1)c1ccccc1	nan
	CHEMBL1409860	32032	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	7	2	6	3.1	O=C(/C=C\Nc1ccc(S(=O)(=O)Nc2ncccn2)cc1)c1ccccc1	nan
	2527257	32085	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	7	2	7	1.7	COc1ccc(C(=O)OCC(=O)Nc2sccc2C(N)=O)cc1OC	nan
	CHEMBL1410234	32085	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	7	2	7	1.7	COc1ccc(C(=O)OCC(=O)Nc2sccc2C(N)=O)cc1OC	nan
	2201015	32095	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	5	1	5	3.3	Cc1ccc(-n2c3c(cc(C(=O)NCC(=O)c4ccccc4)c2=O)C(=O)CCC3)cc1	nan
	CHEMBL1410319	32095	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	5	1	5	3.3	Cc1ccc(-n2c3c(cc(C(=O)NCC(=O)c4ccccc4)c2=O)C(=O)CCC3)cc1	nan
	2135385	32127	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	488	7	1	7	4.1	CCOc1ccc(NC(=O)Cn2cc(C(=O)c3ccc(F)cc3)c(=O)c3cc4c(cc32)OCO4)cc1	nan
	CHEMBL1410565	32127	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	488	7	1	7	4.1	CCOc1ccc(NC(=O)Cn2cc(C(=O)c3ccc(F)cc3)c(=O)c3cc4c(cc32)OCO4)cc1	nan
	1160042	32147	10	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	6	0	5	3.9	Cc1cc(C)c(C#N)c(SCCS(=O)(=O)Cc2ccc(Cl)cc2)n1	nan
	CHEMBL1410783	32147	10	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	6	0	5	3.9	Cc1cc(C)c(C#N)c(SCCS(=O)(=O)Cc2ccc(Cl)cc2)n1	nan
	16232595	32159	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	6	1	6	3.1	Cc1cc(C)c(C#N)c(SCC(=O)Nc2cccc(S(=O)(=O)N3CCCC3)c2)n1	nan
	CHEMBL1410891	32159	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	6	1	6	3.1	Cc1cc(C)c(C#N)c(SCC(=O)Nc2cccc(S(=O)(=O)N3CCCC3)c2)n1	nan
	1963060	32173	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	361	4	0	6	2.6	COCCn1c(-c2ccccc2)nc2c(c(=O)c3ccccc3n2C)c1=O	nan
	CHEMBL1411041	32173	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	361	4	0	6	2.6	COCCn1c(-c2ccccc2)nc2c(c(=O)c3ccccc3n2C)c1=O	nan
	1301263	32215	10	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	7	1	6	4.6	COc1ccc(CC(=O)Nc2ccc(-c3nnc(-c4ccccc4)o3)cc2)cc1OC	nan
	CHEMBL1411349	32215	10	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	7	1	6	4.6	COc1ccc(CC(=O)Nc2ccc(-c3nnc(-c4ccccc4)o3)cc2)cc1OC	nan
	2353143	32392	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	4	1	4	4.4	COc1cc(SC)ccc1C(=O)Nc1ncc(Cl)cc1Cl	nan
	CHEMBL1412778	32392	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	4	1	4	4.4	COc1cc(SC)ccc1C(=O)Nc1ncc(Cl)cc1Cl	nan
	135402203	32469	13	None	-3	3	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	6	1	6	3.5	COc1ccc(OCCSc2nc(O)c3ccccc3n2)cc1	nan
	CHEMBL1413382	32469	13	None	-3	3	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	6	1	6	3.5	COc1ccc(OCCSc2nc(O)c3ccccc3n2)cc1	nan
	8722509	32487	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	7	1	7	3.6	CC(=O)c1ccc(NC(=O)CSc2nnc(-c3ccncc3)n2C2CC2)cc1	nan
	CHEMBL1413558	32487	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	7	1	7	3.6	CC(=O)c1ccc(NC(=O)CSc2nnc(-c3ccncc3)n2C2CC2)cc1	nan
	3240816	32490	4	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	3	0	6	2.0	COC(=O)c1cn(C)c2ccc(S(=O)(=O)N3CC(C)CC(C)C3)cc2c1=O	nan
	CHEMBL1413578	32490	4	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	3	0	6	2.0	COC(=O)c1cn(C)c2ccc(S(=O)(=O)N3CC(C)CC(C)C3)cc2c1=O	nan
	3546772	32524	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	398	8	1	4	5.1	CC(C)OCCCNC(=O)c1cc(Sc2ccc(F)cc2)nc2ccccc12	nan
	CHEMBL1413820	32524	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	398	8	1	4	5.1	CC(C)OCCCNC(=O)c1cc(Sc2ccc(F)cc2)nc2ccccc12	nan
	2216801	32547	16	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	4	1	6	3.2	Cc1cc(NC(=O)CSc2nc3c(cc2C#N)CCCCC3)no1	nan
	CHEMBL1414005	32547	16	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	4	1	6	3.2	Cc1cc(NC(=O)CSc2nc3c(cc2C#N)CCCCC3)no1	nan
	16011480	32594	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	7	1	5	6.1	Cc1cccc(Cn2c(SCc3ccc(C(=O)NC4CCCCC4)cc3)nc3ccncc32)c1	nan
	CHEMBL1414437	32594	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	7	1	5	6.1	Cc1cccc(Cn2c(SCc3ccc(C(=O)NC4CCCCC4)cc3)nc3ccncc32)c1	nan
	3185714	32627	3	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	536	9	3	8	2.9	Cc1cccc(N(C(=O)c2snc(C(N)=O)c2N)C(C(=O)NCC2CCCO2)c2ccc(N(C)C)cc2)c1	nan
	CHEMBL1414702	32627	3	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	536	9	3	8	2.9	Cc1cccc(N(C(=O)c2snc(C(N)=O)c2N)C(C(=O)NCC2CCCO2)c2ccc(N(C)C)cc2)c1	nan
	16024849	32700	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	4	1	4	4.7	CC(NC(=O)C1CCN(c2nc3ccccc3nc2C(F)(F)F)CC1)c1ccccc1	nan
	CHEMBL1415340	32700	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	4	1	4	4.7	CC(NC(=O)C1CCN(c2nc3ccccc3nc2C(F)(F)F)CC1)c1ccccc1	nan
	1997619	32727	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	363	1	0	6	3.4	O=c1nc2sc3ccccc3n2c(=O)n1-c1ccc(Cl)c(Cl)c1	nan
	CHEMBL1415577	32727	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	363	1	0	6	3.4	O=c1nc2sc3ccccc3n2c(=O)n1-c1ccc(Cl)c(Cl)c1	nan
	601275	32754	11	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	5	1	7	2.7	CCc1nnc(NC(=O)CSc2nc(C)cc(C)c2C#N)s1	nan
	CHEMBL1415875	32754	11	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	5	1	7	2.7	CCc1nnc(NC(=O)CSc2nc(C)cc(C)c2C#N)s1	nan
	15988188	32779	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	7	2	4	2.9	CCCCCn1c(=O)[nH]c2cc(C(=O)NCc3ccc(F)cc3)ccc2c1=O	nan
	CHEMBL1416073	32779	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	7	2	4	2.9	CCCCCn1c(=O)[nH]c2cc(C(=O)NCc3ccc(F)cc3)ccc2c1=O	nan
	2135587	32833	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	502	7	1	7	4.2	CCOc1ccc(C(=O)c2cn(CC(=O)Nc3ccc(F)cc3)c3cc4c(cc3c2=O)OCCO4)cc1	nan
	CHEMBL1416515	32833	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	502	7	1	7	4.2	CCOc1ccc(C(=O)c2cn(CC(=O)Nc3ccc(F)cc3)c3cc4c(cc3c2=O)OCCO4)cc1	nan
	1829959	32839	10	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	487	6	1	6	4.6	O=C(Nc1cc[n+](-c2nc3ccccc3nc2[N-]S(=O)(=O)c2ccccc2)cc1)c1cccs1	nan
	CHEMBL1416570	32839	10	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	487	6	1	6	4.6	O=C(Nc1cc[n+](-c2nc3ccccc3nc2[N-]S(=O)(=O)c2ccccc2)cc1)c1cccs1	nan
	4044817	32856	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	457	4	1	6	4.1	CC(OC(=O)c1ccc2c(=O)n3c(nc2c1)CCCCC3)C(=O)Nc1ccc(F)cc1Cl	nan
	CHEMBL1416742	32856	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	457	4	1	6	4.1	CC(OC(=O)c1ccc2c(=O)n3c(nc2c1)CCCCC3)C(=O)Nc1ccc(F)cc1Cl	nan
	16012432	32857	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	3	2	5	3.0	O=C(NCc1cccc(Cl)c1)C(=O)Nc1ccc2nc3n(c(=O)c2c1)CCCCC3	nan
	CHEMBL1416749	32857	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	3	2	5	3.0	O=C(NCc1cccc(Cl)c1)C(=O)Nc1ccc2nc3n(c(=O)c2c1)CCCCC3	nan
	16033988	32873	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	287	2	0	5	2.8	Cc1ccc(-n2ncc3c(N(C)C)ncnc32)cc1Cl	nan
	CHEMBL1416927	32873	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	287	2	0	5	2.8	Cc1ccc(-n2ncc3c(N(C)C)ncnc32)cc1Cl	nan
	16031129	32938	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	447	7	2	6	4.5	COc1ccc(OC)c(CNC(=O)c2ccccc2NC(=O)c2nsc3ccccc23)c1	nan
	CHEMBL1417406	32938	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	447	7	2	6	4.5	COc1ccc(OC)c(CNC(=O)c2ccccc2NC(=O)c2nsc3ccccc23)c1	nan
	16018805	32953	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	396	5	1	6	3.3	COc1ccc(NC(=O)CCn2c(=O)c3cccn3c3cccnc32)cc1Cl	nan
	CHEMBL1417571	32953	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	396	5	1	6	3.3	COc1ccc(NC(=O)CCn2c(=O)c3cccn3c3cccnc32)cc1Cl	nan
	1490637	32996	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	6	2	5	4.5	COc1ccc(NC(=O)c2ccccc2Sc2ccc(NC(C)=O)nc2)cc1	nan
	CHEMBL1417935	32996	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	6	2	5	4.5	COc1ccc(NC(=O)c2ccccc2Sc2ccc(NC(C)=O)nc2)cc1	nan
	5768421	33019	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	9	1	6	3.8	COCCCN1C(=O)C(O)=C(C(=O)c2ccc(OC(C)C)c(C)c2)C1c1ccncc1	nan
	CHEMBL1418118	33019	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	9	1	6	3.8	COCCCN1C(=O)C(O)=C(C(=O)c2ccc(OC(C)C)c(C)c2)C1c1ccncc1	nan
	16025701	33068	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	436	6	1	9	3.7	COc1ccc(-n2nnc(-c3nsc(NC(=O)c4cccc(C)c4)n3)c2C)cc1OC	nan
	CHEMBL1418579	33068	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	436	6	1	9	3.7	COc1ccc(-n2nnc(-c3nsc(NC(=O)c4cccc(C)c4)n3)c2C)cc1OC	nan
	1248279	33091	18	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	347	4	2	7	3.9	COc1ccccc1Nc1nc(N)nc(-c2oc3ccccc3c2C)n1	nan
	CHEMBL1418732	33091	18	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	347	4	2	7	3.9	COc1ccccc1Nc1nc(N)nc(-c2oc3ccccc3c2C)n1	nan
	2082778	33126	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	345	3	2	3	3.6	COc1ccc(Br)c(C(=O)Nc2nc3ccccc3[nH]2)c1	nan
	CHEMBL1419051	33126	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	345	3	2	3	3.6	COc1ccc(Br)c(C(=O)Nc2nc3ccccc3[nH]2)c1	nan
	7708945	33144	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	320	2	1	4	4.3	Nc1c(-c2ccc(Cl)cc2)cnc2c(-c3ccccc3)cnn12	nan
	CHEMBL1419219	33144	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	320	2	1	4	4.3	Nc1c(-c2ccc(Cl)cc2)cnc2c(-c3ccccc3)cnn12	nan
	656027	33237	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	8	1	7	4.2	COc1ccc(CCN2C(=O)C(O)=C(C(=O)c3ccco3)C2c2cccs2)cc1OC	nan
	CHEMBL1420005	33237	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	8	1	7	4.2	COc1ccc(CCN2C(=O)C(O)=C(C(=O)c3ccco3)C2c2cccs2)cc1OC	nan
	16457257	33253	15	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	292	1	1	5	3.5	Cc1ccccc1-c1nc2c3ccccc3nc(S)n2n1	nan
	CHEMBL1420123	33253	15	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	292	1	1	5	3.5	Cc1ccccc1-c1nc2c3ccccc3nc(S)n2n1	nan
	5049250	33267	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	4	3	4	2.6	O=C(COc1cccc2cccnc12)NNC(=S)Nc1ccccc1	nan
	CHEMBL1420194	33267	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	4	3	4	2.6	O=C(COc1cccc2cccnc12)NNC(=S)Nc1ccccc1	nan
	2518728	33321	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	4	1	6	4.3	Cc1nn(Cc2ccc(F)cc2)c2sc(C(=O)Nc3nccs3)cc12	nan
	CHEMBL1420654	33321	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	4	1	6	4.3	Cc1nn(Cc2ccc(F)cc2)c2sc(C(=O)Nc3nccs3)cc12	nan
	1975568	33506	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	436	5	0	6	4.4	COc1ccc2c(c1)c1nc3ccccc3nc1n2CCCN1C(=O)c2ccccc2C1=O	nan
	CHEMBL1422285	33506	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	436	5	0	6	4.4	COc1ccc2c(c1)c1nc3ccccc3nc1n2CCCN1C(=O)c2ccccc2C1=O	nan
	2952481	33626	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	7	2	5	3.6	CCCC(=O)Nc1ccc(C(=O)Nc2ccc([N+](=O)[O-])cc2OC)cc1	nan
	CHEMBL1423274	33626	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	7	2	5	3.6	CCCC(=O)Nc1ccc(C(=O)Nc2ccc([N+](=O)[O-])cc2OC)cc1	nan
	4204373	33708	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	5	2	6	3.5	COc1cc2nc(S)nc(NCc3ccccc3)c2cc1OC	nan
	CHEMBL1423864	33708	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	5	2	6	3.5	COc1cc2nc(S)nc(NCc3ccccc3)c2cc1OC	nan
	3208003	33734	5	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	5	1	5	4.1	CCc1cc2cc(C)ccc2nc1SCC(=O)Nc1cc(C)on1	nan
	CHEMBL1424112	33734	5	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	5	1	5	4.1	CCc1cc2cc(C)ccc2nc1SCC(=O)Nc1cc(C)on1	nan
	4329755	33857	13	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	5	1	3	6.3	O=C(Cc1sc(-c2ccccc2Cl)nc1-c1ccccc1)Nc1ccccc1	nan
	CHEMBL1425135	33857	13	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	5	1	3	6.3	O=C(Cc1sc(-c2ccccc2Cl)nc1-c1ccccc1)Nc1ccccc1	nan
	2293921	33907	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	6	3	5	1.5	NS(=O)(=O)c1ccc(NS(=O)(=O)c2ccc(NC(=O)C3CC3)cc2)cc1	nan
	CHEMBL1425666	33907	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	6	3	5	1.5	NS(=O)(=O)c1ccc(NS(=O)(=O)c2ccc(NC(=O)C3CC3)cc2)cc1	nan
	2009311	33926	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	4	1	6	4.6	O=C(O)CSc1ncnc2c1sc1nc(-c3ccccc3)c3c(c12)CCC3	nan
	CHEMBL1425879	33926	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	4	1	6	4.6	O=C(O)CSc1ncnc2c1sc1nc(-c3ccccc3)c3c(c12)CCC3	nan
	3434681	34039	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	441	7	3	5	3.9	COc1ccccc1NS(=O)(=O)c1cccc(NC(=O)c2[nH]c(C)c(C(C)=O)c2C)c1	nan
	CHEMBL1426649	34039	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	441	7	3	5	3.9	COc1ccccc1NS(=O)(=O)c1cccc(NC(=O)c2[nH]c(C)c(C(C)=O)c2C)c1	nan
	3430748	34042	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	3	3	5	2.1	COc1ccc2c3c([nH]c2c1)C1CC2C(CC(O)C(OC)C2CO)CN1CC3	nan
	CHEMBL1426665	34042	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	3	3	5	2.1	COc1ccc2c3c([nH]c2c1)C1CC2C(CC(O)C(OC)C2CO)CN1CC3	nan
	16195448	34103	0	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	351	2	1	3	4.7	Cc1cccc(NC(=O)c2ccc3c(Cl)c4c(nc3c2)CCCC4)n1	nan
	CHEMBL1427245	34103	0	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	351	2	1	3	4.7	Cc1cccc(NC(=O)c2ccc3c(Cl)c4c(nc3c2)CCCC4)n1	nan
	1206713	34233	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	5	2	5	2.9	Cc1cccc2cc(C#N)c(SCC(=O)NNC(=O)Cc3ccccc3)nc12	nan
	CHEMBL1428460	34233	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	5	2	5	2.9	Cc1cccc2cc(C#N)c(SCC(=O)NNC(=O)Cc3ccccc3)nc12	nan
	2085163	34264	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	313	4	1	5	3.7	CCOc1ncccc1C(=O)Nc1ccc2nc(C)sc2c1	nan
	CHEMBL1428703	34264	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	313	4	1	5	3.7	CCOc1ncccc1C(=O)Nc1ccc2nc(C)sc2c1	nan
	3138587	34296	4	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	6	5	10	-2.3	CN(C)c1ccc2nc3c(=O)[nH]c(=O)nc-3n(CC(O)C(O)C(O)CO)c2c1	nan
	CHEMBL1428985	34296	4	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	6	5	10	-2.3	CN(C)c1ccc2nc3c(=O)[nH]c(=O)nc-3n(CC(O)C(O)C(O)CO)c2c1	nan
	1454920	34387	3	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	5	1	5	4.7	CCc1ccc2c(c1)cc(CN(C(S)=Nc1ccccc1C)C1CC1)c1nnnn12	nan
	CHEMBL1429692	34387	3	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	5	1	5	4.7	CCc1ccc2c(c1)cc(CN(C(S)=Nc1ccccc1C)C1CC1)c1nnnn12	nan
	748627	34414	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	3	1	4	4.7	Cc1ccc(Nc2nc(-c3ccncc3)nc3ccccc23)cc1	nan
	CHEMBL1429854	34414	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	3	1	4	4.7	Cc1ccc(Nc2nc(-c3ccncc3)nc3ccccc23)cc1	nan
	1478328	34479	18	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	297	2	0	5	3.0	CCc1nc2oc3ccc(C)cc3c(=O)c2cc1C(=O)OC	nan
	CHEMBL1430305	34479	18	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	297	2	0	5	3.0	CCc1nc2oc3ccc(C)cc3c(=O)c2cc1C(=O)OC	nan
	2950980	34533	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	410	4	4	6	3.8	O=C(O)c1cc(S(=O)(=O)O)cc(Nc2c3ccccc3nc3ccccc23)c1O	nan
	CHEMBL1430778	34533	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	410	4	4	6	3.8	O=C(O)c1cc(S(=O)(=O)O)cc(Nc2c3ccccc3nc3ccccc23)c1O	nan
	3452486	34620	16	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	4	1	5	4.4	Cc1cccc(NC(=O)CSc2ncnc3c2oc2ccccc23)c1	nan
	CHEMBL1431571	34620	16	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	4	1	5	4.4	Cc1cccc(NC(=O)CSc2ncnc3c2oc2ccccc23)c1	nan
	2031268	34653	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	2	0	5	4.2	Cc1cccc(-c2nc3c(c(=O)c4ccccc4n3C)c(=O)n2-c2ccccc2)c1	nan
	CHEMBL1431855	34653	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	2	0	5	4.2	Cc1cccc(-c2nc3c(c(=O)c4ccccc4n3C)c(=O)n2-c2ccccc2)c1	nan
	16030582	34850	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	7	2	7	4.1	Cc1ccc2[nH]c(CSc3nnc(NC(=O)COc4ccccc4F)s3)cc(=O)c2c1	nan
	CHEMBL1433463	34850	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	7	2	7	4.1	Cc1ccc2[nH]c(CSc3nnc(NC(=O)COc4ccccc4F)s3)cc(=O)c2c1	nan
	16014372	34864	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	6	1	4	4.7	Cc1ccc(CSc2ncc(Cl)c(C(=O)NCc3ccccc3)n2)cc1	nan
	CHEMBL1433681	34864	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	6	1	4	4.7	Cc1ccc(CSc2ncc(Cl)c(C(=O)NCc3ccccc3)n2)cc1	nan
	24980276	34894	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	10	2	8	2.9	CCOC(=O)c1c(NC(=O)COC(=O)CCOc2ccccc2C)sc(C(=O)NC)c1C	nan
	CHEMBL1434167	34894	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	10	2	8	2.9	CCOC(=O)c1c(NC(=O)COC(=O)CCOc2ccccc2C)sc(C(=O)NC)c1C	nan
	17757032	34897	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	1	0	4	4.6	Clc1ccc2c(c1)-c1c(cnc3cc(-c4ccccc4)nn13)CO2	nan
	CHEMBL1434219	34897	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	1	0	4	4.6	Clc1ccc2c(c1)-c1c(cnc3cc(-c4ccccc4)nn13)CO2	nan
	16018775	34898	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	4	1	5	3.7	Cc1cc(NC(=O)CCn2c(=O)c3cccn3c3cccnc32)ccc1Br	nan
	CHEMBL1434221	34898	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	4	1	5	3.7	Cc1cc(NC(=O)CCn2c(=O)c3cccn3c3cccnc32)ccc1Br	nan
	16018825	34909	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	9	1	8	2.4	COc1ccc(CCNC(=O)CCn2c(=O)c3cccn3c3cccnc32)c(OC)c1OC	nan
	CHEMBL1434453	34909	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	9	1	8	2.4	COc1ccc(CCNC(=O)CCn2c(=O)c3cccn3c3cccnc32)c(OC)c1OC	nan
	15989503	34916	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	497	8	1	7	3.2	Cc1cccc(NC(=O)Cn2c(=O)n(CCCS(=O)(=O)C3CCCCC3)c(=O)c3ccccc32)c1	nan
	CHEMBL1434580	34916	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	497	8	1	7	3.2	Cc1cccc(NC(=O)Cn2c(=O)n(CCCS(=O)(=O)C3CCCCC3)c(=O)c3ccccc32)c1	nan
	16034196	34917	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	518	9	2	7	5.2	CCOC(=O)c1ccc(N2CCN(c3cccc(OC)c3)CC2)c(NC(=O)Nc2ccc(OCC)cc2)c1	nan
	CHEMBL1434618	34917	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	518	9	2	7	5.2	CCOC(=O)c1ccc(N2CCN(c3cccc(OC)c3)CC2)c(NC(=O)Nc2ccc(OCC)cc2)c1	nan
	16030773	34926	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	6	1	4	5.0	Cc1cccc(OCC(=O)Nc2cc(-c3ccccc3F)nn2-c2ccccc2)c1	nan
	CHEMBL1434674	34926	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	6	1	4	5.0	Cc1cccc(OCC(=O)Nc2cc(-c3ccccc3F)nn2-c2ccccc2)c1	nan
	4153411	34954	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	5	1	4	5.6	Cc1cc(C)cc(OCC(=O)Nc2ccc(-c3nc4ccccc4s3)cc2)c1	nan
	CHEMBL1435020	34954	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	5	1	4	5.6	Cc1cc(C)cc(OCC(=O)Nc2ccc(-c3nc4ccccc4s3)cc2)c1	nan
	9516939	34955	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	303	3	1	6	3.2	COc1ccc2oc(C(=O)Nc3nnc(C)s3)c(C)c2c1	nan
	CHEMBL1435035	34955	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	303	3	1	6	3.2	COc1ccc2oc(C(=O)Nc3nnc(C)s3)c(C)c2c1	nan
	16016693	34970	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	447	5	2	4	5.5	CC(C)Oc1ccc(CNC(=O)Nc2ccc3c(c2)N(C)C(=O)c2ccccc2S3)cc1	nan
	CHEMBL1435186	34970	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	447	5	2	4	5.5	CC(C)Oc1ccc(CNC(=O)Nc2ccc3c(c2)N(C)C(=O)c2ccccc2S3)cc1	nan
	16026116	34987	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	6	1	9	1.7	COc1cccc(CNC(=O)c2cnc3sc(N4CCCC4)nn3c2=O)c1OC	nan
	CHEMBL1435357	34987	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	6	1	9	1.7	COc1cccc(CNC(=O)c2cnc3sc(N4CCCC4)nn3c2=O)c1OC	nan
	1821611	34997	15	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	7	2	5	5.9	COc1ccc(NC(=O)c2c(NC(=O)COc3ccc(Cl)cc3)sc3c2CCCCC3)cc1	nan
	CHEMBL1435471	34997	15	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	7	2	5	5.9	COc1ccc(NC(=O)c2c(NC(=O)COc3ccc(Cl)cc3)sc3c2CCCCC3)cc1	nan
	1251337	35005	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	4	1	6	3.2	COc1ccc(CNC(=O)c2cc3c(=O)n4cccc(C)c4nc3s2)cc1	nan
	CHEMBL1435587	35005	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	4	1	6	3.2	COc1ccc(CNC(=O)c2cc3c(=O)n4cccc(C)c4nc3s2)cc1	nan
	16010614	35030	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	4	1	5	5.2	Cc1ccc(CNc2nc3ccccc3c3nc(-c4cccc(C)c4)nn23)cc1	nan
	CHEMBL1435932	35030	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	4	1	5	5.2	Cc1ccc(CNc2nc3ccccc3c3nc(-c4cccc(C)c4)nn23)cc1	nan
	16025971	35033	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	5	2	6	4.1	Cc1ccc(NC(=O)CSc2nc(-c3ccccc3Cl)nc3cc(=O)[nH]n23)c(C)c1	nan
	CHEMBL1436000	35033	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	5	2	6	4.1	Cc1ccc(NC(=O)CSc2nc(-c3ccccc3Cl)nc3cc(=O)[nH]n23)c(C)c1	nan
	16023620	35042	0	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	481	7	3	5	3.4	Cc1ccc(CNC(=O)c2ccc3c(c2)NC(=O)C(CS(=O)(=O)Cc2cccc(F)c2)N3)cc1	nan
	CHEMBL1436076	35042	0	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	481	7	3	5	3.4	Cc1ccc(CNC(=O)c2ccc3c(c2)NC(=O)C(CS(=O)(=O)Cc2cccc(F)c2)N3)cc1	nan
	16001329	35063	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	490	5	0	7	4.9	COc1ccc(-c2nn(C)c3sc(C(=O)N4CCN(c5cccc(C)c5C)CC4)cc23)cc1OC	nan
	CHEMBL1436335	35063	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	490	5	0	7	4.9	COc1ccc(-c2nn(C)c3sc(C(=O)N4CCN(c5cccc(C)c5C)CC4)cc23)cc1OC	nan
	16015802	35069	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	5	1	4	6.5	Cc1ccc(SCC(=O)Nc2cccc(-c3nc4cc(Cl)ccc4o3)c2C)cc1	nan
	CHEMBL1436447	35069	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	5	1	4	6.5	Cc1ccc(SCC(=O)Nc2cccc(-c3nc4cc(Cl)ccc4o3)c2C)cc1	nan
	16008886	35074	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	5	1	6	4.3	COc1ccc(CNC(=O)c2cc3c(=O)oc4ccc(C)cc4c3s2)c(OC)c1	nan
	CHEMBL1436510	35074	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	5	1	6	4.3	COc1ccc(CNC(=O)c2cc3c(=O)oc4ccc(C)cc4c3s2)c(OC)c1	nan
	16024495	35113	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	485	9	1	7	3.3	COc1ccc(CCNC(=O)Cn2cc(C(=O)c3ccccc3)c(=O)c3ccc(C)nc32)cc1OC	nan
	CHEMBL1437062	35113	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	485	9	1	7	3.3	COc1ccc(CCNC(=O)Cn2cc(C(=O)c3ccccc3)c(=O)c3ccc(C)nc32)cc1OC	nan
	16019037	35122	3	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	6	0	6	4.6	CCOC(=O)c1cnc2cc(-c3ccc(OCC)cc3)nn2c1-c1ccccc1	nan
	CHEMBL1437136	35122	3	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	6	0	6	4.6	CCOC(=O)c1cnc2cc(-c3ccc(OCC)cc3)nn2c1-c1ccccc1	nan
	16030417	35146	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	7	1	6	3.9	Cc1cccc(OCC(=O)Nc2ccccc2OCc2cc(=O)n3cc(C)ccc3n2)c1	nan
	CHEMBL1437458	35146	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	7	1	6	3.9	Cc1cccc(OCC(=O)Nc2ccccc2OCc2cc(=O)n3cc(C)ccc3n2)c1	nan
	15987619	35149	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	4	0	4	5.7	CCCN(C(=O)c1cc2c(=O)oc3ccccc3c2s1)c1cccc(Cl)c1	nan
	CHEMBL1437513	35149	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	4	0	4	5.7	CCCN(C(=O)c1cc2c(=O)oc3ccccc3c2s1)c1cccc(Cl)c1	nan
	16027516	35157	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	7	1	9	3.6	COc1ccccc1C(=O)Nc1cccc(C(=O)OCc2cc(=O)n3nc(C4CC4)sc3n2)c1	nan
	CHEMBL1437665	35157	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	7	1	9	3.6	COc1ccccc1C(=O)Nc1cccc(C(=O)OCc2cc(=O)n3nc(C4CC4)sc3n2)c1	nan
	2986974	35161	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	373	5	1	5	4.5	Cc1cc(-c2nc3ncccc3o2)ccc1NC(=O)COc1ccccc1C	nan
	CHEMBL1437693	35161	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	373	5	1	5	4.5	Cc1cc(-c2nc3ncccc3o2)ccc1NC(=O)COc1ccccc1C	nan
	16025598	35218	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	490	6	1	7	4.1	CCOc1ccc(NC(=O)CSc2ncc3c(n2)-c2cc(Cl)ccc2N(C)S3(=O)=O)cc1	nan
	CHEMBL1438111	35218	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	490	6	1	7	4.1	CCOc1ccc(NC(=O)CSc2ncc3c(n2)-c2cc(Cl)ccc2N(C)S3(=O)=O)cc1	nan
	16012435	35231	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	335	3	0	4	3.7	CCc1nn(Cc2cccc(F)c2)c(=O)c2cc3cc(C)ccc3n12	nan
	CHEMBL1438209	35231	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	335	3	0	4	3.7	CCc1nn(Cc2cccc(F)c2)c(=O)c2cc3cc(C)ccc3n12	nan
	16014909	35321	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	292	3	1	2	3.7	Cc1ccc2c(c1)cc(C(=O)NCc1ccccc1C)n2C	nan
	CHEMBL1439084	35321	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	292	3	1	2	3.7	Cc1ccc2c(c1)cc(C(=O)NCc1ccccc1C)n2C	nan
	992393	35343	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	8	1	6	5.0	CCOC(=O)c1cnc2c(C)cc(Cl)cc2c1NCCc1ccc(OC)c(OC)c1	nan
	CHEMBL1439287	35343	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	8	1	6	5.0	CCOC(=O)c1cnc2c(C)cc(Cl)cc2c1NCCc1ccc(OC)c(OC)c1	nan
	2767956	35370	15	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	325	4	1	3	4.9	CSc1cc(-c2ccc(Cl)cc2)c(C(=O)NC(C)C)s1	nan
	CHEMBL1439494	35370	15	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	325	4	1	3	4.9	CSc1cc(-c2ccc(Cl)cc2)c(C(=O)NC(C)C)s1	nan
	3116122	35399	15	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	5	2	7	2.1	COc1ccc(NC(=O)CSc2nc(N)c(C#N)cc2C#N)cc1	nan
	CHEMBL1439707	35399	15	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	5	2	7	2.1	COc1ccc(NC(=O)CSc2nc(N)c(C#N)cc2C#N)cc1	nan
	16016094	35444	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	6	1	7	5.1	COc1ccc(-c2noc(-c3ccc(NC4CCCCC4)c([N+](=O)[O-])c3)n2)cc1	nan
	CHEMBL1440140	35444	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	6	1	7	5.1	COc1ccc(-c2noc(-c3ccc(NC4CCCCC4)c([N+](=O)[O-])c3)n2)cc1	nan
	1630787	35490	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	486	5	2	7	3.3	CC(C)(C)NS(=O)(=O)c1ccc2nc(NC(=O)c3ccc(N4C(=O)CCC4=O)cc3)sc2c1	nan
	CHEMBL1440595	35490	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	486	5	2	7	3.3	CC(C)(C)NS(=O)(=O)c1ccc2nc(NC(=O)c3ccc(N4C(=O)CCC4=O)cc3)sc2c1	nan
	16014413	35500	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	6	1	4	4.7	Cc1ccccc1CSc1ncc(Cl)c(C(=O)NCc2ccccc2)n1	nan
	CHEMBL1440676	35500	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	6	1	4	4.7	Cc1ccccc1CSc1ncc(Cl)c(C(=O)NCc2ccccc2)n1	nan
	15989176	35595	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	9	1	5	3.2	CCCCNC(=O)CCCn1c(=O)c2ccccc2n(Cc2ccccc2C)c1=O	nan
	CHEMBL1441599	35595	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	9	1	5	3.2	CCCCNC(=O)CCCn1c(=O)c2ccccc2n(Cc2ccccc2C)c1=O	nan
	16008898	35617	1	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	4	1	6	3.5	CCOC(=O)c1cccc(NC(=O)c2cc3c(=O)n(C)c4ccccc4c3n2C)c1	nan
	CHEMBL1441757	35617	1	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	4	1	6	3.5	CCOC(=O)c1cccc(NC(=O)c2cc3c(=O)n(C)c4ccccc4c3n2C)c1	nan
	1374312	35627	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	6	2	6	2.6	COc1ccc2cc(C#N)c(SCC(=O)NNC(=O)Cc3ccccc3)nc2c1	nan
	CHEMBL1441823	35627	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	6	2	6	2.6	COc1ccc2cc(C#N)c(SCC(=O)NNC(=O)Cc3ccccc3)nc2c1	nan
	979004	35631	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	4	0	10	2.6	CC(C)(C)c1nnc2sc(SCC(=O)c3ccc4c(c3)OCCO4)nn2c1=O	nan
	CHEMBL1441873	35631	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	4	0	10	2.6	CC(C)(C)c1nnc2sc(SCC(=O)c3ccc4c(c3)OCCO4)nn2c1=O	nan
	1860569	35654	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	2	0	5	4.2	Cc1ccc(-c2nc3c(c(=O)c4ccccc4n3C)c(=O)n2-c2ccccc2)cc1	nan
	CHEMBL1442098	35654	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	2	0	5	4.2	Cc1ccc(-c2nc3c(c(=O)c4ccccc4n3C)c(=O)n2-c2ccccc2)cc1	nan
	5302651	35844	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	7	1	5	3.7	CCc1ccc(NC(=O)CSc2nc(C)cc(COC)c2C#N)cc1	nan
	CHEMBL1443840	35844	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	7	1	5	3.7	CCc1ccc(NC(=O)CSc2nc(C)cc(COC)c2C#N)cc1	nan
	12006099	35882	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	498	13	1	7	4.1	CCCN(CCC)C(=O)Cn1c(=O)n(CCCCCC(=O)Nc2ccccc2)c(=O)c2sccc21	nan
	CHEMBL1444172	35882	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	498	13	1	7	4.1	CCCN(CCC)C(=O)Cn1c(=O)n(CCCCCC(=O)Nc2ccccc2)c(=O)c2sccc21	nan
	16019024	35916	0	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	7	1	6	2.5	COCCCNC(=O)c1ccc(Cn2c(=O)c3cccn3c3cccnc32)cc1	nan
	CHEMBL1444500	35916	0	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	7	1	6	2.5	COCCCNC(=O)c1ccc(Cn2c(=O)c3cccn3c3cccnc32)cc1	nan
	16034708	35919	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	5	1	5	3.6	Cc1ccc2c(=O)c(C(=O)c3ccccc3)cn(CC(=O)Nc3ccccc3)c2n1	nan
	CHEMBL1444524	35919	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	5	1	5	3.6	Cc1ccc2c(=O)c(C(=O)c3ccccc3)cn(CC(=O)Nc3ccccc3)c2n1	nan
	16016687	35939	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	5	2	5	4.8	COc1ccc(CNC(=O)Nc2ccc3c(c2)N(C)C(=O)c2ccccc2S3)cc1OC	nan
	CHEMBL1444758	35939	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	5	2	5	4.8	COc1ccc(CNC(=O)Nc2ccc3c(c2)N(C)C(=O)c2ccccc2S3)cc1OC	nan
	3238164	35964	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	345	5	1	3	3.1	O=C(CCN1CCN(c2ccc(F)cc2)CC1)Nc1ccc(F)cc1	nan
	CHEMBL1444967	35964	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	345	5	1	3	3.1	O=C(CCN1CCN(c2ccc(F)cc2)CC1)Nc1ccc(F)cc1	nan
	2296239	35965	13	None	-2	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	8	1	6	2.7	CCn1c(SCC(=O)NCCOc2ccccc2)nc2ccccc2c1=O	nan
	CHEMBL1444971	35965	13	None	-2	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	8	1	6	2.7	CCn1c(SCC(=O)NCCOc2ccccc2)nc2ccccc2c1=O	nan
	657584	35976	8	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	446	5	0	5	3.9	CC(C)Cc1nc(N2CCN(C(=O)Cc3ccccc3)CC2)c(C#N)c2c1COC(C)(C)C2	nan
	CHEMBL1445051	35976	8	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	446	5	0	5	3.9	CC(C)Cc1nc(N2CCN(C(=O)Cc3ccccc3)CC2)c(C#N)c2c1COC(C)(C)C2	nan
	15988979	36029	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	496	8	2	7	3.2	O=C(CCn1c(=O)c2sccc2n(CC(=O)Nc2ccccc2)c1=O)NCc1ccccc1Cl	nan
	CHEMBL1445545	36029	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	496	8	2	7	3.2	O=C(CCn1c(=O)c2sccc2n(CC(=O)Nc2ccccc2)c1=O)NCc1ccccc1Cl	nan
	16023569	36054	3	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	489	6	0	8	3.1	CC(=O)c1ccc(N2CCN(C(=O)CCn3cnc4onc(-c5ccc(F)cc5)c4c3=O)CC2)cc1	nan
	CHEMBL1445781	36054	3	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	489	6	0	8	3.1	CC(=O)c1ccc(N2CCN(C(=O)CCn3cnc4onc(-c5ccc(F)cc5)c4c3=O)CC2)cc1	nan
	7157939	36079	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	334	2	2	3	3.1	O=C(Nc1ccc2c(c1)C(=O)NC2=O)c1cc(Cl)ccc1Cl	nan
	CHEMBL1446030	36079	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	334	2	2	3	3.1	O=C(Nc1ccc2c(c1)C(=O)NC2=O)c1cc(Cl)ccc1Cl	nan
	1480468	36141	15	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	315	4	1	5	3.9	CC(C)Nc1nc(-c2ccncc2)nc(-c2ccccc2)c1C#N	nan
	CHEMBL1446611	36141	15	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	315	4	1	5	3.9	CC(C)Nc1nc(-c2ccncc2)nc(-c2ccccc2)c1C#N	nan
	2195706	36167	5	None	-1	3	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	344	5	1	8	2.8	CCOC(=O)CSc1nc(N)c(C#N)c(-c2cccs2)c1C#N	nan
	CHEMBL1446861	36167	5	None	-1	3	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	344	5	1	8	2.8	CCOC(=O)CSc1nc(N)c(C#N)c(-c2cccs2)c1C#N	nan
	16010637	36205	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	4	1	3	4.7	CCN(Cc1ccccc1)C(=O)c1cc2c(=O)[nH]c3ccc(C)cc3c2s1	nan
	CHEMBL1447092	36205	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	4	1	3	4.7	CCN(Cc1ccccc1)C(=O)c1cc2c(=O)[nH]c3ccc(C)cc3c2s1	nan
	2130696	36303	15	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	5	1	5	4.9	N#C/C(C(=O)NCc1ccco1)=C1/SC=C(c2ccccc2)N1c1ccccc1	nan
	CHEMBL1447960	36303	15	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	5	1	5	4.9	N#C/C(C(=O)NCc1ccco1)=C1/SC=C(c2ccccc2)N1c1ccccc1	nan
	4583349	36350	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	347	4	2	5	2.2	Cc1ccc(NC(=O)CCn2c(=O)[nH]c3ccsc3c2=O)cc1F	nan
	CHEMBL1448388	36350	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	347	4	2	5	2.2	Cc1ccc(NC(=O)CCn2c(=O)[nH]c3ccsc3c2=O)cc1F	nan
	5396132	36432	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	5	0	5	3.7	COc1cc(/C=C2/C(=O)ON=C2C)ccc1OCc1ccccc1F	nan
	CHEMBL1448972	36432	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	5	0	5	3.7	COc1cc(/C=C2/C(=O)ON=C2C)ccc1OCc1ccccc1F	nan
	1201887	36458	8	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	280	3	0	3	4.0	Cc1cccc(CSc2nc3c(cc2C#N)CCC3)c1	nan
	CHEMBL1449126	36458	8	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	280	3	0	3	4.0	Cc1cccc(CSc2nc3c(cc2C#N)CCC3)c1	nan
	649163	36462	9	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	6	0	5	3.0	CCN(CC)S(=O)(=O)c1ccc(Cl)c(C(=O)Oc2cccnc2)c1	nan
	CHEMBL1449162	36462	9	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	6	0	5	3.0	CCN(CC)S(=O)(=O)c1ccc(Cl)c(C(=O)Oc2cccnc2)c1	nan
	16019152	36519	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	440	4	0	7	4.0	Cc1ccccc1Cn1c(=O)n(Cc2ccc3c(c2)OCO3)c(=O)c2oc3ccccc3c21	nan
	CHEMBL1449607	36519	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	440	4	0	7	4.0	Cc1ccccc1Cn1c(=O)n(Cc2ccc3c(c2)OCO3)c(=O)c2oc3ccccc3c21	nan
	16017274	36537	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	6	1	6	2.6	CCN(CC)c1ccc(NC(=O)Cn2nc(C)n3cccc3c2=O)c(C)c1	nan
	CHEMBL1449789	36537	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	6	1	6	2.6	CCN(CC)c1ccc(NC(=O)Cn2nc(C)n3cccc3c2=O)c(C)c1	nan
	15996185	36545	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	7	2	4	4.7	CCC(C)NC(=O)CCC(=O)Nc1ccc2nc(N3CC(C)CC(C)C3)cc(C)c2c1	nan
	CHEMBL1449862	36545	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	7	2	4	4.7	CCC(C)NC(=O)CCC(=O)Nc1ccc2nc(N3CC(C)CC(C)C3)cc(C)c2c1	nan
	15989912	36549	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	5	1	7	5.4	Cc1cc(C)n(-c2nc3ccccc3nc2Nc2ccc(Cl)c(C(=O)OC(C)C)c2)n1	nan
	CHEMBL1449881	36549	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	5	1	7	5.4	Cc1cc(C)n(-c2nc3ccccc3nc2Nc2ccc(Cl)c(C(=O)OC(C)C)c2)n1	nan
	16020571	36710	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	4	0	5	4.2	CCn1cc(S(=O)(=O)c2cc(C)cc(C)c2)c(=O)c2cc(F)c(N3CCCC3)cc21	nan
	CHEMBL1451264	36710	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	4	0	5	4.2	CCn1cc(S(=O)(=O)c2cc(C)cc(C)c2)c(=O)c2cc(F)c(N3CCCC3)cc21	nan
	5058847	36853	9	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	6	1	6	3.0	COc1cc(NC(=O)Cn2c(C)cc3ccccc3c2=O)cc(OC)c1OC	nan
	CHEMBL1452293	36853	9	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	6	1	6	3.0	COc1cc(NC(=O)Cn2c(C)cc3ccccc3c2=O)cc(OC)c1OC	nan
	15988482	36983	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	4	0	4	4.4	Cc1ccc(C(=O)c2cn(Cc3ccc(F)cc3)c3nc(C)ccc3c2=O)cc1	nan
	CHEMBL1453340	36983	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	4	0	4	4.4	Cc1ccc(C(=O)c2cn(Cc3ccc(F)cc3)c3nc(C)ccc3c2=O)cc1	nan
	16019909	36991	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	5	0	8	3.8	COc1cc(-c2noc(-c3cc4cccc(C)c4oc3=O)n2)cc(OC)c1OC	nan
	CHEMBL1453424	36991	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	5	0	8	3.8	COc1cc(-c2noc(-c3cc4cccc(C)c4oc3=O)n2)cc(OC)c1OC	nan
	16024781	37032	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	5	0	4	1.9	O=C1C(=O)N(C2CCN(S(=O)(=O)c3ccc(F)cc3)CC2)CCN1Cc1ccccc1	nan
	CHEMBL1453815	37032	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	5	0	4	1.9	O=C1C(=O)N(C2CCN(S(=O)(=O)c3ccc(F)cc3)CC2)CCN1Cc1ccccc1	nan
	16024608	37042	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	503	9	1	7	3.5	COc1ccc(CCNC(=O)Cn2cc(C(=O)c3ccc(F)cc3)c(=O)c3ccc(C)nc32)cc1OC	nan
	CHEMBL1453881	37042	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	503	9	1	7	3.5	COc1ccc(CCNC(=O)Cn2cc(C(=O)c3ccc(F)cc3)c(=O)c3ccc(C)nc32)cc1OC	nan
	3940076	37055	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	301	3	1	5	3.3	Cc1ccc(CNc2nc3nc(C)c(Cl)c(C)n3n2)cc1	nan
	CHEMBL1453947	37055	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	301	3	1	5	3.3	Cc1ccc(CNc2nc3nc(C)c(Cl)c(C)n3n2)cc1	nan
	1604929	37060	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	441	7	0	5	4.6	CCCCn1cc[n+](-c2nc3ccccc3nc2[N-]S(=O)(=O)c2ccc(Cl)cc2)c1	nan
	CHEMBL1453974	37060	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	441	7	0	5	4.6	CCCCn1cc[n+](-c2nc3ccccc3nc2[N-]S(=O)(=O)c2ccc(Cl)cc2)c1	nan
	707946	37085	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	315	3	1	5	3.0	O=C(Nc1nc2nccc(-c3ccccc3)n2n1)c1ccccc1	nan
	CHEMBL1454141	37085	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	315	3	1	5	3.0	O=C(Nc1nc2nccc(-c3ccccc3)n2n1)c1ccccc1	nan
	16010581	37101	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	6	1	6	2.9	Cc1cc(C)cc(NC(=O)Cn2c(=O)n(CCC(C)C)c(=O)c3cccnc32)c1	nan
	CHEMBL1454246	37101	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	6	1	6	2.9	Cc1cc(C)cc(NC(=O)Cn2c(=O)n(CCC(C)C)c(=O)c3cccnc32)c1	nan
	15988208	37169	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	5	1	9	1.7	COC(=O)c1cccnc1-n1c(=O)c2cccnc2n(CC(=O)Nc2cccc(C)c2)c1=O	nan
	CHEMBL1454833	37169	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	5	1	9	1.7	COC(=O)c1cccnc1-n1c(=O)c2cccnc2n(CC(=O)Nc2cccc(C)c2)c1=O	nan
	5123668	37225	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	494	10	1	7	5.2	CCc1ccc(NC(=O)CSc2nc3c(sc4ccccc43)c(=O)n2CCN(CC)CC)cc1	nan
	CHEMBL1455415	37225	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	494	10	1	7	5.2	CCc1ccc(NC(=O)CSc2nc3c(sc4ccccc43)c(=O)n2CCN(CC)CC)cc1	nan
	135421575	37280	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	305	2	2	4	3.3	CCn1c(=O)c(-c2nc3ccccc3[nH]2)c(O)c2ccccc21	nan
	CHEMBL1455904	37280	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	305	2	2	4	3.3	CCn1c(=O)c(-c2nc3ccccc3[nH]2)c(O)c2ccccc21	nan
	914701	37307	8	None	-7	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	303	1	0	4	4.3	CCc1nc2sc3c(Cl)ncnc3c2c2c1CCCC2	nan
	CHEMBL1456130	37307	8	None	-7	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	303	1	0	4	4.3	CCc1nc2sc3c(Cl)ncnc3c2c2c1CCCC2	nan
	2023595	37431	15	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	5	1	6	4.1	COc1cccc(NC(=O)CSc2ncnc3c2oc2ccccc23)c1	nan
	CHEMBL1457309	37431	15	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	5	1	6	4.1	COc1cccc(NC(=O)CSc2ncnc3c2oc2ccccc23)c1	nan
	16024557	37467	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	5	1	5	4.0	Cc1ccc2c(=O)c(C(=O)c3ccc(Cl)cc3)cn(CC(=O)NC3CCCCC3)c2n1	nan
	CHEMBL1457615	37467	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	5	1	5	4.0	Cc1ccc2c(=O)c(C(=O)c3ccc(Cl)cc3)cn(CC(=O)NC3CCCCC3)c2n1	nan
	20920344	37490	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	6	1	7	4.4	Cc1ccc(-n2nc3c(N4CCC(C(=O)NCCc5cccs5)CC4)nnc(C)c3c2C)cc1	nan
	CHEMBL1457782	37490	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	6	1	7	4.4	Cc1ccc(-n2nc3c(N4CCC(C(=O)NCCc5cccs5)CC4)nnc(C)c3c2C)cc1	nan
	3245484	37620	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	466	8	2	7	1.9	COc1cc2[nH]c(=O)n(CCC(=O)NC3CCN(Cc4ccccc4)CC3)c(=O)c2cc1OC	nan
	CHEMBL1458892	37620	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	466	8	2	7	1.9	COc1cc2[nH]c(=O)n(CCC(=O)NC3CCN(Cc4ccccc4)CC3)c(=O)c2cc1OC	nan
	2467173	37642	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	441	9	1	11	1.4	C=CCn1c(SCC(=O)c2c(N)n(CCC)c(=O)n(C)c2=O)nnc1-c1ccncc1	nan
	CHEMBL1459057	37642	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	441	9	1	11	1.4	C=CCn1c(SCC(=O)c2c(N)n(CCC)c(=O)n(C)c2=O)nnc1-c1ccncc1	nan
	3185309	37669	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	567	10	3	9	3.7	COc1ccc(OC)c(C(C(=O)NC2CCCCC2)N(C(=O)c2snc(C(N)=O)c2N)c2ccccc2OC)c1	nan
	CHEMBL1459257	37669	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	567	10	3	9	3.7	COc1ccc(OC)c(C(C(=O)NC2CCCCC2)N(C(=O)c2snc(C(N)=O)c2N)c2ccccc2OC)c1	nan
	2910207	37686	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	7	1	6	3.9	O=C(C1=C(O)C(=O)N(CCCn2ccnc2)C1c1cccc(Br)c1)c1ccco1	nan
	CHEMBL1459409	37686	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	7	1	6	3.9	O=C(C1=C(O)C(=O)N(CCCn2ccnc2)C1c1cccc(Br)c1)c1ccco1	nan
	2138506	37819	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	5	2	6	3.0	CCOC(=O)c1[nH]c2ccc(OC)cc2c1N=C(S)N1CCN(C(=O)OCC)CC1	nan
	CHEMBL1460540	37819	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	5	2	6	3.0	CCOC(=O)c1[nH]c2ccc(OC)cc2c1N=C(S)N1CCN(C(=O)OCC)CC1	nan
	1995746	37832	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	6	3	8	0.9	NC(=O)c1ccc(NC(=O)CSc2nnc(-c3ccccn3)n2N)cc1	nan
	CHEMBL1460633	37832	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	6	3	8	0.9	NC(=O)c1ccc(NC(=O)CSc2nnc(-c3ccccn3)n2N)cc1	nan
	1511731	37860	18	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	3	1	6	2.9	COc1ccc(C(=O)Nc2nc(C)c3cc4c(cc3n2)OCO4)cc1	nan
	CHEMBL1460863	37860	18	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	3	1	6	2.9	COc1ccc(C(=O)Nc2nc(C)c3cc4c(cc3n2)OCO4)cc1	nan
	4340474	37910	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	6	2	6	2.1	CCCCNC(=O)CCn1c(=S)[nH]c2cc3c(cc2c1=O)OCO3	nan
	CHEMBL1461327	37910	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	6	2	6	2.1	CCCCNC(=O)CCn1c(=S)[nH]c2cc3c(cc2c1=O)OCO3	nan
	2331607	37940	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	2	1	5	2.7	O=C(Nc1ccccn1)c1ccc2c(c1)S(=O)(=O)c1ccccc1C2=O	nan
	CHEMBL1461642	37940	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	2	1	5	2.7	O=C(Nc1ccccn1)c1ccc2c(c1)S(=O)(=O)c1ccccc1C2=O	nan
	4594455	38000	16	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	446	5	0	7	3.9	CSc1nc(N2CCN(c3ccccc3)CC2)cc(N2CCN(c3ccccc3)CC2)n1	nan
	CHEMBL1462148	38000	16	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	446	5	0	7	3.9	CSc1nc(N2CCN(c3ccccc3)CC2)cc(N2CCN(c3ccccc3)CC2)n1	nan
	661296	38031	11	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	267	2	2	1	3.2	CCc1c(C(=O)O)[nH]c2ccc(Br)cc12	nan
	CHEMBL1462380	38031	11	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	267	2	2	1	3.2	CCc1c(C(=O)O)[nH]c2ccc(Br)cc12	nan
	3183779	38061	5	None	-2	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	472	5	1	9	3.7	Oc1nc2cc3c(cc2cc1C(c1nnnn1Cc1ccccc1)N1CCCCCC1)OCCO3	nan
	CHEMBL1462671	38061	5	None	-2	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	472	5	1	9	3.7	Oc1nc2cc3c(cc2cc1C(c1nnnn1Cc1ccccc1)N1CCCCCC1)OCCO3	nan
	5418960	38080	9	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	309	1	1	4	3.3	O=c1c2cc3c(nc2[nH]c(=S)n1-c1ccccc1)CCCC3	nan
	CHEMBL1462820	38080	9	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	309	1	1	4	3.3	O=c1c2cc3c(nc2[nH]c(=S)n1-c1ccccc1)CCCC3	nan
	2766000	38112	14	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	10	1	8	3.9	COCCCn1c(SCc2ccc(OC)cc2)nc2cc(OC)c(OC)cc2c1=N	nan
	CHEMBL1463048	38112	14	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	10	1	8	3.9	COCCCn1c(SCc2ccc(OC)cc2)nc2cc(OC)c(OC)cc2c1=N	nan
	16188024	38135	2	None	-2	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	2	1	4	5.0	Cc1ccc2nc(O)c3cc(C(=O)N(C)c4ccccc4C)sc3c2c1	nan
	CHEMBL1463271	38135	2	None	-2	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	2	1	4	5.0	Cc1ccc2nc(O)c3cc(C(=O)N(C)c4ccccc4C)sc3c2c1	nan
	4429285	38148	3	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	4	1	7	3.7	COC(=O)c1ccc(Nc2ncnc3c2cnn3-c2cccc(C)c2)cc1	nan
	CHEMBL1463413	38148	3	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	4	1	7	3.7	COC(=O)c1ccc(Nc2ncnc3c2cnn3-c2cccc(C)c2)cc1	nan
	1738267	38153	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	8	1	4	5.2	O=C(CCC(=O)OCC(=O)c1ccc(-c2ccccc2)cc1)Nc1cccc(Cl)c1	nan
	CHEMBL1463488	38153	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	8	1	4	5.2	O=C(CCC(=O)OCC(=O)c1ccc(-c2ccccc2)cc1)Nc1cccc(Cl)c1	nan
	3761375	38277	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	299	3	0	4	4.3	CSc1nc(C)c2c(n1)N(c1ccc(C(C)C)cc1)CC2	nan
	CHEMBL1464437	38277	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	299	3	0	4	4.3	CSc1nc(C)c2c(n1)N(c1ccc(C(C)C)cc1)CC2	nan
	2044631	38332	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	4	2	4	4.3	Cc1cc(C)c(NC(=O)CSc2nc3cc(Br)c[nH]c-3n2)c(C)c1	nan
	CHEMBL1464810	38332	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	4	2	4	4.3	Cc1cc(C)c(NC(=O)CSc2nc3cc(Br)c[nH]c-3n2)c(C)c1	nan
	2372173	38378	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	4	1	4	4.4	CC(=O)c1sc(NC(=O)c2ccccc2F)nc1-c1ccccc1	nan
	CHEMBL1465138	38378	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	4	1	4	4.4	CC(=O)c1sc(NC(=O)c2ccccc2F)nc1-c1ccccc1	nan
	2988623	38600	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	5	0	6	3.2	CCOc1ccc(C(=O)N2CCN(c3cnn(-c4ccccc4)c(=O)c3Cl)CC2)cc1	nan
	CHEMBL1466802	38600	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	5	0	6	3.2	CCOc1ccc(C(=O)N2CCN(c3cnn(-c4ccccc4)c(=O)c3Cl)CC2)cc1	nan
	2428874	38620	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	301	2	2	4	1.9	O=C(Nc1cccc2c1C(=O)NC2=O)c1cccnc1Cl	nan
	CHEMBL1466996	38620	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	301	2	2	4	1.9	O=C(Nc1cccc2c1C(=O)NC2=O)c1cccnc1Cl	nan
	3574259	38640	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	5	2	6	3.1	O=C(CCn1c(=S)[nH]c2cc3c(cc2c1=O)OCO3)NCc1cccc(Cl)c1	nan
	CHEMBL1467198	38640	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	5	2	6	3.1	O=C(CCn1c(=S)[nH]c2cc3c(cc2c1=O)OCO3)NCc1cccc(Cl)c1	nan
	16007702	38672	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	441	7	1	5	2.6	CCn1cc(C(=O)NCCc2ccc(C)cc2)c(=O)c2cc(S(=O)(=O)N(C)C)ccc21	nan
	CHEMBL1467433	38672	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	441	7	1	5	2.6	CCn1cc(C(=O)NCCc2ccc(C)cc2)c(=O)c2cc(S(=O)(=O)N(C)C)ccc21	nan
	663318	38685	16	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	4	0	6	4.3	CC1CCN(c2nc3ccccc3nc2C(C#N)C(=O)OC2CCCCC2)CC1	nan
	CHEMBL1467520	38685	16	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	4	0	6	4.3	CC1CCN(c2nc3ccccc3nc2C(C#N)C(=O)OC2CCCCC2)CC1	nan
	2820576	38784	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	6	1	6	5.4	Cc1csc2sc(-c3ccnc(SCC(=O)NCc4ccccc4)n3)c(C)c12	nan
	CHEMBL1468435	38784	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	6	1	6	5.4	Cc1csc2sc(-c3ccnc(SCC(=O)NCc4ccccc4)n3)c(C)c12	nan
	970728	38802	10	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	325	2	2	2	5.0	Cc1cc(C)nc(NC(S)=Nc2cccc(Cl)c2Cl)c1	nan
	CHEMBL1468575	38802	10	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	325	2	2	2	5.0	Cc1cc(C)nc(NC(S)=Nc2cccc(Cl)c2Cl)c1	nan
	4294342	38805	13	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	299	3	2	2	3.6	Cc1cc2cc(CNC(=O)NC3CCCCC3)ccc2n1C	nan
	CHEMBL1468608	38805	13	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	299	3	2	2	3.6	Cc1cc2cc(CNC(=O)NC3CCCCC3)ccc2n1C	nan
	648454	38812	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	3	1	4	3.4	Cc1cc(C)nc(N2CCC(C(=O)Nc3ccc4c(c3)CCC4)CC2)n1	nan
	CHEMBL1468653	38812	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	3	1	4	3.4	Cc1cc(C)nc(N2CCC(C(=O)Nc3ccc4c(c3)CCC4)CC2)n1	nan
	7202588	38895	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	6	1	7	2.9	COC(=O)c1ccc2nc(NC(=O)CCS(=O)(=O)c3ccccc3)sc2c1	nan
	CHEMBL1469363	38895	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	6	1	7	2.9	COC(=O)c1ccc2nc(NC(=O)CCS(=O)(=O)c3ccccc3)sc2c1	nan
	1073207	39035	8	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	6	0	9	2.4	COc1ccc(-n2nnnc2SCC(=O)c2ccc3c(c2)OCCO3)cc1	nan
	CHEMBL1470594	39035	8	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	6	0	9	2.4	COc1ccc(-n2nnnc2SCC(=O)c2ccc3c(c2)OCCO3)cc1	nan
	3615142	39036	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	286	2	1	3	4.0	Cc1c(C(=O)Nc2cccnc2Cl)oc2ccccc12	nan
	CHEMBL1470599	39036	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	286	2	1	3	4.0	Cc1c(C(=O)Nc2cccnc2Cl)oc2ccccc12	nan
	16009952	39273	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	5	1	7	0.9	Cc1ccc(NC(=O)CN(C)S(=O)(=O)c2ccc3c(c2)n(C)c(=O)c(=O)n3C)cc1F	nan
	CHEMBL1472658	39273	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	5	1	7	0.9	Cc1ccc(NC(=O)CN(C)S(=O)(=O)c2ccc3c(c2)n(C)c(=O)c(=O)n3C)cc1F	nan
	1892783	39281	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	3	1	5	4.8	Cc1ccc(-c2nnc3c4ccccc4c(C)nn23)cc1NC(=O)c1ccccc1	nan
	CHEMBL1472759	39281	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	3	1	5	4.8	Cc1ccc(-c2nnc3c4ccccc4c(C)nn23)cc1NC(=O)c1ccccc1	nan
	16008277	39285	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	495	4	1	5	5.8	Cc1cc(N2CCC(C(=O)Nc3ccc(F)cc3F)CC2)n2nc(C)c(-c3ccc(Cl)cc3)c2n1	nan
	CHEMBL1472790	39285	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	495	4	1	5	5.8	Cc1cc(N2CCC(C(=O)Nc3ccc(F)cc3F)CC2)n2nc(C)c(-c3ccc(Cl)cc3)c2n1	nan
	16015830	39288	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	5	1	4	5.1	O=C(COc1ccccc1F)Nc1ccc(-c2nc3ccccc3s2)cc1	nan
	CHEMBL1472798	39288	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	5	1	4	5.1	O=C(COc1ccccc1F)Nc1ccc(-c2nc3ccccc3s2)cc1	nan
	16030736	39298	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	3	1	3	5.3	CC(C)(C)C(=O)Nc1cc(-c2cccc(Br)c2)nn1-c1ccccc1	nan
	CHEMBL1472994	39298	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	3	1	3	5.3	CC(C)(C)C(=O)Nc1cc(-c2cccc(Br)c2)nn1-c1ccccc1	nan
	16015144	39301	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	347	4	1	5	4.6	O=C(/C=C/c1ccc(Cl)cc1)Nc1nc(-c2cccs2)ns1	nan
	CHEMBL1472998	39301	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	347	4	1	5	4.6	O=C(/C=C/c1ccc(Cl)cc1)Nc1nc(-c2cccs2)ns1	nan
	16010790	39328	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	6	1	7	2.7	COc1ccc(Cn2c(=O)c3cccnc3n(CC(=O)Nc3ccc(C)c(F)c3)c2=O)cc1	nan
	CHEMBL1473410	39328	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	6	1	7	2.7	COc1ccc(Cn2c(=O)c3cccnc3n(CC(=O)Nc3ccc(C)c(F)c3)c2=O)cc1	nan
	16009809	39330	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	6	2	5	5.9	COc1ccc(NC(=O)c2oc3ccccc3c2NC(=O)C23CC4CC(CC(C4)C2)C3)c(OC)c1	nan
	CHEMBL1473436	39330	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	6	2	5	5.9	COc1ccc(NC(=O)c2oc3ccccc3c2NC(=O)C23CC4CC(CC(C4)C2)C3)c(OC)c1	nan
	16009067	39335	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	358	2	1	3	5.5	Cc1ccc2nc(Cl)c3cc(C(=O)NC4CCCCC4)sc3c2c1	nan
	CHEMBL1473455	39335	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	358	2	1	3	5.5	Cc1ccc2nc(Cl)c3cc(C(=O)NC4CCCCC4)sc3c2c1	nan
	864758	39342	18	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	307	4	1	6	2.1	CC(=O)c1ccc(NC(=O)c2ccc(-n3cnnn3)cc2)cc1	nan
	CHEMBL1473580	39342	18	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	307	4	1	6	2.1	CC(=O)c1ccc(NC(=O)c2ccc(-n3cnnn3)cc2)cc1	nan
	16010866	39343	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	7	1	7	2.9	COc1ccc(NC(=O)Cn2c(=O)n(CCC(C)C)c(=O)c3cccnc32)cc1Cl	nan
	CHEMBL1473610	39343	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	7	1	7	2.9	COc1ccc(NC(=O)Cn2c(=O)n(CCC(C)C)c(=O)c3cccnc32)cc1Cl	nan
	16008902	39345	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	373	4	1	4	3.3	Cc1cccc(CCNC(=O)c2cc3c(=O)n(C)c4ccccc4c3n2C)c1	nan
	CHEMBL1473624	39345	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	373	4	1	4	3.3	Cc1cccc(CCNC(=O)c2cc3c(=O)n(C)c4ccccc4c3n2C)c1	nan
	4425770	39351	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	5	1	5	4.4	Cc1cccc(-c2nnc(SCC(=O)Nc3ccc(C)c(C)c3)o2)c1	nan
	CHEMBL1473697	39351	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	5	1	5	4.4	Cc1cccc(-c2nnc(SCC(=O)Nc3ccc(C)c(C)c3)o2)c1	nan
	16025407	39356	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	538	6	1	6	5.2	Cc1ccc(NC(=O)CSc2ncc3c(n2)-c2ccccc2N(Cc2cccc(F)c2)S3(=O)=O)cc1F	nan
	CHEMBL1473728	39356	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	538	6	1	6	5.2	Cc1ccc(NC(=O)CSc2ncc3c(n2)-c2ccccc2N(Cc2cccc(F)c2)S3(=O)=O)cc1F	nan
	15989780	39402	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	4	1	5	4.9	Clc1ccc(CCNc2nc3cc(Cl)c(Cl)cc3n3cnnc23)cc1	nan
	CHEMBL1474477	39402	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	4	1	5	4.9	Clc1ccc(CCNc2nc3cc(Cl)c(Cl)cc3n3cnnc23)cc1	nan
	16034729	39414	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	467	5	1	7	5.0	COc1ccc(-c2cn3nc(N4CCC(C(=O)Nc5cccc(Cl)c5)CC4)sc3n2)cc1	nan
	CHEMBL1474594	39414	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	467	5	1	7	5.0	COc1ccc(-c2cn3nc(N4CCC(C(=O)Nc5cccc(Cl)c5)CC4)sc3n2)cc1	nan
	16012452	39426	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	3	2	5	2.4	O=C(NCc1ccccc1)C(=O)Nc1ccc2nc3n(c(=O)c2c1)CCCCC3	nan
	CHEMBL1474806	39426	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	3	2	5	2.4	O=C(NCc1ccccc1)C(=O)Nc1ccc2nc3n(c(=O)c2c1)CCCCC3	nan
	16020997	39428	0	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	6	1	5	4.9	Cc1ccc(NC(=O)Cn2c(SCc3ccc(F)cc3)nc3cccnc32)cc1F	nan
	CHEMBL1474813	39428	0	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	6	1	5	4.9	Cc1ccc(NC(=O)Cn2c(SCc3ccc(F)cc3)nc3cccnc32)cc1F	nan
	16012520	39456	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	441	6	2	5	4.9	CC(=O)Nc1ccc(NC(=O)CCc2c(C)nc3c(c(C)nn3-c3ccccc3)c2C)cc1	nan
	CHEMBL1475217	39456	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	441	6	2	5	4.9	CC(=O)Nc1ccc(NC(=O)CCc2c(C)nc3c(c(C)nn3-c3ccccc3)c2C)cc1	nan
	16008390	39461	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	400	6	1	4	4.2	CCc1ccc(CNC(=O)CSc2cc(=O)n(C)c3ccc(Cl)cc23)cc1	nan
	CHEMBL1475336	39461	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	400	6	1	4	4.2	CCc1ccc(CNC(=O)CSc2cc(=O)n(C)c3ccc(Cl)cc23)cc1	nan
	3225367	39465	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	4	1	3	5.8	Cc1cccc(C)c1NC(=O)c1cc2sccc2n1Cc1ccc(F)cc1	nan
	CHEMBL1475367	39465	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	4	1	3	5.8	Cc1cccc(C)c1NC(=O)c1cc2sccc2n1Cc1ccc(F)cc1	nan
	1983981	39473	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	2	0	4	5.2	Cc1ccc(-c2nn3c(-c4ccc(C)cc4)nnc3c3ccccc23)cc1	nan
	CHEMBL1475431	39473	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	2	0	4	5.2	Cc1ccc(-c2nn3c(-c4ccc(C)cc4)nnc3c3ccccc23)cc1	nan
	16030137	39487	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	465	7	1	7	3.6	CCOc1ccccc1CNC(=O)Cn1nc(C)c2nn(-c3ccc(Cl)cc3)c(C)c2c1=O	nan
	CHEMBL1475622	39487	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	465	7	1	7	3.6	CCOc1ccccc1CNC(=O)Cn1nc(C)c2nn(-c3ccc(Cl)cc3)c(C)c2c1=O	nan
	16016540	39489	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	306	2	2	2	3.7	Cc1cc(=O)c2cc(C(=O)Nc3cccc(C)c3C)ccc2[nH]1	nan
	CHEMBL1475643	39489	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	306	2	2	2	3.7	Cc1cc(=O)c2cc(C(=O)Nc3cccc(C)c3C)ccc2[nH]1	nan
	16026533	39497	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	446	6	1	7	4.0	COc1ccc(OC)c(NC(=O)C(C)n2c(=O)cc(C)c3c(C)nn(-c4ccccc4)c32)c1	nan
	CHEMBL1475722	39497	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	446	6	1	7	4.0	COc1ccc(OC)c(NC(=O)C(C)n2c(=O)cc(C)c3c(C)nn(-c4ccccc4)c32)c1	nan
	16030897	39501	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	6	1	6	4.8	COc1ccc(-c2cn3nc(SCC(=O)Nc4cccc(C)c4C)ccc3n2)cc1	nan
	CHEMBL1475786	39501	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	6	1	6	4.8	COc1ccc(-c2cn3nc(SCC(=O)Nc4cccc(C)c4C)ccc3n2)cc1	nan
	16012637	39522	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	4	0	10	3.3	Cc1ccc2nc3c(cc(C#N)c(=O)n3-c3nnc(SCc4ccccc4)s3)c(=O)n2c1	nan
	CHEMBL1476168	39522	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	4	0	10	3.3	Cc1ccc2nc3c(cc(C#N)c(=O)n3-c3nnc(SCc4ccccc4)s3)c(=O)n2c1	nan
	16009819	39532	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	495	6	1	8	4.3	COc1ccc(NC(=O)Cn2c(=O)n(Cc3ccco3)c(=O)c3sc4ccccc4c32)cc1Cl	nan
	CHEMBL1476323	39532	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	495	6	1	8	4.3	COc1ccc(NC(=O)Cn2c(=O)n(Cc3ccco3)c(=O)c3sc4ccccc4c32)cc1Cl	nan
	16009801	39538	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	491	7	1	9	3.7	COc1ccc(NC(=O)Cn2c(=O)n(Cc3ccco3)c(=O)c3sc4ccccc4c32)c(OC)c1	nan
	CHEMBL1476410	39538	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	491	7	1	9	3.7	COc1ccc(NC(=O)Cn2c(=O)n(Cc3ccco3)c(=O)c3sc4ccccc4c32)c(OC)c1	nan
	15987507	39543	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	3	1	4	6.1	Cc1cc(C)c2oc(-c3ccc(Cl)c(NC(=O)c4cccs4)c3)nc2c1	nan
	CHEMBL1476493	39543	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	3	1	4	6.1	Cc1cc(C)c2oc(-c3ccc(Cl)c(NC(=O)c4cccs4)c3)nc2c1	nan
	16030393	39551	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	5	0	4	5.2	Cc1ccc(Cc2nc3ccccc3nc2SCC(=O)N2CCc3ccccc32)cc1	nan
	CHEMBL1476572	39551	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	425	5	0	4	5.2	Cc1ccc(Cc2nc3ccccc3nc2SCC(=O)N2CCc3ccccc32)cc1	nan
	16010862	39558	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	6	1	6	2.9	Cc1ccc(NC(=O)Cn2c(=O)n(CCC(C)C)c(=O)c3cccnc32)cc1C	nan
	CHEMBL1476637	39558	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	6	1	6	2.9	Cc1ccc(NC(=O)Cn2c(=O)n(CCC(C)C)c(=O)c3cccnc32)cc1C	nan
	4154280	39571	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	6	1	5	5.9	CCc1ccccc1NC(=O)C(CC)Sc1ncnc2c1sc1ccccc12	nan
	CHEMBL1476806	39571	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	6	1	5	5.9	CCc1ccccc1NC(=O)C(CC)Sc1ncnc2c1sc1ccccc12	nan
	7184887	39585	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	3	0	8	3.4	CC1CCN(c2nc3c(S(=O)(=O)c4ccccc4)nnn3c3ccsc23)CC1	nan
	CHEMBL1476979	39585	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	3	0	8	3.4	CC1CCN(c2nc3c(S(=O)(=O)c4ccccc4)nnn3c3ccsc23)CC1	nan
	666072	39686	8	None	-5	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	3	1	6	4.6	CSc1ccc(-c2c(C#N)c(N)nc3c2c(C)nn3-c2ccccc2)cc1	nan
	CHEMBL1477886	39686	8	None	-5	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	3	1	6	4.6	CSc1ccc(-c2c(C#N)c(N)nc3c2c(C)nn3-c2ccccc2)cc1	nan
	2810062	39701	6	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	292	2	1	6	2.9	Cc1csc2c(=O)sc(NC(=O)c3ccco3)nc12	nan
	CHEMBL1478110	39701	6	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	292	2	1	6	2.9	Cc1csc2c(=O)sc(NC(=O)c3ccco3)nc12	nan
	16014364	39733	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	6	1	4	4.8	Cc1ccc(CNC(=O)c2nc(SCc3ccc(F)cc3)ncc2Cl)cc1	nan
	CHEMBL1478416	39733	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	6	1	4	4.8	Cc1ccc(CNC(=O)c2nc(SCc3ccc(F)cc3)ncc2Cl)cc1	nan
	947086	39756	8	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	326	2	0	4	4.1	COc1ccc(-c2c(C#N)c(C)nc3c2C(=O)c2ccccc2-3)cc1	nan
	CHEMBL1478573	39756	8	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	326	2	0	4	4.1	COc1ccc(-c2c(C#N)c(C)nc3c2C(=O)c2ccccc2-3)cc1	nan
	15990421	39767	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	477	3	1	4	5.9	Cc1cc(Br)ccc1NC(=O)c1cn(C2CCCC2)c(=O)c2c1c1ccccc1n2C	nan
	CHEMBL1478684	39767	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	477	3	1	4	5.9	Cc1cc(Br)ccc1NC(=O)c1cn(C2CCCC2)c(=O)c2c1c1ccccc1n2C	nan
	2150494	39779	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	423	7	1	7	3.8	COCCn1c(SCC(=O)Nc2ccc(C)cc2)nc2c(oc3ccccc32)c1=O	nan
	CHEMBL1478802	39779	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	423	7	1	7	3.8	COCCn1c(SCC(=O)Nc2ccc(C)cc2)nc2c(oc3ccccc32)c1=O	nan
	9267240	39787	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	316	3	1	4	3.3	O=C(Nc1ccc(Cl)cc1F)c1ccc(-n2cncn2)cc1	nan
	CHEMBL1478883	39787	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	316	3	1	4	3.3	O=C(Nc1ccc(Cl)cc1F)c1ccc(-n2cncn2)cc1	nan
	16015604	39827	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	466	7	1	6	6.3	CCOc1ccc(C(=O)c2oc3ccccc3c2NC(=O)c2cc(-c3ccc(C)cc3)on2)cc1	nan
	CHEMBL1479260	39827	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	466	7	1	6	6.3	CCOc1ccc(C(=O)c2oc3ccccc3c2NC(=O)c2cc(-c3ccc(C)cc3)on2)cc1	nan
	4050786	39899	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	5	1	7	2.8	COCCn1/c(=N/C(=O)c2ccc3c(c2)OCCO3)sc2cc(NC(C)=O)ccc21	nan
	CHEMBL1479784	39899	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	5	1	7	2.8	COCCn1/c(=N/C(=O)c2ccc3c(c2)OCCO3)sc2cc(NC(C)=O)ccc21	nan
	16009694	39901	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	8	1	8	4.6	COc1ccc(-c2nnn3c2nc(NCCc2ccc(OC)c(OC)c2)c2ccccc23)cc1	nan
	CHEMBL1479788	39901	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	8	1	8	4.6	COc1ccc(-c2nnn3c2nc(NCCc2ccc(OC)c(OC)c2)c2ccccc23)cc1	nan
	2140519	40061	17	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	5	3	6	1.2	COC(=O)CCC(=O)NC(=S)Nc1sc(C)c(C)c1C(N)=O	nan
	CHEMBL1481122	40061	17	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	5	3	6	1.2	COC(=O)CCC(=O)NC(=S)Nc1sc(C)c(C)c1C(N)=O	nan
	16189596	40074	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	7	1	4	4.5	CCN1CCCc2cc(CN(CCN3CCOCC3)C(S)=Nc3ccccc3C)ccc21	nan
	CHEMBL1481195	40074	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	7	1	4	4.5	CCN1CCCc2cc(CN(CCN3CCOCC3)C(S)=Nc3ccccc3C)ccc21	nan
	6324455	40158	14	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	330	4	1	4	3.1	CCN(CC)S(=O)(=O)c1ccc2nc(O)c3ccccc3c2c1	nan
	CHEMBL1482015	40158	14	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	330	4	1	4	3.1	CCN(CC)S(=O)(=O)c1ccc2nc(O)c3ccccc3c2c1	nan
	4898982	40183	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	4	1	5	2.9	COc1ccc2cc(C(=O)N3CCN(Cc4ccc5c(c4)OCO5)CC3)[nH]c2c1	nan
	CHEMBL1482223	40183	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	4	1	5	2.9	COc1ccc2cc(C(=O)N3CCN(Cc4ccc5c(c4)OCO5)CC3)[nH]c2c1	nan
	16194617	40193	9	None	-2	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	5	1	6	4.4	CCOc1ncccc1C(=O)Nc1cccc(-c2nc3cccnc3s2)c1	nan
	CHEMBL1482332	40193	9	None	-2	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	5	1	6	4.4	CCOc1ncccc1C(=O)Nc1cccc(-c2nc3cccnc3s2)c1	nan
	7598416	40297	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	4	1	6	2.6	Cc1cccc(Cn2cccc(C(=O)Nc3nnc(C)s3)c2=O)c1	nan
	CHEMBL1483270	40297	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	340	4	1	6	2.6	Cc1cccc(Cn2cccc(C(=O)Nc3nnc(C)s3)c2=O)c1	nan
	16033878	40309	3	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	2	1	6	4.0	Cc1c(Cl)cccc1Nc1nn2c(=O)c3ccccc3nc2s1	nan
	CHEMBL1483384	40309	3	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	2	1	6	4.0	Cc1c(Cl)cccc1Nc1nn2c(=O)c3ccccc3nc2s1	nan
	5033969	40353	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	5	2	4	3.0	CC(=O)c1c(C)[nH]c(C(=O)Nc2ccc(Cl)c(S(=O)(=O)N(C)C)c2)c1C	nan
	CHEMBL1483695	40353	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	5	2	4	3.0	CC(=O)c1c(C)[nH]c(C(=O)Nc2ccc(Cl)c(S(=O)(=O)N(C)C)c2)c1C	nan
	2346667	40363	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	313	6	0	5	2.8	COc1ccc(C(=O)COC(=O)c2ccc(N(C)C)cc2)cc1	nan
	CHEMBL1483762	40363	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	313	6	0	5	2.8	COc1ccc(C(=O)COC(=O)c2ccc(N(C)C)cc2)cc1	nan
	4199549	40384	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	477	9	0	6	4.9	CCOc1ccccc1C(=O)N1CCc2cc(OC)c(OC)cc2C1COc1ccc(OC)cc1	nan
	CHEMBL1483991	40384	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	477	9	0	6	4.9	CCOc1ccccc1C(=O)N1CCc2cc(OC)c(OC)cc2C1COc1ccc(OC)cc1	nan
	135399202	40449	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	313	2	1	5	3.1	NC1=C(c2nc3ccccc3s2)C(=O)CN1C1CCCCC1	nan
	CHEMBL1484439	40449	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	313	2	1	5	3.1	NC1=C(c2nc3ccccc3s2)C(=O)CN1C1CCCCC1	nan
	2377756	40485	21	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	3	1	6	3.4	O=C(O)c1cccnc1Sc1ncnc2sc3c(c12)CCC3	nan
	CHEMBL1484807	40485	21	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	3	1	6	3.4	O=C(O)c1cccnc1Sc1ncnc2sc3c(c12)CCC3	nan
	135410529	40524	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	5	2	6	4.7	CCS(=O)(=O)c1cccc(C(=O)Nc2ccc(-c3nc4ccccc4s3)c(O)c2)c1	nan
	CHEMBL1485170	40524	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	5	2	6	4.7	CCS(=O)(=O)c1cccc(C(=O)Nc2ccc(-c3nc4ccccc4s3)c(O)c2)c1	nan
	135521955	40563	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	7	2	7	4.7	Cc1cc(-n2c(SCC(=O)NCCC3=CCCCC3)nc3nnc(C)c-3c2N)ccc1Cl	nan
	CHEMBL1485562	40563	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	7	2	7	4.7	Cc1cc(-n2c(SCC(=O)NCCC3=CCCCC3)nc3nnc(C)c-3c2N)ccc1Cl	nan
	15989053	40575	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	519	8	1	8	4.0	Cc1cc(C)c(Cn2c(=O)n(CCCC(=O)NCc3ccc4c(c3)OCO4)c(=O)c3sccc32)c(C)c1	nan
	CHEMBL1485622	40575	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	519	8	1	8	4.0	Cc1cc(C)c(Cn2c(=O)n(CCCC(=O)NCc3ccc4c(c3)OCO4)c(=O)c3sccc32)c(C)c1	nan
	4277738	40587	1	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	358	4	1	3	4.8	Sc1nc(-c2ccc(Br)cc2)cn1CCc1ccccc1	nan
	CHEMBL1485734	40587	1	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	358	4	1	3	4.8	Sc1nc(-c2ccc(Br)cc2)cn1CCc1ccccc1	nan
	16012072	40623	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	477	11	1	6	3.8	CCCCN(C)CCCNC(=O)Cn1ncc2c3ccccc3n(Cc3ccccc3F)c2c1=O	nan
	CHEMBL1486036	40623	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	477	11	1	6	3.8	CCCCN(C)CCCNC(=O)Cn1ncc2c3ccccc3n(Cc3ccccc3F)c2c1=O	nan
	1273744	40653	11	None	-6	3	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	5	1	7	3.8	Cc1cc(C)c(C#N)c(SCC(=O)Nc2nnc(-c3ccccc3)s2)n1	nan
	CHEMBL1486391	40653	11	None	-6	3	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	5	1	7	3.8	Cc1cc(C)c(C#N)c(SCC(=O)Nc2nnc(-c3ccccc3)s2)n1	nan
	16021806	40676	0	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	4	1	4	5.1	CSc1ncc(C(=O)Nc2ccccc2C(F)(F)F)c(-c2ccccc2)n1	nan
	CHEMBL1486543	40676	0	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	4	1	4	5.1	CSc1ncc(C(=O)Nc2ccccc2C(F)(F)F)c(-c2ccccc2)n1	nan
	5339079	40705	14	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	313	2	1	4	4.4	Cc1nc(-c2ccccc2)nc2nc(-c3ccccc3)cc(O)c12	nan
	CHEMBL1486764	40705	14	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	313	2	1	4	4.4	Cc1nc(-c2ccccc2)nc2nc(-c3ccccc3)cc(O)c12	nan
	702036	40782	13	None	-19	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	1	0	5	4.2	N#Cc1c2c(c(-n3cnc4ccccc43)n3c1nc1ccccc13)CCC2	nan
	CHEMBL1487421	40782	13	None	-19	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	1	0	5	4.2	N#Cc1c2c(c(-n3cnc4ccccc43)n3c1nc1ccccc13)CCC2	nan
	15989752	40802	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	4	1	5	3.9	Cc1ccc2nc(NCCc3ccc(Cl)cc3)c3nncn3c2c1	nan
	CHEMBL1487625	40802	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	4	1	5	3.9	Cc1ccc2nc(NCCc3ccc(Cl)cc3)c3nncn3c2c1	nan
	16008663	40815	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	5	1	8	1.6	COC(=O)c1ccc(NC(=O)CCc2c(C)nc3c(c2C)c(=O)n(C)c(=O)n3C)cc1	nan
	CHEMBL1487699	40815	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	5	1	8	1.6	COC(=O)c1ccc(NC(=O)CCc2c(C)nc3c(c2C)c(=O)n(C)c(=O)n3C)cc1	nan
	16025367	40911	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	570	7	1	7	5.4	COc1ccc(NC(=O)CSc2ncc3c(n2)-c2cc(Cl)ccc2N(Cc2ccccc2F)S3(=O)=O)cc1	nan
	CHEMBL1488348	40911	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	570	7	1	7	5.4	COc1ccc(NC(=O)CSc2ncc3c(n2)-c2cc(Cl)ccc2N(Cc2ccccc2F)S3(=O)=O)cc1	nan
	4611609	40917	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	6	1	3	6.2	CCc1ccc(OCC(=O)Nc2ccc3c(c2)c2ccccc2n3CC)c(Br)c1	nan
	CHEMBL1488388	40917	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	6	1	3	6.2	CCc1ccc(OCC(=O)Nc2ccc3c(c2)c2ccccc2n3CC)c(Br)c1	nan
	1726407	40938	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	5	1	4	6.4	CCOc1cccc(C(=O)Nc2ccc3oc(-c4ccc(C(C)(C)C)cc4)nc3c2)c1	nan
	CHEMBL1488581	40938	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	5	1	4	6.4	CCOc1cccc(C(=O)Nc2ccc3oc(-c4ccc(C(C)(C)C)cc4)nc3c2)c1	nan
	16030737	40974	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	5	1	10	2.0	Cc1ccc(-c2nc(SCC(=O)Nc3cc(C)on3)c3c(=O)n(C)c(=O)n(C)c3n2)cc1	nan
	CHEMBL1488787	40974	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	5	1	10	2.0	Cc1ccc(-c2nc(SCC(=O)Nc3cc(C)on3)c3c(=O)n(C)c(=O)n(C)c3n2)cc1	nan
	824820	41023	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	326	2	1	5	3.1	Cc1ccc(-n2c(N)c(C#N)c(-c3ccccc3)c(C#N)c2=O)cc1	nan
	CHEMBL1489157	41023	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	326	2	1	5	3.1	Cc1ccc(-n2c(N)c(C#N)c(-c3ccccc3)c(C#N)c2=O)cc1	nan
	2036296	41064	14	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	4	0	6	4.0	CCCCn1c(-c2cccs2)nc2oc3ccccc3c(=O)c2c1=O	nan
	CHEMBL1489469	41064	14	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	4	0	6	4.0	CCCCn1c(-c2cccs2)nc2oc3ccccc3c(=O)c2c1=O	nan
	3448820	41120	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	6	0	4	4.8	COc1cc2c(cc1OC)C(COc1ccc(F)cc1)N(C(=O)c1ccccc1F)CC2	nan
	CHEMBL1489934	41120	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	6	0	4	4.8	COc1cc2c(cc1OC)C(COc1ccc(F)cc1)N(C(=O)c1ccccc1F)CC2	nan
	655760	41195	14	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	3	1	4	3.0	Cc1ccc(C)c(NC(=O)Cn2nc(C)c3ccccc3c2=O)c1	nan
	CHEMBL1490512	41195	14	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	3	1	4	3.0	Cc1ccc(C)c(NC(=O)Cn2nc(C)c3ccccc3c2=O)c1	nan
	16007588	41227	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	515	7	1	5	4.1	CN(C1CCCCC1)S(=O)(=O)c1ccc2c(c1)c(=O)c(C(=O)NCCc1ccc(Cl)cc1)cn2C	nan
	CHEMBL1490705	41227	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	515	7	1	5	4.1	CN(C1CCCCC1)S(=O)(=O)c1ccc2c(c1)c(=O)c(C(=O)NCCc1ccc(Cl)cc1)cn2C	nan
	1483825	41234	14	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	336	2	0	4	4.3	FC(F)(F)c1cnc(-c2cnc(-c3cccnc3)nc2)c(Cl)c1	nan
	CHEMBL1490743	41234	14	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	336	2	0	4	4.3	FC(F)(F)c1cnc(-c2cnc(-c3cccnc3)nc2)c(Cl)c1	nan
	16194118	41260	6	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	5	1	8	2.0	CCOC(=O)c1ccc(NC(=S)N2CCN(c3ccc(N4CCOCC4)nn3)CC2)cc1	nan
	CHEMBL1490926	41260	6	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	5	1	8	2.0	CCOC(=O)c1ccc(NC(=S)N2CCN(c3ccc(N4CCOCC4)nn3)CC2)cc1	nan
	4578555	41281	17	None	-7	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	4	1	5	3.9	O=C(CSc1ncnc2c1oc1ccccc12)NC1CCCCC1	nan
	CHEMBL1491054	41281	17	None	-7	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	4	1	5	3.9	O=C(CSc1ncnc2c1oc1ccccc12)NC1CCCCC1	nan
	1147591	41342	18	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	4	1	6	3.0	COc1ccc(C(=O)Nc2nc3ccc(S(C)(=O)=O)cc3s2)cc1	nan
	CHEMBL1491533	41342	18	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	4	1	6	3.0	COc1ccc(C(=O)Nc2nc3ccc(S(C)(=O)=O)cc3s2)cc1	nan
	761949	41474	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	2	0	4	3.7	CC(=O)c1cnc2cc(-c3cccc(Br)c3)nn2c1C	nan
	CHEMBL1492474	41474	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	329	2	0	4	3.7	CC(=O)c1cnc2cc(-c3cccc(Br)c3)nn2c1C	nan
	16031672	41522	1	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	447	4	2	4	2.8	O=C(Nc1ccc(F)cc1F)C1CCN(S(=O)(=O)c2ccc3[nH]c(=O)ccc3c2)CC1	nan
	CHEMBL1492791	41522	1	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	447	4	2	4	2.8	O=C(Nc1ccc(F)cc1F)C1CCN(S(=O)(=O)c2ccc3[nH]c(=O)ccc3c2)CC1	nan
	3496289	41554	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	471	11	2	7	3.7	CCOc1cc2[nH]c(=S)n(Cc3ccc(C(=O)NCCCOC)cc3)c(=O)c2cc1OCC	nan
	CHEMBL1493174	41554	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	471	11	2	7	3.7	CCOc1cc2[nH]c(=S)n(Cc3ccc(C(=O)NCCCOC)cc3)c(=O)c2cc1OCC	nan
	16033055	41567	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	530	10	0	11	3.4	CCOc1ccc(C(=O)Cn2c(=O)n3nc(CCn4nc(C)cc4C)nc3c3cc(OC)c(OC)cc32)cc1	nan
	CHEMBL1493282	41567	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	530	10	0	11	3.4	CCOc1ccc(C(=O)Cn2c(=O)n3nc(CCn4nc(C)cc4C)nc3c3cc(OC)c(OC)cc32)cc1	nan
	6324582	41621	9	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	4	2	3	3.7	Cc1ccc2cc(CCNC(=O)CC(C)(C)C)c(O)nc2c1C	nan
	CHEMBL1493825	41621	9	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	4	2	3	3.7	Cc1ccc2cc(CCNC(=O)CC(C)(C)C)c(O)nc2c1C	nan
	2337492	41691	20	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	423	5	1	5	5.2	CCOC(=O)c1c(C)oc2c1cc(NS(=O)(=O)c1ccc(C)cc1)c1ccccc12	nan
	CHEMBL1494522	41691	20	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	423	5	1	5	5.2	CCOC(=O)c1c(C)oc2c1cc(NS(=O)(=O)c1ccc(C)cc1)c1ccccc12	nan
	16030367	41759	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	8	1	5	5.5	CCc1ccccc1NC(=O)CSc1nc2ccccc2nc1Cc1cccc(OC)c1	nan
	CHEMBL1495193	41759	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	8	1	5	5.5	CCc1ccccc1NC(=O)CSc1nc2ccccc2nc1Cc1cccc(OC)c1	nan
	659270	41765	14	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	6	1	8	2.7	CCOC(=O)CSc1nc(N)c(C#N)c(-c2ccc(OC)cc2)c1C#N	nan
	CHEMBL1495223	41765	14	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	6	1	8	2.7	CCOC(=O)CSc1nc(N)c(C#N)c(-c2ccc(OC)cc2)c1C#N	nan
	1473491	41766	14	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	4	0	4	4.3	O=C1c2ccccc2C(=O)N1CCc1csc(-c2cccc(Cl)c2)n1	nan
	CHEMBL1495238	41766	14	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	4	0	4	4.3	O=C1c2ccccc2C(=O)N1CCc1csc(-c2cccc(Cl)c2)n1	nan
	803577	41789	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	304	3	1	6	2.6	CC(=O)c1sc(NC(=O)c2ccc3c(c2)OCO3)nc1C	nan
	CHEMBL1495561	41789	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	304	3	1	6	2.6	CC(=O)c1sc(NC(=O)c2ccc3c(c2)OCO3)nc1C	nan
	16015766	41796	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	4	2	2	4.9	CC(C)CC(=O)Nc1ccc(Cl)c(-c2nc3ccccc3[nH]2)c1	nan
	CHEMBL1495596	41796	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	4	2	2	4.9	CC(C)CC(=O)Nc1ccc(Cl)c(-c2nc3ccccc3[nH]2)c1	nan
	1394903	41806	6	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	519	6	0	5	4.9	O=S(=O)([N-]c1nc2ccccc2nc1-[n+]1ccn(Cc2ccccc2)c1)c1ccc(Br)cc1	nan
	CHEMBL1495702	41806	6	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	519	6	0	5	4.9	O=S(=O)([N-]c1nc2ccccc2nc1-[n+]1ccn(Cc2ccccc2)c1)c1ccc(Br)cc1	nan
	9550975	41889	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	5	1	6	4.1	COc1ccccc1CNC(=O)c1nn(-c2ccc(C)cc2)c(=O)c2c1c1ccccc1n2C	nan
	CHEMBL1496499	41889	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	5	1	6	4.1	COc1ccccc1CNC(=O)c1nn(-c2ccc(C)cc2)c(=O)c2c1c1ccccc1n2C	nan
	7190533	41926	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	4	0	6	3.8	Cc1ccccc1CSc1ccc2nnc(-c3ccccn3)n2n1	nan
	CHEMBL1496795	41926	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	4	0	6	3.8	Cc1ccccc1CSc1ccc2nnc(-c3ccccn3)n2n1	nan
	22548523	41939	1	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	4	1	4	2.8	CN(Cc1ccccc1)S(=O)(=O)c1ccc2nc(O)ccc2c1	nan
	CHEMBL1496881	41939	1	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	4	1	4	2.8	CN(Cc1ccccc1)S(=O)(=O)c1ccc2nc(O)ccc2c1	nan
	16030464	41954	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	6	2	4	5.1	COc1ccccc1C(=O)Nc1ccccc1SCc1cc(=O)c2ccccc2[nH]1	nan
	CHEMBL1497018	41954	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	6	2	4	5.1	COc1ccccc1C(=O)Nc1ccccc1SCc1cc(=O)c2ccccc2[nH]1	nan
	3282397	41984	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	5	1	5	3.8	CCOc1ccc(-n2nc(C(=O)NC3CCCCC3)c3ccccc3c2=O)cc1	nan
	CHEMBL1497244	41984	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	391	5	1	5	3.8	CCOc1ccc(-n2nc(C(=O)NC3CCCCC3)c3ccccc3c2=O)cc1	nan
	2190255	41990	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	4	3	6	-0.1	CCN1C(=O)/C(=C/Nc2ccc(S(N)(=O)=O)cc2)C(=O)NC1=S	nan
	CHEMBL1497307	41990	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	4	3	6	-0.1	CCN1C(=O)/C(=C/Nc2ccc(S(N)(=O)=O)cc2)C(=O)NC1=S	nan
	860457	42061	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	4	0	6	2.6	CSc1nnc(-c2ccc(S(=O)(=O)N3CCCCC3)cc2)o1	nan
	CHEMBL1497958	42061	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	4	0	6	2.6	CSc1nnc(-c2ccc(S(=O)(=O)N3CCCCC3)cc2)o1	nan
	2815318	42140	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	317	3	0	7	2.2	CCOC(=O)Cn1cnc2c(sc3nc(C)cc(C)c32)c1=O	nan
	CHEMBL1498797	42140	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	317	3	0	7	2.2	CCOC(=O)Cn1cnc2c(sc3nc(C)cc(C)c32)c1=O	nan
	2126242	42144	7	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	373	5	1	5	4.3	COc1ccc2c(C)cc(SCC(=O)Nc3cccnc3Cl)nc2c1	nan
	CHEMBL1498813	42144	7	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	373	5	1	5	4.3	COc1ccc2c(C)cc(SCC(=O)Nc3cccnc3Cl)nc2c1	nan
	1105537	42233	10	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	8	1	6	3.2	CCOC(=O)/C(C#N)=C/c1ccc(OCC(=O)Nc2ccccc2)c(OC)c1	nan
	CHEMBL1499500	42233	10	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	8	1	6	3.2	CCOC(=O)/C(C#N)=C/c1ccc(OCC(=O)Nc2ccccc2)c(OC)c1	nan
	649649	42246	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	4	1	6	2.0	Cc1ccnc(N2CCC(C(=O)NCc3ccc4c(c3)OCO4)CC2)n1	nan
	CHEMBL1499616	42246	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	4	1	6	2.0	Cc1ccnc(N2CCC(C(=O)NCc3ccc4c(c3)OCO4)CC2)n1	nan
	866361	42247	20	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	2	1	5	2.8	O=c1c2ccccc2[nH]c(=S)n1Cc1ccc2c(c1)OCO2	nan
	CHEMBL1499629	42247	20	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	2	1	5	2.8	O=c1c2ccccc2[nH]c(=S)n1Cc1ccc2c(c1)OCO2	nan
	2764824	42273	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	3	2	2	2.8	CNC(=O)c1cc(C(=O)c2ccc(C(F)(F)F)cc2F)c[nH]1	nan
	CHEMBL1499851	42273	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	3	2	2	2.8	CNC(=O)c1cc(C(=O)c2ccc(C(F)(F)F)cc2F)c[nH]1	nan
	852955	42308	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	332	3	1	4	5.0	Cc1sc2nc(Cc3ccccc3)nc(O)c2c1-c1ccccc1	nan
	CHEMBL1500159	42308	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	332	3	1	4	5.0	Cc1sc2nc(Cc3ccccc3)nc(O)c2c1-c1ccccc1	nan
	135415434	42464	7	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	5	1	7	2.3	Cc1ccc(S(=O)(=O)N2CCN(C(=O)CSc3nc(O)c4ccccc4n3)CC2)cc1	nan
	CHEMBL1501602	42464	7	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	5	1	7	2.3	Cc1ccc(S(=O)(=O)N2CCN(C(=O)CSc3nc(O)c4ccccc4n3)CC2)cc1	nan
	54676936	42485	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	2	2	4	3.0	O=C(Nc1cccc(F)c1)c1c(O)c2cccc3c2n(c1=O)CCC3	nan
	CHEMBL1501763	42485	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	2	2	4	3.0	O=C(Nc1cccc(F)c1)c1c(O)c2cccc3c2n(c1=O)CCC3	nan
	1176241	42541	5	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	485	8	1	6	4.5	CCOc1ccc2nc(SCC(=O)Nc3ccc(S(=O)(=O)N4CCCC4)cc3)c(C)cc2c1	nan
	CHEMBL1502202	42541	5	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	485	8	1	6	4.5	CCOc1ccc2nc(SCC(=O)Nc3ccc(S(=O)(=O)N4CCCC4)cc3)c(C)cc2c1	nan
	734457	42640	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	257	3	1	5	2.6	COC(=O)c1ccc(Nc2nc(C)cc(C)n2)cc1	nan
	CHEMBL1503104	42640	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	257	3	1	5	2.6	COC(=O)c1ccc(Nc2nc(C)cc(C)n2)cc1	nan
	2515869	42664	1	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	6	1	5	2.9	CCC(=O)c1ccc(OCC(=O)c2ccc3c(c2)NC(=O)CO3)cc1	nan
	CHEMBL1503299	42664	1	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	6	1	5	2.9	CCC(=O)c1ccc(OCC(=O)c2ccc3c(c2)NC(=O)CO3)cc1	nan
	5310469	42694	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	6	0	8	3.3	COc1ccc(-c2nnc3ccc(SCC(=O)N4CCCCCC4)nn23)cc1OC	nan
	CHEMBL1503498	42694	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	6	0	8	3.3	COc1ccc(-c2nnc3ccc(SCC(=O)N4CCCCCC4)nn23)cc1OC	nan
	3574258	42702	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	5	2	6	3.1	O=C(CCn1c(=S)[nH]c2cc3c(cc2c1=O)OCO3)NCc1ccc(Cl)cc1	nan
	CHEMBL1503560	42702	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	5	2	6	3.1	O=C(CCn1c(=S)[nH]c2cc3c(cc2c1=O)OCO3)NCc1ccc(Cl)cc1	nan
	1859366	42707	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	5	1	4	5.0	Cc1ccc(S(=O)(=O)N(Cc2cc3ccc(C)cc3nc2O)c2ccccc2)cc1	nan
	CHEMBL1503583	42707	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	5	1	4	5.0	Cc1ccc(S(=O)(=O)N(Cc2cc3ccc(C)cc3nc2O)c2ccccc2)cc1	nan
	664334	42812	14	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	2	0	4	4.2	O=C1CC(c2ccc(F)cc2)Cc2nc(N3CCc4ccccc43)ncc21	nan
	CHEMBL1504653	42812	14	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	2	0	4	4.2	O=C1CC(c2ccc(F)cc2)Cc2nc(N3CCc4ccccc43)ncc21	nan
	2980439	42871	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	7	2	4	3.2	CCc1ccc(N2CCN(CCNC(=O)Nc3ccc(OC)cc3)CC2)cc1	nan
	CHEMBL1505203	42871	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	7	2	4	3.2	CCc1ccc(N2CCN(CCNC(=O)Nc3ccc(OC)cc3)CC2)cc1	nan
	661657	42881	18	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	3	0	7	3.3	O=C1c2ccccc2C(=O)N1Cc1nn2c(-c3ccc(Cl)cc3)nnc2s1	nan
	CHEMBL1505268	42881	18	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	3	0	7	3.3	O=C1c2ccccc2C(=O)N1Cc1nn2c(-c3ccc(Cl)cc3)nnc2s1	nan
	12006071	42899	9	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	4	0	6	4.5	O=C(CSc1ccc2nnc(-c3ccc(Cl)cc3)n2n1)N1CCCc2ccccc21	nan
	CHEMBL1505466	42899	9	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	4	0	6	4.5	O=C(CSc1ccc2nnc(-c3ccc(Cl)cc3)n2n1)N1CCCc2ccccc21	nan
	834457	42963	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	4	2	3	2.7	NS(=O)(=O)c1ccc(NCc2c(F)cccc2Cl)cc1	nan
	CHEMBL1505860	42963	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	4	2	3	2.7	NS(=O)(=O)c1ccc(NCc2c(F)cccc2Cl)cc1	nan
	1804684	42969	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	6	1	5	3.8	COCc1cc(C)nc(SCC(=O)Nc2cccc(C)c2C)c1C#N	nan
	CHEMBL1505914	42969	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	6	1	5	3.8	COCc1cc(C)nc(SCC(=O)Nc2cccc(C)c2C)c1C#N	nan
	3882765	42998	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	268	2	2	1	3.9	Cc1ccc2[nH]c(C(=O)Nc3ccc(F)cc3)cc2c1	nan
	CHEMBL1506222	42998	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	268	2	2	1	3.9	Cc1ccc2[nH]c(C(=O)Nc3ccc(F)cc3)cc2c1	nan
	3795359	43037	16	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	3	1	6	3.8	CCC(C)c1ccc(-n2c(=O)c3ccccc3n3c(S)nnc23)cc1	nan
	CHEMBL1506487	43037	16	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	3	1	6	3.8	CCC(C)c1ccc(-n2c(=O)c3ccccc3n3c(S)nnc23)cc1	nan
	4118928	43042	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	363	7	2	5	2.1	CCCCOCCCN1C(C)=CC(=C2C(=O)NC(=S)NC2=O)C=C1C	nan
	CHEMBL1506535	43042	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	363	7	2	5	2.1	CCCCOCCCN1C(C)=CC(=C2C(=O)NC(=S)NC2=O)C=C1C	nan
	1078308	43098	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	5	1	6	4.4	COc1ccccc1NC(=O)c1sc2ncn(Cc3ccccc3C)c(=O)c2c1C	nan
	CHEMBL1507058	43098	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	5	1	6	4.4	COc1ccccc1NC(=O)c1sc2ncn(Cc3ccccc3C)c(=O)c2c1C	nan
	1390207	43106	6	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	475	6	0	5	4.8	O=S(=O)([N-]c1nc2ccccc2nc1-[n+]1ccn(Cc2ccccc2)c1)c1ccc(Cl)cc1	nan
	CHEMBL1507117	43106	6	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	475	6	0	5	4.8	O=S(=O)([N-]c1nc2ccccc2nc1-[n+]1ccn(Cc2ccccc2)c1)c1ccc(Cl)cc1	nan
	9550860	43124	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	292	3	2	3	2.0	Cc1ccc(OC(=O)c2ccccc2P(=O)(O)O)cc1	nan
	CHEMBL1507343	43124	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	292	3	2	3	2.0	Cc1ccc(OC(=O)c2ccccc2P(=O)(O)O)cc1	nan
	2810073	43136	6	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	308	2	1	6	3.3	Cc1csc2c(=O)sc(NC(=O)c3cccs3)nc12	nan
	CHEMBL1507430	43136	6	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	308	2	1	6	3.3	Cc1csc2c(=O)sc(NC(=O)c3cccs3)nc12	nan
	20874463	43201	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	317	3	1	5	4.1	Cc1ccc(-c2nnn3c2nc(NC(C)C)c2ccccc23)cc1	nan
	CHEMBL1507945	43201	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	317	3	1	5	4.1	Cc1ccc(-c2nnn3c2nc(NC(C)C)c2ccccc23)cc1	nan
	5875901	43220	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	4	0	4	3.8	CCOC(=O)CN1C(=O)/C(=C/c2cccc(Br)c2)Oc2ccccc21	nan
	CHEMBL1508095	43220	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	4	0	4	3.8	CCOC(=O)CN1C(=O)/C(=C/c2cccc(Br)c2)Oc2ccccc21	nan
	649082	43251	2	None	-1	3	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	6	2	7	2.6	O=C(Cn1nnc(-c2ccccc2NC(=O)c2ccco2)n1)NC1CCCCC1	nan
	CHEMBL1508376	43251	2	None	-1	3	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	6	2	7	2.6	O=C(Cn1nnc(-c2ccccc2NC(=O)c2ccco2)n1)NC1CCCCC1	nan
	1735895	43552	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	7	2	7	3.2	CCc1ccc(OCC(=O)NNC(=O)CSc2ncnc3sc(C)c(C)c23)cc1	nan
	CHEMBL1511120	43552	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	7	2	7	3.2	CCc1ccc(OCC(=O)NNC(=O)CSc2ncnc3sc(C)c(C)c23)cc1	nan
	1186303	43577	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	6	2	6	3.3	CN(C)c1ccc(C(=O)Nc2ccc(S(=O)(=O)Nc3nccs3)cc2)cc1	nan
	CHEMBL1511271	43577	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	6	2	6	3.3	CN(C)c1ccc(C(=O)Nc2ccc(S(=O)(=O)Nc3nccs3)cc2)cc1	nan
	2815635	43613	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	351	3	2	4	5.7	O=C(Nc1ccccc1)Nc1sccc1-c1nc2ccccc2s1	nan
	CHEMBL1511507	43613	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	351	3	2	4	5.7	O=C(Nc1ccccc1)Nc1sccc1-c1nc2ccccc2s1	nan
	661880	43615	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	269	1	0	6	2.3	N#CCc1nc2c3c4c(sc3ncn2n1)CCCC4	nan
	CHEMBL1511519	43615	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	269	1	0	6	2.3	N#CCc1nc2c3c4c(sc3ncn2n1)CCCC4	nan
	4604131	43656	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	7	1	7	3.9	COc1ccc(-n2c(SCC(=O)NCc3ccccc3)nc3ccsc3c2=O)cc1	nan
	CHEMBL1512120	43656	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	7	1	7	3.9	COc1ccc(-n2c(SCC(=O)NCc3ccccc3)nc3ccsc3c2=O)cc1	nan
	16027453	43688	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	6	1	8	3.7	COc1ccccc1C(=O)Nc1ccccc1C(=O)OCc1cc(=O)n2c(C)csc2n1	nan
	CHEMBL1512551	43688	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	6	1	8	3.7	COc1ccccc1C(=O)Nc1ccccc1C(=O)OCc1cc(=O)n2c(C)csc2n1	nan
	16018474	43690	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	4	1	4	5.8	CCc1ccc(-c2cn3c(n2)sc2cc(C(=O)NC4CCCCC4)ccc23)cc1	nan
	CHEMBL1512597	43690	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	4	1	4	5.8	CCc1ccc(-c2cn3c(n2)sc2cc(C(=O)NC4CCCCC4)ccc23)cc1	nan
	16030606	43692	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	5	1	5	4.1	Cc1cccc(C(=O)Nc2cccc(OCc3cc(=O)n4cccc(C)c4n3)c2)c1	nan
	CHEMBL1512611	43692	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	5	1	5	4.1	Cc1cccc(C(=O)Nc2cccc(OCc3cc(=O)n4cccc(C)c4n3)c2)c1	nan
	16030447	43693	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	5	1	5	4.5	Cc1ccc2nc(COc3cccc(NC(=O)c4ccccc4Cl)c3)cc(=O)n2c1	nan
	CHEMBL1512613	43693	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	5	1	5	4.5	Cc1ccc2nc(COc3cccc(NC(=O)c4ccccc4Cl)c3)cc(=O)n2c1	nan
	7245878	43700	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	346	4	0	6	2.6	COc1ccc(S(=O)(=O)c2cc3cc(OC)ccc3oc2=O)cc1	nan
	CHEMBL1512705	43700	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	346	4	0	6	2.6	COc1ccc(S(=O)(=O)c2cc3cc(OC)ccc3oc2=O)cc1	nan
	16020157	43720	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	7	0	9	3.6	CCOC(=O)CSc1nc2cc(OC)c(OC)cc2c2nc(-c3ccccc3)nn12	nan
	CHEMBL1512982	43720	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	7	0	9	3.6	CCOC(=O)CSc1nc2cc(OC)c(OC)cc2c2nc(-c3ccccc3)nn12	nan
	16023839	43721	0	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	487	3	0	6	4.0	CN1CCN(C(=O)c2cnn(-c3cccc(Cl)c3)c2C2CCN(C(=O)OC(C)(C)C)CC2)CC1	nan
	CHEMBL1513006	43721	0	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	487	3	0	6	4.0	CN1CCN(C(=O)c2cnn(-c3cccc(Cl)c3)c2C2CCN(C(=O)OC(C)(C)C)CC2)CC1	nan
	3402023	43723	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	8	2	5	5.4	COc1ccc(CNC(=O)c2ccc(Sc3ccc(Cl)cc3)c(NC(C)=O)c2)c(OC)c1	nan
	CHEMBL1513023	43723	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	8	2	5	5.4	COc1ccc(CNC(=O)c2ccc(Sc3ccc(Cl)cc3)c(NC(C)=O)c2)c(OC)c1	nan
	16014785	43724	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	7	2	6	4.5	COC(=O)c1ccc(NC(=O)CSc2nc(C)cc(C)c2C(=O)Nc2ccccc2)cc1	nan
	CHEMBL1513057	43724	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	7	2	6	4.5	COC(=O)c1ccc(NC(=O)CSc2nc(C)cc(C)c2C(=O)Nc2ccccc2)cc1	nan
	16021019	43726	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	7	1	5	6.0	O=C(NC1CCCCC1)c1ccc(CSc2nc3cccnc3n2Cc2ccc(F)cc2)cc1	nan
	CHEMBL1513070	43726	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	7	1	5	6.0	O=C(NC1CCCCC1)c1ccc(CSc2nc3cccnc3n2Cc2ccc(F)cc2)cc1	nan
	16008530	43732	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	486	8	1	5	6.0	CSc1ccc(CCNC(=O)CCc2c(C)nc3c(c(C)nn3-c3ccc(C)c(C)c3)c2C)cc1	nan
	CHEMBL1513168	43732	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	486	8	1	5	6.0	CSc1ccc(CCNC(=O)CCc2c(C)nc3c(c(C)nn3-c3ccc(C)c(C)c3)c2C)cc1	nan
	16018739	43743	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	5	1	5	3.0	O=C(CCn1c(=O)c2cccn2c2cccnc21)NCc1ccc(Cl)cc1	nan
	CHEMBL1513371	43743	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	5	1	5	3.0	O=C(CCn1c(=O)c2cccn2c2cccnc21)NCc1ccc(Cl)cc1	nan
	16030719	43746	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	6	1	9	2.0	Cc1cccc(-c2nc(SCC(=O)NCc3ccco3)c3c(=O)n(C)c(=O)n(C)c3n2)c1	nan
	CHEMBL1513435	43746	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	6	1	9	2.0	Cc1cccc(-c2nc(SCC(=O)NCc3ccco3)c3c(=O)n(C)c(=O)n(C)c3n2)c1	nan
	16025371	43748	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	568	6	1	6	6.0	Cc1ccc(C)c(NC(=O)CSc2ncc3c(n2)-c2cc(Cl)ccc2N(Cc2ccccc2F)S3(=O)=O)c1	nan
	CHEMBL1513466	43748	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	568	6	1	6	6.0	Cc1ccc(C)c(NC(=O)CSc2ncc3c(n2)-c2cc(Cl)ccc2N(Cc2ccccc2F)S3(=O)=O)c1	nan
	16026779	43752	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	6	1	8	2.8	O=C(CNC(=O)c1ccc(F)cc1)OCc1cc(=O)n2nc(C3CCCCC3)sc2n1	nan
	CHEMBL1513507	43752	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	444	6	1	8	2.8	O=C(CNC(=O)c1ccc(F)cc1)OCc1cc(=O)n2nc(C3CCCCC3)sc2n1	nan
	16024940	43754	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	5	1	4	4.9	O=C(NCCc1ccccc1Cl)C1CCN(c2nc3ccccc3nc2C(F)(F)F)CC1	nan
	CHEMBL1513535	43754	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	5	1	4	4.9	O=C(NCCc1ccccc1Cl)C1CCN(c2nc3ccccc3nc2C(F)(F)F)CC1	nan
	1316309	43766	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	4	1	3	5.6	Cc1ccc2oc(-c3ccc(Cl)c(NC(=O)Cc4ccccc4)c3)nc2c1	nan
	CHEMBL1513652	43766	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	4	1	3	5.6	Cc1ccc2oc(-c3ccc(Cl)c(NC(=O)Cc4ccccc4)c3)nc2c1	nan
	16025593	43781	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	3	0	8	3.9	Cc1c(-c2nc(-c3ccc4c(c3)OCO4)no2)nnn1-c1ccc(Br)cc1F	nan
	CHEMBL1514000	43781	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	3	0	8	3.9	Cc1c(-c2nc(-c3ccc4c(c3)OCO4)no2)nnn1-c1ccc(Br)cc1F	nan
	15989077	43796	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	547	10	1	8	4.8	Cc1cc(C)c(Cn2c(=O)n(CCCCCC(=O)NCc3ccc4c(c3)OCO4)c(=O)c3sccc32)c(C)c1	nan
	CHEMBL1514246	43796	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	547	10	1	8	4.8	Cc1cc(C)c(Cn2c(=O)n(CCCCCC(=O)NCc3ccc4c(c3)OCO4)c(=O)c3sccc32)c(C)c1	nan
	2689697	43801	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	6	1	5	3.2	COc1ccc(C(=O)OCC(=O)c2c[nH]c3ccccc23)cc1OC	nan
	CHEMBL1514340	43801	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	339	6	1	5	3.2	COc1ccc(C(=O)OCC(=O)c2c[nH]c3ccccc23)cc1OC	nan
	24982480	43814	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	8	0	5	2.3	CCN(Cc1ccccc1)C(=O)Cc1ccc(OC)c(S(=O)(=O)N2CCOCC2)c1	nan
	CHEMBL1514540	43814	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	8	0	5	2.3	CCN(Cc1ccccc1)C(=O)Cc1ccc(OC)c(S(=O)(=O)N2CCOCC2)c1	nan
	16015735	43839	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	3	3	9	2.5	COC(=O)c1c(C)sc(-c2c(-c3ccc4c(c3)OCCO4)[nH]c3c2c(=O)[nH]c(=O)n3C)c1O	nan
	CHEMBL1514818	43839	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	3	3	9	2.5	COC(=O)c1c(C)sc(-c2c(-c3ccc4c(c3)OCCO4)[nH]c3c2c(=O)[nH]c(=O)n3C)c1O	nan
	16022151	43843	1	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	2	0	6	2.5	COc1ccc2c(c1)c1c(c(=O)n(-c3ccccc3C)c(=O)n1C)n2C	nan
	CHEMBL1514879	43843	1	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	2	0	6	2.5	COc1ccc2c(c1)c1c(c(=O)n(-c3ccccc3C)c(=O)n1C)n2C	nan
	16009667	43851	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	398	4	0	5	4.5	O=c1c2sc3ccccc3c2n(Cc2ccccc2)c(=O)n1Cc1ccccc1	nan
	CHEMBL1515036	43851	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	398	4	0	5	4.5	O=c1c2sc3ccccc3c2n(Cc2ccccc2)c(=O)n1Cc1ccccc1	nan
	5167801	43854	1	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	345	4	2	3	5.0	O=C(NC1CCCCC1)c1cc(Nc2ccccc2)nc2ccccc12	nan
	CHEMBL1515050	43854	1	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	345	4	2	3	5.0	O=C(NC1CCCCC1)c1cc(Nc2ccccc2)nc2ccccc12	nan
	16030854	43856	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	5	2	4	5.0	CC(NC(=O)c1ccc(NC(=O)c2nsc3ccccc23)cc1)c1ccccc1	nan
	CHEMBL1515130	43856	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	5	2	4	5.0	CC(NC(=O)c1ccc(NC(=O)c2nsc3ccccc23)cc1)c1ccccc1	nan
	135416423	43877	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	4	2	4	4.7	CCc1ccc2oc(-c3cc(NC(=O)C(C)C)cc(C)c3O)nc2c1	nan
	CHEMBL1515394	43877	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	338	4	2	4	4.7	CCc1ccc2oc(-c3cc(NC(=O)C(C)C)cc(C)c3O)nc2c1	nan
	8057488	43898	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	4	0	4	5.4	Cc1cc2nc(-c3ccc(OCc4ccccc4F)cc3)cc(C(F)(F)F)n2n1	nan
	CHEMBL1515771	43898	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	4	0	4	5.4	Cc1cc2nc(-c3ccc(OCc4ccccc4F)cc3)cc(C(F)(F)F)n2n1	nan
	4154278	43900	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	4	1	5	5.2	Cc1ccc(NC(=O)CSc2ncnc3c2sc2ccccc23)cc1C	nan
	CHEMBL1515779	43900	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	4	1	5	5.2	Cc1ccc(NC(=O)CSc2ncnc3c2sc2ccccc23)cc1C	nan
	16017003	43926	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	6	1	4	4.5	CCOc1ccccc1NC(=O)C(=O)c1cc(C)n(-c2ccc(F)cc2)c1C	nan
	CHEMBL1516117	43926	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	380	6	1	4	4.5	CCOc1ccccc1NC(=O)C(=O)c1cc(C)n(-c2ccc(F)cc2)c1C	nan
	7343169	43937	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	4	0	5	4.9	CCOC(=O)c1cnc2cc(-c3ccc(Cl)cc3)nn2c1-c1ccccc1	nan
	CHEMBL1516275	43937	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	4	0	5	4.9	CCOC(=O)c1cnc2cc(-c3ccc(Cl)cc3)nn2c1-c1ccccc1	nan
	3586950	43945	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	485	6	1	6	4.6	O=C(CSc1nc2ccsc2c(=O)n1-c1ccc(Br)cc1)NCc1ccccc1	nan
	CHEMBL1516478	43945	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	485	6	1	6	4.6	O=C(CSc1nc2ccsc2c(=O)n1-c1ccc(Br)cc1)NCc1ccccc1	nan
	3206747	44086	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	344	4	1	5	3.5	COc1cccc(CC(=O)Nc2nc3c(s2)C(=O)CC(C)(C)C3)c1	nan
	CHEMBL1517888	44086	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	344	4	1	5	3.5	COc1cccc(CC(=O)Nc2nc3c(s2)C(=O)CC(C)(C)C3)c1	nan
	985821	44090	9	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	3	1	3	5.0	O=C(Nc1cc(F)cc(F)c1)c1sc(Cl)nc1-c1ccccc1	nan
	CHEMBL1517907	44090	9	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	3	1	3	5.0	O=C(Nc1cc(F)cc(F)c1)c1sc(Cl)nc1-c1ccccc1	nan
	1093907	44091	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	396	5	2	7	1.5	CNS(=O)(=O)c1ccc(NC(=O)c2nc3nc(C)cc(C(F)F)n3n2)cc1	nan
	CHEMBL1517917	44091	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	396	5	2	7	1.5	CNS(=O)(=O)c1ccc(NC(=O)c2nc3nc(C)cc(C(F)F)n3n2)cc1	nan
	15991337	44114	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	478	4	0	7	4.8	CCc1ccc(C2c3c(oc4ccc(F)cc4c3=O)C(=O)N2c2nc(C)c(C(=O)OC)s2)cc1	nan
	CHEMBL1518140	44114	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	478	4	0	7	4.8	CCc1ccc(C2c3c(oc4ccc(F)cc4c3=O)C(=O)N2c2nc(C)c(C(=O)OC)s2)cc1	nan
	16011836	44156	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	7	1	6	5.0	COc1ccc(CSc2nc3ccncc3n2CC(=O)Nc2cc(C)cc(C)c2)cc1	nan
	CHEMBL1518592	44156	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	7	1	6	5.0	COc1ccc(CSc2nc3ccncc3n2CC(=O)Nc2cc(C)cc(C)c2)cc1	nan
	1086869	44205	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	6	1	6	3.4	COc1ccc(C(=O)Nc2nnc(Cc3ccccc3)s2)c(OC)c1	nan
	CHEMBL1518977	44205	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	6	1	6	3.4	COc1ccc(C(=O)Nc2nnc(Cc3ccccc3)s2)c(OC)c1	nan
	730225	44218	10	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	274	3	2	6	2.2	N#CCc1c(C#N)c(N)nc(Nc2ccccc2)c1C#N	nan
	CHEMBL1519080	44218	10	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	274	3	2	6	2.2	N#CCc1c(C#N)c(N)nc(Nc2ccccc2)c1C#N	nan
	1008965	44230	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	4	1	4	6.1	CC(=O)c1cccc(NC(=O)c2cc(-c3ccc(Cl)s3)nc3ccccc23)c1	nan
	CHEMBL1519196	44230	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	4	1	4	6.1	CC(=O)c1cccc(NC(=O)c2cc(-c3ccc(Cl)s3)nc3ccccc23)c1	nan
	16025959	44313	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	5	1	8	1.6	O=C(NCCc1ccc(Cl)cc1)c1cnc2sc(N3CCOCC3)nn2c1=O	nan
	CHEMBL1519916	44313	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	5	1	8	1.6	O=C(NCCc1ccc(Cl)cc1)c1cnc2sc(N3CCOCC3)nn2c1=O	nan
	2740242	44320	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	2	2	4	3.1	Cc1noc(C(F)(F)F)c1C(=O)NNC(=O)c1cccc(C(F)(F)F)c1	nan
	CHEMBL1519973	44320	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	2	2	4	3.1	Cc1noc(C(F)(F)F)c1C(=O)NNC(=O)c1cccc(C(F)(F)F)c1	nan
	16020184	44412	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	508	8	0	9	5.3	COc1cc2nc(SCc3cccc(Cl)c3)n3nc(CCn4nc(C)cc4C)nc3c2cc1OC	nan
	CHEMBL1520786	44412	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	508	8	0	9	5.3	COc1cc2nc(SCc3cccc(Cl)c3)n3nc(CCn4nc(C)cc4C)nc3c2cc1OC	nan
	15989989	44415	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	8	2	9	3.4	COc1ccc(CCNC(=O)c2ccc(Nc3nc4ccccc4n4nnnc34)cc2)cc1OC	nan
	CHEMBL1520796	44415	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	8	2	9	3.4	COc1ccc(CCNC(=O)c2ccc(Nc3nc4ccccc4n4nnnc34)cc2)cc1OC	nan
	742057	44456	14	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	289	3	1	6	3.1	O=C(Nc1nc2ccc([N+](=O)[O-])cc2s1)c1ccco1	nan
	CHEMBL1521136	44456	14	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	289	3	1	6	3.1	O=C(Nc1nc2ccc([N+](=O)[O-])cc2s1)c1ccco1	nan
	16026879	44484	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	7	1	6	4.4	COc1ccc(Cn2ccc3nc(C)c(C(=O)NCc4ccc(SC)cc4)cc3c2=O)cc1	nan
	CHEMBL1521365	44484	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	7	1	6	4.4	COc1ccc(Cn2ccc3nc(C)c(C(=O)NCc4ccc(SC)cc4)cc3c2=O)cc1	nan
	1164118	44497	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	6	0	7	3.4	COc1ccc(-c2nnc(SCC(=O)N3CCc4ccccc43)o2)cc1OC	nan
	CHEMBL1521488	44497	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	6	0	7	3.4	COc1ccc(-c2nnc(SCC(=O)N3CCc4ccccc43)o2)cc1OC	nan
	3146504	44551	16	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	320	5	1	6	2.9	CCOC(=O)c1sc(NC(=O)c2ccc(OC)cc2)nc1C	nan
	CHEMBL1521972	44551	16	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	320	5	1	6	2.9	CCOC(=O)c1sc(NC(=O)c2ccc(OC)cc2)nc1C	nan
	16021952	44583	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	496	7	1	7	3.9	CCc1cccc(NC(=O)Cn2c(=O)n(Cc3ccccc3)c(=O)c3c2c2cc(OC)ccc2n3C)c1	nan
	CHEMBL1522220	44583	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	496	7	1	7	3.9	CCc1cccc(NC(=O)Cn2c(=O)n(Cc3ccccc3)c(=O)c3c2c2cc(OC)ccc2n3C)c1	nan
	4090626	44634	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	7	2	4	5.8	CCOc1ccc(NC(=O)c2c(NC(=O)Cc3ccccc3)sc3c2CCCCC3)cc1	nan
	CHEMBL1522769	44634	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	7	2	4	5.8	CCOc1ccc(NC(=O)c2c(NC(=O)Cc3ccccc3)sc3c2CCCCC3)cc1	nan
	3148294	44640	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	7	1	6	4.1	CC(C)CNC(=O)CCSc1nc(-c2ccc3c(c2)OCO3)cc(C(F)(F)F)n1	nan
	CHEMBL1522819	44640	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	7	1	6	4.1	CC(C)CNC(=O)CCSc1nc(-c2ccc3c(c2)OCO3)cc(C(F)(F)F)n1	nan
	16030650	44664	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	501	5	0	8	3.0	O=c1cc(CN2CCN(S(=O)(=O)c3ccccc3)CC2)nc2sc(-c3ccccc3Cl)nn12	nan
	CHEMBL1522977	44664	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	501	5	0	8	3.0	O=c1cc(CN2CCN(S(=O)(=O)c3ccccc3)CC2)nc2sc(-c3ccccc3Cl)nn12	nan
	16026964	44706	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	6	0	9	3.1	O=C(COc1ccccc1F)OCc1cc(=O)n2nc(-c3cccs3)sc2n1	nan
	CHEMBL1523393	44706	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	6	0	9	3.1	O=C(COc1ccccc1F)OCc1cc(=O)n2nc(-c3cccs3)sc2n1	nan
	16027395	44730	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	9	1	10	3.4	CCOCCc1nn2c(=O)cc(COC(=O)c3ccccc3NC(=O)c3cccs3)nc2s1	nan
	CHEMBL1523585	44730	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	9	1	10	3.4	CCOCCc1nn2c(=O)cc(COC(=O)c3ccccc3NC(=O)c3cccs3)nc2s1	nan
	2465708	44739	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	518	6	1	9	4.8	COc1ccccc1-n1c(=O)c(C#N)c(-c2ccc([N+](=O)[O-])cc2)c2cc(C(=O)c3ccccc3O)cnc21	nan
	CHEMBL1523696	44739	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	518	6	1	9	4.8	COc1ccccc1-n1c(=O)c(C#N)c(-c2ccc([N+](=O)[O-])cc2)c2cc(C(=O)c3ccccc3O)cnc21	nan
	1465904	44756	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	6	1	7	4.8	CCc1nnc(NC(=O)CSc2nc(C3CCCCC3)nc3ccccc23)s1	nan
	CHEMBL1523892	44756	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	6	1	7	4.8	CCc1nnc(NC(=O)CSc2nc(C3CCCCC3)nc3ccccc23)s1	nan
	7422674	44757	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	4	1	3	4.2	O=C(Nc1ccccc1C(F)(F)F)c1cccn(Cc2ccccc2)c1=O	nan
	CHEMBL1523907	44757	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	4	1	3	4.2	O=C(Nc1ccccc1C(F)(F)F)c1cccn(Cc2ccccc2)c1=O	nan
	15989150	44801	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	471	9	1	6	3.6	COc1ccccc1CNC(=O)CCCn1c(=O)c2ccccc2n(Cc2ccc(C)cc2)c1=O	nan
	CHEMBL1524350	44801	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	471	9	1	6	3.6	COc1ccccc1CNC(=O)CCCn1c(=O)c2ccccc2n(Cc2ccc(C)cc2)c1=O	nan
	2548636	44884	6	None	-2	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	6	3	7	2.5	Cc1nc(SCC(=O)Nc2cc(C(N)=O)cc(C(N)=O)c2)c2c(C)c(C)sc2n1	nan
	CHEMBL1525189	44884	6	None	-2	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	6	3	7	2.5	Cc1nc(SCC(=O)Nc2cc(C(N)=O)cc(C(N)=O)c2)c2c(C)c(C)sc2n1	nan
	15989883	44888	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	3	1	3	5.4	Cc1c(C(=O)OC2CCCCC2)[nH]c2c1C(=O)CC(c1ccccc1Cl)C2	nan
	CHEMBL1525262	44888	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	3	1	3	5.4	Cc1c(C(=O)OC2CCCCC2)[nH]c2c1C(=O)CC(c1ccccc1Cl)C2	nan
	1186420	44931	10	None	-31	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	4	1	7	3.8	Clc1ccc(-n2ncc3c(NCc4ccc5c(c4)OCO5)ncnc32)cc1	nan
	CHEMBL1525610	44931	10	None	-31	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	4	1	7	3.8	Clc1ccc(-n2ncc3c(NCc4ccc5c(c4)OCO5)ncnc32)cc1	nan
	4154665	44935	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	457	10	2	7	3.3	CCOc1cc2[nH]c(=S)n(Cc3ccc(C(=O)NCCOC)cc3)c(=O)c2cc1OCC	nan
	CHEMBL1525634	44935	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	457	10	2	7	3.3	CCOc1cc2[nH]c(=S)n(Cc3ccc(C(=O)NCCOC)cc3)c(=O)c2cc1OCC	nan
	135460528	44990	8	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	478	3	2	5	3.5	Cc1ccc(N2C(=O)NC(=O)/C(=C/Nc3ncc(Br)cc3Br)C2=O)cc1	nan
	CHEMBL1526117	44990	8	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	478	3	2	5	3.5	Cc1ccc(N2C(=O)NC(=O)/C(=C/Nc3ncc(Br)cc3Br)C2=O)cc1	nan
	579848	45048	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	336	4	1	3	4.7	O=C(Nc1ccc(-c2ccc([N+](=O)[O-])cc2)cc1)c1ccccc1F	nan
	CHEMBL1526496	45048	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	336	4	1	3	4.7	O=C(Nc1ccc(-c2ccc([N+](=O)[O-])cc2)cc1)c1ccccc1F	nan
	16018883	45108	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	6	1	4	4.6	Cc1ccc(C)c(NC(=O)CCCN2C(=O)C(c3ccccc3)Oc3cccnc32)c1	nan
	CHEMBL1527105	45108	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	6	1	4	4.6	Cc1ccc(C)c(NC(=O)CCCN2C(=O)C(c3ccccc3)Oc3cccnc32)c1	nan
	2765322	45154	22	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	305	2	1	7	1.1	N#Cc1cc(C#N)c(N2CCN(c3ccccn3)CC2)nc1N	nan
	CHEMBL1527484	45154	22	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	305	2	1	7	1.1	N#Cc1cc(C#N)c(N2CCN(c3ccccn3)CC2)nc1N	nan
	16009430	45187	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	7	1	6	3.7	CCC(CC)C(=O)Nc1ccc(OCc2cc(=O)n3ccsc3n2)cc1	nan
	CHEMBL1527797	45187	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	7	1	6	3.7	CCC(CC)C(=O)Nc1ccc(OCc2cc(=O)n3ccsc3n2)cc1	nan
	16015678	45188	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	7	1	5	5.1	CCC(=O)Nc1ccc2nc(SCCOc3ccc(C)cc3)sc2c1	nan
	CHEMBL1527810	45188	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	7	1	5	5.1	CCC(=O)Nc1ccc2nc(SCCOc3ccc(C)cc3)sc2c1	nan
	16009490	45236	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	5	1	6	4.2	Cc1cccc(C(=O)Nc2cccc(OCc3cc(=O)n4c(C)csc4n3)c2)c1	nan
	CHEMBL1528261	45236	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	5	1	6	4.2	Cc1cccc(C(=O)Nc2cccc(OCc3cc(=O)n4c(C)csc4n3)c2)c1	nan
	16016701	45239	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	5	1	5	2.6	COC(=O)c1ccccc1NC(=O)CCC(=O)N1CCOc2ccccc21	nan
	CHEMBL1528274	45239	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	5	1	5	2.6	COC(=O)c1ccccc1NC(=O)CCC(=O)N1CCOc2ccccc21	nan
	16391033	45255	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	292	3	1	3	3.8	COc1cc2ccccc2cc1C(=O)Nc1ccc(C)cn1	nan
	CHEMBL1528436	45255	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	292	3	1	3	3.8	COc1cc2ccccc2cc1C(=O)Nc1ccc(C)cn1	nan
	7185472	45277	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	6	2	6	2.6	CCOC(=O)c1ccccc1NC(=O)CSc1nc(=O)[nH]c2c1CCCC2	nan
	CHEMBL1528587	45277	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	6	2	6	2.6	CCOC(=O)c1ccccc1NC(=O)CSc1nc(=O)[nH]c2c1CCCC2	nan
	5310045	45331	9	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	3	1	5	4.2	Cc1c(C(=O)Nc2ccncc2)sc2nc(-c3ccc(F)cc3)cn12	nan
	CHEMBL1529086	45331	9	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	3	1	5	4.2	Cc1c(C(=O)Nc2ccncc2)sc2nc(-c3ccc(F)cc3)cn12	nan
	5146627	45369	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	9	0	6	5.1	COCCN(CCOC)c1ncnc2c1c(-c1ccccc1)cn2-c1ccc(C)c(Cl)c1	nan
	CHEMBL1529403	45369	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	9	0	6	5.1	COCCN(CCOC)c1ncnc2c1c(-c1ccccc1)cn2-c1ccc(C)c(Cl)c1	nan
	5181996	45383	18	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	271	4	0	6	1.0	CCOC(=O)Cc1nc2ccccc2n(CC#N)c1=O	nan
	CHEMBL1529516	45383	18	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	271	4	0	6	1.0	CCOC(=O)Cc1nc2ccccc2n(CC#N)c1=O	nan
	2099952	45410	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	3	1	4	4.9	Oc1nc(Cc2ccc(F)cc2)nc2scc(-c3ccc(F)cc3)c12	nan
	CHEMBL1529751	45410	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	3	1	4	4.9	Oc1nc(Cc2ccc(F)cc2)nc2scc(-c3ccc(F)cc3)c12	nan
	4373285	45438	1	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	472	4	1	4	6.7	COc1ccc(C(=O)Nc2ccc3oc(-c4ccc5ccccc5c4)nc3c2)cc1Br	nan
	CHEMBL1529998	45438	1	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	472	4	1	4	6.7	COc1ccc(C(=O)Nc2ccc3oc(-c4ccc5ccccc5c4)nc3c2)cc1Br	nan
	16024591	45482	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	7	1	5	3.4	Cc1ccc2c(=O)c(C(=O)c3ccc(F)cc3)cn(CC(=O)NCCc3ccccc3)c2n1	nan
	CHEMBL1530480	45482	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	7	1	5	3.4	Cc1ccc2c(=O)c(C(=O)c3ccc(F)cc3)cn(CC(=O)NCCc3ccccc3)c2n1	nan
	4994836	45631	1	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	345	4	2	3	5.0	Cc1ccccc1Nc1cc(C(=O)NC2CCCC2)c2ccccc2n1	nan
	CHEMBL1531717	45631	1	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	345	4	2	3	5.0	Cc1ccccc1Nc1cc(C(=O)NC2CCCC2)c2ccccc2n1	nan
	982830	45676	21	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	400	4	1	5	4.7	Cc1cc2nnc(SCC(=O)Nc3ccc(F)c(Cl)c3)n2c2ccccc12	nan
	CHEMBL1532117	45676	21	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	400	4	1	5	4.7	Cc1cc2nnc(SCC(=O)Nc3ccc(F)c(Cl)c3)n2c2ccccc12	nan
	895668	45692	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	307	3	1	4	3.2	CC(=O)c1cccc(NC(=O)c2cc(=O)c3ccccc3o2)c1	nan
	CHEMBL1532290	45692	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	307	3	1	4	3.2	CC(=O)c1cccc(NC(=O)c2cc(=O)c3ccccc3o2)c1	nan
	2078424	45758	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	344	5	2	4	2.9	COc1cccc(CC(=O)Nc2sc3c(c2C(N)=O)CCCC3)c1	nan
	CHEMBL1532835	45758	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	344	5	2	4	2.9	COc1cccc(CC(=O)Nc2sc3c(c2C(N)=O)CCCC3)c1	nan
	718477	45761	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	227	1	0	6	2.1	COc1nc(C)nc2c1sc(=S)n2C	nan
	CHEMBL1532843	45761	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	227	1	0	6	2.1	COc1nc(C)nc2c1sc(=S)n2C	nan
	3239288	45800	1	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	332	5	1	6	2.9	CCC(Sc1ccc2nnc(-c3ccc(F)cc3)n2n1)C(=O)O	nan
	CHEMBL1533246	45800	1	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	332	5	1	6	2.9	CCC(Sc1ccc2nnc(-c3ccc(F)cc3)n2n1)C(=O)O	nan
	16025355	45839	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	530	7	1	6	5.5	CCc1ccccc1NC(=O)CSc1ncc2c(n1)-c1ccccc1N(Cc1ccc(C)cc1)S2(=O)=O	nan
	CHEMBL1533601	45839	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	530	7	1	6	5.5	CCc1ccccc1NC(=O)CSc1ncc2c(n1)-c1ccccc1N(Cc1ccc(C)cc1)S2(=O)=O	nan
	3214708	45859	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	475	5	2	8	2.5	CC(=O)Nc1ccc(S(=O)(=O)N2CCN(Cc3nc(O)c4c(C)c(C)sc4n3)CC2)cc1	nan
	CHEMBL1533736	45859	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	475	5	2	8	2.5	CC(=O)Nc1ccc(S(=O)(=O)N2CCN(Cc3nc(O)c4c(C)c(C)sc4n3)CC2)cc1	nan
	16028279	45875	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	8	1	8	3.2	CCOc1ccc(NC(=O)Cn2ccn3nc(-c4ccc(OC)c(OC)c4)cc3c2=O)cc1	nan
	CHEMBL1533861	45875	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	448	8	1	8	3.2	CCOc1ccc(NC(=O)Cn2ccn3nc(-c4ccc(OC)c(OC)c4)cc3c2=O)cc1	nan
	4046943	45892	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	4	1	6	2.5	Cc1cc(NC(=O)CSc2nc3c(cc2C#N)CCC3)no1	nan
	CHEMBL1534012	45892	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	4	1	6	2.5	Cc1cc(NC(=O)CSc2nc3c(cc2C#N)CCC3)no1	nan
	3932775	45908	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	4	1	5	3.8	CCc1ccc2nc(NC(=O)c3ccc(N4C(=O)CCC4=O)cc3)sc2c1	nan
	CHEMBL1534252	45908	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	4	1	5	3.8	CCc1ccc2nc(NC(=O)c3ccc(N4C(=O)CCC4=O)cc3)sc2c1	nan
	4658600	45943	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	506	7	1	6	6.0	CCN(CC)C(=O)c1sc(NC(=O)C2c3ccccc3Oc3ccccc32)c(C(=O)OC(C)C)c1C	nan
	CHEMBL1534562	45943	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	506	7	1	6	6.0	CCN(CC)C(=O)c1sc(NC(=O)C2c3ccccc3Oc3ccccc32)c(C(=O)OC(C)C)c1C	nan
	16025630	45989	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	5	1	7	3.7	COc1cccc(NC(=O)CSc2ncc3c(n2)-c2ccc(Cl)cc2N(C)S3(=O)=O)c1	nan
	CHEMBL1535077	45989	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	5	1	7	3.7	COc1cccc(NC(=O)CSc2ncc3c(n2)-c2ccc(Cl)cc2N(C)S3(=O)=O)c1	nan
	3185711	46002	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	522	9	3	8	2.6	CN(C)c1ccc(C(C(=O)NCC2CCCO2)N(C(=O)c2snc(C(N)=O)c2N)c2ccccc2)cc1	nan
	CHEMBL1535224	46002	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	522	9	3	8	2.6	CN(C)c1ccc(C(C(=O)NCC2CCCO2)N(C(=O)c2snc(C(N)=O)c2N)c2ccccc2)cc1	nan
	54677757	46039	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	283	2	1	4	3.4	Cn1c(=O)c(Sc2ccccc2)c(O)c2ccccc21	nan
	CHEMBL1535623	46039	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	283	2	1	4	3.4	Cn1c(=O)c(Sc2ccccc2)c(O)c2ccccc21	nan
	4792884	46072	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	440	4	1	6	2.9	COc1ccc(Br)cc1-c1nc2c(c(=O)[nH]c(=O)n2Cc2ccccc2)n1C	nan
	CHEMBL1535940	46072	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	440	4	1	6	2.9	COc1ccc(Br)cc1-c1nc2c(c(=O)[nH]c(=O)n2Cc2ccccc2)n1C	nan
	135516269	46103	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	8	2	8	3.1	CCOc1ccc(-n2c(SCC(=O)NC(C)CC)nc3nnc(C)c-3c2N)cc1	nan
	CHEMBL1536353	46103	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	8	2	8	3.1	CCOc1ccc(-n2c(SCC(=O)NC(C)CC)nc3nnc(C)c-3c2N)cc1	nan
	3208311	46123	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	400	5	3	9	2.5	CCc1cc2cc3c(cc2nc1SCC(=O)Nc1cnc(O)nc1O)OCO3	nan
	CHEMBL1536575	46123	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	400	5	3	9	2.5	CCc1cc2cc3c(cc2nc1SCC(=O)Nc1cnc(O)nc1O)OCO3	nan
	1965061	46178	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	7	0	6	4.0	CCCCCc1nc2c(c(=O)c3ccccc3n2C)c(=O)n1Cc1ccc(OC)cc1	nan
	CHEMBL1536987	46178	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	7	0	6	4.0	CCCCCc1nc2c(c(=O)c3ccccc3n2C)c(=O)n1Cc1ccc(OC)cc1	nan
	2296181	46220	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	304	4	2	3	2.4	O=C(CNC(=S)NC(=O)C1CCCCC1)c1ccccc1	nan
	CHEMBL1537419	46220	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	304	4	2	3	2.4	O=C(CNC(=S)NC(=O)C1CCCCC1)c1ccccc1	nan
	4358102	46252	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	498	7	1	7	3.8	O=C(CCCCCn1c(=S)[nH]c2cc3c(cc2c1=O)OCO3)N1CCN(c2ccc(F)cc2)CC1	nan
	CHEMBL1537648	46252	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	498	7	1	7	3.8	O=C(CCCCCn1c(=S)[nH]c2cc3c(cc2c1=O)OCO3)N1CCN(c2ccc(F)cc2)CC1	nan
	16194098	46271	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	4	1	6	3.6	CSc1ccc(CNc2nc3ccccc3n3cnnc23)cc1	nan
	CHEMBL1537791	46271	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	4	1	6	3.6	CSc1ccc(CNc2nc3ccccc3n3cnnc23)cc1	nan
	1272394	46372	10	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	361	6	1	7	3.5	COc1ccc(C(=O)Nc2nnc(Cc3cccs3)s2)cc1OC	nan
	CHEMBL1538560	46372	10	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	361	6	1	7	3.5	COc1ccc(C(=O)Nc2nnc(Cc3cccs3)s2)cc1OC	nan
	921484	46468	13	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	315	3	1	4	4.1	O=C(Nc1ccc2oc(-c3ccncc3)nc2c1)c1ccccc1	nan
	CHEMBL1539494	46468	13	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	315	3	1	4	4.1	O=C(Nc1ccc2oc(-c3ccncc3)nc2c1)c1ccccc1	nan
	664170	46539	8	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	3	0	8	3.5	CCOC(=O)N1CCN(c2nc(SC)nc3sc4c(c23)CC(C)(C)OC4)CC1	nan
	CHEMBL1540011	46539	8	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	3	0	8	3.5	CCOC(=O)N1CCN(c2nc(SC)nc3sc4c(c23)CC(C)(C)OC4)CC1	nan
	6621296	46622	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	4	1	6	3.3	O=C(NCc1ccccc1)C1CCCN(c2nc3ccsc3c(=O)s2)C1	nan
	CHEMBL1540762	46622	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	385	4	1	6	3.3	O=C(NCc1ccccc1)C1CCCN(c2nc3ccsc3c(=O)s2)C1	nan
	2855521	46687	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	5	2	4	3.2	COc1ccc(COC(=O)C2=C(C)NC(=O)NC2c2ccc(F)cc2)cc1	nan
	CHEMBL1541261	46687	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	5	2	4	3.2	COc1ccc(COC(=O)C2=C(C)NC(=O)NC2c2ccc(F)cc2)cc1	nan
	687554	46715	23	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	295	3	1	4	3.1	CC(=O)Oc1ccc2oc(-c3ccccc3)c(C(N)=O)c2c1	nan
	CHEMBL1541470	46715	23	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	295	3	1	4	3.1	CC(=O)Oc1ccc2oc(-c3ccccc3)c(C(N)=O)c2c1	nan
	16746196	46895	0	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	10	3	5	3.2	CCCCNc1ccc(C(CC(N)=O)NC(=O)c2ccccc2)cc1[N+](=O)[O-]	nan
	CHEMBL1543039	46895	0	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	384	10	3	5	3.2	CCCCNc1ccc(C(CC(N)=O)NC(=O)c2ccccc2)cc1[N+](=O)[O-]	nan
	654907	46909	15	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	5	1	6	4.5	COc1ccc(C(=O)Nc2cccc(-c3nc4ncccc4o3)c2C)cc1OC	nan
	CHEMBL1543164	46909	15	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	5	1	6	4.5	COc1ccc(C(=O)Nc2cccc(-c3nc4ncccc4o3)c2C)cc1OC	nan
	899145	46937	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	348	2	0	5	4.1	Cc1cnn(C(=O)c2cc(-c3ccccn3)nc3ccc(Cl)cc23)c1	nan
	CHEMBL1543380	46937	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	348	2	0	5	4.1	Cc1cnn(C(=O)c2cc(-c3ccccn3)nc3ccc(Cl)cc23)c1	nan
	1337412	46941	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	5	1	6	4.2	CCOc1ccc(-c2nn(-c3ccccc3)cc2/C=C2\SC(N)=NC2=O)cc1C	nan
	146674638	46941	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	5	1	6	4.2	CCOc1ccc(-c2nn(-c3ccccc3)cc2/C=C2\SC(N)=NC2=O)cc1C	nan
	CHEMBL1543421	46941	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	5	1	6	4.2	CCOc1ccc(-c2nn(-c3ccccc3)cc2/C=C2\SC(N)=NC2=O)cc1C	nan
	1773311	46986	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	6	1	7	3.1	CCN(CC)C(=O)CSc1nc(N)c(C#N)c(-c2cccs2)c1C#N	nan
	CHEMBL1543838	46986	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	6	1	7	3.1	CCN(CC)C(=O)CSc1nc(N)c(C#N)c(-c2cccs2)c1C#N	nan
	22553577	47057	3	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	6	1	5	3.5	O=C(CCCn1c(=O)c2cccn2c2cccnc21)NCc1cccc(Br)c1	nan
	CHEMBL1544274	47057	3	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	6	1	5	3.5	O=C(CCCn1c(=O)c2cccn2c2cccnc21)NCc1cccc(Br)c1	nan
	2150501	47237	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	8	1	8	3.5	COCCn1c(SCC(=O)Nc2ccc(OC)cc2)nc2c(oc3ccccc32)c1=O	nan
	CHEMBL1545636	47237	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	8	1	8	3.5	COCCn1c(SCC(=O)Nc2ccc(OC)cc2)nc2c(oc3ccccc32)c1=O	nan
	1131000	47245	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	4	2	5	3.2	COC(=O)c1c(NC(C)=O)sc(C(=O)Nc2ccccc2F)c1C	nan
	CHEMBL1545709	47245	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	4	2	5	3.2	COC(=O)c1c(NC(C)=O)sc(C(=O)Nc2ccccc2F)c1C	nan
	4975679	47341	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	310	1	1	1	4.0	O=C(c1cc2cc(Cl)ccc2[nH]1)N1CCc2ccccc2C1	nan
	CHEMBL1546589	47341	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	310	1	1	1	4.0	O=C(c1cc2cc(Cl)ccc2[nH]1)N1CCc2ccccc2C1	nan
	4099286	47388	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	366	8	1	4	3.8	CCOc1ccc(CNC(=O)CCc2cn(C)c3ccccc23)cc1OC	nan
	CHEMBL1547036	47388	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	366	8	1	4	3.8	CCOc1ccc(CNC(=O)CCc2cn(C)c3ccccc23)cc1OC	nan
	246421	47397	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	283	3	3	6	3.0	CSc1nc(O)c(Nc2cccc(Cl)c2)c(O)n1	nan
	CHEMBL1547116	47397	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	283	3	3	6	3.0	CSc1nc(O)c(Nc2cccc(Cl)c2)c(O)n1	nan
	3179963	47507	3	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	8	3	7	2.3	CCC(C(=O)NC1CCCC1)N(C(=O)c1snc(C(N)=O)c1N)c1ccc(OC)cc1	nan
	CHEMBL1548213	47507	3	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	8	3	7	2.3	CCC(C(=O)NC1CCCC1)N(C(=O)c1snc(C(N)=O)c1N)c1ccc(OC)cc1	nan
	16608827	47526	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	479	7	1	5	3.8	COc1ccc(S(=O)(=O)N2CCN(C(c3ccccc3)c3ccccc3)CC2)cc1NC(C)=O	nan
	CHEMBL1548379	47526	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	479	7	1	5	3.8	COc1ccc(S(=O)(=O)N2CCN(C(c3ccccc3)c3ccccc3)CC2)cc1NC(C)=O	nan
	1711150	47634	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	8	1	6	3.6	COc1cc(/C=C/C(=O)OCC(=O)Nc2ccccc2Cl)cc(OC)c1OC	nan
	CHEMBL1549297	47634	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	8	1	6	3.6	COc1cc(/C=C/C(=O)OCC(=O)Nc2ccccc2Cl)cc(OC)c1OC	nan
	4371420	47639	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	5	0	4	2.9	O=C(COC(=O)c1ccc(N2CCCC2=O)cc1)c1ccccc1	nan
	CHEMBL1549350	47639	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	5	0	4	2.9	O=C(COC(=O)c1ccc(N2CCCC2=O)cc1)c1ccccc1	nan
	650104	47767	2	None	-3	3	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	6	1	6	3.8	CCc1cc2ccc(OC)cc2nc1SCC(=O)Nc1cc(C)on1	nan
	CHEMBL1550363	47767	2	None	-3	3	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	6	1	6	3.8	CCc1cc2ccc(OC)cc2nc1SCC(=O)Nc1cc(C)on1	nan
	891743	47812	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	3	1	3	4.5	Cc1nc(-c2ccc(C(=O)Nc3ccc(F)cc3)cc2)cs1	nan
	CHEMBL1550704	47812	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	3	1	3	4.5	Cc1nc(-c2ccc(C(=O)Nc3ccc(F)cc3)cc2)cs1	nan
	135437051	47857	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	6	3	6	4.1	CCc1ccccc1NC(=O)CSc1nc2[nH]nc(C)c2c(=N)n1-c1cccc(C)c1	nan
	CHEMBL1551159	47857	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	6	3	6	4.1	CCc1ccccc1NC(=O)CSc1nc2[nH]nc(C)c2c(=N)n1-c1cccc(C)c1	nan
	16030615	47861	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	505	6	0	9	3.1	COc1ccc(C(=O)N2CCN(Cc3cc(=O)n4nc(-c5ccccc5C)sc4n3)CC2)cc1OC	nan
	CHEMBL1551229	47861	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	505	6	0	9	3.1	COc1ccc(C(=O)N2CCN(Cc3cc(=O)n4nc(-c5ccccc5C)sc4n3)CC2)cc1OC	nan
	16018080	47864	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	8	1	6	3.5	COc1cccc(CNC(=O)CCCn2c(=O)c3cccn3c3ccc(F)cc32)c1OC	nan
	CHEMBL1551250	47864	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	8	1	6	3.5	COc1cccc(CNC(=O)CCCn2c(=O)c3cccn3c3ccc(F)cc32)c1OC	nan
	16012980	47873	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	3	1	3	5.3	Cc1ccc2nc(O)c(CN(C(=O)c3cccc(Cl)c3)C(C)(C)C)cc2c1	nan
	CHEMBL1551350	47873	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	3	1	3	5.3	Cc1ccc2nc(O)c(CN(C(=O)c3cccc(Cl)c3)C(C)(C)C)cc2c1	nan
	3534311	47880	16	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	363	5	2	6	2.0	NS(=O)(=O)c1ccc2nc(NC(=O)COc3ccccc3)sc2c1	nan
	CHEMBL1551511	47880	16	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	363	5	2	6	2.0	NS(=O)(=O)c1ccc2nc(NC(=O)COc3ccccc3)sc2c1	nan
	16030318	47882	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	7	1	9	3.5	CCOc1ccc(C(=O)Nc2nnc(SCc3cc(=O)n4ccccc4n3)s2)cc1	nan
	CHEMBL1551529	47882	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	7	1	9	3.5	CCOc1ccc(C(=O)Nc2nnc(SCc3cc(=O)n4ccccc4n3)s2)cc1	nan
	16031341	47888	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	260	2	1	5	1.9	Cc1ccccc1C(=O)Nc1nnc2n1CCS2	nan
	CHEMBL1551637	47888	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	260	2	1	5	1.9	Cc1ccccc1C(=O)Nc1nnc2n1CCS2	nan
	16012572	47892	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	5	1	5	4.4	Cc1cc(C)c2c(n1)nn1c(C)c(CCC(=O)NCc3ccc(Cl)cc3)c(C)nc21	nan
	CHEMBL1551773	47892	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	5	1	5	4.4	Cc1cc(C)c2c(n1)nn1c(C)c(CCC(=O)NCc3ccc(Cl)cc3)c(C)nc21	nan
	4112916	47906	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	5	0	5	5.2	CCOc1nc(-c2ccccc2)ccc1-c1noc(-c2ccc(C)cc2)n1	nan
	CHEMBL1551932	47906	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	5	0	5	5.2	CCOc1nc(-c2ccccc2)ccc1-c1noc(-c2ccc(C)cc2)n1	nan
	16030647	47908	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	509	6	0	8	3.6	CC(Oc1ccccc1)C(=O)N1CCN(Cc2cc(=O)n3nc(-c4ccccc4Cl)sc3n2)CC1	nan
	CHEMBL1551961	47908	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	509	6	0	8	3.6	CC(Oc1ccccc1)C(=O)N1CCN(Cc2cc(=O)n3nc(-c4ccccc4Cl)sc3n2)CC1	nan
	4069977	47916	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	7	1	4	6.3	CCOc1ccc(Sc2cc(C(=O)NC(C)c3ccccc3)c3ccccc3n2)cc1	nan
	CHEMBL1552026	47916	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	7	1	4	6.3	CCOc1ccc(Sc2cc(C(=O)NC(C)c3ccccc3)c3ccccc3n2)cc1	nan
	16027075	47924	0	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	6	0	8	4.8	COc1ccc(-c2nc(Cn3c(=O)cc(C)c4c(C)nn(-c5ccccc5)c43)c(C)o2)cc1OC	nan
	CHEMBL1552119	47924	0	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	6	0	8	4.8	COc1ccc(-c2nc(Cn3c(=O)cc(C)c4c(C)nn(-c5ccccc5)c43)c(C)o2)cc1OC	nan
	24792649	47928	0	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	310	0	0	3	3.5	Cn1c2ccccc2c(=O)c2ccc(C#Cc3ccccn3)cc21	nan
	CHEMBL1552163	47928	0	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	310	0	0	3	3.5	Cn1c2ccccc2c(=O)c2ccc(C#Cc3ccccn3)cc21	nan
	16020555	47950	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	480	5	0	5	4.8	O=c1c(S(=O)(=O)c2ccccc2)cn(Cc2cccc(F)c2)c2cc(N3CCCC3)c(F)cc12	nan
	CHEMBL1552450	47950	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	480	5	0	5	4.8	O=c1c(S(=O)(=O)c2ccccc2)cn(Cc2cccc(F)c2)c2cc(N3CCCC3)c(F)cc12	nan
	7217107	47953	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	6	2	8	2.4	Cc1ccc(NC(=O)c2cnc(SCC(=O)Nc3cc(C)on3)n(C)c2=O)cc1	nan
	CHEMBL1552487	47953	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	6	2	8	2.4	Cc1ccc(NC(=O)c2cnc(SCC(=O)Nc3cc(C)on3)n(C)c2=O)cc1	nan
	3666941	47954	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	499	6	1	6	4.9	Cc1ccc(CNC(=O)CSc2nc3ccsc3c(=O)n2-c2ccc(Br)cc2)cc1	nan
	CHEMBL1552556	47954	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	499	6	1	6	4.9	Cc1ccc(CNC(=O)CSc2nc3ccsc3c(=O)n2-c2ccc(Br)cc2)cc1	nan
	16010970	47967	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	4	0	7	3.6	CCc1cc2c(cc3c(=O)n(CC(=O)N4CCN(c5cc(Cl)ccc5C)CC4)ncn32)s1	nan
	CHEMBL1552740	47967	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	4	0	7	3.6	CCc1cc2c(cc3c(=O)n(CC(=O)N4CCN(c5cc(Cl)ccc5C)CC4)ncn32)s1	nan
	16021520	47970	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	5	1	4	4.6	CSc1ncc(C(=O)NCc2cccc(Br)c2)c(-c2ccccc2)n1	nan
	CHEMBL1552765	47970	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	5	1	4	4.6	CSc1ncc(C(=O)NCc2cccc(Br)c2)c(-c2ccccc2)n1	nan
	16024485	47989	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	5	1	5	3.9	Cc1ccc2c(=O)c(C(=O)c3ccccc3)cn(CC(=O)Nc3ccccc3C)c2n1	nan
	CHEMBL1553018	47989	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	5	1	5	3.9	Cc1ccc2c(=O)c(C(=O)c3ccccc3)cn(CC(=O)Nc3ccccc3C)c2n1	nan
	3160964	47993	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	4	1	5	3.6	Cc1cccc(OCC(=O)Nc2c(C)ccc3nsnc23)c1C	nan
	CHEMBL1553050	47993	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	4	1	5	3.6	Cc1cccc(OCC(=O)Nc2c(C)ccc3nsnc23)c1C	nan
	16012361	48041	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	6	1	5	4.2	CCc1ccccc1NC(=O)Cn1ncc2c(C)n(Cc3ccccc3F)c(C)c2c1=O	nan
	CHEMBL1553757	48041	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	6	1	5	4.2	CCc1ccccc1NC(=O)Cn1ncc2c(C)n(Cc3ccccc3F)c(C)c2c1=O	nan
	16027446	48057	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	464	6	1	8	3.8	O=C(OCc1cc(=O)n2nc(C3CC3)sc2n1)c1ccc(NC(=O)c2ccccc2F)cc1	nan
	CHEMBL1553997	48057	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	464	6	1	8	3.8	O=C(OCc1cc(=O)n2nc(C3CC3)sc2n1)c1ccc(NC(=O)c2ccccc2F)cc1	nan
	16030862	48084	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	398	4	1	3	3.1	CC(=O)N1CCc2cc(CNS(=O)(=O)c3ccccc3C(F)(F)F)ccc21	nan
	CHEMBL1554375	48084	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	398	4	1	3	3.1	CC(=O)N1CCc2cc(CNS(=O)(=O)c3ccccc3C(F)(F)F)ccc21	nan
	16030106	48093	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	6	1	7	3.2	COc1ccc(CNC(=O)Cn2nc(C)c3nn(-c4ccc(Cl)cc4)c(C)c3c2=O)cc1	nan
	CHEMBL1554505	48093	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	6	1	7	3.2	COc1ccc(CNC(=O)Cn2nc(C)c3nn(-c4ccc(Cl)cc4)c(C)c3c2=O)cc1	nan
	4074992	48099	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	7	1	4	5.9	CCOc1ccc(Sc2cc(C(=O)NCc3ccc(F)cc3)c3ccccc3n2)cc1	nan
	CHEMBL1554644	48099	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	7	1	4	5.9	CCOc1ccc(Sc2cc(C(=O)NCc3ccc(F)cc3)c3ccccc3n2)cc1	nan
	5058559	48111	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	5	1	5	2.9	CC(=O)c1cccc(NC(=O)c2ccc(S(=O)(=O)N3CC(C)OC(C)C3)cc2)c1	nan
	CHEMBL1554762	48111	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	5	1	5	2.9	CC(=O)c1cccc(NC(=O)c2ccc(S(=O)(=O)N3CC(C)OC(C)C3)cc2)c1	nan
	16026882	48112	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	6	0	8	3.5	O=C(COc1ccc(F)cc1)OCc1cc(=O)n2nc(C3CCCCC3)sc2n1	nan
	CHEMBL1554822	48112	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	417	6	0	8	3.5	O=C(COc1ccc(F)cc1)OCc1cc(=O)n2nc(C3CCCCC3)sc2n1	nan
	4289361	48126	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	7	1	5	5.3	CCOc1cccc(C(=O)Nc2c(C(=O)c3ccc(OC)cc3)oc3ccccc23)c1	nan
	CHEMBL1555049	48126	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	7	1	5	5.3	CCOc1cccc(C(=O)Nc2c(C(=O)c3ccc(OC)cc3)oc3ccccc23)c1	nan
	3282564	48133	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	347	3	1	4	4.6	Cc1ccc(-c2nnc(NC(=O)c3c(F)cccc3Cl)s2)cc1	nan
	CHEMBL1555127	48133	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	347	3	1	4	4.6	Cc1ccc(-c2nnc(NC(=O)c3c(F)cccc3Cl)s2)cc1	nan
	16009325	48144	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	5	1	7	3.2	O=C(Cn1cc(S(=O)(=O)c2ccccc2)c(=O)c2cc3c(cc21)OCO3)Nc1ccccc1	nan
	CHEMBL1555288	48144	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	5	1	7	3.2	O=C(Cn1cc(S(=O)(=O)c2ccccc2)c(=O)c2cc3c(cc21)OCO3)Nc1ccccc1	nan
	135416425	48147	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	358	3	2	4	5.1	Cc1ccccc1C(=O)Nc1cc(C)c(O)c(-c2nc3ccccc3o2)c1	nan
	CHEMBL1555312	48147	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	358	3	2	4	5.1	Cc1ccccc1C(=O)Nc1cc(C)c(O)c(-c2nc3ccccc3o2)c1	nan
	16023840	48197	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	5	1	6	4.3	CCOC(=O)c1c(C)oc2nc(C)nc(NCc3ccccc3Cl)c12	nan
	CHEMBL1555863	48197	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	5	1	6	4.3	CCOC(=O)c1c(C)oc2nc(C)nc(NCc3ccccc3Cl)c12	nan
	4432211	48206	9	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	2	1	6	2.5	CC(=O)N1CCc2c(sc(NC(=O)c3ccc4c(c3)OCCO4)c2C#N)C1	nan
	CHEMBL1555967	48206	9	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	383	2	1	6	2.5	CC(=O)N1CCc2c(sc(NC(=O)c3ccc4c(c3)OCCO4)c2C#N)C1	nan
	929959	48241	12	None	-2	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	2	1	8	0.8	COc1ccc(-c2c(C#N)c(N)nc3c2c(=O)n(C)c(=O)n3C)cc1	nan
	CHEMBL1556274	48241	12	None	-2	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	2	1	8	0.8	COc1ccc(-c2c(C#N)c(N)nc3c2c(=O)n(C)c(=O)n3C)cc1	nan
	1718133	48269	10	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	6	2	5	4.3	CCCCCC(=O)NC(=S)Nc1cccc(-c2nc3ncccc3o2)c1	nan
	CHEMBL1556586	48269	10	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	6	2	5	4.3	CCCCCC(=O)NC(=S)Nc1cccc(-c2nc3ncccc3o2)c1	nan
	1475314	48280	14	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	251	2	1	4	3.2	Cc1nc(N)ncc1Sc1ccc(Cl)cc1	nan
	CHEMBL1556672	48280	14	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	251	2	1	4	3.2	Cc1nc(N)ncc1Sc1ccc(Cl)cc1	nan
	1829088	48332	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	6	1	5	2.5	COCCNC(=O)Cn1nc(-c2ccc(Cl)cc2)c2ccccc2c1=O	nan
	CHEMBL1557090	48332	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	6	1	5	2.5	COCCNC(=O)Cn1nc(-c2ccc(Cl)cc2)c2ccccc2c1=O	nan
	16008924	48342	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	3	1	4	3.6	Cn1c(C(=O)NCc2ccc(Cl)cc2)cc2c(=O)n(C)c3ccccc3c21	nan
	CHEMBL1557189	48342	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	379	3	1	4	3.6	Cn1c(C(=O)NCc2ccc(Cl)cc2)cc2c(=O)n(C)c3ccccc3c21	nan
	20868637	48385	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	4	1	5	3.8	CCOc1ccc2ncc(S(=O)(=O)c3ccc(C)c(C)c3)c(O)c2c1	nan
	CHEMBL1557551	48385	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	4	1	5	3.8	CCOc1ccc2ncc(S(=O)(=O)c3ccc(C)c(C)c3)c(O)c2c1	nan
	16030924	48401	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	6	1	6	5.1	COc1ccc(-c2cn3nc(SCC(=O)Nc4ccc(C)c(Cl)c4)ccc3n2)cc1	nan
	CHEMBL1557656	48401	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	438	6	1	6	5.1	COc1ccc(-c2cn3nc(SCC(=O)Nc4ccc(C)c(Cl)c4)ccc3n2)cc1	nan
	899391	48406	12	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	296	3	1	4	2.8	O=C(Cc1ccccc1)Nc1nc(=O)c2ccccc2s1	nan
	CHEMBL1557721	48406	12	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	296	3	1	4	2.8	O=C(Cc1ccccc1)Nc1nc(=O)c2ccccc2s1	nan
	3846782	48408	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	534	4	1	7	4.1	Cc1ccc(Cn2c(=N)c(S(=O)(=O)c3ccc(Br)cc3)cc3c(=O)n4ccccc4nc32)cc1	nan
	CHEMBL1557740	48408	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	534	4	1	7	4.1	Cc1ccc(Cn2c(=N)c(S(=O)(=O)c3ccc(Br)cc3)cc3c(=O)n4ccccc4nc32)cc1	nan
	1485561	48430	12	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	3	0	5	4.4	O=S(=O)(c1ccccc1)c1cnn2c(C(F)(F)F)cc(-c3ccc(F)cc3)nc12	nan
	CHEMBL1557929	48430	12	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	3	0	5	4.4	O=S(=O)(c1ccccc1)c1cnn2c(C(F)(F)F)cc(-c3ccc(F)cc3)nc12	nan
	54706216	48486	15	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	2	3	4	3.5	O=C(NC1CCCCCCC1)c1c(O)nc2ccccc2c1O	nan
	CHEMBL1558469	48486	15	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	314	2	3	4	3.5	O=C(NC1CCCCCCC1)c1c(O)nc2ccccc2c1O	nan
	5185520	48497	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	310	4	2	4	2.5	Nc1cc(Cl)ccc1C(=O)OCC(=O)NC1CCCCC1	nan
	CHEMBL1558534	48497	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	310	4	2	4	2.5	Nc1cc(Cl)ccc1C(=O)OCC(=O)NC1CCCCC1	nan
	666603	48531	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	2	1	6	4.1	Cc1nn(-c2ccc(F)cc2)c2nc(N)c(C#N)c(-c3cccs3)c12	nan
	CHEMBL1558784	48531	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	2	1	6	4.1	Cc1nn(-c2ccc(F)cc2)c2nc(N)c(C#N)c(-c3cccs3)c12	nan
	15991438	48539	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	5	1	6	3.8	Cc1cccc(NC(=O)CSc2nc3ccccc3nc2N2CCOCC2)c1C	nan
	CHEMBL1558859	48539	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	5	1	6	3.8	Cc1cccc(NC(=O)CSc2nc3ccccc3nc2N2CCOCC2)c1C	nan
	950988	48555	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	4	2	5	4.8	COc1cccc(Nc2nc(-c3ccccc3O)nc3ccccc23)c1	nan
	CHEMBL1558977	48555	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	4	2	5	4.8	COc1cccc(Nc2nc(-c3ccccc3O)nc3ccccc23)c1	nan
	4345257	48566	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	6	2	6	3.2	Cc1cc(C)cc(NC(=O)CSc2nnc(NC(=O)C3CC3)s2)c1	nan
	CHEMBL1559060	48566	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	6	2	6	3.2	Cc1cc(C)cc(NC(=O)CSc2nnc(NC(=O)C3CC3)s2)c1	nan
	900716	48578	19	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	326	3	1	5	3.6	COC(=O)c1ccc(NC(=O)c2ccc3nc(C)sc3c2)cc1	nan
	CHEMBL1559158	48578	19	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	326	3	1	5	3.6	COC(=O)c1ccc(NC(=O)c2ccc3nc(C)sc3c2)cc1	nan
	2156049	48648	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	4	1	4	5.5	Cc1ccc(-n2c(SCc3ccccc3)nc3c([nH]c4ccccc43)c2=O)cc1	nan
	CHEMBL1559857	48648	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	4	1	4	5.5	Cc1ccc(-n2c(SCc3ccccc3)nc3c([nH]c4ccccc43)c2=O)cc1	nan
	3138574	48651	10	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	4	3	4	3.6	O=C(NNc1c2ccccc2nc2ccccc12)C(O)c1ccccc1	nan
	CHEMBL1559872	48651	10	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	4	3	4	3.6	O=C(NNc1c2ccccc2nc2ccccc12)C(O)c1ccccc1	nan
	16017814	48669	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	5	1	6	2.9	COc1ccc(Cl)cc1NC(=O)Cn1ccn(-c2cc(C)cc(C)c2)c(=O)c1=O	nan
	CHEMBL1560031	48669	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	5	1	6	2.9	COc1ccc(Cl)cc1NC(=O)Cn1ccn(-c2cc(C)cc(C)c2)c(=O)c1=O	nan
	2028031	48743	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	1	0	5	3.5	Cc1nc2c(c(=O)c3ccccc3n2C)c(=O)n1C1CCCCCC1	nan
	CHEMBL1560823	48743	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	1	0	5	3.5	Cc1nc2c(c(=O)c3ccccc3n2C)c(=O)n1C1CCCCCC1	nan
	4690835	48746	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	4	1	5	4.8	COc1ccc2oc(-c3cccc(NC(=O)c4ccc(C#N)cc4F)c3)nc2c1	nan
	CHEMBL1560860	48746	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	387	4	1	5	4.8	COc1ccc2oc(-c3cccc(NC(=O)c4ccc(C#N)cc4F)c3)nc2c1	nan
	15990056	48918	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	3	1	5	4.4	CCc1nnc2c3ccccc3nc(Nc3ccc(F)c(Cl)c3)n12	nan
	CHEMBL1562390	48918	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	3	1	5	4.4	CCc1nnc2c3ccccc3nc(Nc3ccc(F)c(Cl)c3)n12	nan
	5299641	48922	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	4	1	4	4.6	Cc1ccc(Cl)cc1NC(=O)CSc1nc(C)c(C)c(C)c1C#N	nan
	CHEMBL1562426	48922	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	4	1	4	4.6	Cc1ccc(Cl)cc1NC(=O)CSc1nc(C)c(C)c(C)c1C#N	nan
	135496880	48925	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	4	2	9	3.5	Oc1nc(SCc2nc(O)c3cnn(-c4ccccc4)c3n2)nc2ccccc12	nan
	CHEMBL1562459	48925	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	4	2	9	3.5	Oc1nc(SCc2nc(O)c3cnn(-c4ccccc4)c3n2)nc2ccccc12	nan
	1176245	48971	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	6	1	6	4.0	CCOc1ccc2nc(SCC(=O)Nc3cc(C)on3)c(C)cc2c1	nan
	CHEMBL1562840	48971	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	6	1	6	4.0	CCOc1ccc2nc(SCC(=O)Nc3cc(C)on3)c(C)cc2c1	nan
	16030293	48974	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	483	7	1	5	6.0	COc1ccccc1Cc1nc2ccccc2nc1SCC(=O)Nc1ccccc1C(F)(F)F	nan
	CHEMBL1562857	48974	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	483	7	1	5	6.0	COc1ccccc1Cc1nc2ccccc2nc1SCC(=O)Nc1ccccc1C(F)(F)F	nan
	16008836	49053	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	482	6	1	5	5.2	O=C(NCCCN1CCN(c2ccc(F)cc2)CC1)c1cc2c(Cl)nc3ccccc3c2s1	nan
	CHEMBL1563658	49053	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	482	6	1	5	5.2	O=C(NCCCN1CCN(c2ccc(F)cc2)CC1)c1cc2c(Cl)nc3ccccc3c2s1	nan
	258436	49123	41	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	211	1	0	2	2.5	CN1C=CC(=CC=C2C=CC(=O)C=C2)C=C1	nan
	CHEMBL1564141	49123	41	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	211	1	0	2	2.5	CN1C=CC(=CC=C2C=CC(=O)C=C2)C=C1	nan
	16030542	49142	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	7	1	6	3.9	Cc1ccc(OCC(=O)Nc2cccc(OCc3cc(=O)n4ccccc4n3)c2)cc1C	nan
	CHEMBL1564400	49142	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	7	1	6	3.9	Cc1ccc(OCC(=O)Nc2cccc(OCc3cc(=O)n4ccccc4n3)c2)cc1C	nan
	2819137	49202	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	272	3	1	6	2.3	COc1cccc(-c2nc(N)nc(SC)c2C#N)c1	nan
	CHEMBL1564918	49202	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	272	3	1	6	2.3	COc1cccc(-c2nc(N)nc(SC)c2C#N)c1	nan
	3244591	49206	1	None	-100	3	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	5	0	6	4.3	CC(C)CCn1c(SCC#N)nc2c(sc3ccccc32)c1=O	nan
	CHEMBL1564940	49206	1	None	-100	3	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	5	0	6	4.3	CC(C)CCn1c(SCC#N)nc2c(sc3ccccc32)c1=O	nan
	16010206	49218	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	5	1	7	1.6	CCc1ccc(NC(=O)C2CCCN2S(=O)(=O)c2ccc3c(c2)n(C)c(=O)c(=O)n3C)cc1	nan
	CHEMBL1565063	49218	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	470	5	1	7	1.6	CCc1ccc(NC(=O)C2CCCN2S(=O)(=O)c2ccc3c(c2)n(C)c(=O)c(=O)n3C)cc1	nan
	1147655	49221	20	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	5	1	7	3.0	COc1ccc(C(=O)Nc2nc3ccc(S(C)(=O)=O)cc3s2)cc1OC	nan
	CHEMBL1565079	49221	20	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	392	5	1	7	3.0	COc1ccc(C(=O)Nc2nc3ccc(S(C)(=O)=O)cc3s2)cc1OC	nan
	694360	49270	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	315	5	1	5	3.1	N#Cc1c(-c2cccs2)cc(C2CC2)nc1SCC(N)=O	nan
	CHEMBL1565417	49270	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	315	5	1	5	3.1	N#Cc1c(-c2cccs2)cc(C2CC2)nc1SCC(N)=O	nan
	16021091	49313	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	486	8	1	6	5.8	COc1ccc(Cn2c(SCc3ccc(C(=O)NC4CCCCC4)cc3)nc3cccnc32)cc1	nan
	CHEMBL1565772	49313	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	486	8	1	6	5.8	COc1ccc(Cn2c(SCc3ccc(C(=O)NC4CCCCC4)cc3)nc3cccnc32)cc1	nan
	16019049	49397	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	7	1	7	3.6	COc1ccc(CNC(=O)c2ccc(Cn3c(=O)c4cccn4c4cccnc43)cc2)c(OC)c1	nan
	CHEMBL1566421	49397	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	7	1	7	3.6	COc1ccc(CNC(=O)c2ccc(Cn3c(=O)c4cccn4c4cccnc43)cc2)c(OC)c1	nan
	2810064	49405	6	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	332	4	1	7	2.5	COc1cc2nc(NC(=O)c3ccco3)sc(=O)c2cc1OC	nan
	CHEMBL1566488	49405	6	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	332	4	1	7	2.5	COc1cc2nc(NC(=O)c3ccco3)sc(=O)c2cc1OC	nan
	15988926	49558	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	12	1	7	3.0	CCN(CC)C(=O)Cn1c(=O)n(CCCCCC(=O)NCc2ccccc2)c(=O)c2sccc21	nan
	CHEMBL1567696	49558	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	12	1	7	3.0	CCN(CC)C(=O)Cn1c(=O)n(CCCCCC(=O)NCc2ccccc2)c(=O)c2sccc21	nan
	16017081	49647	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	5	1	6	4.5	CCC(C(=O)Nc1ccccc1OC)n1nc(C)c2sc3ccccc3c2c1=O	nan
	CHEMBL1568421	49647	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	5	1	6	4.5	CCC(C(=O)Nc1ccccc1OC)n1nc(C)c2sc3ccccc3c2c1=O	nan
	16030322	49698	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	6	1	8	2.9	CCCC(=O)Nc1nnc(SCc2cc(=O)n3cccc(C)c3n2)s1	nan
	CHEMBL1568901	49698	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	6	1	8	2.9	CCCC(=O)Nc1nnc(SCc2cc(=O)n3cccc(C)c3n2)s1	nan
	713644	49714	14	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	283	2	0	5	1.4	Cc1cn(C(=O)CN2C(=O)c3ccccc3C2=O)c(C)n1	nan
	CHEMBL1569010	49714	14	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	283	2	0	5	1.4	Cc1cn(C(=O)CN2C(=O)c3ccccc3C2=O)c(C)n1	nan
	16024577	49753	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	475	7	1	7	3.7	COc1cc(NC(=O)Cn2cc(C(=O)c3ccc(F)cc3)c(=O)c3ccc(C)nc32)cc(OC)c1	nan
	CHEMBL1569365	49753	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	475	7	1	7	3.7	COc1cc(NC(=O)Cn2cc(C(=O)c3ccc(F)cc3)c(=O)c3ccc(C)nc32)cc(OC)c1	nan
	1146106	49777	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	467	7	1	5	5.2	COc1ccc(-c2cc(C(F)(F)F)nc(SCC(=O)NCc3ccc(Cl)cc3)n2)cc1	nan
	CHEMBL1569521	49777	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	467	7	1	5	5.2	COc1ccc(-c2cc(C(F)(F)F)nc(SCC(=O)NCc3ccc(Cl)cc3)n2)cc1	nan
	1433832	49799	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	283	4	1	4	2.5	N#Cc1cc2ccccc2nc1SCC(=O)NC1CC1	nan
	CHEMBL1569775	49799	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	283	4	1	4	2.5	N#Cc1cc2ccccc2nc1SCC(=O)NC1CC1	nan
	660750	49803	8	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	3	1	5	2.9	Cn1nnnc1-c1cc(Br)ccc1NC(=O)c1ccccc1	nan
	CHEMBL1569814	49803	8	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	357	3	1	5	2.9	Cn1nnnc1-c1cc(Br)ccc1NC(=O)c1ccccc1	nan
	16020020	49862	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	351	5	0	5	4.2	CCOC(=O)CCc1c(C)nc2c(c(C)nn2-c2ccc(C)cc2)c1C	nan
	CHEMBL1570342	49862	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	351	5	0	5	4.2	CCOC(=O)CCc1c(C)nc2c(c(C)nn2-c2ccc(C)cc2)c1C	nan
	893344	49863	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	301	2	2	4	3.3	Cn1nnc2cc(NC(=O)Nc3cccc(Cl)c3)ccc21	nan
	CHEMBL1570344	49863	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	301	2	2	4	3.3	Cn1nnc2cc(NC(=O)Nc3cccc(Cl)c3)ccc21	nan
	7692920	49930	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	5	1	6	3.0	O=C(Nc1nnc(S(=O)(=O)Cc2ccc(F)cc2)s1)c1ccccc1F	nan
	CHEMBL1570825	49930	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	5	1	6	3.0	O=C(Nc1nnc(S(=O)(=O)Cc2ccc(F)cc2)s1)c1ccccc1F	nan
	16015598	49994	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	7	1	6	6.0	CCOc1ccc(C(=O)c2oc3ccccc3c2NC(=O)c2cc(-c3ccccc3)on2)cc1	nan
	CHEMBL1571539	49994	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	7	1	6	6.0	CCOc1ccc(C(=O)c2oc3ccccc3c2NC(=O)c2cc(-c3ccccc3)on2)cc1	nan
	16015076	50057	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	6	1	6	4.0	COC(=O)c1ccccc1NC(=O)CSc1cc(-c2ccccc2)nc(C)n1	nan
	CHEMBL1572102	50057	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	6	1	6	4.0	COC(=O)c1ccccc1NC(=O)CSc1cc(-c2ccccc2)nc(C)n1	nan
	663126	50119	9	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	4	0	6	5.1	Clc1ccc(OCc2nn3c(C4CCCCC4)nnc3s2)c(Cl)c1	nan
	CHEMBL1572687	50119	9	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	4	0	6	5.1	Clc1ccc(OCc2nn3c(C4CCCCC4)nnc3s2)c(Cl)c1	nan
	2318048	50143	14	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	6	1	7	3.7	COc1ccc(-c2csc(NC(=O)c3ccc(N4C(=O)CCC4=O)cc3)n2)cc1OC	nan
	CHEMBL1572874	50143	14	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	6	1	7	3.7	COc1ccc(-c2csc(NC(=O)c3ccc(N4C(=O)CCC4=O)cc3)n2)cc1OC	nan
	135492018	50165	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	317	3	1	4	3.4	O=C1N=C(Nc2ccccn2)SC1Cc1ccccc1Cl	nan
	135635832	50165	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	317	3	1	4	3.4	O=C1N=C(Nc2ccccn2)SC1Cc1ccccc1Cl	nan
	135914561	50165	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	317	3	1	4	3.4	O=C1N=C(Nc2ccccn2)SC1Cc1ccccc1Cl	nan
	CHEMBL1573000	50165	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	317	3	1	4	3.4	O=C1N=C(Nc2ccccn2)SC1Cc1ccccc1Cl	nan
	135870946	50189	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	8	1	8	1.6	COc1ccc(C(=O)COC(=O)CCNC2=NS(=O)(=O)c3ccccc32)c(OC)c1	nan
	CHEMBL1573236	50189	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	8	1	8	1.6	COc1ccc(C(=O)COC(=O)CCNC2=NS(=O)(=O)c3ccccc32)c(OC)c1	nan
	16011872	50193	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	494	6	0	6	7.1	Cc1cccc(-c2nc(Cn3c(SCc4cccc(C(F)(F)F)c4)nc4ccncc43)c(C)o2)c1	nan
	CHEMBL1573276	50193	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	494	6	0	6	7.1	Cc1cccc(-c2nc(Cn3c(SCc4cccc(C(F)(F)F)c4)nc4ccncc43)c(C)o2)c1	nan
	16019020	50206	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	436	6	1	5	4.0	Cc1ccc(CCNC(=O)c2ccc(Cn3c(=O)c4cccn4c4cccnc43)cc2)cc1	nan
	CHEMBL1573442	50206	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	436	6	1	5	4.0	Cc1ccc(CCNC(=O)c2ccc(Cn3c(=O)c4cccn4c4cccnc43)cc2)cc1	nan
	4599423	50252	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	3	3	1	5.2	S=C(NCc1ccc2[nH]c3c(c2c1)CCCC3)Nc1ccccc1Cl	nan
	CHEMBL1573942	50252	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	3	3	1	5.2	S=C(NCc1ccc2[nH]c3c(c2c1)CCCC3)Nc1ccccc1Cl	nan
	16014814	50295	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	6	1	4	5.2	Cc1cccc(NC(=O)c2c(C)cc(C)nc2SCC(=O)c2ccccc2)c1	nan
	CHEMBL1574276	50295	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	6	1	4	5.2	Cc1cccc(NC(=O)c2c(C)cc(C)nc2SCC(=O)c2ccccc2)c1	nan
	921918	50412	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	346	2	0	5	4.8	Fc1ccc(-n2c(-c3cccs3)nc3nc4ccccc4nc32)cc1	nan
	CHEMBL1575663	50412	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	346	2	0	5	4.8	Fc1ccc(-n2c(-c3cccs3)nc3nc4ccccc4nc32)cc1	nan
	1960193	50467	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	3	1	4	3.9	Cn1c(NC(=O)c2ccccc2)c(-c2ccccn2)c(=O)c2ccccc21	nan
	CHEMBL1576207	50467	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	3	1	4	3.9	Cn1c(NC(=O)c2ccccc2)c(-c2ccccn2)c(=O)c2ccccc21	nan
	5846704	50476	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	324	9	1	5	3.9	CCN(CC)CCCNc1oc(/C=C/c2ccccc2)nc1C#N	nan
	CHEMBL1576280	50476	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	324	9	1	5	3.9	CCN(CC)CCCNc1oc(/C=C/c2ccccc2)nc1C#N	nan
	935443	50486	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	3	3	2	5.1	Cc1ccc(NC(S)=Nc2cc(-c3ccccc3)[nH]n2)cc1Cl	nan
	CHEMBL1576343	50486	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	342	3	3	2	5.1	Cc1ccc(NC(S)=Nc2cc(-c3ccccc3)[nH]n2)cc1Cl	nan
	3228917	50555	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	6	2	5	4.7	CCc1cccc(C)c1NC(=O)CSc1[nH]c(-c2ccccc2F)nc2ncnc1-2	nan
	CHEMBL1576889	50555	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	6	2	5	4.7	CCc1cccc(C)c1NC(=O)CSc1[nH]c(-c2ccccc2F)nc2ncnc1-2	nan
	709545	50590	11	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	4	1	6	2.9	Cc1cc(NC(=O)CSc2nc3c(cc2C#N)CCCC3)no1	nan
	CHEMBL1577228	50590	11	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	4	1	6	2.9	Cc1cc(NC(=O)CSc2nc3c(cc2C#N)CCCC3)no1	nan
	3917007	50698	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	7	1	6	2.9	O=C1COc2ccc(C(=O)COC(=O)CCSc3ccccc3)cc2N1	nan
	CHEMBL1578153	50698	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	371	7	1	6	2.9	O=C1COc2ccc(C(=O)COC(=O)CCSc3ccccc3)cc2N1	nan
	20884721	50885	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	5	1	7	1.7	COc1cccc2c1cc1c(=O)n(CC(=O)NCc3ccccn3)nc(C)n12	nan
	CHEMBL1579740	50885	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	5	1	7	1.7	COc1cccc2c1cc1c(=O)n(CC(=O)NCc3ccccn3)nc(C)n12	nan
	1292507	50929	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	6	1	7	4.4	Cc1ccc(-n2c(SCC(=O)NCc3ccco3)nc3sc(C)c(C)c3c2=O)cc1	nan
	CHEMBL1580140	50929	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	6	1	7	4.4	Cc1ccc(-n2c(SCC(=O)NCc3ccco3)nc3sc(C)c(C)c3c2=O)cc1	nan
	2347564	51149	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	3	1	9	1.6	Cc1nn(-c2ccccc2)c2sc(C(=O)c3c(N)n(C)c(=O)n(C)c3=O)cc12	nan
	CHEMBL1581991	51149	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	3	1	9	1.6	Cc1nn(-c2ccccc2)c2sc(C(=O)c3c(N)n(C)c(=O)n(C)c3=O)cc12	nan
	1454917	51179	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	5	1	5	4.7	CCc1ccc2c(c1)cc(CN(C(S)=Nc1cccc(C)c1)C1CC1)c1nnnn12	nan
	CHEMBL1582197	51179	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	5	1	5	4.7	CCc1ccc2c(c1)cc(CN(C(S)=Nc1cccc(C)c1)C1CC1)c1nnnn12	nan
	7080789	51245	1	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	373	5	3	4	3.3	Cc1ccc2cc(CCNC(=O)C(=O)c3c[nH]c4ccccc34)c(O)nc2c1	nan
	CHEMBL1582792	51245	1	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	373	5	3	4	3.3	Cc1ccc2cc(CCNC(=O)C(=O)c3c[nH]c4ccccc34)c(O)nc2c1	nan
	1420394	51263	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	4	1	4	5.2	Cc1ccc2cc(CN(C(=O)c3cccs3)c3ccccc3)c(O)nc2c1	nan
	CHEMBL1583002	51263	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	4	1	4	5.2	Cc1ccc2cc(CN(C(=O)c3cccs3)c3ccccc3)c(O)nc2c1	nan
	2012958	51310	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	363	5	1	5	4.1	Cc1nc(SCC(=O)NCc2ccccc2)c2oc3ccccc3c2n1	nan
	CHEMBL1583344	51310	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	363	5	1	5	4.1	Cc1nc(SCC(=O)NCc2ccccc2)c2oc3ccccc3c2n1	nan
	2810452	51336	4	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	3	0	6	3.5	Cc1cc(C)c(-n2nnnc2SC2Cc3ccccc3C2=O)c(C)c1	nan
	CHEMBL1583573	51336	4	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	350	3	0	6	3.5	Cc1cc(C)c(-n2nnnc2SC2Cc3ccccc3C2=O)c(C)c1	nan
	4102688	51422	14	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	299	2	1	5	2.6	Cc1cccc(NC(=O)c2cnc3sccn3c2=O)c1C	nan
	CHEMBL1584232	51422	14	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	299	2	1	5	2.6	Cc1cccc(NC(=O)c2cnc3sccn3c2=O)c1C	nan
	15944711	51425	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	5	1	5	3.9	Cc1ccc(NC(=O)Cn2cc(S(=O)(=O)c3ccccc3)c(=O)c3cc(F)ccc32)cc1	nan
	CHEMBL1584268	51425	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	5	1	5	3.9	Cc1ccc(NC(=O)Cn2cc(S(=O)(=O)c3ccccc3)c(=O)c3cc(F)ccc32)cc1	nan
	2981373	51675	15	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	335	2	1	4	4.3	Cc1nc(Nc2cccc(C(F)(F)F)c2)nc2c1C(=O)CC(C)C2	nan
	CHEMBL1586327	51675	15	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	335	2	1	4	4.3	Cc1nc(Nc2cccc(C(F)(F)F)c2)nc2c1C(=O)CC(C)C2	nan
	6404569	51814	13	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	4	0	3	5.4	c1ccc(Cc2nnc(Sc3ccccc3)c3ccccc23)cc1	nan
	CHEMBL1587518	51814	13	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	328	4	0	3	5.4	c1ccc(Cc2nnc(Sc3ccccc3)c3ccccc23)cc1	nan
	16189382	51966	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	2	1	4	5.0	Cc1cccc(N(C)C(=O)c2cc3c(O)nc4ccc(C)cc4c3s2)c1	nan
	CHEMBL1588813	51966	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	2	1	4	5.0	Cc1cccc(N(C)C(=O)c2cc3c(O)nc4ccc(C)cc4c3s2)c1	nan
	5770860	52008	4	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	373	7	2	6	2.4	CCOC(=O)CNC(=O)c1sc(NC(=O)/C=C/c2ccccc2)nc1C	nan
	CHEMBL1589172	52008	4	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	373	7	2	6	2.4	CCOC(=O)CNC(=O)c1sc(NC(=O)/C=C/c2ccccc2)nc1C	nan
	2428876	52011	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	346	4	2	4	2.7	O=C(COc1ccc2ccccc2c1)Nc1cccc2c1C(=O)NC2=O	nan
	CHEMBL1589183	52011	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	346	4	2	4	2.7	O=C(COc1ccc2ccccc2c1)Nc1cccc2c1C(=O)NC2=O	nan
	16007870	52094	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	8	1	4	4.9	Cc1ccc(CCNC(=O)CSCc2nc(-c3ccc(C)cc3)oc2C)cc1	nan
	CHEMBL1589908	52094	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	394	8	1	4	4.9	Cc1ccc(CCNC(=O)CSCc2nc(-c3ccc(C)cc3)oc2C)cc1	nan
	6418319	52111	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	6	1	5	5.7	O=C(CSc1nnc(-c2ccc(Cl)cc2)c(-c2ccc(Cl)cc2)n1)NC1CCCC1	nan
	CHEMBL1590097	52111	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	6	1	5	5.7	O=C(CSc1nnc(-c2ccc(Cl)cc2)c(-c2ccc(Cl)cc2)n1)NC1CCCC1	nan
	16025990	52122	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	3	1	8	2.2	Cc1c(Cl)cccc1NC(=O)c1cnc2sc(N3CCOCC3)nn2c1=O	nan
	CHEMBL1590252	52122	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	405	3	1	8	2.2	Cc1c(Cl)cccc1NC(=O)c1cnc2sc(N3CCOCC3)nn2c1=O	nan
	16030611	52139	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	6	0	5	5.3	COc1cccc(Cc2nc3ccccc3nc2SCC(=O)N2CCCc3ccccc32)c1	nan
	CHEMBL1590504	52139	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	6	0	5	5.3	COc1cccc(Cc2nc3ccccc3nc2SCC(=O)N2CCCc3ccccc32)c1	nan
	16009482	52140	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	6	1	7	3.9	COc1ccccc1C(=O)Nc1ccccc1OCc1cc(=O)n2c(C)csc2n1	nan
	CHEMBL1590536	52140	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	6	1	7	3.9	COc1ccccc1C(=O)Nc1ccccc1OCc1cc(=O)n2c(C)csc2n1	nan
	16015095	52141	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	426	8	1	6	5.5	CCOc1ccccc1NC(=O)c1sc(-n2nc(C)c(CCC(C)C)c2C)nc1C	nan
	CHEMBL1590548	52141	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	426	8	1	6	5.5	CCOc1ccccc1NC(=O)c1sc(-n2nc(C)c(CCC(C)C)c2C)nc1C	nan
	16019575	52149	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	505	5	1	9	4.6	O=S(=O)(c1ccc(Br)cc1)c1nnn2c1nc(NCc1cccs1)c1sccc12	nan
	CHEMBL1590659	52149	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	505	5	1	9	4.6	O=S(=O)(c1ccc(Br)cc1)c1nnn2c1nc(NCc1cccs1)c1sccc12	nan
	4249793	52156	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	296	3	2	4	1.8	COc1ccccc1C(=O)Nc1ccc2c(c1)C(=O)NC2=O	nan
	CHEMBL1590747	52156	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	296	3	2	4	1.8	COc1ccccc1C(=O)Nc1ccc2c(c1)C(=O)NC2=O	nan
	16016850	52164	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	7	2	3	5.9	COc1ccc2c(Sc3ccccc3)c(C(=O)NCC(C)c3ccccc3)[nH]c2c1	nan
	CHEMBL1590842	52164	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	7	2	3	5.9	COc1ccc2c(Sc3ccccc3)c(C(=O)NCC(C)c3ccccc3)[nH]c2c1	nan
	16025801	52198	3	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	7	1	7	2.9	COc1cccc(CNc2nccn(-c3ccc(OC)c(OC)c3)c2=O)c1	nan
	CHEMBL1591265	52198	3	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	7	1	7	2.9	COc1cccc(CNc2nccn(-c3ccc(OC)c(OC)c3)c2=O)c1	nan
	7533419	52237	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	8	1	6	3.5	CCOc1ccc(-c2nnc(SCC(=O)NCc3ccccc3)o2)cc1	nan
	CHEMBL1591699	52237	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	369	8	1	6	3.5	CCOc1ccc(-c2nnc(SCC(=O)NCc3ccccc3)o2)cc1	nan
	16030248	52258	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	5	1	5	3.7	O=C(CSc1nnc(-c2ccccc2Cl)[nH]1)N1CCN(c2ccc(F)cc2)CC1	nan
	CHEMBL1591982	52258	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	5	1	5	3.7	O=C(CSc1nnc(-c2ccccc2Cl)[nH]1)N1CCN(c2ccc(F)cc2)CC1	nan
	16021788	52268	3	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	5	2	7	3.3	O=C(NCc1ccccc1)c1cccc(Nc2nc3ccccc3n3nnnc23)c1	nan
	CHEMBL1592133	52268	3	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	5	2	7	3.3	O=C(NCc1ccccc1)c1cccc(Nc2nc3ccccc3n3nnnc23)c1	nan
	16008534	52307	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	512	9	1	6	5.2	CCOC(=O)C(Cc1ccccc1)NC(=O)CCc1c(C)nc2c(c(C)nn2-c2ccc(C)c(C)c2)c1C	nan
	CHEMBL1592680	52307	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	512	9	1	6	5.2	CCOC(=O)C(Cc1ccccc1)NC(=O)CCc1c(C)nc2c(c(C)nn2-c2ccc(C)c(C)c2)c1C	nan
	16012042	52309	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	488	7	1	5	4.6	O=C(Cn1ncc2c3ccccc3n(Cc3ccccc3F)c2c1=O)NCCc1ccc(Cl)cc1	nan
	CHEMBL1592702	52309	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	488	7	1	5	4.6	O=C(Cn1ncc2c3ccccc3n(Cc3ccccc3F)c2c1=O)NCCc1ccc(Cl)cc1	nan
	15991036	52322	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	4	1	4	6.7	COc1ccc(Cl)cc1C(=O)Nc1ccc2oc(-c3ccc(C(C)(C)C)cc3)nc2c1	nan
	CHEMBL1592855	52322	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	4	1	4	6.7	COc1ccc(Cl)cc1C(=O)Nc1ccc2oc(-c3ccc(C(C)(C)C)cc3)nc2c1	nan
	16026106	52337	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	5	1	5	3.9	CC1=C(c2ccc(C(C)C)cc2)S(=O)(=O)N=C1N1CCC(C(=O)NCc2ccco2)CC1	nan
	CHEMBL1593080	52337	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	5	1	5	3.9	CC1=C(c2ccc(C(C)C)cc2)S(=O)(=O)N=C1N1CCC(C(=O)NCc2ccco2)CC1	nan
	16009361	52340	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	494	7	1	6	4.3	CCOc1ccc(NC(=O)Cn2cc(S(=O)(=O)c3ccc(C)cc3)c(=O)c3cc(F)ccc32)cc1	nan
	CHEMBL1593099	52340	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	494	7	1	6	4.3	CCOc1ccc(NC(=O)Cn2cc(S(=O)(=O)c3ccc(C)cc3)c(=O)c3cc(F)ccc32)cc1	nan
	16030919	52345	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	7	1	6	4.7	CCc1ccc(NC(=O)CSc2ccc3nc(-c4ccc(OC)cc4)cn3n2)cc1	nan
	CHEMBL1593184	52345	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	7	1	6	4.7	CCc1ccc(NC(=O)CSc2ccc3nc(-c4ccc(OC)cc4)cn3n2)cc1	nan
	16033356	52350	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	5	1	4	5.5	COc1ccc(CC(=O)Nc2ccc(-c3nc4ccccc4s3)c(C)c2)cc1	nan
	CHEMBL1593249	52350	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	5	1	4	5.5	COc1ccc(CC(=O)Nc2ccc(-c3nc4ccccc4s3)c(C)c2)cc1	nan
	16015767	52379	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	7	0	5	3.9	Cc1ccc(CN(C(=O)COc2ccccc2[N+](=O)[O-])c2ccccn2)cc1	nan
	CHEMBL1593732	52379	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	7	0	5	3.9	Cc1ccc(CN(C(=O)COc2ccccc2[N+](=O)[O-])c2ccccn2)cc1	nan
	15990880	52384	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	6	2	3	5.6	Cc1ccc(Nc2cc(C(=O)NCCc3ccccc3)c3ccccc3n2)c(C)c1	nan
	CHEMBL1593807	52384	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	395	6	2	3	5.6	Cc1ccc(Nc2cc(C(=O)NCCc3ccccc3)c3ccccc3n2)c(C)c1	nan
	3623411	52396	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	7	1	4	6.0	CCOc1ccc(Sc2cc(C(=O)NCc3ccc(C)cc3)c3ccccc3n2)cc1	nan
	CHEMBL1593971	52396	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	7	1	4	6.0	CCOc1ccc(Sc2cc(C(=O)NCc3ccc(C)cc3)c3ccccc3n2)cc1	nan
	16030473	52467	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	5	1	5	4.5	Cc1ccc2nc(COc3cccc(NC(=O)c4cccc(Cl)c4)c3)cc(=O)n2c1	nan
	CHEMBL1594609	52467	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	5	1	5	4.5	Cc1ccc2nc(COc3cccc(NC(=O)c4cccc(Cl)c4)c3)cc(=O)n2c1	nan
	2328630	52481	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	6	1	6	2.9	CCOC(=O)c1c(C)[nH]c(C(=O)CSc2nccc(C)n2)c1C	nan
	CHEMBL1594696	52481	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	6	1	6	2.9	CCOC(=O)c1c(C)[nH]c(C(=O)CSc2nccc(C)n2)c1C	nan
	16027342	52535	0	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	3	0	4	4.1	Cc1cc(=O)n(Cc2cccc(F)c2)c2c1c(C)nn2-c1cccc(F)c1	nan
	CHEMBL1595156	52535	0	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	365	3	0	4	4.1	Cc1cc(=O)n(Cc2cccc(F)c2)c2c1c(C)nn2-c1cccc(F)c1	nan
	16021494	52542	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	5	1	4	3.9	CSc1ncc(C(=O)NCc2ccc(F)cc2)c(-c2ccccc2)n1	nan
	CHEMBL1595189	52542	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	5	1	4	3.9	CSc1ncc(C(=O)NCc2ccc(F)cc2)c(-c2ccccc2)n1	nan
	4584398	52644	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	318	2	1	2	4.7	Cn1c(C(=O)Nc2ccc(Cl)cc2)cc2cc(Cl)ccc21	nan
	CHEMBL1596148	52644	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	318	2	1	2	4.7	Cn1c(C(=O)Nc2ccc(Cl)cc2)cc2cc(Cl)ccc21	nan
	16016964	52676	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	5	1	4	4.7	Cc1cc(C)c2c(-n3cccc3)c(C(=O)NCCc3ccccc3)sc2n1	nan
	CHEMBL1596415	52676	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	5	1	4	4.7	Cc1cc(C)c2c(-n3cccc3)c(C(=O)NCCc3ccccc3)sc2n1	nan
	891582	52701	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	2	0	5	3.8	Cc1cccc(-n2ncc3c(N4CCc5ccccc54)ncnc32)c1	nan
	CHEMBL1596656	52701	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	327	2	0	5	3.8	Cc1cccc(-n2ncc3c(N4CCc5ccccc54)ncnc32)c1	nan
	2138637	52704	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	5	2	6	3.5	CC(=O)NCCNc1nc2c(-c3cccc(C(F)(F)F)c3)nnn2c2ccccc12	nan
	CHEMBL1596664	52704	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	414	5	2	6	3.5	CC(=O)NCCNc1nc2c(-c3cccc(C(F)(F)F)c3)nnn2c2ccccc12	nan
	4062063	52770	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	8	3	8	-0.4	CN(CCO)S(=O)(=O)c1ccc2c(c1)C(=NN)c1cc(S(=O)(=O)N(C)CCO)ccc1-2	nan
	CHEMBL1597275	52770	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	8	3	8	-0.4	CN(CCO)S(=O)(=O)c1ccc2c(c1)C(=NN)c1cc(S(=O)(=O)N(C)CCO)ccc1-2	nan
	1611638	52863	16	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	7	2	10	3.2	CCOC(=O)Cc1csc(NC(=O)CSc2nc(N)c3c(C)c(C)sc3n2)n1	nan
	CHEMBL1598169	52863	16	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	7	2	10	3.2	CCOC(=O)Cc1csc(NC(=O)CSc2nc(N)c3c(C)c(C)sc3n2)n1	nan
	16010773	52866	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	6	1	7	3.2	COc1ccc(Cn2c(=O)c3cccnc3n(CC(=O)Nc3c(C)cc(C)cc3C)c2=O)cc1	nan
	CHEMBL1598197	52866	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	458	6	1	7	3.2	COc1ccc(Cn2c(=O)c3cccnc3n(CC(=O)Nc3c(C)cc(C)cc3C)c2=O)cc1	nan
	2958808	52868	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	4	2	4	3.7	Cc1nc(NC(=S)NC(=O)COc2ccccc2Cl)ccc1Br	nan
	CHEMBL1598226	52868	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	4	2	4	3.7	Cc1nc(NC(=S)NC(=O)COc2ccccc2Cl)ccc1Br	nan
	921716	52925	10	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	316	2	1	4	4.9	Cc1ccc(O)c(C2=Nc3ccccc3N=C(c3ccco3)C2)c1	nan
	CHEMBL1598745	52925	10	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	316	2	1	4	4.9	Cc1ccc(O)c(C2=Nc3ccccc3N=C(c3ccco3)C2)c1	nan
	3284133	52933	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	534	10	2	6	4.2	CC(C)CN(CC(C)C)S(=O)(=O)c1ccc(C(=O)Nc2sc3c(c2C(N)=O)CCN(C(C)C)C3)cc1	nan
	CHEMBL1598836	52933	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	534	10	2	6	4.2	CC(C)CN(CC(C)C)S(=O)(=O)c1ccc(C(=O)Nc2sc3c(c2C(N)=O)CCN(C(C)C)C3)cc1	nan
	7326265	52984	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	366	6	2	5	3.5	CC(=O)Nc1ccc(C(=O)Nc2nnc(CCc3ccccc3)s2)cc1	nan
	CHEMBL1599247	52984	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	366	6	2	5	3.5	CC(=O)Nc1ccc(C(=O)Nc2nnc(CCc3ccccc3)s2)cc1	nan
	16009345	52999	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	5	0	6	4.0	COc1cccc(OCc2cc(=O)n3c(-c4ccccc4)csc3n2)c1	nan
	CHEMBL1599358	52999	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	364	5	0	6	4.0	COc1cccc(OCc2cc(=O)n3c(-c4ccccc4)csc3n2)c1	nan
	16024944	53038	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	447	5	2	4	4.8	Cc1cccc(N2CCN(c3ccc(C(=O)O)cc3NC(=O)c3ccccc3F)CC2C)c1	nan
	CHEMBL1599731	53038	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	447	5	2	4	4.8	Cc1cccc(N2CCN(c3ccc(C(=O)O)cc3NC(=O)c3ccccc3F)CC2C)c1	nan
	6536107	53083	3	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	5	1	5	5.2	Cc1ccc(-c2csc(/C=C3\SC(C)C(=O)N3CC(=O)Nc3ccccc3F)n2)cc1	nan
	CHEMBL1600183	53083	3	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	5	1	5	5.2	Cc1ccc(-c2csc(/C=C3\SC(C)C(=O)N3CC(=O)Nc3ccccc3F)n2)cc1	nan
	733979	53093	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	300	2	1	4	2.5	CC(=O)c1ccc(NC2=NS(=O)(=O)c3ccccc32)cc1	nan
	CHEMBL1600285	53093	13	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	300	2	1	4	2.5	CC(=O)c1ccc(NC2=NS(=O)(=O)c3ccccc32)cc1	nan
	2999237	53098	4	None	-1	3	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	332	6	1	6	2.8	CCCCn1c(-c2ccsc2)nc2c1c(=O)[nH]c(=O)n2CCC	nan
	CHEMBL1600302	53098	4	None	-1	3	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	332	6	1	6	2.8	CCCCn1c(-c2ccsc2)nc2c1c(=O)[nH]c(=O)n2CCC	nan
	3946061	53140	12	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	4	1	7	3.2	CC1(C)Cc2nc3sc4c(=O)n(CC(=O)NCc5ccccc5)cnc4c3cc2CO1	nan
	CHEMBL1600688	53140	12	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	4	1	7	3.2	CC1(C)Cc2nc3sc4c(=O)n(CC(=O)NCc5ccccc5)cnc4c3cc2CO1	nan
	16019821	53143	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	6	2	6	3.4	CCOc1ccc(NC(=O)C2CCCN(S(=O)(=O)c3ccc4nc(O)ccc4c3)C2)cc1	nan
	CHEMBL1600701	53143	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	6	2	6	3.4	CCOc1ccc(NC(=O)C2CCCN(S(=O)(=O)c3ccc4nc(O)ccc4c3)C2)cc1	nan
	648853	53151	16	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	296	2	1	4	3.2	Cc1ccc(C(=O)Nc2nc3ccccc3c(=O)s2)cc1	nan
	CHEMBL1600749	53151	16	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	296	2	1	4	3.2	Cc1ccc(C(=O)Nc2nc3ccccc3c(=O)s2)cc1	nan
	1326969	53211	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	5	1	4	5.1	Cc1ccc(OCC(=O)Nc2ccc(-c3nc4ccccc4o3)cc2)c(C)c1	nan
	CHEMBL1601297	53211	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	372	5	1	4	5.1	Cc1ccc(OCC(=O)Nc2ccc(-c3nc4ccccc4o3)cc2)c(C)c1	nan
	20949434	53214	1	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	442	4	2	6	1.7	CC(=O)c1ccc(N2CCN(S(=O)(=O)c3ccc4c(c3)NC(=O)CC(=O)N4)CC2)cc1	nan
	CHEMBL1601336	53214	1	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	442	4	2	6	1.7	CC(=O)c1ccc(N2CCN(S(=O)(=O)c3ccc4c(c3)NC(=O)CC(=O)N4)CC2)cc1	nan
	16015783	53225	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	472	6	1	6	6.2	COc1ccc(-c2cc(C(=O)Nc3c(C(=O)c4ccc(Cl)cc4)oc4ccccc34)no2)cc1	nan
	CHEMBL1601476	53225	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	472	6	1	6	6.2	COc1ccc(-c2cc(C(=O)Nc3c(C(=O)c4ccc(Cl)cc4)oc4ccccc34)no2)cc1	nan
	3579351	53264	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	5	0	7	4.2	COc1ccc(-n2c(SCC(=O)C(C)(C)C)nc3ccsc3c2=O)cc1	nan
	CHEMBL1601921	53264	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	5	0	7	4.2	COc1ccc(-n2c(SCC(=O)C(C)(C)C)nc3ccsc3c2=O)cc1	nan
	16034721	53330	3	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	441	5	2	7	4.3	Cc1ccccc1Nc1nn2c(=O)c3ccc(C(=O)NCc4ccccc4)cc3nc2s1	nan
	CHEMBL1602585	53330	3	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	441	5	2	7	4.3	Cc1ccccc1Nc1nn2c(=O)c3ccc(C(=O)NCc4ccccc4)cc3nc2s1	nan
	3938730	53370	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	483	5	2	4	6.4	Cc1cc(C)c2c(NC(=O)c3ccccc3Cl)c(C(=O)NCc3ccc(Cl)cc3)sc2n1	nan
	CHEMBL1602945	53370	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	483	5	2	4	6.4	Cc1cc(C)c2c(NC(=O)c3ccccc3Cl)c(C(=O)NCc3ccc(Cl)cc3)sc2n1	nan
	3343394	53450	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	2	1	6	5.1	CC1(C)Cc2c(sc3c2c(N)nc(=S)n3Cc2ccc(Br)cc2)CO1	nan
	CHEMBL1603651	53450	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	2	1	6	5.1	CC1(C)Cc2c(sc3c2c(N)nc(=S)n3Cc2ccc(Br)cc2)CO1	nan
	5223767	53451	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	5	1	4	3.3	Cc1cc2cc(CNC(=O)Cc3ccc([N+](=O)[O-])cc3)ccc2n1C	nan
	CHEMBL1603656	53451	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	337	5	1	4	3.3	Cc1cc2cc(CNC(=O)Cc3ccc([N+](=O)[O-])cc3)ccc2n1C	nan
	16030948	53468	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	5	1	5	5.1	O=C(CSc1ccc2nc(-c3ccccc3)cn2n1)Nc1ccccc1C(F)(F)F	nan
	CHEMBL1603757	53468	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	5	1	5	5.1	O=C(CSc1ccc2nc(-c3ccccc3)cn2n1)Nc1ccccc1C(F)(F)F	nan
	2791873	53500	12	None	-2	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	5	2	5	3.0	CCOC(=O)c1cnc2ccc(Br)cc2c1NCC(C)O	nan
	CHEMBL1603951	53500	12	None	-2	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	5	2	5	3.0	CCOC(=O)c1cnc2ccc(Br)cc2c1NCC(C)O	nan
	16014801	53612	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	4	1	5	4.1	Cc1cccc(CSc2nc(=O)c3c(n2C)NC(=O)CC3c2cc(F)cc(F)c2)c1	nan
	CHEMBL1605009	53612	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	4	1	5	4.1	Cc1cccc(CSc2nc(=O)c3c(n2C)NC(=O)CC3c2cc(F)cc(F)c2)c1	nan
	135435545	53627	20	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	290	2	2	4	2.3	NC1=C(c2nc3ccccc3[nH]2)C(=O)CN1c1ccccc1	nan
	CHEMBL1605162	53627	20	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	290	2	2	4	2.3	NC1=C(c2nc3ccccc3[nH]2)C(=O)CN1c1ccccc1	nan
	1511904	53642	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	3	1	4	3.8	O=C(O)c1cn(-c2ccc(N3CCCC3)c(F)c2)c2c(F)c(F)c(F)cc2c1=O	nan
	CHEMBL1605292	53642	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	3	1	4	3.8	O=C(O)c1cn(-c2ccc(N3CCCC3)c(F)c2)c2c(F)c(F)c(F)cc2c1=O	nan
	1961588	53719	9	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	3	0	6	4.9	Cn1c2ccccc2c(=O)c2c(=O)n(Cc3ccco3)c(-c3ccc(Cl)cc3Cl)nc21	nan
	CHEMBL1605870	53719	9	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	451	3	0	6	4.9	Cn1c2ccccc2c(=O)c2c(=O)n(Cc3ccco3)c(-c3ccc(Cl)cc3Cl)nc21	nan
	16001902	53734	3	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	4	1	6	3.3	Cc1ccc(NC(=O)C2CCCN(S(=O)(=O)c3cccc4nsnc34)C2)cc1C	nan
	CHEMBL1605982	53734	3	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	4	1	6	3.3	Cc1ccc(NC(=O)C2CCCN(S(=O)(=O)c3cccc4nsnc34)C2)cc1C	nan
	16031132	53822	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	6	2	5	4.5	CN(C)c1ccc(CNC(=O)c2ccccc2NC(=O)c2nsc3ccccc23)cc1	nan
	CHEMBL1606681	53822	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	430	6	2	5	4.5	CN(C)c1ccc(CNC(=O)c2ccccc2NC(=O)c2nsc3ccccc23)cc1	nan
	2931173	53828	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	324	5	2	3	4.9	CCCCn1c(N=C(S)Nc2ccccc2)nc2ccccc21	nan
	CHEMBL1606716	53828	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	324	5	2	3	4.9	CCCCn1c(N=C(S)Nc2ccccc2)nc2ccccc21	nan
	1481761	53944	22	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	348	3	1	5	4.1	COc1ccc(-c2c(C)nc3c(-c4ccc(F)cc4)cnn3c2N)cc1	nan
	CHEMBL1607515	53944	22	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	348	3	1	5	4.1	COc1ccc(-c2c(C)nc3c(-c4ccc(F)cc4)cnn3c2N)cc1	nan
	16030158	53980	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	464	6	1	7	3.2	Cc1nn(CC(=O)NCc2ccc(N(C)C)cc2)c(=O)c2c(C)n(-c3ccc(Cl)cc3)nc12	nan
	CHEMBL1607845	53980	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	464	6	1	7	3.2	Cc1nn(CC(=O)NCc2ccc(N(C)C)cc2)c(=O)c2c(C)n(-c3ccc(Cl)cc3)nc12	nan
	786570	53994	36	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	332	1	1	3	3.8	O=c1c2cc(Br)ccc2[nH]c(=S)n1-c1ccccc1	nan
	CHEMBL1608028	53994	36	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	332	1	1	3	3.8	O=c1c2cc(Br)ccc2[nH]c(=S)n1-c1ccccc1	nan
	744022	54091	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	281	4	1	4	3.8	COCc1cc(C)nc(Nc2ccc(C)c(C)c2)c1C#N	nan
	CHEMBL1608862	54091	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	281	4	1	4	3.8	COCc1cc(C)nc(Nc2ccc(C)c(C)c2)c1C#N	nan
	20868577	54108	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	3	0	5	4.5	CC(=O)c1ccc(N2CCN(C(=O)c3cc4c(C)nc5ccccc5c4o3)CC2)cc1	nan
	CHEMBL1609003	54108	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	413	3	0	5	4.5	CC(=O)c1ccc(N2CCN(C(=O)c3cc4c(C)nc5ccccc5c4o3)CC2)cc1	nan
	16015522	54114	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	6	1	7	3.5	COc1ccc(C(=O)Nc2ccc3nc(SCC(=O)N4CCOCC4)sc3c2)cc1	nan
	CHEMBL1609032	54114	6	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	443	6	1	7	3.5	COc1ccc(C(=O)Nc2ccc3nc(SCC(=O)N4CCOCC4)sc3c2)cc1	nan
	3128209	54202	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	335	4	2	8	1.5	NS(=O)(=O)c1ccc(Nc2ccc([N+](=O)[O-])c3nonc23)cc1	nan
	CHEMBL1609744	54202	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	335	4	2	8	1.5	NS(=O)(=O)c1ccc(Nc2ccc([N+](=O)[O-])c3nonc23)cc1	nan
	16026888	54272	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	5	0	8	3.6	COc1ccccc1C(=O)OCc1cc(=O)n2nc(C3CCCCC3)sc2n1	nan
	CHEMBL1610338	54272	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	5	0	8	3.6	COc1ccccc1C(=O)OCc1cc(=O)n2nc(C3CCCCC3)sc2n1	nan
	16015736	54296	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	7	0	4	3.3	Cc1ccc(C(C)C)c(OCC(=O)N2CCN(CCc3ccncc3)CC2)c1	nan
	CHEMBL1610516	54296	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	7	0	4	3.3	Cc1ccc(C(C)C)c(OCC(=O)N2CCN(CCc3ccncc3)CC2)c1	nan
	2220915	54370	11	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	447	7	1	5	4.9	COc1ccc(CCNC(=O)c2cc(-c3ccccn3)nc3c(Cl)cccc23)cc1OC	nan
	CHEMBL1611237	54370	11	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	447	7	1	5	4.9	COc1ccc(CCNC(=O)c2cc(-c3ccccn3)nc3c(Cl)cccc23)cc1OC	nan
	16030297	54398	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	441	6	0	5	4.9	COc1ccccc1Cc1nc2ccccc2nc1SCC(=O)N1CCc2ccccc21	nan
	CHEMBL1611407	54398	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	441	6	0	5	4.9	COc1ccccc1Cc1nc2ccccc2nc1SCC(=O)N1CCc2ccccc21	nan
	903550	54442	18	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	266	4	1	5	2.5	CCOC(=O)c1sc(NC(=O)CC)c(C#N)c1C	nan
	CHEMBL1611829	54442	18	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	266	4	1	5	2.5	CCOC(=O)c1sc(NC(=O)CC)c(C#N)c1C	nan
	2804057	54470	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	206	0	2	2	3.1	Cc1c(C)c(C)c2[nH]c(S)nc2c1C	nan
	CHEMBL1612138	54470	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	206	0	2	2	3.1	Cc1c(C)c(C)c2[nH]c(S)nc2c1C	nan
	16019436	54537	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	8	1	7	3.6	Cc1ccc(C)c(CSc2ccc3nnc(CCNS(=O)(=O)c4ccccc4)n3n2)c1	nan
	CHEMBL1612674	54537	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	8	1	7	3.6	Cc1ccc(C)c(CSc2ccc3nnc(CCNS(=O)(=O)c4ccccc4)n3n2)c1	nan
	4152434	54551	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	5	1	5	5.7	CC(C)c1ccc(NC(=O)CSc2ncnc3c2sc2ccccc23)cc1	nan
	CHEMBL1612783	54551	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	393	5	1	5	5.7	CC(C)c1ccc(NC(=O)CSc2ncnc3c2sc2ccccc23)cc1	nan
	16034221	54587	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	498	8	1	7	1.1	CCOC(=O)N1CCN(S(=O)(=O)N2CCCC(C(=O)NCc3cc(OC)ccc3OC)C2)CC1	nan
	CHEMBL1613162	54587	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	498	8	1	7	1.1	CCOC(=O)N1CCN(S(=O)(=O)N2CCCC(C(=O)NCc3cc(OC)ccc3OC)C2)CC1	nan
	3238969	54591	2	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	3	1	4	5.6	O=C(Nc1ccc2oc(-c3ccccc3Cl)nc2c1)c1cncc(Br)c1	nan
	CHEMBL1613230	54591	2	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	3	1	4	5.6	O=C(Nc1ccc2oc(-c3ccccc3Cl)nc2c1)c1cncc(Br)c1	nan
	16033448	54602	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	3	1	4	4.8	Cc1cc(C)c(NC(=O)c2nc3ccccc3nc2N2CCCCC2)c(C)c1	nan
	CHEMBL1613324	54602	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	374	3	1	4	4.8	Cc1cc(C)c(NC(=O)c2nc3ccccc3nc2N2CCCCC2)c(C)c1	nan
	2138172	54607	16	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	332	6	1	6	3.1	C=CCOC(=O)c1sc(NC(=O)c2ccc(OC)cc2)nc1C	nan
	CHEMBL1613374	54607	16	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	332	6	1	6	3.1	C=CCOC(=O)c1sc(NC(=O)c2ccc(OC)cc2)nc1C	nan
	17585635	54886	5	None	-11	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	283	2	0	1	3.8	Cn1cc(/C=C/c2cc[n+](C)cc2)c2cc(Cl)ccc21	nan
	73401607	54886	5	None	-11	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	283	2	0	1	3.8	Cn1cc(/C=C/c2cc[n+](C)cc2)c2cc(Cl)ccc21	nan
	CHEMBL1311226	54886	5	None	-11	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	283	2	0	1	3.8	Cn1cc(/C=C/c2cc[n+](C)cc2)c2cc(Cl)ccc21	nan
	CHEMBL1617414	54886	5	None	-11	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	283	2	0	1	3.8	Cn1cc(/C=C/c2cc[n+](C)cc2)c2cc(Cl)ccc21	nan
	424003	55022	28	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	202	1	1	2	1.8	NCc1cc2c3c(c1)CCCN3CCC2	nan
	CHEMBL1359356	55022	28	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	202	1	1	2	1.8	NCc1cc2c3c(c1)CCCN3CCC2	nan
	CHEMBL1618556	55022	28	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	202	1	1	2	1.8	NCc1cc2c3c(c1)CCCN3CCC2	nan
	719481	55032	14	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	316	3	1	4	4.5	COc1ccc(-n2cc(-c3ccc(Cl)cc3)nc2S)cc1	nan
	CHEMBL1379055	55032	14	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	316	3	1	4	4.5	COc1ccc(-n2cc(-c3ccc(Cl)cc3)nc2S)cc1	nan
	CHEMBL1618658	55032	14	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	316	3	1	4	4.5	COc1ccc(-n2cc(-c3ccc(Cl)cc3)nc2S)cc1	nan
	1453026	55379	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	8	2	7	3.6	COc1ccc(C(=O)Nc2ccc(NC(=O)c3cc(OC)c(OC)c(OC)c3)cn2)cc1	nan
	CHEMBL1442637	55379	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	8	2	7	3.6	COc1ccc(C(=O)Nc2ccc(NC(=O)c3cc(OC)c(OC)c(OC)c3)cn2)cc1	nan
	CHEMBL1621750	55379	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	8	2	7	3.6	COc1ccc(C(=O)Nc2ccc(NC(=O)c3cc(OC)c(OC)c(OC)c3)cn2)cc1	nan
	5044272	55627	5	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	9	1	7	4.8	CCN(CC)CCn1c(SCC(=O)Nc2ccc(F)cc2)nc2c(sc3ccccc32)c1=O	nan
	CHEMBL1524152	55627	5	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	9	1	7	4.8	CCN(CC)CCn1c(SCC(=O)Nc2ccc(F)cc2)nc2c(sc3ccccc32)c1=O	nan
	CHEMBL1623691	55627	5	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	484	9	1	7	4.8	CCN(CC)CCn1c(SCC(=O)Nc2ccc(F)cc2)nc2c(sc3ccccc32)c1=O	nan
	3149296	55659	6	None	-2	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	2	0	3	6.1	CCN1/C(=C/c2ccc3cc(C)ccc3[n+]2C)Sc2ccc3sccc3c21	nan
	5768586	55659	6	None	-2	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	2	0	3	6.1	CCN1/C(=C/c2ccc3cc(C)ccc3[n+]2C)Sc2ccc3sccc3c21	nan
	CHEMBL1508982	55659	6	None	-2	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	2	0	3	6.1	CCN1/C(=C/c2ccc3cc(C)ccc3[n+]2C)Sc2ccc3sccc3c21	nan
	CHEMBL1623968	55659	6	None	-2	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	389	2	0	3	6.1	CCN1/C(=C/c2ccc3cc(C)ccc3[n+]2C)Sc2ccc3sccc3c21	nan
	1956404	55684	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	5	1	7	3.5	COCCN1CCn2c(nc3cc(Nc4nnc(C)c5ccccc45)ccc32)C1	nan
	CHEMBL1556245	55684	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	5	1	7	3.5	COCCN1CCn2c(nc3cc(Nc4nnc(C)c5ccccc45)ccc32)C1	nan
	CHEMBL1624228	55684	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	5	1	7	3.5	COCCN1CCn2c(nc3cc(Nc4nnc(C)c5ccccc45)ccc32)C1	nan
	3602384	55818	1	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	5	1	3	4.5	Cc1ccc(CNC(=O)c2cc3c(s2)CN(Cc2ccccc2)C3)cc1	nan
	CHEMBL1602214	55818	1	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	5	1	3	4.5	Cc1ccc(CNC(=O)c2cc3c(s2)CN(Cc2ccccc2)C3)cc1	nan
	CHEMBL1625426	55818	1	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	5	1	3	4.5	Cc1ccc(CNC(=O)c2cc3c(s2)CN(Cc2ccccc2)C3)cc1	nan
	2151347	71637	10	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	316	2	0	4	3.3	C#CCn1/c(=N/C(=O)c2ccco2)sc2cccc(Cl)c21	nan
	CHEMBL1973713	71637	10	None	-3	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	316	2	0	4	3.3	C#CCn1/c(=N/C(=O)c2ccco2)sc2cccc(Cl)c21	nan
	741794	71943	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	304	1	1	4	3.1	Cc1c(C(C)(C)C)s/c(=N/C(=O)c2ccccc2O)n1C	nan
	CHEMBL1983034	71943	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	304	1	1	4	3.1	Cc1c(C(C)(C)C)s/c(=N/C(=O)c2ccccc2O)n1C	nan
	9583974	72204	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	6	2	7	5.1	COc1cccc(/C=N/NC(=O)c2oc3nc(-c4ccccc4)cc(-c4ccco4)c3c2N)c1	nan
	CHEMBL1991618	72204	2	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	6	2	7	5.1	COc1cccc(/C=N/NC(=O)c2oc3nc(-c4ccccc4)cc(-c4ccco4)c3c2N)c1	nan
	135498048	72287	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	246	3	2	6	0.8	Cc1nonc1C(=O)N/N=C/c1ccc(O)cc1	nan
	CHEMBL1994596	72287	7	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	246	3	2	6	0.8	Cc1nonc1C(=O)N/N=C/c1ccc(O)cc1	nan
	1362920	95326	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	6	1	5	5.1	COc1ccc(OCC(=O)Nc2ccc(-c3nc4cc(C)cc(C)c4o3)cc2)cc1	nan
	CHEMBL258549	95326	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	6	1	5	5.1	COc1ccc(OCC(=O)Nc2ccc(-c3nc4cc(C)cc(C)c4o3)cc2)cc1	nan
	2150885	107131	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	334	3	0	5	3.3	COc1ccc(OC)c2c1s/c(=N\C(=O)C1CCCCC1)n2C	nan
	CHEMBL3189890	107131	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	334	3	0	5	3.3	COc1ccc(OC)c2c1s/c(=N\C(=O)C1CCCCC1)n2C	nan
	3604296	107293	13	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	5	0	7	2.1	CCOC(=O)Cn1/c(=N/C(=O)CSC(C)=O)sc2cc(F)ccc21	nan
	CHEMBL3191753	107293	13	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	5	0	7	2.1	CCOC(=O)Cn1/c(=N/C(=O)CSC(C)=O)sc2cc(F)ccc21	nan
	1389664	107489	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	7	0	8	3.2	COc1cc(/C=c2\sc3nc(=O)c(-c4ccccc4)nn3c2=O)ccc1OCCC(C)C	nan
	CHEMBL3193918	107489	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	7	0	8	3.2	COc1cc(/C=c2\sc3nc(=O)c(-c4ccccc4)nn3c2=O)ccc1OCCC(C)C	nan
	2321009	107563	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	288	1	0	4	3.4	Cc1ccc2c(c1)s/c(=N/C(=O)c1cccs1)n2C	nan
	CHEMBL3194826	107563	8	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	288	1	0	4	3.4	Cc1ccc2c(c1)s/c(=N/C(=O)c1cccs1)n2C	nan
	3245289	107568	11	None	-31	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	6	0	8	2.0	CCOC(=O)Cn1/c(=N/C(=O)CSC(C)=O)sc2cc(OC)ccc21	nan
	CHEMBL3194890	107568	11	None	-31	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	6	0	8	2.0	CCOC(=O)Cn1/c(=N/C(=O)CSC(C)=O)sc2cc(OC)ccc21	nan
	4668650	107840	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	5	1	8	1.5	COCCn1/c(=N/C(=O)c2ccc3c(c2)OCCO3)sc2cc(S(N)(=O)=O)ccc21	nan
	CHEMBL3197833	107840	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	5	1	8	1.5	COCCn1/c(=N/C(=O)c2ccc3c(c2)OCCO3)sc2cc(S(N)(=O)=O)ccc21	nan
	2150918	107895	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	3	0	6	3.0	COc1ccc(C)c2s/c(=N\C(=O)c3cccc(N4C(=O)CCC4=O)c3)n(C)c12	nan
	CHEMBL3198311	107895	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	409	3	0	6	3.0	COc1ccc(C)c2s/c(=N\C(=O)c3cccc(N4C(=O)CCC4=O)c3)n(C)c12	nan
	135460447	107908	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	263	3	3	6	1.9	Nc1c(Cl)ncnc1N/N=C/c1ccc(O)cc1	nan
	CHEMBL3198494	107908	5	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	263	3	3	6	1.9	Nc1c(Cl)ncnc1N/N=C/c1ccc(O)cc1	nan
	6184027	108186	1	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	497	12	1	9	0.8	COCCCn1c(=O)/c(=C\c2ccc(OC(F)F)c(OC)c2)s/c1=C(/C#N)C(=O)NCCOC	nan
	CHEMBL3207685	108186	1	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	497	12	1	9	0.8	COCCCn1c(=O)/c(=C\c2ccc(OC(F)F)c(OC)c2)s/c1=C(/C#N)C(=O)NCCOC	nan
	2150849	108218	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	5	0	7	3.3	COc1cc(C(=O)/N=c2\sc3c(C)ccc(OC)c3n2C)cc(OC)c1OC	nan
	CHEMBL3208227	108218	9	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	5	0	7	3.3	COc1cc(C(=O)/N=c2\sc3c(C)ccc(OC)c3n2C)cc(OC)c1OC	nan
	5122885	108347	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	3	0	5	3.1	CCOC(=O)c1s/c(=N\C(=O)c2ccccc2Br)n(C)c1C	nan
	CHEMBL3209816	108347	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	3	0	5	3.1	CCOC(=O)c1s/c(=N\C(=O)c2ccccc2Br)n(C)c1C	nan
	9631393	108440	5	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	3	1	4	3.2	O=C(N/N=C/c1ccc2nccnc2c1)c1ccc(Br)cc1	nan
	CHEMBL3211205	108440	5	None	-1	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	3	1	4	3.2	O=C(N/N=C/c1ccc2nccnc2c1)c1ccc(Br)cc1	nan
	4128025	108454	14	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	3	0	6	2.4	COc1cccc(C(=O)/N=c2\sc3cc(S(C)(=O)=O)ccc3n2C)c1	nan
	CHEMBL3211378	108454	14	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	3	0	6	2.4	COc1cccc(C(=O)/N=c2\sc3cc(S(C)(=O)=O)ccc3n2C)c1	nan
	7161820	108474	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	320	4	0	5	2.7	CCOC(=O)Cn1/c(=N/C(=O)CC)sc2c(C)cc(C)cc21	nan
	CHEMBL3211674	108474	10	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	320	4	0	5	2.7	CCOC(=O)Cn1/c(=N/C(=O)CC)sc2c(C)cc(C)cc21	nan
	2150987	108684	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	294	4	0	5	2.5	CCCC(=O)/N=c1\sc2c(OC)ccc(OC)c2n1C	nan
	CHEMBL3214516	108684	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	294	4	0	5	2.5	CCCC(=O)/N=c1\sc2c(OC)ccc(OC)c2n1C	nan
	3213263	112114	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	5	0	7	3.1	COCC/N=C1\Sc2nc3cc4c(cc3cc2CN1CC1CCCO1)OCO4	nan
	CHEMBL3197118	112114	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	5	0	7	3.1	COCC/N=C1\Sc2nc3cc4c(cc3cc2CN1CC1CCCO1)OCO4	nan
	CHEMBL3302243	112114	4	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	401	5	0	7	3.1	COCC/N=C1\Sc2nc3cc4c(cc3cc2CN1CC1CCCO1)OCO4	nan
	6540428	184281	1	None	-37	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	4	2	4	1.9	CCC(CO)NC(=O)[C@@H]1C=C2c3cccc4c3c(cn4C)C[C@H]2N(C)C1	nan
	CHEMBL3989558	184281	1	None	-37	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	4	2	4	1.9	CCC(CO)NC(=O)[C@@H]1C=C2c3cccc4c3c(cn4C)C[C@H]2N(C)C1	nan
	CHEMBL485253	184281	1	None	-37	2	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	4	2	4	1.9	CCC(CO)NC(=O)[C@@H]1C=C2c3cccc4c3c(cn4C)C[C@H]2N(C)C1	nan
	846186	192769	24	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	263	1	3	3	3.0	Cc1nc2ccc(-c3nc4cc(N)ccc4[nH]3)cc2[nH]1	nan
	CHEMBL525103	192769	24	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	263	1	3	3	3.0	Cc1nc2ccc(-c3nc4cc(N)ccc4[nH]3)cc2[nH]1	nan
	2850154	196219	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	204	1	2	1	2.1	CC1=CC(c2ccccc2)NC(=S)N1	nan
	CHEMBL572806	196219	12	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	204	1	2	1	2.1	CC1=CC(c2ccccc2)NC(=S)N1	nan
	138884	198319	15	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	6	2	4	4.2	COc1cccc(NC(=O)c2cccc(C(=O)Nc3cccc(OC)c3)c2)c1	nan
	CHEMBL595273	198319	15	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	6	2	4	4.2	COc1cccc(NC(=O)c2cccc(C(=O)Nc3cccc(OC)c3)c2)c1	nan
	16020583	200691	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	3	0	5	4.2	Cn1cc(S(=O)(=O)c2cccc(Cl)c2)c(=O)c2cc(F)c(N3CCCCC3)cc21	nan
	CHEMBL610622	200691	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	434	3	0	5	4.2	Cn1cc(S(=O)(=O)c2cccc(Cl)c2)c(=O)c2cc(F)c(N3CCCCC3)cc21	nan
	1361408	21197	8	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	3	1	4	6.1	O=C(Nc1ccc(-c2nc3cc(Cl)ccc3o2)cc1)c1cc2ccccc2o1	nan
	CHEMBL1314585	21197	8	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	3	1	4	6.1	O=C(Nc1ccc(-c2nc3cc(Cl)ccc3o2)cc1)c1cc2ccccc2o1	nan
	1369231	21322	7	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	5	2	5	5.5	O=C(COc1ccc(Cl)cc1)Nc1ccc(-c2nc3cc(Cl)ccc3o2)c(O)c1	nan
	CHEMBL1316173	21322	7	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	5	2	5	5.5	O=C(COc1ccc(Cl)cc1)Nc1ccc(-c2nc3cc(Cl)ccc3o2)c(O)c1	nan
	16033420	21717	3	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	3	1	5	2.4	CC(=O)c1ccc(NC(=O)c2nc3ccccc3n(C)c2=O)cc1	nan
	CHEMBL1320318	21717	3	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	321	3	1	5	2.4	CC(=O)c1ccc(NC(=O)c2nc3ccccc3n(C)c2=O)cc1	nan
	16019599	22208	12	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	4	1	8	4.5	Cc1ccc(Nc2nc3c(S(=O)(=O)c4ccccc4)nnn3c3ccsc23)c(C)c1	nan
	CHEMBL1324615	22208	12	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	4	1	8	4.5	Cc1ccc(Nc2nc3c(S(=O)(=O)c4ccccc4)nnn3c3ccsc23)c(C)c1	nan
	16033879	22277	6	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	366	4	1	8	3.2	CCOC(=O)c1ccc(Nc2nn3c(=O)c4ccccc4nc3s2)cc1	nan
	CHEMBL1325210	22277	6	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	366	4	1	8	3.2	CCOC(=O)c1ccc(Nc2nn3c(=O)c4ccccc4nc3s2)cc1	nan
	1115824	23002	14	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	5	1	5	6.1	N#Cc1c(C(F)(F)F)cc(-c2cccs2)nc1SCC(=O)Nc1ccc(Cl)cc1	nan
	CHEMBL1331382	23002	14	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	5	1	5	6.1	N#Cc1c(C(F)(F)F)cc(-c2cccs2)nc1SCC(=O)Nc1ccc(Cl)cc1	nan
	460749	23346	9	None	-11	6	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	303	1	0	7	0.7	Cn1nc(-c2ccc(Cl)cc2)nc2c(=O)n(C)c(=O)nc1-2	nan
	CHEMBL1334062	23346	9	None	-11	6	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	303	1	0	7	0.7	Cn1nc(-c2ccc(Cl)cc2)nc2c(=O)n(C)c(=O)nc1-2	nan
	16746586	24329	0	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	5	3	8	0.2	CCCN=C1C(=O)C2=C(C(O)=C1C)N1CC3NC3[C@@]1(OC)C2COC(N)=O	nan
	CHEMBL1342436	24329	0	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	5	3	8	0.2	CCCN=C1C(=O)C2=C(C(O)=C1C)N1CC3NC3[C@@]1(OC)C2COC(N)=O	nan
	2128809	26838	7	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	317	5	1	6	3.2	Cc1cc(C)c(C(=O)CSc2nnc(O)n2C2CC2)cc1C	nan
	CHEMBL1365084	26838	7	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	317	5	1	6	3.2	Cc1cc(C)c(C(=O)CSc2nnc(O)n2C2CC2)cc1C	nan
	15988395	26966	12	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	344	2	2	3	3.4	CC1(C)CC(=O)c2cc(C(=O)Nc3ccc(Cl)cc3)c(=O)[nH]c2C1	nan
	CHEMBL1366158	26966	12	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	344	2	2	3	3.4	CC1(C)CC(=O)c2cc(C(=O)Nc3ccc(Cl)cc3)c(=O)[nH]c2C1	nan
	2168191	27870	14	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	4	1	5	5.8	Cc1sc(NC(=O)C2c3ccccc3Oc3ccccc32)c(C(=O)OC(C)C)c1C	nan
	CHEMBL1372901	27870	14	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	421	4	1	5	5.8	Cc1sc(NC(=O)C2c3ccccc3Oc3ccccc32)c(C(=O)OC(C)C)c1C	nan
	4578108	28882	8	None	1	2	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	2	2	5	2.4	O=C(Nc1ccc2c(c1)C(=O)NC2=O)c1ccc2ncsc2c1	nan
	CHEMBL1381180	28882	8	None	1	2	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	323	2	2	5	2.4	O=C(Nc1ccc2c(c1)C(=O)NC2=O)c1ccc2ncsc2c1	nan
	15988012	29789	6	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	6	1	8	2.6	COc1ccccc1NC(=O)CCCc1nnc2n(C)c(=O)c3sccc3n12	nan
	CHEMBL1388847	29789	6	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	397	6	1	8	2.6	COc1ccccc1NC(=O)CCCc1nnc2n(C)c(=O)c3sccc3n12	nan
	16024702	32084	5	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	493	9	1	7	4.3	COCCn1c(SCC(=O)c2ccc(C)cc2C)nc2cc(C(=O)NC3CCCC3)ccc2c1=O	nan
	CHEMBL1410231	32084	5	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	493	9	1	7	4.3	COCCn1c(SCC(=O)c2ccc(C)cc2C)nc2cc(C(=O)NC3CCCC3)ccc2c1=O	nan
	16025307	32975	5	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	566	8	1	7	4.9	COc1ccccc1CNC(=O)CSc1ncc2c(n1)-c1ccc(Cl)cc1N(Cc1ccccc1)S2(=O)=O	nan
	CHEMBL1417794	32975	5	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	566	8	1	7	4.9	COc1ccccc1CNC(=O)CSc1ncc2c(n1)-c1ccc(Cl)cc1N(Cc1ccccc1)S2(=O)=O	nan
	4658659	35151	11	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	400	5	0	5	4.9	CCOC(=O)CSc1nc(-c2ccc(Cl)cc2)cc(C(F)(F)F)c1C#N	nan
	CHEMBL1437587	35151	11	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	400	5	0	5	4.9	CCOC(=O)CSc1nc(-c2ccc(Cl)cc2)cc(C(F)(F)F)c1C#N	nan
	16018194	40379	6	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	6	1	4	4.1	O=C(CCCn1c(=O)c2cccn2c2ccccc21)NCc1ccccc1Br	nan
	CHEMBL1483956	40379	6	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	437	6	1	4	4.1	O=C(CCCn1c(=O)c2cccn2c2ccccc21)NCc1ccccc1Br	nan
	1046621	40453	11	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	3	1	6	5.4	Cc1c(Cl)cccc1NC(=O)c1cc2nc(-c3ccc4c(c3)OCO4)cc(C(F)(F)F)n2n1	nan
	CHEMBL1484483	40453	11	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	3	1	6	5.4	Cc1c(Cl)cccc1NC(=O)c1cc2nc(-c3ccc4c(c3)OCO4)cc(C(F)(F)F)n2n1	nan
	16025305	43871	5	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	566	8	1	7	4.9	COc1ccc(CNC(=O)CSc2ncc3c(n2)-c2ccc(Cl)cc2N(Cc2ccccc2)S3(=O)=O)cc1	nan
	CHEMBL1515325	43871	5	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	566	8	1	7	4.9	COc1ccc(CNC(=O)CSc2ncc3c(n2)-c2ccc(Cl)cc2N(Cc2ccccc2)S3(=O)=O)cc1	nan
	2119988	44354	14	None	2	2	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	4	1	6	4.7	CCOC(=O)c1sc2nc(Cc3ccc(Cl)cc3)nc(S)c2c1C	nan
	CHEMBL1520325	44354	14	None	2	2	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	4	1	6	4.7	CCOC(=O)c1sc2nc(Cc3ccc(Cl)cc3)nc(S)c2c1C	nan
	3368526	46934	16	None	2	2	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	4	1	6	3.9	Cc1ccc(C(=O)C2=C(O)C(=O)N(c3ncccn3)C2c2ccc(Br)cc2)o1	nan
	CHEMBL1543365	46934	16	None	2	2	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	4	1	6	3.9	Cc1ccc(C(=O)C2=C(O)C(=O)N(c3ncccn3)C2c2ccc(Br)cc2)o1	nan
	16020714	52095	10	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	7	0	6	3.8	CCN(CC)c1cc2c(cc1F)c(=O)c(S(=O)(=O)c1ccc(OC)cc1)cn2CC	nan
	CHEMBL1589919	52095	10	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	432	7	0	6	3.8	CCN(CC)c1cc2c(cc1F)c(=O)c(S(=O)(=O)c1ccc(OC)cc1)cn2CC	nan
	1164393	52113	10	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	398	7	2	6	2.9	CCOc1ccccc1C(=O)Nc1ccc(S(=O)(=O)Nc2ncccn2)cc1	nan
	CHEMBL1590134	52113	10	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	398	7	2	6	2.9	CCOc1ccccc1C(=O)Nc1ccc(S(=O)(=O)Nc2ncccn2)cc1	nan
	2254266	107588	11	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	423	5	0	6	4.7	C=CCN1C(=O)/C(=C2/Sc3ccc(OC)cc3N2C)S/C1=N\Cc1ccccc1	nan
	CHEMBL3195210	107588	11	None	-	1	Human	5.4	pPotency	=	5.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	423	5	0	6	4.7	C=CCN1C(=O)/C(=C2/Sc3ccc(OC)cc3N2C)S/C1=N\Cc1ccccc1	nan
	7424526	40162	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	5	2	7	0.0	COCCNC(=O)C(=O)Nc1c2c(nn1-c1ccccc1)CS(=O)(=O)C2	nan
	CHEMBL1482031	40162	11	None	-	1	Human	4.4	pPotency	=	4.4	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	378	5	2	7	0.0	COCCNC(=O)C(=O)Nc1c2c(nn1-c1ccccc1)CS(=O)(=O)C2	nan
	4890321	19508	8	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	2	2	6	3.7	Cc1ccc(NC2=NC(c3ccc(F)cc3)n3c(nc(C)cc3=O)N2)c(C)c1	nan
	CHEMBL1300954	19508	8	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	377	2	2	6	3.7	Cc1ccc(NC2=NC(c3ccc(F)cc3)n3c(nc(C)cc3=O)N2)c(C)c1	nan
	7119211	21272	12	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	6	1	4	4.6	COc1ccc(-c2nc(CCNC(=O)c3c(F)cccc3Cl)cs2)cc1	nan
	CHEMBL1315624	21272	12	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	6	1	4	4.6	COc1ccc(-c2nc(CCNC(=O)c3c(F)cccc3Cl)cs2)cc1	nan
	16028928	21399	4	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	6	2	6	3.0	COC(=O)c1ccc(NC(=O)C(=O)NCCc2csc(-c3ccc(F)cc3)n2)cc1	nan
	CHEMBL1317331	21399	4	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	6	2	6	3.0	COC(=O)c1ccc(NC(=O)C(=O)NCCc2csc(-c3ccc(F)cc3)n2)cc1	nan
	16009640	21977	9	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	485	7	1	7	4.5	CCOc1ccc(NC(=O)Cn2c(=O)n(Cc3ccccc3)c(=O)c3sc4ccccc4c32)cc1	nan
	CHEMBL1322592	21977	9	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	485	7	1	7	4.5	CCOc1ccc(NC(=O)Cn2c(=O)n(Cc3ccccc3)c(=O)c3sc4ccccc4c32)cc1	nan
	15988993	22211	6	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	5	1	4	5.7	COc1ccc(CNC(=O)c2cc(-c3ccc(Br)s3)nc3ccccc23)cc1	nan
	CHEMBL1324637	22211	6	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	452	5	1	4	5.7	COc1ccc(CNC(=O)c2cc(-c3ccc(Br)s3)nc3ccccc23)cc1	nan
	682221	25179	17	None	1	2	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	244	4	3	8	0.2	CC(C)OC(=O)CNc1nnc(S)nc1O	nan
	CHEMBL1349621	25179	17	None	1	2	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	244	4	3	8	0.2	CC(C)OC(=O)CNc1nnc(S)nc1O	nan
	16009655	25875	9	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	5	1	6	4.4	Cc1ccc(NC(=O)Cn2c(=O)n(Cc3ccccc3)c(=O)c3sc4ccccc4c32)cc1	nan
	CHEMBL1355671	25875	9	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	5	1	6	4.4	Cc1ccc(NC(=O)Cn2c(=O)n(Cc3ccccc3)c(=O)c3sc4ccccc4c32)cc1	nan
	16019300	27011	12	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	501	6	1	10	4.6	COc1cc(Nc2nc3c(S(=O)(=O)c4cccc(Cl)c4)nnn3c3ccsc23)cc(OC)c1	nan
	CHEMBL1366490	27011	12	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	501	6	1	10	4.6	COc1cc(Nc2nc3c(S(=O)(=O)c4cccc(Cl)c4)nnn3c3ccsc23)cc(OC)c1	nan
	16024750	29026	5	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	436	4	0	5	3.7	O=S(=O)(c1ccc2nc(N3CCN(c4ccccc4)CC3)ccc2c1)N1CCCCC1	nan
	CHEMBL1382499	29026	5	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	436	4	0	5	3.7	O=S(=O)(c1ccc2nc(N3CCN(c4ccccc4)CC3)ccc2c1)N1CCCCC1	nan
	5302633	30744	12	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	493	6	2	5	6.6	CCc1ccc(NC(=O)c2sc3nc(C)c(Cl)c(C)c3c2NC(=O)c2ccccc2OC)cc1	nan
	CHEMBL1398493	30744	12	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	493	6	2	5	6.6	CCc1ccc(NC(=O)c2sc3nc(C)c(Cl)c(C)c3c2NC(=O)c2ccccc2OC)cc1	nan
	16009653	35400	5	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	6	2	4	5.2	Cc1ccccc1OCC(=O)Nc1c(C(=O)Nc2ccccc2F)oc2ccccc12	nan
	CHEMBL1439712	35400	5	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	418	6	2	4	5.2	Cc1ccccc1OCC(=O)Nc1c(C(=O)Nc2ccccc2F)oc2ccccc12	nan
	3522635	38782	7	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	498	7	1	7	2.8	CCN(CC)S(=O)(=O)c1ccc(N2CCN(C)CC2)c(NC(=O)c2cc(=O)c3ccccc3o2)c1	nan
	CHEMBL1468421	38782	7	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	498	7	1	7	2.8	CCN(CC)S(=O)(=O)c1ccc(N2CCN(C)CC2)c(NC(=O)c2cc(=O)c3ccccc3o2)c1	nan
	16018176	39770	5	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	461	6	1	5	5.2	COc1ccc(CNC(=O)c2oc3c(c2C)-c2nn(Cc4ccc(Cl)cc4)cc2CC3)cc1	nan
	CHEMBL1478735	39770	5	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	461	6	1	5	5.2	COc1ccc(CNC(=O)c2oc3c(c2C)-c2nn(Cc4ccc(Cl)cc4)cc2CC3)cc1	nan
	3432810	39927	10	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	3	2	4	5.7	O=C(Nc1ccc(-c2nc3ccccc3s2)c(O)c1)c1ccc(Br)cc1	nan
	CHEMBL1479998	39927	10	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	424	3	2	4	5.7	O=C(Nc1ccc(-c2nc3ccccc3s2)c(O)c1)c1ccc(Br)cc1	nan
	1234246	41106	10	None	-1	2	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	270	1	1	5	3.0	Cc1ccc(-n2nc3c(S)nnc(C)c3c2C)cc1	nan
	CHEMBL1489869	41106	10	None	-1	2	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	270	1	1	5	3.0	Cc1ccc(-n2nc3c(S)nnc(C)c3c2C)cc1	nan
	6800739	44302	3	None	1	2	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	5	1	4	4.6	CCc1ccc2n(-c3ccc(OC)cc3)c([S-])c(C(=O)Nc3cc(C)cc(C)c3)[n+]2c1	nan
	CHEMBL1519802	44302	3	None	1	2	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	431	5	1	4	4.6	CCc1ccc2n(-c3ccc(OC)cc3)c([S-])c(C(=O)Nc3cc(C)cc(C)c3)[n+]2c1	nan
	1744296	48127	22	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	6	1	4	6.7	N#Cc1c(-c2ccccc2)cc(-c2ccccc2)nc1SCC(=O)Nc1ccc(Cl)cc1	nan
	CHEMBL1555056	48127	22	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	455	6	1	4	6.7	N#Cc1c(-c2ccccc2)cc(-c2ccccc2)nc1SCC(=O)Nc1ccc(Cl)cc1	nan
	15988419	52265	6	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	2	2	3	3.5	CC1(C)CC(=O)c2cc(C(=O)Nc3ccc(Br)cc3)c(=O)[nH]c2C1	nan
	CHEMBL1592108	52265	6	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	388	2	2	3	3.5	CC1(C)CC(=O)c2cc(C(=O)Nc3ccc(Br)cc3)c(=O)[nH]c2C1	nan
	1863779	71890	15	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	5	2	8	2.4	CC1=CC=CN2C(=O)C(=C\c3sc(S)nc3O)/C(=N/CCCN3CCOCC3)N=C12	nan
	CHEMBL1981539	71890	15	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	445	5	2	8	2.4	CC1=CC=CN2C(=O)C(=C\c3sc(S)nc3O)/C(=N/CCCN3CCOCC3)N=C12	nan
	755656	172121	46	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	2	1	3	4.4	O=C(O)c1cc(-c2cccs2)nc2ccc(Br)cc12	nan
	CHEMBL450135	172121	46	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	2	1	3	4.4	O=C(O)c1cc(-c2cccs2)nc2ccc(Br)cc12	nan
	5808	176206	20	None	-1	5	Human	6.3	pPotency	=	6.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	211	4	4	4	1.1	CC(C)NC[C@@H](O)c1ccc(O)c(O)c1	nan
	CHEMBL1257092	176206	20	None	-1	5	Human	6.3	pPotency	=	6.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	211	4	4	4	1.1	CC(C)NC[C@@H](O)c1ccc(O)c(O)c1	nan
	CHEMBL460574	176206	20	None	-1	5	Human	6.3	pPotency	=	6.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	211	4	4	4	1.1	CC(C)NC[C@@H](O)c1ccc(O)c(O)c1	nan
	4905097	26732	10	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	316	6	1	5	2.2	CCCC(=O)Nc1ccc2c(c1)nc1n2CCN(CCOC)C1	nan
	CHEMBL1364140	26732	10	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	316	6	1	5	2.2	CCCC(=O)Nc1ccc2c(c1)nc1n2CCN(CCOC)C1	nan
	995260	30852	13	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	3	1	3	5.3	CCc1ccc(-c2nc3ccc(Br)cc3c(C(=O)O)c2C)s1	nan
	CHEMBL1399507	30852	13	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	3	1	3	5.3	CCc1ccc(-c2nc3ccc(Br)cc3c(C(=O)O)c2C)s1	nan
	15990423	32040	6	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	5	1	5	5.3	CCOc1ccccc1NC(=O)c1cn(C2CCCC2)c(=O)c2c1c1ccccc1n2C	nan
	CHEMBL1409911	32040	6	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	5	1	5	5.3	CCOc1ccccc1NC(=O)c1cn(C2CCCC2)c(=O)c2c1c1ccccc1n2C	nan
	16024826	32712	5	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	4	0	5	4.1	CC1CCN(S(=O)(=O)c2ccc3nc(N4CCN(c5ccc(F)cc5)CC4)ccc3c2)CC1	nan
	CHEMBL1415463	32712	5	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	468	4	0	5	4.1	CC1CCN(S(=O)(=O)c2ccc3nc(N4CCN(c5ccc(F)cc5)CC4)ccc3c2)CC1	nan
	3242125	38698	5	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	5	1	4	1.7	COc1ccc(OC)c(CNC(=O)C2CCN(C(=O)N(C)C)CC2)c1	nan
	CHEMBL1467628	38698	5	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	349	5	1	4	1.7	COc1ccc(OC)c(CNC(=O)C2CCN(C(=O)N(C)C)CC2)c1	nan
	3501359	42515	17	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	6	2	8	2.6	COc1ccc(CNC(=O)c2cc3c(=O)n4cccc(C)c4nc3n(CC3CCCO3)c2=N)cc1	nan
	CHEMBL1501993	42515	17	None	-	1	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	473	6	2	8	2.6	COc1ccc(CNC(=O)c2cc3c(=O)n4cccc(C)c4nc3n(CC3CCCO3)c2=N)cc1	nan
	1234242	46307	3	None	1	2	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	300	3	1	6	3.1	CCOc1ccc(-n2nc3c(S)nnc(C)c3c2C)cc1	nan
	CHEMBL1538068	46307	3	None	1	2	Human	5.3	pPotency	=	5.3	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	300	3	1	6	3.1	CCOc1ccc(-n2nc3c(S)nnc(C)c3c2C)cc1	nan
	20921619	23380	5	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	8	1	8	2.9	COc1ccc(CN(C)S(=O)(=O)c2nnc(NC(=O)c3ccc(C)cc3)s2)cc1OC	nan
	CHEMBL1334300	23380	5	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	8	1	8	2.9	COc1ccc(CN(C)S(=O)(=O)c2nnc(NC(=O)c3ccc(C)cc3)s2)cc1OC	nan
	16024792	24883	7	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	4	0	5	4.0	CC1CCN(S(=O)(=O)c2ccc3nc(N4CCN(c5ccccc5)CC4)ccc3c2)CC1	nan
	CHEMBL1347118	24883	7	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	4	0	5	4.0	CC1CCN(S(=O)(=O)c2ccc3nc(N4CCN(c5ccccc5)CC4)ccc3c2)CC1	nan
	5762489	25211	5	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	6	1	3	4.6	N#C/C(=C/c1ccc(OCc2ccccc2)cc1)C(=O)NC1CCCCC1	nan
	CHEMBL1349947	25211	5	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	360	6	1	3	4.6	N#C/C(=C/c1ccc(OCc2ccccc2)cc1)C(=O)NC1CCCCC1	nan
	652632	26790	5	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	8	0	8	3.7	COc1cccc(C(=O)CSc2nnc(-c3cc(OC)cc(OC)c3)o2)c1	nan
	CHEMBL1364667	26790	5	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	386	8	0	8	3.7	COc1cccc(C(=O)CSc2nnc(-c3cc(OC)cc(OC)c3)o2)c1	nan
	4137748	27222	1	None	3	2	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	348	2	1	4	4.0	Cc1cc(NC(=O)c2ccccc2F)nc2c1c(=O)oc1ccccc12	nan
	CHEMBL1368254	27222	1	None	3	2	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	348	2	1	4	4.0	Cc1cc(NC(=O)c2ccccc2F)nc2c1c(=O)oc1ccccc12	nan
	701063	28038	17	None	-1	2	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	242	2	1	5	2.7	COc1ccc(Cl)cc1-c1nnc(S)o1	nan
	CHEMBL1374054	28038	17	None	-1	2	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	242	2	1	5	2.7	COc1ccc(Cl)cc1-c1nnc(S)o1	nan
	16024750	29026	5	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	436	4	0	5	3.7	O=S(=O)(c1ccc2nc(N3CCN(c4ccccc4)CC3)ccc2c1)N1CCCCC1	nan
	CHEMBL1382499	29026	5	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	436	4	0	5	3.7	O=S(=O)(c1ccc2nc(N3CCN(c4ccccc4)CC3)ccc2c1)N1CCCCC1	nan
	1051489	29151	14	None	1	2	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	457	6	1	5	5.7	COc1ccc(NC(=O)CSc2nc(-c3ccc(C)cc3)cc(C(F)(F)F)c2C#N)cc1	nan
	CHEMBL1383601	29151	14	None	1	2	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	457	6	1	5	5.7	COc1ccc(NC(=O)CSc2nc(-c3ccc(C)cc3)cc(C(F)(F)F)c2C#N)cc1	nan
	2185557	29493	9	None	-1	2	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	3	0	6	3.7	COc1ccc(C(=O)/C=C2/Sc3cc4c(cc3N2C)OCO4)cc1	nan
	CHEMBL1386474	29493	9	None	-1	2	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	341	3	0	6	3.7	COc1ccc(C(=O)/C=C2/Sc3cc4c(cc3N2C)OCO4)cc1	nan
	16017568	30449	6	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	6	1	6	2.9	Cc1cccc(C(=O)Nc2nnc(S(=O)(=O)N(C)Cc3ccccc3)s2)c1	nan
	CHEMBL1394623	30449	6	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	402	6	1	6	2.9	Cc1cccc(C(=O)Nc2nnc(S(=O)(=O)N(C)Cc3ccccc3)s2)c1	nan
	16025297	30483	10	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	582	8	1	8	5.3	COc1cc(NC(=O)CSc2ncc3c(n2)-c2ccc(Cl)cc2N(Cc2ccccc2)S3(=O)=O)cc(OC)c1	nan
	CHEMBL1395000	30483	10	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	582	8	1	8	5.3	COc1cc(NC(=O)CSc2ncc3c(n2)-c2ccc(Cl)cc2N(Cc2ccccc2)S3(=O)=O)cc(OC)c1	nan
	2092877	31005	6	None	-1	2	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	4	1	6	3.1	CS(=O)(=O)c1ccc2nc(NC(=O)c3ccc(N4CCCC4=O)cc3)sc2c1	nan
	CHEMBL1400998	31005	6	None	-1	2	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	415	4	1	6	3.1	CS(=O)(=O)c1ccc2nc(NC(=O)c3ccc(N4CCCC4=O)cc3)sc2c1	nan
	681250	33645	15	None	3	2	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	266	3	0	3	3.7	N#Cc1cc2c(nc1SCc1ccccc1)CCC2	nan
	CHEMBL1423417	33645	15	None	3	2	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	266	3	0	3	3.7	N#Cc1cc2c(nc1SCc1ccccc1)CCC2	nan
	2994363	37316	9	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	2	1	4	2.3	CN1C(=O)c2ccc(C(=O)Nc3ccc(Br)cn3)cc2C1=O	nan
	CHEMBL1456212	37316	9	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	359	2	1	4	2.3	CN1C(=O)c2ccc(C(=O)Nc3ccc(Br)cn3)cc2C1=O	nan
	54679694	37926	6	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	442	8	2	6	3.5	C=CCn1c(=O)c(C(=O)NCCc2ccc(Cl)cc2)c(O)c2cc(OC)c(OC)cc21	nan
	CHEMBL1461466	37926	6	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	442	8	2	6	3.5	C=CCn1c(=O)c(C(=O)NCCc2ccc(Cl)cc2)c(O)c2cc(OC)c(OC)cc21	nan
	16814136	38549	8	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	7	1	11	1.1	CCCc1nc(SCC(=O)Nc2nnc(CC)s2)c2c(=O)n(C)c(=O)n(C)c2n1	nan
	CHEMBL1466491	38549	8	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	435	7	1	11	1.1	CCCc1nc(SCC(=O)Nc2nnc(CC)s2)c2c(=O)n(C)c(=O)n(C)c2n1	nan
	16017049	39451	4	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	464	4	0	6	4.4	CCC(C(=O)N1CCN(c2ccccc2F)CC1)n1nc(C)c2sc3ccccc3c2c1=O	nan
	CHEMBL1475149	39451	4	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	464	4	0	6	4.4	CCC(C(=O)N1CCN(c2ccccc2F)CC1)n1nc(C)c2sc3ccccc3c2c1=O	nan
	655498	40375	3	None	-1	2	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	7	1	5	3.5	CCOc1ccc2cc(C#N)c(SCC(=O)NC(C)CC)nc2c1	nan
	CHEMBL1483885	40375	3	None	-1	2	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	7	1	5	3.5	CCOc1ccc2cc(C#N)c(SCC(=O)NC(C)CC)nc2c1	nan
	16019676	40817	0	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	373	5	1	7	2.4	Cn1c(=O)c2sccc2n2c(CCCC(=O)NC3CCCCC3)nnc12	nan
	CHEMBL1487718	40817	0	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	373	5	1	7	2.4	Cn1c(=O)c2sccc2n2c(CCCC(=O)NC3CCCCC3)nnc12	nan
	1305684	40829	12	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	461	6	1	5	5.5	COc1ccc(-c2cc(C(F)(F)F)c(C#N)c(SCC(=O)Nc3ccccc3F)n2)cc1	nan
	CHEMBL1487797	40829	12	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	461	6	1	5	5.5	COc1ccc(-c2cc(C(F)(F)F)c(C#N)c(SCC(=O)Nc3ccccc3F)n2)cc1	nan
	4008999	40919	8	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	7	1	4	6.7	CCCCOc1ccc(C(=O)Nc2ccc(-c3nc4ccccc4s3)cc2C)cc1	nan
	CHEMBL1488396	40919	8	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	416	7	1	4	6.7	CCCCOc1ccc(C(=O)Nc2ccc(-c3nc4ccccc4s3)cc2C)cc1	nan
	976779	41300	14	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	292	4	1	4	2.5	COc1ccc(S(=O)(=O)Nc2ccccn2)c(C)c1C	nan
	CHEMBL1491184	41300	14	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	292	4	1	4	2.5	COc1ccc(S(=O)(=O)Nc2ccccn2)c(C)c1C	nan
	1457998	42240	9	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	319	4	1	6	2.3	Cc1cc(C)n2c(SCC(=O)NC3CCCCC3)nnc2n1	nan
	CHEMBL1499565	42240	9	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	319	4	1	6	2.3	Cc1cc(C)n2c(SCC(=O)NC3CCCCC3)nnc2n1	nan
	1555503	43467	19	None	1	2	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	258	6	3	8	0.6	CCCCOC(=O)CNc1nnc(S)nc1O	nan
	CHEMBL1510408	43467	19	None	1	2	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	258	6	3	8	0.6	CCCCOC(=O)CNc1nnc(S)nc1O	nan
	1484666	43589	13	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	304	4	0	6	4.2	COc1ccc(Oc2nc(SC)nc3ccsc23)cc1	nan
	CHEMBL1511350	43589	13	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	304	4	0	6	4.2	COc1ccc(Oc2nc(SC)nc3ccsc23)cc1	nan
	23760140	44120	1	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	304	9	5	5	-1.6	CC(=O)N[C@@H](CC(=O)N[C@H](CCC(=O)O)C(=O)O)C(=O)O	nan
	CHEMBL1518212	44120	1	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	304	9	5	5	-1.6	CC(=O)N[C@@H](CC(=O)N[C@H](CCC(=O)O)C(=O)O)C(=O)O	nan
	4385342	44428	8	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	348	7	1	6	3.2	CCOC(=O)c1sc(NC(=O)CCc2ccc(OC)cc2)nc1C	nan
	CHEMBL1520883	44428	8	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	348	7	1	6	3.2	CCOC(=O)c1sc(NC(=O)CCc2ccc(OC)cc2)nc1C	nan
	2552702	46335	6	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	316	4	0	7	2.2	O=C(OCc1cc([N+](=O)[O-])cc2c1OCOC2)c1ccccn1	nan
	CHEMBL1538293	46335	6	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	316	4	0	7	2.2	O=C(OCc1cc([N+](=O)[O-])cc2c1OCOC2)c1ccccn1	nan
	16021074	48026	4	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	2	1	4	4.3	Cc1cc(C)cc(NC(=O)c2cn3c4c(ccc(Cl)c4c2=O)OC(C)C3)c1	nan
	CHEMBL1553439	48026	4	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	2	1	4	4.3	Cc1cc(C)cc(NC(=O)c2cn3c4c(ccc(Cl)c4c2=O)OC(C)C3)c1	nan
	16034749	48027	4	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	2	1	4	4.7	CC1Cn2cc(C(=O)Nc3ccccc3C(F)(F)F)c(=O)c3c(Cl)ccc(c32)O1	nan
	CHEMBL1553466	48027	4	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	422	2	1	4	4.7	CC1Cn2cc(C(=O)Nc3ccccc3C(F)(F)F)c(=O)c3c(Cl)ccc(c32)O1	nan
	16019427	48050	11	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	479	6	1	9	5.0	COc1ccccc1Nc1nc2c(S(=O)(=O)c3ccc(C(C)C)cc3)nnn2c2ccsc12	nan
	CHEMBL1553892	48050	11	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	479	6	1	9	5.0	COc1ccccc1Nc1nc2c(S(=O)(=O)c3ccc(C(C)C)cc3)nnn2c2ccsc12	nan
	16024639	49517	5	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	7	1	5	4.1	CCc1ccc(C(=O)c2cn(CC(=O)NCc3ccc(C)cc3)c3nc(C)ccc3c2=O)cc1	nan
	CHEMBL1567298	49517	5	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	453	7	1	5	4.1	CCc1ccc(C(=O)c2cn(CC(=O)NCc3ccc(C)cc3)c3nc(C)ccc3c2=O)cc1	nan
	16017791	50279	4	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	4	0	5	2.6	Cc1cc(C)cc(-n2ccn(CC(=O)c3ccc(F)cc3)c(=O)c2=O)c1	nan
	CHEMBL1574186	50279	4	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	352	4	0	5	2.6	Cc1cc(C)cc(-n2ccn(CC(=O)c3ccc(F)cc3)c(=O)c2=O)c1	nan
	935556	51004	10	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	326	6	1	5	3.7	O=C(O)c1cccc(CSc2nnc(Cc3ccccc3)o2)c1	nan
	CHEMBL1580776	51004	10	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	326	6	1	5	3.7	O=C(O)c1cccc(CSc2nnc(Cc3ccccc3)o2)c1	nan
	3441236	52342	3	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	2	1	6	3.2	O=c1c2ccccc2nc2sc(Nc3ccc(F)cc3)nn12	nan
	CHEMBL1593132	52342	3	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	312	2	1	6	3.2	O=c1c2ccccc2nc2sc(Nc3ccc(F)cc3)nn12	nan
	7199916	52528	10	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	400	5	1	8	3.5	Cc1cc(NC(=O)CSc2ncnc3c2cnn3-c2cccc(Cl)c2)no1	nan
	CHEMBL1595048	52528	10	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	400	5	1	8	3.5	Cc1cc(NC(=O)CSc2ncnc3c2cnn3-c2cccc(Cl)c2)no1	nan
	865684	53881	12	None	1	2	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	289	3	1	4	4.2	COc1ccccc1Nc1nc2cc(C)ccc2cc1C#N	nan
	CHEMBL1607092	53881	12	None	1	2	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	289	3	1	4	4.2	COc1ccccc1Nc1nc2cc(C)ccc2cc1C#N	nan
	135421676	108577	8	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	313	4	1	5	2.8	Cc1ccccc1CC1SC(N/N=C/c2ccco2)=NC1=O	nan
	135599408	108577	8	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	313	4	1	5	2.8	Cc1ccccc1CC1SC(N/N=C/c2ccco2)=NC1=O	nan
	137179849	108577	8	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	313	4	1	5	2.8	Cc1ccccc1CC1SC(N/N=C/c2ccco2)=NC1=O	nan
	CHEMBL3212907	108577	8	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	313	4	1	5	2.8	Cc1ccccc1CC1SC(N/N=C/c2ccco2)=NC1=O	nan
	23874512	55109	1	None	-	1	Human	6.2	pPotency	=	6.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	7	2	11	1.9	CCCC(=O)Nc1ncnc2c1ncn2[C@@H]1O[C@@H]2OP(=O)(O)OC[C@H]2[C@H]1OC(=O)CCC	nan
	CHEMBL1397465	55109	1	None	-	1	Human	6.2	pPotency	=	6.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	7	2	11	1.9	CCCC(=O)Nc1ncnc2c1ncn2[C@@H]1O[C@@H]2OP(=O)(O)OC[C@H]2[C@H]1OC(=O)CCC	nan
	CHEMBL1619312	55109	1	None	-	1	Human	6.2	pPotency	=	6.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	469	7	2	11	1.9	CCCC(=O)Nc1ncnc2c1ncn2[C@@H]1O[C@@H]2OP(=O)(O)OC[C@H]2[C@H]1OC(=O)CCC	nan
	16019610	10763	10	None	-50	2	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	461	4	1	8	5.0	O=S(=O)(c1cccc(Cl)c1)c1nnn2c1nc(NC1CCCCCC1)c1sccc12	nan
	CHEMBL1172404	10763	10	None	-50	2	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	461	4	1	8	5.0	O=S(=O)(c1cccc(Cl)c1)c1nnn2c1nc(NC1CCCCCC1)c1sccc12	nan
	20923126	22915	2	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	5	0	6	2.5	COc1ccc(CN2C(=O)c3cccnc3C2=O)cc1S(=O)(=O)N1CCCCC1C	nan
	CHEMBL1330832	22915	2	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	5	0	6	2.5	COc1ccc(CN2C(=O)c3cccnc3C2=O)cc1S(=O)(=O)N1CCCCC1C	nan
	1425004	23068	11	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	216	3	3	8	-0.5	COC(=O)CNc1nnc(S)nc1O	nan
	CHEMBL1331930	23068	11	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	216	3	3	8	-0.5	COC(=O)CNc1nnc(S)nc1O	nan
	16024792	24883	7	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	4	0	5	4.0	CC1CCN(S(=O)(=O)c2ccc3nc(N4CCN(c5ccccc5)CC4)ccc3c2)CC1	nan
	CHEMBL1347118	24883	7	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	450	4	0	5	4.0	CC1CCN(S(=O)(=O)c2ccc3nc(N4CCN(c5ccccc5)CC4)ccc3c2)CC1	nan
	15989825	25883	6	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	304	3	1	6	2.9	Cc1ccc(CNc2nc3ccc(C)cc3n3nnnc23)cc1	nan
	CHEMBL1355740	25883	6	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	304	3	1	6	2.9	Cc1ccc(CNc2nc3ccc(C)cc3n3nnnc23)cc1	nan
	930238	26561	9	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	301	1	1	5	4.1	CC(C)c1nc2sc3c(S)ncnc3c2c2c1CCC2	nan
	CHEMBL1362595	26561	9	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	301	1	1	5	4.1	CC(C)c1nc2sc3c(S)ncnc3c2c2c1CCC2	nan
	15988284	27472	6	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	5	1	7	1.9	Cn1c(=O)c2sccc2n2c(CCC(=O)NCc3ccccc3)nnc12	nan
	CHEMBL1370040	27472	6	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	5	1	7	1.9	Cn1c(=O)c2sccc2n2c(CCC(=O)NCc3ccccc3)nnc12	nan
	7245805	30629	10	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	5	1	5	1.8	Cc1ccc(CNC(=O)Cn2ccn(-c3ccc(F)cc3)c(=O)c2=O)cc1	nan
	CHEMBL1396990	30629	10	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	5	1	5	1.8	Cc1ccc(CNC(=O)Cn2ccn(-c3ccc(F)cc3)c(=O)c2=O)cc1	nan
	16025341	30732	5	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	550	8	1	6	5.0	O=C(CSc1ncc2c(n1)-c1cc(Cl)ccc1N(Cc1ccccc1)S2(=O)=O)NCCc1ccccc1	nan
	CHEMBL1398424	30732	5	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	550	8	1	6	5.0	O=C(CSc1ncc2c(n1)-c1cc(Cl)ccc1N(Cc1ccccc1)S2(=O)=O)NCCc1ccccc1	nan
	995260	30852	13	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	3	1	3	5.3	CCc1ccc(-c2nc3ccc(Br)cc3c(C(=O)O)c2C)s1	nan
	CHEMBL1399507	30852	13	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	375	3	1	3	5.3	CCc1ccc(-c2nc3ccc(Br)cc3c(C(=O)O)c2C)s1	nan
	3243282	34432	2	None	2	2	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	308	3	1	4	4.3	CCCCn1c(=S)[nH]c2c(oc3ccc(Cl)cc32)c1=O	nan
	CHEMBL1429998	34432	2	None	2	2	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	308	3	1	4	4.3	CCCCn1c(=S)[nH]c2c(oc3ccc(Cl)cc32)c1=O	nan
	1007107	35540	14	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	3	1	4	5.8	Cc1ccc(-c2nc3cc(NC(=O)c4cc5ccccc5o4)ccc3o2)cc1	nan
	CHEMBL1441054	35540	14	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	368	3	1	4	5.8	Cc1ccc(-c2nc3cc(NC(=O)c4cc5ccccc5o4)ccc3o2)cc1	nan
	16800714	38731	6	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	7	1	9	0.4	CCCc1nc(SCC(=O)NCC2CCCO2)c2c(=O)n(C)c(=O)n(C)c2n1	nan
	CHEMBL1468004	38731	6	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	407	7	1	9	0.4	CCCc1nc(SCC(=O)NCC2CCCO2)c2c(=O)n(C)c(=O)n(C)c2n1	nan
	814519	39195	24	None	-1	2	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	201	0	2	3	2.4	Sc1[nH]cnc2c3ccccc3nc1-2	nan
	CHEMBL1471924	39195	24	None	-1	2	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	201	0	2	3	2.4	Sc1[nH]cnc2c3ccccc3nc1-2	nan
	44142305	39409	0	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	348	1	1	5	3.1	Cn1cncc1C#Cc1ccc2cc(C3(O)CCCCC3)oc(=O)c2c1	nan
	CHEMBL1474528	39409	0	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	348	1	1	5	3.1	Cn1cncc1C#Cc1ccc2cc(C3(O)CCCCC3)oc(=O)c2c1	nan
	2138538	48619	12	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	7	1	7	4.9	COc1ccc(CCNc2nc3c(-c4cccc(C)c4)nnn3c3ccccc23)cc1OC	nan
	CHEMBL1559550	48619	12	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	439	7	1	7	4.9	COc1ccc(CCNc2nc3c(-c4cccc(C)c4)nnn3c3ccccc23)cc1OC	nan
	16028162	49151	7	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	3	2	3	3.7	O=C1CC(c2ccccc2)Cc2[nH]c(=O)c(C(=O)Nc3ccc(F)cc3)cc21	nan
	CHEMBL1564507	49151	7	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	3	2	3	3.7	O=C1CC(c2ccccc2)Cc2[nH]c(=O)c(C(=O)Nc3ccc(F)cc3)cc21	nan
	7720817	51088	0	None	1	2	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	241	0	1	5	2.9	Sc1nncn2c1cc1oc3ccccc3c12	nan
	CHEMBL1581464	51088	0	None	1	2	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	241	0	1	5	2.9	Sc1nncn2c1cc1oc3ccccc3c12	nan
	1909591	51820	9	None	-1	2	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	2	1	5	3.4	Oc1c2nc3ccc(Br)cc3c-2ncn1Cc1ccncc1	nan
	CHEMBL1587545	51820	9	None	-1	2	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	354	2	1	5	3.4	Oc1c2nc3ccc(Br)cc3c-2ncn1Cc1ccncc1	nan
	15988964	52233	6	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	9	1	4	5.6	CCCCN(C)CCCNC(=O)c1cc(-c2ccc(Br)s2)nc2ccccc12	nan
	CHEMBL1591653	52233	6	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	459	9	1	4	5.6	CCCCN(C)CCCNC(=O)c1cc(-c2ccc(Br)s2)nc2ccccc12	nan
	44143234	52381	0	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	588	16	3	12	2.5	CCCC[N+](CCCC)(CCCC)CCCC.Nc1ncnc2c1ncn2[C@@H]1O[C@H](COS(=O)(=O)[O-])[C@@H](O)[C@H]1O	nan
	CHEMBL1593759	52381	0	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	588	16	3	12	2.5	CCCC[N+](CCCC)(CCCC)CCCC.Nc1ncnc2c1ncn2[C@@H]1O[C@H](COS(=O)(=O)[O-])[C@@H](O)[C@H]1O	nan
	660350	55156	6	None	-70	2	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	265	2	0	3	2.6	O=C(OC1CN2CCC1CC2)c1cccc(Cl)c1	nan
	CHEMBL1413816	55156	6	None	-70	2	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	265	2	0	3	2.6	O=C(OC1CN2CCC1CC2)c1cccc(Cl)c1	nan
	CHEMBL1619747	55156	6	None	-70	2	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	265	2	0	3	2.6	O=C(OC1CN2CCC1CC2)c1cccc(Cl)c1	nan
	24892704	71452	7	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	8	0	8	2.4	COCCn1/c(=N\C(=O)CCS(=O)(=O)c2ccccc2)sc2cc(C(=O)OC)ccc21	nan
	CHEMBL1967784	71452	7	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	462	8	0	8	2.4	COCCn1/c(=N\C(=O)CCS(=O)(=O)c2ccccc2)sc2cc(C(=O)OC)ccc21	nan
	2815701	104970	9	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	4	2	4	2.6	Cc1ccc(S(=O)(=O)NC(=O)Nc2ccc(N(C)C)cc2)cc1	nan
	CHEMBL312032	104970	9	None	-	1	Human	5.2	pPotency	=	5.2	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	333	4	2	4	2.6	Cc1ccc(S(=O)(=O)NC(=O)Nc2ccc(N(C)C)cc2)cc1	nan
	664514	46209	11	None	3	2	Human	6.1	pPotency	=	6.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	330	6	0	7	3.0	CCOC(=O)CC(=O)CSc1ncnc2c1oc1ccccc12	nan
	CHEMBL1537230	46209	11	None	3	2	Human	6.1	pPotency	=	6.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	330	6	0	7	3.0	CCOC(=O)CC(=O)CSc1ncnc2c1oc1ccccc12	nan
	4679126	22464	14	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	482	7	1	9	4.3	CCOc1ccc(C2C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2c2nc(C)c(C(=O)OC)s2)cc1	nan
	CHEMBL1327057	22464	14	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	482	7	1	9	4.3	CCOc1ccc(C2C(C(=O)c3ccc(C)o3)=C(O)C(=O)N2c2nc(C)c(C(=O)OC)s2)cc1	nan
	16030531	23912	5	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	8	1	4	4.9	CCCCNC(=O)CSc1nc2ccccc2nc1Cc1ccc(Cl)cc1	nan
	CHEMBL1338691	23912	5	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	399	8	1	4	4.9	CCCCNC(=O)CSc1nc2ccccc2nc1Cc1ccc(Cl)cc1	nan
	1371049	24191	11	None	1	2	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	396	4	1	6	3.6	COc1ccc(Cl)cc1C(=O)Nc1nc2ccc(S(C)(=O)=O)cc2s1	nan
	CHEMBL1341278	24191	11	None	1	2	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	396	4	1	6	3.6	COc1ccc(Cl)cc1C(=O)Nc1nc2ccc(S(C)(=O)=O)cc2s1	nan
	3236027	24908	10	None	-1	2	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	5	1	7	3.9	COc1ccc(N2CCN(c3ccc(NC(=O)c4ccc5c(c4)OCO5)cc3C#N)CC2)cc1	nan
	CHEMBL1347313	24908	10	None	-1	2	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	5	1	7	3.9	COc1ccc(N2CCN(c3ccc(NC(=O)c4ccc5c(c4)OCO5)cc3C#N)CC2)cc1	nan
	1208330	25119	16	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	6	0	5	4.6	CCN(CC)CCn1c2ccccc2c2nc3ccc([N+](=O)[O-])cc3cc21	nan
	CHEMBL1349151	25119	16	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	6	0	5	4.6	CCN(CC)CCn1c2ccccc2c2nc3ccc([N+](=O)[O-])cc3cc21	nan
	3414203	26002	12	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	3	0	5	2.9	Cn1/c(=N\C(=O)c2ccc(S(=O)(=O)N3CCCC3)cc2)sc2cc(F)ccc21	nan
	CHEMBL1357194	26002	12	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	3	0	5	2.9	Cn1/c(=N\C(=O)c2ccc(S(=O)(=O)N3CCCC3)cc2)sc2cc(F)ccc21	nan
	1920995	26664	8	None	-2	2	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	4	2	3	4.1	Cc1ccc(OCC(=O)NC(=S)Nc2ccc3c4c(cccc24)CC3)cc1	nan
	CHEMBL1363550	26664	8	None	-2	2	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	4	2	3	4.1	Cc1ccc(OCC(=O)NC(=S)Nc2ccc3c4c(cccc24)CC3)cc1	nan
	15988900	28011	8	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	6	1	7	5.1	CCOC(=O)c1c(NC(=O)c2cc(-c3ccc(Br)cc3)on2)sc(C(C)=O)c1C	nan
	CHEMBL1373810	28011	8	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	476	6	1	7	5.1	CCOC(=O)c1c(NC(=O)c2cc(-c3ccc(Br)cc3)on2)sc(C(C)=O)c1C	nan
	1450216	29874	5	None	-1	2	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	5	1	5	4.2	Cc1ccc(C)c2nc(SCC(=O)NCc3cccs3)c(C#N)cc12	nan
	CHEMBL1389491	29874	5	None	-1	2	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	367	5	1	5	4.2	Cc1ccc(C)c2nc(SCC(=O)NCc3cccs3)c(C#N)cc12	nan
	3330912	30543	12	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	475	7	1	5	5.9	CCOc1ccc(NC(=O)CSc2nc(-c3ccc(F)cc3)cc(C(F)(F)F)c2C#N)cc1	nan
	CHEMBL1395727	30543	12	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	475	7	1	5	5.9	CCOc1ccc(NC(=O)CSc2nc(-c3ccc(F)cc3)cc(C(F)(F)F)c2C#N)cc1	nan
	16033852	30894	0	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	2	1	6	4.1	O=c1c2ccccc2nc2sc(Nc3cccc(C(F)(F)F)c3)nn12	nan
	CHEMBL1399988	30894	0	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	362	2	1	6	4.1	O=c1c2ccccc2nc2sc(Nc3cccc(C(F)(F)F)c3)nn12	nan
	20923127	30916	4	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	5	0	6	2.3	COc1ccc(CN2C(=O)c3cccnc3C2=O)cc1S(=O)(=O)N1CCCC(C)C1	nan
	CHEMBL1400119	30916	4	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	429	5	0	6	2.3	COc1ccc(CN2C(=O)c3cccnc3C2=O)cc1S(=O)(=O)N1CCCC(C)C1	nan
	692203	31398	16	None	1	2	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	332	2	0	5	4.5	O=C(Oc1ccccc1)Oc1ccc2c(c1)oc(=O)c1ccccc12	nan
	CHEMBL1404472	31398	16	None	1	2	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	332	2	0	5	4.5	O=C(Oc1ccccc1)Oc1ccc2c(c1)oc(=O)c1ccccc12	nan
	16745677	31828	0	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	581	9	0	9	6.0	CCCCC1=CC2=C(c3ccco3)C(=O)C(C)(OC(=O)c3ccc(OC)cc3)C(=O)C2=CN1Cc1ccc2c(c1)OCO2	nan
	CHEMBL1408237	31828	0	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	581	9	0	9	6.0	CCCCC1=CC2=C(c3ccco3)C(=O)C(C)(OC(=O)c3ccc(OC)cc3)C(=O)C2=CN1Cc1ccc2c(c1)OCO2	nan
	16010801	34882	6	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	488	8	1	8	3.1	COc1ccc(CCn2c(=O)c3cccnc3n(CC(=O)Nc3c(C)cccc3C)c2=O)cc1OC	nan
	CHEMBL1433929	34882	6	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	488	8	1	8	3.1	COc1ccc(CCn2c(=O)c3cccnc3n(CC(=O)Nc3c(C)cccc3C)c2=O)cc1OC	nan
	4107570	39556	6	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	3	1	4	4.8	COc1ccc2c(c1)-c1nc(NC(=O)c3ccc(Cl)cc3)sc1CC2	nan
	CHEMBL1476611	39556	6	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	370	3	1	4	4.8	COc1ccc2c(c1)-c1nc(NC(=O)c3ccc(Cl)cc3)sc1CC2	nan
	16009524	39582	4	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	7	1	7	4.3	Cc1ccc(OCC(=O)Nc2ccc(OCc3cc(=O)n4c(C)csc4n3)cc2)cc1C	nan
	CHEMBL1476936	39582	4	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	449	7	1	7	4.3	Cc1ccc(OCC(=O)Nc2ccc(OCc3cc(=O)n4c(C)csc4n3)cc2)cc1C	nan
	7184626	40389	8	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	7	1	8	3.0	CCOc1ccc(NC(=O)CCCc2nnc3n(C)c(=O)c4sccc4n23)cc1	nan
	CHEMBL1484029	40389	8	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	411	7	1	8	3.0	CCOc1ccc(NC(=O)CCCc2nnc3n(C)c(=O)c4sccc4n23)cc1	nan
	4423184	43922	11	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	5	0	8	2.6	COCCn1/c(=N/C(=O)c2ccc3c(c2)OCCO3)sc2cc(C(=O)OC)ccc21	nan
	CHEMBL1516075	43922	11	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	428	5	0	8	2.6	COCCn1/c(=N/C(=O)c2ccc3c(c2)OCCO3)sc2cc(C(=O)OC)ccc21	nan
	2946893	44266	12	None	-1	2	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	9	1	7	3.2	CCN(CC)S(=O)(=O)c1ccc(OC)c(NC(=O)COc2ccc3c(C)cc(=O)oc3c2)c1	nan
	CHEMBL1519514	44266	12	None	-1	2	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	474	9	1	7	3.2	CCN(CC)S(=O)(=O)c1ccc(OC)c(NC(=O)COc2ccc3c(C)cc(=O)oc3c2)c1	nan
	2808378	10289	26	None	-2	2	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	289	4	2	4	2.9	CC(=O)c1sccc1NC(=O)c1ccccc1C(=O)O	nan
	CHEMBL1162443	10289	26	None	-2	2	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	289	4	2	4	2.9	CC(=O)c1sccc1NC(=O)c1ccccc1C(=O)O	nan
	2085722	22250	2	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	345	5	1	7	1.6	CCCNC(=O)COC(=O)c1cc2c(=O)n3ccccc3nc2s1	nan
	CHEMBL1324965	22250	2	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	345	5	1	7	1.6	CCCNC(=O)COC(=O)c1cc2c(=O)n3ccccc3nc2s1	nan
	2918454	23851	15	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	5	1	8	4.1	COC(=O)c1sc(N2C(=O)C(O)=C(C(=O)c3ccc(C)o3)C2c2ccc(F)cc2)nc1C	nan
	CHEMBL1338266	23851	15	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	456	5	1	8	4.1	COC(=O)c1sc(N2C(=O)C(O)=C(C(=O)c3ccc(C)o3)C2c2ccc(F)cc2)nc1C	nan
	4902571	24038	10	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	5	1	8	4.3	CSc1nnc(N2C(=O)C(O)=C(C(=O)c3ccc(C)o3)C2c2ccc(C)cc2)s1	nan
	CHEMBL1339921	24038	10	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	427	5	1	8	4.3	CSc1nnc(N2C(=O)C(O)=C(C(=O)c3ccc(C)o3)C2c2ccc(C)cc2)s1	nan
	15990443	25960	6	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	463	4	1	5	5.8	COc1cc(Cl)c(C)cc1NC(=O)c1cn(C2CCCC2)c(=O)c2c1c1ccccc1n2C	nan
	CHEMBL1356755	25960	6	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	463	4	1	5	5.8	COc1cc(Cl)c(C)cc1NC(=O)c1cn(C2CCCC2)c(=O)c2c1c1ccccc1n2C	nan
	3442498	26974	10	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	311	5	1	8	1.9	Cc1nnc(NC(=O)CSc2ccc([N+](=O)[O-])cn2)s1	nan
	CHEMBL1366225	26974	10	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	311	5	1	8	1.9	Cc1nnc(NC(=O)CSc2ccc([N+](=O)[O-])cn2)s1	nan
	18561048	28224	8	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	6	2	8	2.9	CC(=O)Nc1ccc(NC(=O)CSc2ccc3nnc(-c4cccnc4)n3n2)cc1	nan
	CHEMBL1375333	28224	8	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	6	2	8	2.9	CC(=O)Nc1ccc(NC(=O)CSc2ccc3nnc(-c4cccnc4)n3n2)cc1	nan
	5098091	29515	3	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	6	1	4	5.6	COc1ccc(-c2sc(C(=O)c3ccc(Cl)cc3Cl)cc2CC(=O)O)cc1	nan
	CHEMBL1386663	29515	3	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	420	6	1	4	5.6	COc1ccc(-c2sc(C(=O)c3ccc(Cl)cc3Cl)cc2CC(=O)O)cc1	nan
	1112430	36209	18	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	6	1	6	3.3	CCOC(=O)c1cccc(NC(=O)COc2ccc3c(C)cc(=O)oc3c2)c1	nan
	CHEMBL1447146	36209	18	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	381	6	1	6	3.3	CCOC(=O)c1cccc(NC(=O)COc2ccc3c(C)cc(=O)oc3c2)c1	nan
	734580	36811	15	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	226	3	1	4	2.2	CC(=O)c1sc(NC(=O)C(C)C)nc1C	nan
	CHEMBL1451957	36811	15	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	226	3	1	4	2.2	CC(=O)c1sc(NC(=O)C(C)C)nc1C	nan
	18561036	37592	8	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	6	2	8	2.9	CC(=O)Nc1ccc(NC(=O)CSc2ccc3nnc(-c4ccccn4)n3n2)cc1	nan
	CHEMBL1458644	37592	8	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	419	6	2	8	2.9	CC(=O)Nc1ccc(NC(=O)CSc2ccc3nnc(-c4ccccn4)n3n2)cc1	nan
	16195440	38274	0	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	4	1	5	4.7	CCn1c(=O)c2cc(C(=O)Nc3cccc(C(C)=O)c3)sc2c2ccccc21	nan
	CHEMBL1464378	38274	0	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	390	4	1	5	4.7	CCn1c(=O)c2cc(C(=O)Nc3cccc(C(C)=O)c3)sc2c2ccccc21	nan
	16008699	39372	5	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	447	6	1	9	2.5	CCOc1ccc(-c2nc(C(N)=O)c3c(n2)n(-c2ccc4c(c2)OCO4)c(=O)n3CC)cc1	nan
	CHEMBL1474027	39372	5	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	447	6	1	9	2.5	CCOc1ccc(-c2nc(C(N)=O)c3c(n2)n(-c2ccc4c(c2)OCO4)c(=O)n3CC)cc1	nan
	2746740	41558	5	None	2	2	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	5	2	6	5.5	O=C(Nc1ccc(Cl)cc1)Nc1ccccc1Sc1ncc([N+](=O)[O-])s1	nan
	CHEMBL1493199	41558	5	None	2	2	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	406	5	2	6	5.5	O=C(Nc1ccc(Cl)cc1)Nc1ccccc1Sc1ncc([N+](=O)[O-])s1	nan
	17469833	42666	8	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	3	1	6	3.0	COc1ccccc1NC(=O)c1sc2nc3n(c(=O)c2c1C)CCC3	nan
	CHEMBL1503328	42666	8	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	355	3	1	6	3.0	COc1ccccc1NC(=O)c1sc2nc3n(c(=O)c2c1C)CCC3	nan
	17581208	42844	8	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	436	5	1	8	3.1	COc1ccc(NC(=O)Cn2c3ccc(OC)cc3c3nc4n(c(=O)c32)CCS4)cc1	nan
	CHEMBL1505004	42844	8	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	436	5	1	8	3.1	COc1ccc(NC(=O)Cn2c3ccc(OC)cc3c3nc4n(c(=O)c32)CCS4)cc1	nan
	3207506	43101	4	None	1	2	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	5	1	5	3.9	Cc1ccc2nc(SCC(=O)NCc3cccs3)c(C#N)cc2c1	nan
	CHEMBL1507076	43101	4	None	1	2	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	353	5	1	5	3.9	Cc1ccc2nc(SCC(=O)NCc3cccs3)c(C#N)cc2c1	nan
	16018870	44351	5	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	426	4	0	7	6.2	Cc1oc(-c2ccc(Cl)cc2)nc1CSc1nnc(C)n2c1cc1sccc12	nan
	CHEMBL1520274	44351	5	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	426	4	0	7	6.2	Cc1oc(-c2ccc(Cl)cc2)nc1CSc1nnc(C)n2c1cc1sccc12	nan
	1130973	46626	6	None	-2	2	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	6	2	5	5.1	Cc1ccccc1OCC(=O)Nc1sc(C(=O)Nc2cccc(C)c2C)c(C)c1C#N	nan
	CHEMBL1540811	46626	6	None	-2	2	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	433	6	2	5	5.1	Cc1ccccc1OCC(=O)Nc1sc(C(=O)Nc2cccc(C)c2C)c(C)c1C#N	nan
	724891	47051	26	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	302	4	1	5	3.5	O=C(O)CSc1ncnc2scc(-c3ccccc3)c12	nan
	CHEMBL1544233	47051	26	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	302	4	1	5	3.5	O=C(O)CSc1ncnc2scc(-c3ccccc3)c12	nan
	1004390	47572	12	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	8	1	5	4.1	COc1cccc(-c2ccc(C#N)c(SCC(=O)NCCc3ccccc3)n2)c1	nan
	CHEMBL1548754	47572	12	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	403	8	1	5	4.1	COc1cccc(-c2ccc(C#N)c(SCC(=O)NCCc3ccccc3)n2)c1	nan
	1450522	48514	5	None	-1	2	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	4	1	6	3.2	COc1ccc2cc(C#N)c(SCC(=O)N3CC(=O)Nc4ccccc43)nc2c1	nan
	CHEMBL1558667	48514	5	None	-1	2	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	404	4	1	6	3.2	COc1ccc2cc(C#N)c(SCC(=O)N3CC(=O)Nc4ccccc43)nc2c1	nan
	16021094	48855	4	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	3	1	4	4.3	CCc1cccc(NC(=O)c2cn3c4c(ccc(Cl)c4c2=O)OC(C)C3)c1	nan
	CHEMBL1561841	48855	4	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	382	3	1	4	4.3	CCc1cccc(NC(=O)c2cn3c4c(ccc(Cl)c4c2=O)OC(C)C3)c1	nan
	4585955	50290	6	None	-1	2	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	560	6	1	9	4.4	O=C(O)C1CCC(Cn2c(SCc3cc(=O)n4cc(Br)ccc4n3)nc3ccsc3c2=O)CC1	nan
	CHEMBL1574238	50290	6	None	-1	2	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	560	6	1	9	4.4	O=C(O)C1CCC(Cn2c(SCc3cc(=O)n4cc(Br)ccc4n3)nc3ccsc3c2=O)CC1	nan
	16025788	52103	5	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	485	6	1	4	5.7	CCc1ccc(CNC(=O)C2CCN(C(=O)c3ccc(-n4c(C)cc5ccccc54)s3)CC2)cc1	nan
	CHEMBL1590035	52103	5	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	485	6	1	4	5.7	CCc1ccc(CNC(=O)C2CCN(C(=O)c3ccc(-n4c(C)cc5ccccc54)s3)CC2)cc1	nan
	7184644	52207	6	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	7	2	8	0.2	CC(=O)NCCNC(=O)CCCc1nnc2n(C)c(=O)c3sccc3n12	nan
	CHEMBL1591356	52207	6	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	376	7	2	8	0.2	CC(=O)NCCNC(=O)CCCc1nnc2n(C)c(=O)c3sccc3n12	nan
	16010575	52276	4	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	6	1	6	3.2	Cc1cc(C)c(NC(=O)Cn2c(=O)n(CCC(C)C)c(=O)c3cccnc32)c(C)c1	nan
	CHEMBL1592228	52276	4	None	-	1	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	408	6	1	6	3.2	Cc1cc(C)c(NC(=O)Cn2c(=O)n(CCC(C)C)c(=O)c3cccnc32)c(C)c1	nan
	101430	95986	18	None	-1949	5	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	4	4	9	0.2	OC[C@H]1O[C@@H](n2cnc3c(Nc4ccccc4)ncnc32)[C@H](O)[C@@H]1O	nan
	CHEMBL262083	95986	18	None	-1949	5	Human	5.1	pPotency	=	5.1	Functional	PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory) PUBCHEM_BIOASSAY: qHTS Assay for Agonists of the Relaxin Receptor RXFP1. (Class of assay: confirmatory)	ChEMBL	343	4	4	9	0.2	OC[C@H]1O[C@@H](n2cnc3c(Nc4ccccc4)ncnc32)[C@H](O)[C@@H]1O	nan
	12501	3399	0	None	-	1	Human	9.7	pEC50	=	9.7	Functional	Determined in a cell-based cAMP assay.Determined in a cell-based cAMP assay.	Guide to Pharmacology		None	None	None		None	33555858
	12501	3399	0	None	-	1	Human	9.7	pEC50	=	9.7	Functional	Determined in a cell-based cAMP assay.Determined in a cell-based cAMP assay.	Guide to Pharmacology		None	None	None		None	36443381
	1989	3253	0	None	17	3	Human	10.4	pEC50	=	10.4	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	18434306
	56593349	2534	25	None	-	1	Human	7.0	pEC50	=	7.0	Functional	UnclassifiedUnclassified	Guide to Pharmacology	506	7	2	5	5.3	CC(Oc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(c1)S(=O)(=O)C(F)(F)F)C	23764525
	56593349	2534	25	None	-	1	Human	7.0	pEC50	=	7.0	Functional	UnclassifiedUnclassified	Guide to Pharmacology	506	7	2	5	5.3	CC(Oc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(c1)S(=O)(=O)C(F)(F)F)C	23905199
	56593349	2534	25	None	-	1	Human	7.0	pEC50	=	7.0	Functional	UnclassifiedUnclassified	Guide to Pharmacology	506	7	2	5	5.3	CC(Oc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(c1)S(=O)(=O)C(F)(F)F)C	28592882
	8322	2534	25	None	-	1	Human	7.0	pEC50	=	7.0	Functional	UnclassifiedUnclassified	Guide to Pharmacology	506	7	2	5	5.3	CC(Oc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(c1)S(=O)(=O)C(F)(F)F)C	23764525
	8322	2534	25	None	-	1	Human	7.0	pEC50	=	7.0	Functional	UnclassifiedUnclassified	Guide to Pharmacology	506	7	2	5	5.3	CC(Oc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(c1)S(=O)(=O)C(F)(F)F)C	23905199
	8322	2534	25	None	-	1	Human	7.0	pEC50	=	7.0	Functional	UnclassifiedUnclassified	Guide to Pharmacology	506	7	2	5	5.3	CC(Oc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(c1)S(=O)(=O)C(F)(F)F)C	28592882
	CHEMBL3716980	2534	25	None	-	1	Human	7.0	pEC50	=	7.0	Functional	UnclassifiedUnclassified	Guide to Pharmacology	506	7	2	5	5.3	CC(Oc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(c1)S(=O)(=O)C(F)(F)F)C	23764525
	CHEMBL3716980	2534	25	None	-	1	Human	7.0	pEC50	=	7.0	Functional	UnclassifiedUnclassified	Guide to Pharmacology	506	7	2	5	5.3	CC(Oc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(c1)S(=O)(=O)C(F)(F)F)C	23905199
	CHEMBL3716980	2534	25	None	-	1	Human	7.0	pEC50	=	7.0	Functional	UnclassifiedUnclassified	Guide to Pharmacology	506	7	2	5	5.3	CC(Oc1ccccc1C(=O)Nc1ccccc1C(=O)Nc1cccc(c1)S(=O)(=O)C(F)(F)F)C	28592882
	11898	1099	0	None	-	1	Human	7.9	pEC50	=	7.9	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	33555858
	8346	200	0	None	165	2	Human	8.2	pEC50	=	8.2	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	21878627
	11462	3691	0	None	-	1	Human	9.1	pEC50	=	9.1	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	30594862
	134813895	201	0	None	-	1	Human	9.8	pEC50	=	9.8	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	23024363
	8349	201	0	None	-	1	Human	9.8	pEC50	=	9.8	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	23024363
	1988	3254	0	None	-	1	Human	8.8	pEC50	None	8.8	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	16411781
	4371	707	0	None	-	1	Human	6.2	pIC50	=	6.2	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	20043231
	4371	707	0	None	-	1	Human	6.2	pIC50	=	6.2	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	24812057

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Ligands					Receptor			Assay information							Chemical information
Sel. page	Common name	GPCRdb ID	#Vendors	Reference ligand	Fold selectivity (Affinity)	# tested GPCRs (Affinity)	Species	p-value (-log)	Type	Activity Relation	Activity Value	Assay Type	Assay Description	Source	Mol weight	Rot Bonds	H don	H acc	LogP	Smiles	DOI
	162654489	180053	0	None	-	1	Rat	9.3	pEC50	=	9.3	Binding	Agonist activity at rat RXFP1 expressed in human HEK296 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at rat RXFP1 expressed in human HEK296 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	5876	136	86	84	-20.9	CC[C@H](C)[C@@H]1NC(=O)[C@H](C)NC(=O)[C@H]([C@@H](C)CC)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](C(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCSC)NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](CO)NC(=O)[C@@H](N)CC(=O)O)C(C)C)[C@@H](C)CC)CSSC[C@@H]2NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](Cc3ccc(O)cc3)NC(=O)[C@@H](N)CC(C)C)CSCCSC[C@H](NC(=O)CNC(=O)[C@H](C(C)C)NC(=O)[C@H](Cc3cnc[nH]3)NC2=O)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CO)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](Cc2ccccc2)C(=O)NC(C(=O)O)CSSC[C@@H](C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)N[C@@H](CO)C(=O)O)[C@@H](C)O)NC1=O	10.1021/acs.jmedchem.0c01533
	CHEMBL4754949	180053	0	None	-	1	Rat	9.3	pEC50	=	9.3	Binding	Agonist activity at rat RXFP1 expressed in human HEK296 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at rat RXFP1 expressed in human HEK296 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	5876	136	86	84	-20.9	CC[C@H](C)[C@@H]1NC(=O)[C@H](C)NC(=O)[C@H]([C@@H](C)CC)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](C(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCSC)NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](CO)NC(=O)[C@@H](N)CC(=O)O)C(C)C)[C@@H](C)CC)CSSC[C@@H]2NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](Cc3ccc(O)cc3)NC(=O)[C@@H](N)CC(C)C)CSCCSC[C@H](NC(=O)CNC(=O)[C@H](C(C)C)NC(=O)[C@H](Cc3cnc[nH]3)NC2=O)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CO)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](Cc2ccccc2)C(=O)NC(C(=O)O)CSSC[C@@H](C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)N[C@@H](CO)C(=O)O)[C@@H](C)O)NC1=O	10.1021/acs.jmedchem.0c01533
	162672610	182434	0	None	-	0	Rat	9.1	pEC50	=	9.1	Binding	Agonist activity at rat RXFP1 expressed in human HEK296 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at rat RXFP1 expressed in human HEK296 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	4064	171	53	59	-9.7	CCCCCCCCCCCCCCCCC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCCN)NC(=O)CCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCNC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](C)CNC(=O)[C@H](CO)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H](NC(=O)[C@H](CO)NC(=O)[C@H](CCSC)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCC(=O)O)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4793799	182434	0	None	-	0	Rat	9.1	pEC50	=	9.1	Binding	Agonist activity at rat RXFP1 expressed in human HEK296 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at rat RXFP1 expressed in human HEK296 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	4064	171	53	59	-9.7	CCCCCCCCCCCCCCCCC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCCN)NC(=O)CCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCOCCNC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](C)CNC(=O)[C@H](CO)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H](NC(=O)[C@H](CO)NC(=O)[C@H](CCSC)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCC(=O)O)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	162664297	181499	0	None	-	0	Rat	8.3	pEC50	=	8.3	Binding	Agonist activity at rat RXFP1 expressed in human HEK296 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at rat RXFP1 expressed in human HEK296 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	2767	100	45	38	-12.7	CCCC[C@H](NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)NC[C@H](C)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4781560	181499	0	None	-	0	Rat	8.3	pEC50	=	8.3	Binding	Agonist activity at rat RXFP1 expressed in human HEK296 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assayAgonist activity at rat RXFP1 expressed in human HEK296 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins followed by compound addition and measured after 30 mins by HTRF assay	ChEMBL	2767	100	45	38	-12.7	CCCC[C@H](NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](C)CNC(=O)[C@@H](C)CNC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(C)=O)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)NC[C@H](C)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	162654489	180053	0	None	-	1	Human	9.0	pKi	=	9.0	Binding	Displacement of Eu3+-labelled H2 relaxin from human RXFP1 expressed in human HEK-293T cells in presence of 10 % FCS by competition binding assayDisplacement of Eu3+-labelled H2 relaxin from human RXFP1 expressed in human HEK-293T cells in presence of 10 % FCS by competition binding assay	ChEMBL	5876	136	86	84	-20.9	CC[C@H](C)[C@@H]1NC(=O)[C@H](C)NC(=O)[C@H]([C@@H](C)CC)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](C(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCSC)NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](CO)NC(=O)[C@@H](N)CC(=O)O)C(C)C)[C@@H](C)CC)CSSC[C@@H]2NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](Cc3ccc(O)cc3)NC(=O)[C@@H](N)CC(C)C)CSCCSC[C@H](NC(=O)CNC(=O)[C@H](C(C)C)NC(=O)[C@H](Cc3cnc[nH]3)NC2=O)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CO)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](Cc2ccccc2)C(=O)NC(C(=O)O)CSSC[C@@H](C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)N[C@@H](CO)C(=O)O)[C@@H](C)O)NC1=O	10.1021/acs.jmedchem.0c01533
	CHEMBL4754949	180053	0	None	-	1	Human	9.0	pKi	=	9.0	Binding	Displacement of Eu3+-labelled H2 relaxin from human RXFP1 expressed in human HEK-293T cells in presence of 10 % FCS by competition binding assayDisplacement of Eu3+-labelled H2 relaxin from human RXFP1 expressed in human HEK-293T cells in presence of 10 % FCS by competition binding assay	ChEMBL	5876	136	86	84	-20.9	CC[C@H](C)[C@@H]1NC(=O)[C@H](C)NC(=O)[C@H]([C@@H](C)CC)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](C(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCSC)NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](CO)NC(=O)[C@@H](N)CC(=O)O)C(C)C)[C@@H](C)CC)CSSC[C@@H]2NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](Cc3ccc(O)cc3)NC(=O)[C@@H](N)CC(C)C)CSCCSC[C@H](NC(=O)CNC(=O)[C@H](C(C)C)NC(=O)[C@H](Cc3cnc[nH]3)NC2=O)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CO)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](Cc2ccccc2)C(=O)NC(C(=O)O)CSSC[C@@H](C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)N[C@@H](CO)C(=O)O)[C@@H](C)O)NC1=O	10.1021/acs.jmedchem.0c01533
	162662592	181387	0	None	-	1	Human	5.5	pKi	=	5.5	Binding	Displacement of Eu3+-labelled H2 relaxin from human RXFP1 expressed in human HEK-293T cells in presence of 10 % FCS by competition binding assayDisplacement of Eu3+-labelled H2 relaxin from human RXFP1 expressed in human HEK-293T cells in presence of 10 % FCS by competition binding assay	ChEMBL	2985	104	48	42	-13.7	CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CO)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](N)C(C)C)[C@@H](C)CC)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CO)C(=O)N[C@@H](CC(C)C)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	CHEMBL4780098	181387	0	None	-	1	Human	5.5	pKi	=	5.5	Binding	Displacement of Eu3+-labelled H2 relaxin from human RXFP1 expressed in human HEK-293T cells in presence of 10 % FCS by competition binding assayDisplacement of Eu3+-labelled H2 relaxin from human RXFP1 expressed in human HEK-293T cells in presence of 10 % FCS by competition binding assay	ChEMBL	2985	104	48	42	-13.7	CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)[C@H](CO)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](N)C(C)C)[C@@H](C)CC)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)NCC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CO)C(=O)N[C@@H](CC(C)C)C(N)=O)[C@@H](C)O	10.1021/acs.jmedchem.0c01533
	12502	2386	0	None	24	2	Human	10.1	pKd	=	10.1	Binding	Binding affinity determined by SPR.Binding affinity determined by SPR.	Guide to Pharmacology		None	None	None		None	36780899
	12502	2386	0	None	-24	2	Mouse	8.7	pKd	=	8.7	Binding	Binding affinity determined by SPR.Binding affinity determined by SPR.	Guide to Pharmacology		None	None	None		None	36780899
	8346	200	0	None	9	2	Human	7.0	pKd	=	7.0	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	21878627
	3874	1573	0	None	-	1	Human	9.0	pKd	=	9	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	19343240
	3874	1573	0	None	-	1	Human	9.3	pKd	=	9.3	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	22425984
	1993	3250	0	None	-	1	Human	7.3	pKd	None	7.3	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	15649866
	1992	3252	0	None	15	2	Human	9.1	pKd	None	9.1	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	15649866
	1994	3251	0	None	39	2	Human	9.4	pKd	None	9.4	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	15649866
	9321	558	0	None	-	1	Human	5.5	pKi	=	5.5	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	30155023
	9321	558	0	None	-	1	Human	5.5	pKi	=	5.5	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	32295457
	4371	707	0	None	-	1	Human	5.7	pKi	=	5.7	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	20043231
	4371	707	0	None	-	1	Human	5.7	pKi	=	5.7	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	24812057
	1995	2013	0	None	-16982	2	Human	5.7	pKi	=	5.7	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	23303914
	134813895	201	0	None	-	1	Human	9.2	pKi	=	9.2	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	23024363
	8349	201	0	None	-	1	Human	9.2	pKi	=	9.2	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	23024363
	1989	3253	0	None	-1	3	Human	9.7	pKi	=	9.7	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	12506116
	1989	3253	0	None	-1	3	Human	9.7	pKi	=	9.7	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	15649866
	1989	3253	0	None	-1	3	Human	9.7	pKi	=	9.7	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	18434306
	1990	3256	0	None	-14	4	Human	7.8	pKi	None	7.8	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	12506116
	1990	3256	0	None	-14	4	Human	7.8	pKi	None	7.8	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	15649866

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Main reference

Ligand source activities (1 row/activity)