Biased Signaling Atlas

Ligand source activities (1 row/activity)

Potency
Affinity

Get vendors

Ligands (move mouse cursor over ligand name to see structure)					Receptor			Assay information							Chemical information
Sel. page	Common name	GPCRdb ID	#Vendors	Reference ligand	Fold selectivity	# Tested GPCRs	Species	p-value (-log)	Activity Type	Activity Relation	Activity Value	AssayType	Assay Description	Source	Mol weight	Rot Bonds	H don	H acc	LogP	Smiles	DOI
	44314644	13510	0	None	-	1	Rat	9.1	pEC50	=	9.1	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	533	10	2	5	4.2	CCOC(=O)C[C@@H]1CC2(CCN(C(=O)[C@@H](CCCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21	10.1016/S0960-894X(97)00421-6
	CHEMBL1193573	13510	0	None	-	1	Rat	9.1	pEC50	=	9.1	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	533	10	2	5	4.2	CCOC(=O)C[C@@H]1CC2(CCN(C(=O)[C@@H](CCCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21	10.1016/S0960-894X(97)00421-6
	CHEMBL545002	13510	0	None	-	1	Rat	9.1	pEC50	=	9.1	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	533	10	2	5	4.2	CCOC(=O)C[C@@H]1CC2(CCN(C(=O)[C@@H](CCCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21	10.1016/S0960-894X(97)00421-6
	44314965	12914	0	None	-	1	Rat	9.0	pEC50	=	9	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	533	10	2	5	4.2	CCOC(=O)C[C@H]1CC2(CCN(C(=O)[C@@H](CCCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21	10.1016/S0960-894X(97)00421-6
	CHEMBL1189070	12914	0	None	-	1	Rat	9.0	pEC50	=	9	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	533	10	2	5	4.2	CCOC(=O)C[C@H]1CC2(CCN(C(=O)[C@@H](CCCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21	10.1016/S0960-894X(97)00421-6
	CHEMBL538008	12914	0	None	-	1	Rat	9.0	pEC50	=	9	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	533	10	2	5	4.2	CCOC(=O)C[C@H]1CC2(CCN(C(=O)[C@@H](CCCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21	10.1016/S0960-894X(97)00421-6
	9937590	108026	0	None	-	1	Rat	9.0	pEC50	=	9	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	519	9	2	5	3.8	CCOC(=O)[C@H]1CC2(CCN(C(=O)[C@@H](CCCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21	10.1016/S0960-894X(97)00421-6
	CHEMBL319460	108026	0	None	-	1	Rat	9.0	pEC50	=	9	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	519	9	2	5	3.8	CCOC(=O)[C@H]1CC2(CCN(C(=O)[C@@H](CCCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21	10.1016/S0960-894X(97)00421-6
	CHEMBL545465	108026	0	None	-	1	Rat	9.0	pEC50	=	9	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	519	9	2	5	3.8	CCOC(=O)[C@H]1CC2(CCN(C(=O)[C@@H](CCCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21	10.1016/S0960-894X(97)00421-6
	44314574	12913	0	None	-	1	Rat	8.9	pEC50	=	8.9	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	547	11	2	5	4.6	CCOC(=O)CCC1CC2(CCN(C(=O)[C@@H](CCCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21	10.1016/S0960-894X(97)00421-6
	CHEMBL1189066	12913	0	None	-	1	Rat	8.9	pEC50	=	8.9	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	547	11	2	5	4.6	CCOC(=O)CCC1CC2(CCN(C(=O)[C@@H](CCCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21	10.1016/S0960-894X(97)00421-6
	CHEMBL538004	12913	0	None	-	1	Rat	8.9	pEC50	=	8.9	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	547	11	2	5	4.6	CCOC(=O)CCC1CC2(CCN(C(=O)[C@@H](CCCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21	10.1016/S0960-894X(97)00421-6
	178024	1971	33	None	-1	3	Rat	8.8	pEC50	=	8.8	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	528	8	2	6	1.8	O=C([C@H](NC(=O)C(N)(C)C)COCc1ccccc1)N1CCC2(CC1)CN(c1c2cccc1)S(=O)(=O)C	10.1016/S0960-894X(97)00421-6
	5867	1971	33	None	-1	3	Rat	8.8	pEC50	=	8.8	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	528	8	2	6	1.8	O=C([C@H](NC(=O)C(N)(C)C)COCc1ccccc1)N1CCC2(CC1)CN(c1c2cccc1)S(=O)(=O)C	10.1016/S0960-894X(97)00421-6
	CHEMBL13817	1971	33	None	-1	3	Rat	8.8	pEC50	=	8.8	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	528	8	2	6	1.8	O=C([C@H](NC(=O)C(N)(C)C)COCc1ccccc1)N1CCC2(CC1)CN(c1c2cccc1)S(=O)(=O)C	10.1016/S0960-894X(97)00421-6
	22867267	13698	0	None	-	1	Rat	8.7	pEC50	=	8.7	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	505	9	3	4	3.8	CC(C)(N)C(=O)N[C@H](CCCc1ccccc1)C(=O)N1CCC2(CC1)C[C@@H](CC(=O)O)c1ccccc12	10.1016/S0960-894X(97)00421-6
	CHEMBL1194874	13698	0	None	-	1	Rat	8.7	pEC50	=	8.7	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	505	9	3	4	3.8	CC(C)(N)C(=O)N[C@H](CCCc1ccccc1)C(=O)N1CCC2(CC1)C[C@@H](CC(=O)O)c1ccccc12	10.1016/S0960-894X(97)00421-6
	CHEMBL553478	13698	0	None	-	1	Rat	8.7	pEC50	=	8.7	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	505	9	3	4	3.8	CC(C)(N)C(=O)N[C@H](CCCc1ccccc1)C(=O)N1CCC2(CC1)C[C@@H](CC(=O)O)c1ccccc12	10.1016/S0960-894X(97)00421-6
	44293557	101088	0	None	-1	2	Rat	8.0	pEC50	=	8	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	447	7	2	3	3.7	CC(C)(N)C(=O)N[C@H](CCCc1ccccc1)C(=O)N1CCC2(CCc3ccccc32)CC1	10.1016/S0960-894X(97)00421-6
	CHEMBL294923	101088	0	None	-1	2	Rat	8.0	pEC50	=	8	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	447	7	2	3	3.7	CC(C)(N)C(=O)N[C@H](CCCc1ccccc1)C(=O)N1CCC2(CCc3ccccc32)CC1	10.1016/S0960-894X(97)00421-6
	CHEMBL540001	101088	0	None	-1	2	Rat	8.0	pEC50	=	8	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	447	7	2	3	3.7	CC(C)(N)C(=O)N[C@H](CCCc1ccccc1)C(=O)N1CCC2(CCc3ccccc32)CC1	10.1016/S0960-894X(97)00421-6
	9890375	98270	0	None	-1	3	Rat	7.9	pEC50	=	7.9	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	458	5	3	3	3.4	CC(C)(N)C(=O)N[C@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC2(CCc3ccccc32)CC1	10.1016/S0960-894X(97)00421-6
	CHEMBL274599	98270	0	None	-1	3	Rat	7.9	pEC50	=	7.9	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	458	5	3	3	3.4	CC(C)(N)C(=O)N[C@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC2(CCc3ccccc32)CC1	10.1016/S0960-894X(97)00421-6
	CHEMBL558802	98270	0	None	-1	3	Rat	7.9	pEC50	=	7.9	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	458	5	3	3	3.4	CC(C)(N)C(=O)N[C@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC2(CCc3ccccc32)CC1	10.1016/S0960-894X(97)00421-6
	10026738	162769	0	None	-1	2	Rat	7.8	pEC50	=	7.8	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	449	7	2	4	2.9	CC(C)(N)C(=O)N[C@H](COCc1ccccc1)C(=O)N1CCC2(CCc3ccccc32)CC1	10.1016/S0960-894X(97)00421-6
	CHEMBL417182	162769	0	None	-1	2	Rat	7.8	pEC50	=	7.8	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	449	7	2	4	2.9	CC(C)(N)C(=O)N[C@H](COCc1ccccc1)C(=O)N1CCC2(CCc3ccccc32)CC1	10.1016/S0960-894X(97)00421-6
	CHEMBL557206	162769	0	None	-1	2	Rat	7.8	pEC50	=	7.8	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	449	7	2	4	2.9	CC(C)(N)C(=O)N[C@H](COCc1ccccc1)C(=O)N1CCC2(CCc3ccccc32)CC1	10.1016/S0960-894X(97)00421-6
	44315065	13491	0	None	-	1	Rat	8.7	pEC50	=	8.7	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	519	9	2	5	3.8	CCOC(=O)[C@@H]1CC2(CCN(C(=O)[C@@H](CCCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21	10.1016/S0960-894X(97)00421-6
	CHEMBL1193375	13491	0	None	-	1	Rat	8.7	pEC50	=	8.7	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	519	9	2	5	3.8	CCOC(=O)[C@@H]1CC2(CCN(C(=O)[C@@H](CCCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21	10.1016/S0960-894X(97)00421-6
	CHEMBL544769	13491	0	None	-	1	Rat	8.7	pEC50	=	8.7	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	519	9	2	5	3.8	CCOC(=O)[C@@H]1CC2(CCN(C(=O)[C@@H](CCCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21	10.1016/S0960-894X(97)00421-6
	44314651	13604	0	None	-	1	Rat	8.7	pEC50	=	8.7	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	491	8	3	4	3.4	CC(C)(N)C(=O)N[C@H](CCCc1ccccc1)C(=O)N1CCC2(CC1)C[C@H](C(=O)O)c1ccccc12	10.1016/S0960-894X(97)00421-6
	CHEMBL1194179	13604	0	None	-	1	Rat	8.7	pEC50	=	8.7	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	491	8	3	4	3.4	CC(C)(N)C(=O)N[C@H](CCCc1ccccc1)C(=O)N1CCC2(CC1)C[C@H](C(=O)O)c1ccccc12	10.1016/S0960-894X(97)00421-6
	CHEMBL545704	13604	0	None	-	1	Rat	8.7	pEC50	=	8.7	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	491	8	3	4	3.4	CC(C)(N)C(=O)N[C@H](CCCc1ccccc1)C(=O)N1CCC2(CC1)C[C@H](C(=O)O)c1ccccc12	10.1016/S0960-894X(97)00421-6
	22867284	13109	0	None	-	1	Rat	8.6	pEC50	=	8.6	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	505	9	3	4	3.8	CC(C)(N)C(=O)N[C@H](CCCc1ccccc1)C(=O)N1CCC2(CC1)C[C@H](CC(=O)O)c1ccccc12	10.1016/S0960-894X(97)00421-6
	CHEMBL1190399	13109	0	None	-	1	Rat	8.6	pEC50	=	8.6	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	505	9	3	4	3.8	CC(C)(N)C(=O)N[C@H](CCCc1ccccc1)C(=O)N1CCC2(CC1)C[C@H](CC(=O)O)c1ccccc12	10.1016/S0960-894X(97)00421-6
	CHEMBL540805	13109	0	None	-	1	Rat	8.6	pEC50	=	8.6	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	505	9	3	4	3.8	CC(C)(N)C(=O)N[C@H](CCCc1ccccc1)C(=O)N1CCC2(CC1)C[C@H](CC(=O)O)c1ccccc12	10.1016/S0960-894X(97)00421-6
	22867266	13108	0	None	-	1	Rat	8.6	pEC50	=	8.6	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	519	10	3	4	4.1	CC(C)(N)C(=O)N[C@H](CCCc1ccccc1)C(=O)N1CCC2(CC1)CC(CCC(=O)O)c1ccccc12	10.1016/S0960-894X(97)00421-6
	CHEMBL1190394	13108	0	None	-	1	Rat	8.6	pEC50	=	8.6	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	519	10	3	4	4.1	CC(C)(N)C(=O)N[C@H](CCCc1ccccc1)C(=O)N1CCC2(CC1)CC(CCC(=O)O)c1ccccc12	10.1016/S0960-894X(97)00421-6
	CHEMBL540800	13108	0	None	-	1	Rat	8.6	pEC50	=	8.6	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	519	10	3	4	4.1	CC(C)(N)C(=O)N[C@H](CCCc1ccccc1)C(=O)N1CCC2(CC1)CC(CCC(=O)O)c1ccccc12	10.1016/S0960-894X(97)00421-6
	44314888	13684	0	None	-	1	Rat	8.6	pEC50	=	8.6	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	491	8	3	4	3.4	CC(C)(N)C(=O)N[C@H](CCCc1ccccc1)C(=O)N1CCC2(CC1)C[C@@H](C(=O)O)c1ccccc12	10.1016/S0960-894X(97)00421-6
	CHEMBL1194776	13684	0	None	-	1	Rat	8.6	pEC50	=	8.6	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	491	8	3	4	3.4	CC(C)(N)C(=O)N[C@H](CCCc1ccccc1)C(=O)N1CCC2(CC1)C[C@@H](C(=O)O)c1ccccc12	10.1016/S0960-894X(97)00421-6
	CHEMBL553290	13684	0	None	-	1	Rat	8.6	pEC50	=	8.6	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	491	8	3	4	3.4	CC(C)(N)C(=O)N[C@H](CCCc1ccccc1)C(=O)N1CCC2(CC1)C[C@@H](C(=O)O)c1ccccc12	10.1016/S0960-894X(97)00421-6
	44314948	13463	0	None	-	1	Rat	8.5	pEC50	=	8.5	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	521	9	2	6	3.0	CCOC(=O)[C@H]1CC2(CCN(C(=O)[C@@H](COCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21	10.1016/S0960-894X(97)00421-6
	CHEMBL1193173	13463	0	None	-	1	Rat	8.5	pEC50	=	8.5	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	521	9	2	6	3.0	CCOC(=O)[C@H]1CC2(CCN(C(=O)[C@@H](COCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21	10.1016/S0960-894X(97)00421-6
	CHEMBL544536	13463	0	None	-	1	Rat	8.5	pEC50	=	8.5	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	521	9	2	6	3.0	CCOC(=O)[C@H]1CC2(CCN(C(=O)[C@@H](COCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21	10.1016/S0960-894X(97)00421-6
	44314963	13794	0	None	-	1	Rat	7.6	pEC50	=	7.6	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	544	8	3	5	3.9	CCOC(=O)C[C@H]1CC2(CCN(C(=O)[C@@H](Cc3c[nH]c4ccccc34)NC(=O)C(C)(C)N)CC2)c2ccccc21	10.1016/S0960-894X(97)00421-6
	CHEMBL1195548	13794	0	None	-	1	Rat	7.6	pEC50	=	7.6	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	544	8	3	5	3.9	CCOC(=O)C[C@H]1CC2(CCN(C(=O)[C@@H](Cc3c[nH]c4ccccc34)NC(=O)C(C)(C)N)CC2)c2ccccc21	10.1016/S0960-894X(97)00421-6
	CHEMBL554852	13794	0	None	-	1	Rat	7.6	pEC50	=	7.6	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	544	8	3	5	3.9	CCOC(=O)C[C@H]1CC2(CCN(C(=O)[C@@H](Cc3c[nH]c4ccccc34)NC(=O)C(C)(C)N)CC2)c2ccccc21	10.1016/S0960-894X(97)00421-6
	9872740	26465	37	None	-	1	Rat	8.5	pEC50	=	8.5	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	567	10	4	7	3.6	C[C@@H](O)CNC(C)(C)CC(=O)N[C@@H]1CCc2ccccc2N(Cc2ccc(-c3ccccc3-c3nn[nH]n3)cc2)C1=O	10.1016/S0960-894X(97)00421-6
	CHEMBL13600	26465	37	None	-	1	Rat	8.5	pEC50	=	8.5	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	567	10	4	7	3.6	C[C@@H](O)CNC(C)(C)CC(=O)N[C@@H]1CCc2ccccc2N(Cc2ccc(-c3ccccc3-c3nn[nH]n3)cc2)C1=O	10.1016/S0960-894X(97)00421-6
	44314653	13511	0	None	-	1	Rat	8.4	pEC50	=	8.4	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	493	8	3	5	2.6	CC(C)(N)C(=O)N[C@H](COCc1ccccc1)C(=O)N1CCC2(CC1)C[C@H](C(=O)O)c1ccccc12	10.1016/S0960-894X(97)00421-6
	CHEMBL1193574	13511	0	None	-	1	Rat	8.4	pEC50	=	8.4	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	493	8	3	5	2.6	CC(C)(N)C(=O)N[C@H](COCc1ccccc1)C(=O)N1CCC2(CC1)C[C@H](C(=O)O)c1ccccc12	10.1016/S0960-894X(97)00421-6
	CHEMBL545003	13511	0	None	-	1	Rat	8.4	pEC50	=	8.4	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	493	8	3	5	2.6	CC(C)(N)C(=O)N[C@H](COCc1ccccc1)C(=O)N1CCC2(CC1)C[C@H](C(=O)O)c1ccccc12	10.1016/S0960-894X(97)00421-6
	22867262	13978	0	None	-	1	Rat	8.2	pEC50	=	8.2	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	516	7	4	4	3.5	CC(C)(N)C(=O)N[C@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC2(CC1)C[C@@H](CC(=O)O)c1ccccc12	10.1016/S0960-894X(97)00421-6
	CHEMBL1196866	13978	0	None	-	1	Rat	8.2	pEC50	=	8.2	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	516	7	4	4	3.5	CC(C)(N)C(=O)N[C@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC2(CC1)C[C@@H](CC(=O)O)c1ccccc12	10.1016/S0960-894X(97)00421-6
	CHEMBL558422	13978	0	None	-	1	Rat	8.2	pEC50	=	8.2	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	516	7	4	4	3.5	CC(C)(N)C(=O)N[C@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC2(CC1)C[C@@H](CC(=O)O)c1ccccc12	10.1016/S0960-894X(97)00421-6
	44314767	13700	0	None	-	1	Rat	8.2	pEC50	=	8.2	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	530	7	3	5	3.5	CCOC(=O)[C@H]1CC2(CCN(C(=O)[C@@H](Cc3c[nH]c4ccccc34)NC(=O)C(C)(C)N)CC2)c2ccccc21	10.1016/S0960-894X(97)00421-6
	CHEMBL1194891	13700	0	None	-	1	Rat	8.2	pEC50	=	8.2	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	530	7	3	5	3.5	CCOC(=O)[C@H]1CC2(CCN(C(=O)[C@@H](Cc3c[nH]c4ccccc34)NC(=O)C(C)(C)N)CC2)c2ccccc21	10.1016/S0960-894X(97)00421-6
	CHEMBL553507	13700	0	None	-	1	Rat	8.2	pEC50	=	8.2	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	530	7	3	5	3.5	CCOC(=O)[C@H]1CC2(CCN(C(=O)[C@@H](Cc3c[nH]c4ccccc34)NC(=O)C(C)(C)N)CC2)c2ccccc21	10.1016/S0960-894X(97)00421-6
	44314881	13658	0	None	-	1	Rat	8.2	pEC50	=	8.2	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	521	9	2	6	3.0	CCOC(=O)[C@@H]1CC2(CCN(C(=O)[C@@H](COCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21	10.1016/S0960-894X(97)00421-6
	CHEMBL1194592	13658	0	None	-	1	Rat	8.2	pEC50	=	8.2	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	521	9	2	6	3.0	CCOC(=O)[C@@H]1CC2(CCN(C(=O)[C@@H](COCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21	10.1016/S0960-894X(97)00421-6
	CHEMBL552911	13658	0	None	-	1	Rat	8.2	pEC50	=	8.2	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	521	9	2	6	3.0	CCOC(=O)[C@@H]1CC2(CCN(C(=O)[C@@H](COCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21	10.1016/S0960-894X(97)00421-6
	121879	2234	24	None	-1	5	Rat	7.2	pEC50	=	7.2	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	509	7	3	6	3.6	O=C(CC(N)(C)C)N[C@@H]1CCc2c(N(C1=O)Cc1ccc(cc1)c1ccccc1c1nnn[nH]1)cccc2	10.1016/S0960-894X(97)00421-6
	5868	2234	24	None	-1	5	Rat	7.2	pEC50	=	7.2	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	509	7	3	6	3.6	O=C(CC(N)(C)C)N[C@@H]1CCc2c(N(C1=O)Cc1ccc(cc1)c1ccccc1c1nnn[nH]1)cccc2	10.1016/S0960-894X(97)00421-6
	CHEMBL308716	2234	24	None	-1	5	Rat	7.2	pEC50	=	7.2	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	509	7	3	6	3.6	O=C(CC(N)(C)C)N[C@@H]1CCc2c(N(C1=O)Cc1ccc(cc1)c1ccccc1c1nnn[nH]1)cccc2	10.1016/S0960-894X(97)00421-6
	44314642	13638	0	None	-	1	Rat	8.2	pEC50	=	8.2	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	544	8	3	5	3.9	CCOC(=O)C[C@@H]1CC2(CCN(C(=O)[C@@H](Cc3c[nH]c4ccccc34)NC(=O)C(C)(C)N)CC2)c2ccccc21	10.1016/S0960-894X(97)00421-6
	CHEMBL1194442	13638	0	None	-	1	Rat	8.2	pEC50	=	8.2	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	544	8	3	5	3.9	CCOC(=O)C[C@@H]1CC2(CCN(C(=O)[C@@H](Cc3c[nH]c4ccccc34)NC(=O)C(C)(C)N)CC2)c2ccccc21	10.1016/S0960-894X(97)00421-6
	CHEMBL552657	13638	0	None	-	1	Rat	8.2	pEC50	=	8.2	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	544	8	3	5	3.9	CCOC(=O)C[C@@H]1CC2(CCN(C(=O)[C@@H](Cc3c[nH]c4ccccc34)NC(=O)C(C)(C)N)CC2)c2ccccc21	10.1016/S0960-894X(97)00421-6
	44315063	13873	0	None	-	1	Rat	8.1	pEC50	=	8.1	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	530	7	3	5	3.5	CCOC(=O)[C@@H]1CC2(CCN(C(=O)[C@@H](Cc3c[nH]c4ccccc34)NC(=O)C(C)(C)N)CC2)c2ccccc21	10.1016/S0960-894X(97)00421-6
	CHEMBL1196053	13873	0	None	-	1	Rat	8.1	pEC50	=	8.1	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	530	7	3	5	3.5	CCOC(=O)[C@@H]1CC2(CCN(C(=O)[C@@H](Cc3c[nH]c4ccccc34)NC(=O)C(C)(C)N)CC2)c2ccccc21	10.1016/S0960-894X(97)00421-6
	CHEMBL555821	13873	0	None	-	1	Rat	8.1	pEC50	=	8.1	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	530	7	3	5	3.5	CCOC(=O)[C@@H]1CC2(CCN(C(=O)[C@@H](Cc3c[nH]c4ccccc34)NC(=O)C(C)(C)N)CC2)c2ccccc21	10.1016/S0960-894X(97)00421-6
	1104	1792	0	None	-	1	Rat	9.1	pIC50	=	9.1	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	1534126
	1122	2701	0	None	-	1	Rat	10.2	pIC50	None	10.2	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9145431
	1123	2702	0	None	-	1	Rat	10.2	pIC50	None	10.2	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9145431
	1105	1793	0	None	-	1	Rat	8.0	pIC50	None	8	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	1534126
	1103	1791	0	None	-	1	Rat	8.2	pIC50	None	8.2	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	1534126
	CHEMBL440262	1791	0	None	-	1	Rat	8.2	pIC50	None	8.2	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	1534126

Get vendors

Ligands (move mouse cursor over ligand name to see structure)					Receptor			Assay information							Chemical information
Sel. page	Similar- ity	Common name	GPCRdb ID	#Vendors	Reference ligand	Fold selectivity	# Tested GPCRs	Species	p-value (-log)	Activity Type	Activity Relation	Activity Value	Assay Type	Assay Description	Source	Mol weight	Rot Bonds	H don	H acc	LogP	Smiles	DOI
		148124	207099	86	None	-	1	Human	9.9	pIC50	=	9.9	Binding	Displacement of [125I]JV1-42 from GHRH receptor expressed in human MX1 cellsDisplacement of [125I]JV1-42 from GHRH receptor expressed in human MX1 cells	ChEMBL	807	8	5	14	3.3	CC(=O)O[C@@]12CO[C@@H]1C[C@H](O)[C@@]1(C)C(=O)[C@H](O)C3=C(C)[C@@H](OC(=O)[C@H](O)[C@@H](NC(=O)OC(C)(C)C)c4ccccc4)C[C@@](O)([C@@H](OC(=O)c4ccccc4)[C@@H]12)C3(C)C	10.1073/pnas.0610860104
		CHEMBL3545252	207099	86	None	-	1	Human	9.9	pIC50	=	9.9	Binding	Displacement of [125I]JV1-42 from GHRH receptor expressed in human MX1 cellsDisplacement of [125I]JV1-42 from GHRH receptor expressed in human MX1 cells	ChEMBL	807	8	5	14	3.3	CC(=O)O[C@@]12CO[C@@H]1C[C@H](O)[C@@]1(C)C(=O)[C@H](O)C3=C(C)[C@@H](OC(=O)[C@H](O)[C@@H](NC(=O)OC(C)(C)C)c4ccccc4)C[C@@](O)([C@@H](OC(=O)c4ccccc4)[C@@H]12)C3(C)C	10.1073/pnas.0610860104
		CHEMBL92	207099	86	None	-	1	Human	9.9	pIC50	=	9.9	Binding	Displacement of [125I]JV1-42 from GHRH receptor expressed in human MX1 cellsDisplacement of [125I]JV1-42 from GHRH receptor expressed in human MX1 cells	ChEMBL	807	8	5	14	3.3	CC(=O)O[C@@]12CO[C@@H]1C[C@H](O)[C@@]1(C)C(=O)[C@H](O)C3=C(C)[C@@H](OC(=O)[C@H](O)[C@@H](NC(=O)OC(C)(C)C)c4ccccc4)C[C@@](O)([C@@H](OC(=O)c4ccccc4)[C@@H]12)C3(C)C	10.1073/pnas.0610860104
		44387407	141826	0	None	-	0	Rat	9.1	pIC50	=	9.1	Binding	Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates	ChEMBL	3354	116	47	46	-12.4	CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)CC(=O)CCc1ccc(O)cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O	10.1021/jm00088a023
		91928715	141826	0	None	-	0	Rat	9.1	pIC50	=	9.1	Binding	Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates	ChEMBL	3354	116	47	46	-12.4	CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)CC(=O)CCc1ccc(O)cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O	10.1021/jm00088a023
		CHEMBL386366	141826	0	None	-	0	Rat	9.1	pIC50	=	9.1	Binding	Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates	ChEMBL	3354	116	47	46	-12.4	CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)CC(=O)CCc1ccc(O)cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O	10.1021/jm00088a023
		1103	1791	0	None	-	0	Rat	9.1	pIC50	=	9.1	Binding	Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates	ChEMBL		None	None	None		None	10.1021/jm00088a023
		CHEMBL440262	1791	0	None	-	0	Rat	9.1	pIC50	=	9.1	Binding	Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates	ChEMBL		None	None	None		None	10.1021/jm00088a023
		CHEMBL385308	212348	0	None	-	0	Rat	8.7	pIC50	=	8.7	Binding	Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates	ChEMBL		None	None	None		CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@H](Cc1c[nH]cn1)NC(C)=O)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CO)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1c[nH]cn1)C(=O)N[C@@H](CCC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)[C@@H](C)CC)[C@@H](C)O	10.1021/jm00088a023
		CHEMBL412221	212977	0	None	-	0	Rat	6.0	pIC50	=	6	Binding	Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates	ChEMBL		None	None	None		CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O	10.1021/jm00088a023
		CHEMBL269263	210783	0	None	-	0	Rat	6.0	pIC50	=	6	Binding	Compound was tested to Inhibit [125I]GRF in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]GRF in rat adenopituitary homogenates	ChEMBL		None	None	None		CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O	10.1021/jm00088a023
		CHEMBL264522	210624	0	None	-	0	Rat	6.9	pIC50	=	6.9	Binding	Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates	ChEMBL		None	None	None		CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O	10.1021/jm00088a023
		44387431	96521	0	None	-	0	Rat	7.9	pIC50	=	7.9	Binding	Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates	ChEMBL	3441	119	50	48	-15.1	CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CCCN)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O	10.1021/jm00088a023
		91928702	96521	0	None	-	0	Rat	7.9	pIC50	=	7.9	Binding	Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates	ChEMBL	3441	119	50	48	-15.1	CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CCCN)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O	10.1021/jm00088a023
		CHEMBL262750	96521	0	None	-	0	Rat	7.9	pIC50	=	7.9	Binding	Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates	ChEMBL	3441	119	50	48	-15.1	CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CCCN)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O	10.1021/jm00088a023
		44387406	161243	0	None	-	0	Rat	6.9	pIC50	=	6.9	Binding	Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates	ChEMBL	3136	108	44	42	-11.2	CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)CC(=O)CCc1ccc(O)cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O	10.1021/jm00088a023
		91928713	161243	0	None	-	0	Rat	6.9	pIC50	=	6.9	Binding	Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates	ChEMBL	3136	108	44	42	-11.2	CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)CC(=O)CCc1ccc(O)cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O	10.1021/jm00088a023
		CHEMBL411913	161243	0	None	-	0	Rat	6.9	pIC50	=	6.9	Binding	Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates	ChEMBL	3136	108	44	42	-11.2	CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)CC(=O)CCc1ccc(O)cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O	10.1021/jm00088a023
		CHEMBL427794	213384	0	None	-	0	Rat	7.8	pIC50	=	7.8	Binding	Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates	ChEMBL		None	None	None		CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O	10.1021/jm00088a023
		CHEMBL413014	213044	0	None	-	0	Rat	7.8	pIC50	=	7.8	Binding	Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates	ChEMBL		None	None	None		CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(C)=O)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O	10.1021/jm00088a023
		CHEMBL414943	213163	0	None	-	0	Rat	7.7	pIC50	=	7.7	Binding	Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates	ChEMBL		None	None	None		CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O	10.1021/jm00088a023
		CHEMBL437461	213721	0	None	-	0	Rat	7.7	pIC50	=	7.7	Binding	Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates	ChEMBL		None	None	None		CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)C(C)C)[C@@H](C)O	10.1021/jm00088a023
		44387434	168986	0	None	-	0	Rat	7.7	pIC50	=	7.7	Binding	Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates	ChEMBL	3497	123	50	48	-13.5	CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CCCCCCCN)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O	10.1021/jm00088a023
		91928693	168986	0	None	-	0	Rat	7.7	pIC50	=	7.7	Binding	Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates	ChEMBL	3497	123	50	48	-13.5	CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CCCCCCCN)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O	10.1021/jm00088a023
		CHEMBL439108	168986	0	None	-	0	Rat	7.7	pIC50	=	7.7	Binding	Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates	ChEMBL	3497	123	50	48	-13.5	CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CCCCCCCN)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O	10.1021/jm00088a023
		CHEMBL269041	210776	0	None	-	0	Rat	6.7	pIC50	=	6.7	Binding	Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates	ChEMBL		None	None	None		None	10.1021/jm00088a023
		CHEMBL428284	213433	0	None	-	0	Rat	6.5	pIC50	=	6.5	Binding	Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates	ChEMBL		None	None	None		CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](N)CC(=O)O)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O	10.1021/jm00088a023
		CHEMBL439306	213835	0	None	-	0	Rat	6.4	pIC50	=	6.4	Binding	Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates	ChEMBL		None	None	None		CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O	10.1021/jm00088a023
		CHEMBL427665	213363	0	None	-	0	Rat	7.4	pIC50	=	7.4	Binding	Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates	ChEMBL		None	None	None		CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CO)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1c[nH]cn1)C(=O)N[C@@H](CCC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)[C@@H](C)CC)[C@@H](C)O	10.1021/jm00088a023
		CHEMBL262536	210540	0	None	-	0	Rat	7.3	pIC50	=	7.3	Binding	Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates	ChEMBL		None	None	None		CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O	10.1021/jm00088a023
		CHEMBL428135	213418	17	None	-	0	Rat	8.3	pIC50	=	8.3	Binding	Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates	ChEMBL		None	None	None		CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O	10.1021/jm00088a023
		44387430	81895	0	None	-	0	Rat	8.2	pIC50	=	8.2	Binding	Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates	ChEMBL	3469	121	50	48	-14.3	CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CCCCCN)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O	10.1021/jm00088a023
		91928698	81895	0	None	-	0	Rat	8.2	pIC50	=	8.2	Binding	Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates	ChEMBL	3469	121	50	48	-14.3	CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CCCCCN)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O	10.1021/jm00088a023
		CHEMBL216479	81895	0	None	-	0	Rat	8.2	pIC50	=	8.2	Binding	Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates	ChEMBL	3469	121	50	48	-14.3	CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CCCCCN)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O	10.1021/jm00088a023
		CHEMBL438545	213775	0	None	-	0	Rat	8.1	pIC50	=	8.1	Binding	Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates	ChEMBL		None	None	None		CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O	10.1021/jm00088a023
		CHEMBL415373	213186	0	None	-	0	Rat	6.1	pIC50	=	6.1	Binding	Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates	ChEMBL		None	None	None		CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O	10.1021/jm00088a023
		CHEMBL266658	210691	0	None	-	0	Rat	8.0	pIC50	=	8.0	Binding	Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates	ChEMBL		None	None	None		CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O	10.1021/jm00088a023
		CHEMBL265167	210640	13	None	-	0	Rat	8.0	pIC50	=	8.0	Binding	Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates	ChEMBL		None	None	None		CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@@H](N)Cc1c[nH]cn1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CO)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1c[nH]cn1)C(=O)N[C@@H](CCC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)[C@@H](C)CC)[C@@H](C)O	10.1021/jm00088a023
		CHEMBL412558	213003	0	None	-	0	Rat	7.0	pIC50	=	7.0	Binding	Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates	ChEMBL		None	None	None		CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O	10.1021/jm00088a023
		148124	207099	86	None	-	1	Human	8.0	pIC50	=	8.0	Binding	Displacement of [125I]JV1-42 from GHRH receptor expressed in human MX1 cellsDisplacement of [125I]JV1-42 from GHRH receptor expressed in human MX1 cells	Drug Central	807	8	5	14	3.3	CC(=O)O[C@@]12CO[C@@H]1C[C@H](O)[C@@]1(C)C(=O)[C@H](O)C3=C(C)[C@@H](OC(=O)[C@H](O)[C@@H](NC(=O)OC(C)(C)C)c4ccccc4)C[C@@](O)([C@@H](OC(=O)c4ccccc4)[C@@H]12)C3(C)C	None
		CHEMBL3545252	207099	86	None	-	1	Human	8.0	pIC50	=	8.0	Binding	Displacement of [125I]JV1-42 from GHRH receptor expressed in human MX1 cellsDisplacement of [125I]JV1-42 from GHRH receptor expressed in human MX1 cells	Drug Central	807	8	5	14	3.3	CC(=O)O[C@@]12CO[C@@H]1C[C@H](O)[C@@]1(C)C(=O)[C@H](O)C3=C(C)[C@@H](OC(=O)[C@H](O)[C@@H](NC(=O)OC(C)(C)C)c4ccccc4)C[C@@](O)([C@@H](OC(=O)c4ccccc4)[C@@H]12)C3(C)C	None
		CHEMBL92	207099	86	None	-	1	Human	8.0	pIC50	=	8.0	Binding	Displacement of [125I]JV1-42 from GHRH receptor expressed in human MX1 cellsDisplacement of [125I]JV1-42 from GHRH receptor expressed in human MX1 cells	Drug Central	807	8	5	14	3.3	CC(=O)O[C@@]12CO[C@@H]1C[C@H](O)[C@@]1(C)C(=O)[C@H](O)C3=C(C)[C@@H](OC(=O)[C@H](O)[C@@H](NC(=O)OC(C)(C)C)c4ccccc4)C[C@@](O)([C@@H](OC(=O)c4ccccc4)[C@@H]12)C3(C)C	None
		9114	2118	0	None	-	0	Human	9.9	pIC50	=	9.9	Binding	Measuring displacement of [<sup>12</sup>5I]JV-1-42 in a radioligand binding assay.Measuring displacement of [<sup>12</sup>5I]JV-1-42 in a radioligand binding assay.	Guide to Pharmacology		None	None	None		None	17261802
		1109	2159	0	None	-	1	Rat	10.1	pKi	=	10.1	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	10542394
		1109	2159	0	None	-	1	Rat	10.1	pKi	=	10.1	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	14755056
		1109	2159	0	None	-	1	Rat	10.1	pKi	=	10.1	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9892695
		1107	2157	0	None	-	1	Rat	10.3	pKi	=	10.3	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	10542394
		1107	2157	0	None	-	1	Rat	10.3	pKi	=	10.3	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	14755056
		1107	2157	0	None	-	1	Rat	10.3	pKi	=	10.3	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9892695
		1110	2160	0	None	-	1	Rat	10.1	pKi	None	10.1	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9892695
		1115	2165	0	None	-	1	Rat	10.2	pKi	None	10.2	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	14755056
		1116	2166	0	None	-	1	Rat	10.2	pKi	None	10.2	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	14755056
		1121	2700	0	None	-	1	Rat	10.2	pKi	None	10.2	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9145431
		1124	2703	0	None	-	1	Rat	10.2	pKi	None	10.2	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9892695
		1106	2156	0	None	-	1	Rat	10.3	pKi	None	10.3	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9892695
		1118	2696	0	None	-	1	Rat	10.3	pKi	None	10.3	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	7991622
		1108	2158	0	None	-	1	Rat	10.4	pKi	None	10.4	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9892695
		1111	2161	0	None	-	1	Rat	10.4	pKi	None	10.4	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9892695
		1112	2162	0	None	-	1	Rat	10.4	pKi	None	10.4	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9892695
		1113	2163	0	None	-	1	Rat	10.4	pKi	None	10.4	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9892695
		1114	2164	0	None	-	1	Rat	10.4	pKi	None	10.4	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9892695
		1117	2695	0	None	-	1	Rat	10.4	pKi	None	10.4	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	7991622
		1119	2697	0	None	-	1	Rat	10.4	pKi	None	10.4	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	7991622
		1125	281	0	None	-	1	Rat	8.4	pKi	None	8.4	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	14755056
		1125	281	0	None	-	1	Rat	8.4	pKi	None	8.4	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	7991622
		1125	281	0	None	-	1	Rat	8.4	pKi	None	8.4	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9145431
		1125	281	0	None	-	1	Rat	8.4	pKi	None	8.4	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9892695
		1120	2699	0	None	-	1	Rat	9.9	pKi	None	9.9	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	7991622
		1120	2699	0	None	-	1	Rat	9.9	pKi	None	9.9	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9145431

Join us

Cite us

Main reference

Ligand source activities (1 row/activity)