Ligand source activities (1 row/activity)





Ligands (move mouse cursor over ligand name to see structure) Receptor Assay information Chemical information
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DOI

44314644 20282 0 None - 1 Rat 9.1 pEC50 = 9.1 Functional
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 533 10 2 5 4.2 CCOC(=O)C[C@@H]1CC2(CCN(C(=O)[C@@H](CCCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21 10.1016/S0960-894X(97)00421-6
CHEMBL1193573 20282 0 None - 1 Rat 9.1 pEC50 = 9.1 Functional
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 533 10 2 5 4.2 CCOC(=O)C[C@@H]1CC2(CCN(C(=O)[C@@H](CCCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21 10.1016/S0960-894X(97)00421-6
CHEMBL545002 20282 0 None - 1 Rat 9.1 pEC50 = 9.1 Functional
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 533 10 2 5 4.2 CCOC(=O)C[C@@H]1CC2(CCN(C(=O)[C@@H](CCCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21 10.1016/S0960-894X(97)00421-6
44314965 19686 0 None - 1 Rat 9.0 pEC50 = 9 Functional
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 533 10 2 5 4.2 CCOC(=O)C[C@H]1CC2(CCN(C(=O)[C@@H](CCCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21 10.1016/S0960-894X(97)00421-6
CHEMBL1189070 19686 0 None - 1 Rat 9.0 pEC50 = 9 Functional
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 533 10 2 5 4.2 CCOC(=O)C[C@H]1CC2(CCN(C(=O)[C@@H](CCCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21 10.1016/S0960-894X(97)00421-6
CHEMBL538008 19686 0 None - 1 Rat 9.0 pEC50 = 9 Functional
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 533 10 2 5 4.2 CCOC(=O)C[C@H]1CC2(CCN(C(=O)[C@@H](CCCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21 10.1016/S0960-894X(97)00421-6
9937590 114803 0 None - 1 Rat 9.0 pEC50 = 9 Functional
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 519 9 2 5 3.8 CCOC(=O)[C@H]1CC2(CCN(C(=O)[C@@H](CCCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21 10.1016/S0960-894X(97)00421-6
CHEMBL319460 114803 0 None - 1 Rat 9.0 pEC50 = 9 Functional
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 519 9 2 5 3.8 CCOC(=O)[C@H]1CC2(CCN(C(=O)[C@@H](CCCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21 10.1016/S0960-894X(97)00421-6
CHEMBL545465 114803 0 None - 1 Rat 9.0 pEC50 = 9 Functional
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 519 9 2 5 3.8 CCOC(=O)[C@H]1CC2(CCN(C(=O)[C@@H](CCCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21 10.1016/S0960-894X(97)00421-6
44314574 19685 0 None - 1 Rat 8.9 pEC50 = 8.9 Functional
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 547 11 2 5 4.6 CCOC(=O)CCC1CC2(CCN(C(=O)[C@@H](CCCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21 10.1016/S0960-894X(97)00421-6
CHEMBL1189066 19685 0 None - 1 Rat 8.9 pEC50 = 8.9 Functional
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 547 11 2 5 4.6 CCOC(=O)CCC1CC2(CCN(C(=O)[C@@H](CCCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21 10.1016/S0960-894X(97)00421-6
CHEMBL538004 19685 0 None - 1 Rat 8.9 pEC50 = 8.9 Functional
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 547 11 2 5 4.6 CCOC(=O)CCC1CC2(CCN(C(=O)[C@@H](CCCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21 10.1016/S0960-894X(97)00421-6
178024 8752 33 None -1 3 Rat 8.8 pEC50 = 8.8 Functional
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 528 8 2 6 1.8 O=C([C@H](NC(=O)C(N)(C)C)COCc1ccccc1)N1CCC2(CC1)CN(c1c2cccc1)S(=O)(=O)C 10.1016/S0960-894X(97)00421-6
5867 8752 33 None -1 3 Rat 8.8 pEC50 = 8.8 Functional
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 528 8 2 6 1.8 O=C([C@H](NC(=O)C(N)(C)C)COCc1ccccc1)N1CCC2(CC1)CN(c1c2cccc1)S(=O)(=O)C 10.1016/S0960-894X(97)00421-6
CHEMBL13817 8752 33 None -1 3 Rat 8.8 pEC50 = 8.8 Functional
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 528 8 2 6 1.8 O=C([C@H](NC(=O)C(N)(C)C)COCc1ccccc1)N1CCC2(CC1)CN(c1c2cccc1)S(=O)(=O)C 10.1016/S0960-894X(97)00421-6
22867267 20470 0 None - 1 Rat 8.7 pEC50 = 8.7 Functional
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 505 9 3 4 3.8 CC(C)(N)C(=O)N[C@H](CCCc1ccccc1)C(=O)N1CCC2(CC1)C[C@@H](CC(=O)O)c1ccccc12 10.1016/S0960-894X(97)00421-6
CHEMBL1194874 20470 0 None - 1 Rat 8.7 pEC50 = 8.7 Functional
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 505 9 3 4 3.8 CC(C)(N)C(=O)N[C@H](CCCc1ccccc1)C(=O)N1CCC2(CC1)C[C@@H](CC(=O)O)c1ccccc12 10.1016/S0960-894X(97)00421-6
CHEMBL553478 20470 0 None - 1 Rat 8.7 pEC50 = 8.7 Functional
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 505 9 3 4 3.8 CC(C)(N)C(=O)N[C@H](CCCc1ccccc1)C(=O)N1CCC2(CC1)C[C@@H](CC(=O)O)c1ccccc12 10.1016/S0960-894X(97)00421-6
44293557 107865 0 None -1 2 Rat 8.0 pEC50 = 8 Functional
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 447 7 2 3 3.7 CC(C)(N)C(=O)N[C@H](CCCc1ccccc1)C(=O)N1CCC2(CCc3ccccc32)CC1 10.1016/S0960-894X(97)00421-6
CHEMBL294923 107865 0 None -1 2 Rat 8.0 pEC50 = 8 Functional
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 447 7 2 3 3.7 CC(C)(N)C(=O)N[C@H](CCCc1ccccc1)C(=O)N1CCC2(CCc3ccccc32)CC1 10.1016/S0960-894X(97)00421-6
CHEMBL540001 107865 0 None -1 2 Rat 8.0 pEC50 = 8 Functional
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 447 7 2 3 3.7 CC(C)(N)C(=O)N[C@H](CCCc1ccccc1)C(=O)N1CCC2(CCc3ccccc32)CC1 10.1016/S0960-894X(97)00421-6
9890375 105046 0 None -1 3 Rat 7.9 pEC50 = 7.9 Functional
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 458 5 3 3 3.4 CC(C)(N)C(=O)N[C@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC2(CCc3ccccc32)CC1 10.1016/S0960-894X(97)00421-6
CHEMBL274599 105046 0 None -1 3 Rat 7.9 pEC50 = 7.9 Functional
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 458 5 3 3 3.4 CC(C)(N)C(=O)N[C@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC2(CCc3ccccc32)CC1 10.1016/S0960-894X(97)00421-6
CHEMBL558802 105046 0 None -1 3 Rat 7.9 pEC50 = 7.9 Functional
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 458 5 3 3 3.4 CC(C)(N)C(=O)N[C@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC2(CCc3ccccc32)CC1 10.1016/S0960-894X(97)00421-6
10026738 169548 0 None -1 2 Rat 7.8 pEC50 = 7.8 Functional
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 449 7 2 4 2.9 CC(C)(N)C(=O)N[C@H](COCc1ccccc1)C(=O)N1CCC2(CCc3ccccc32)CC1 10.1016/S0960-894X(97)00421-6
CHEMBL417182 169548 0 None -1 2 Rat 7.8 pEC50 = 7.8 Functional
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 449 7 2 4 2.9 CC(C)(N)C(=O)N[C@H](COCc1ccccc1)C(=O)N1CCC2(CCc3ccccc32)CC1 10.1016/S0960-894X(97)00421-6
CHEMBL557206 169548 0 None -1 2 Rat 7.8 pEC50 = 7.8 Functional
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 449 7 2 4 2.9 CC(C)(N)C(=O)N[C@H](COCc1ccccc1)C(=O)N1CCC2(CCc3ccccc32)CC1 10.1016/S0960-894X(97)00421-6
44315065 20263 0 None - 1 Rat 8.7 pEC50 = 8.7 Functional
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 519 9 2 5 3.8 CCOC(=O)[C@@H]1CC2(CCN(C(=O)[C@@H](CCCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21 10.1016/S0960-894X(97)00421-6
CHEMBL1193375 20263 0 None - 1 Rat 8.7 pEC50 = 8.7 Functional
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 519 9 2 5 3.8 CCOC(=O)[C@@H]1CC2(CCN(C(=O)[C@@H](CCCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21 10.1016/S0960-894X(97)00421-6
CHEMBL544769 20263 0 None - 1 Rat 8.7 pEC50 = 8.7 Functional
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 519 9 2 5 3.8 CCOC(=O)[C@@H]1CC2(CCN(C(=O)[C@@H](CCCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21 10.1016/S0960-894X(97)00421-6
44314651 20376 0 None - 1 Rat 8.7 pEC50 = 8.7 Functional
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 491 8 3 4 3.4 CC(C)(N)C(=O)N[C@H](CCCc1ccccc1)C(=O)N1CCC2(CC1)C[C@H](C(=O)O)c1ccccc12 10.1016/S0960-894X(97)00421-6
CHEMBL1194179 20376 0 None - 1 Rat 8.7 pEC50 = 8.7 Functional
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 491 8 3 4 3.4 CC(C)(N)C(=O)N[C@H](CCCc1ccccc1)C(=O)N1CCC2(CC1)C[C@H](C(=O)O)c1ccccc12 10.1016/S0960-894X(97)00421-6
CHEMBL545704 20376 0 None - 1 Rat 8.7 pEC50 = 8.7 Functional
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 491 8 3 4 3.4 CC(C)(N)C(=O)N[C@H](CCCc1ccccc1)C(=O)N1CCC2(CC1)C[C@H](C(=O)O)c1ccccc12 10.1016/S0960-894X(97)00421-6
22867284 19881 0 None - 1 Rat 8.6 pEC50 = 8.6 Functional
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 505 9 3 4 3.8 CC(C)(N)C(=O)N[C@H](CCCc1ccccc1)C(=O)N1CCC2(CC1)C[C@H](CC(=O)O)c1ccccc12 10.1016/S0960-894X(97)00421-6
CHEMBL1190399 19881 0 None - 1 Rat 8.6 pEC50 = 8.6 Functional
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 505 9 3 4 3.8 CC(C)(N)C(=O)N[C@H](CCCc1ccccc1)C(=O)N1CCC2(CC1)C[C@H](CC(=O)O)c1ccccc12 10.1016/S0960-894X(97)00421-6
CHEMBL540805 19881 0 None - 1 Rat 8.6 pEC50 = 8.6 Functional
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 505 9 3 4 3.8 CC(C)(N)C(=O)N[C@H](CCCc1ccccc1)C(=O)N1CCC2(CC1)C[C@H](CC(=O)O)c1ccccc12 10.1016/S0960-894X(97)00421-6
22867266 19880 0 None - 1 Rat 8.6 pEC50 = 8.6 Functional
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 519 10 3 4 4.1 CC(C)(N)C(=O)N[C@H](CCCc1ccccc1)C(=O)N1CCC2(CC1)CC(CCC(=O)O)c1ccccc12 10.1016/S0960-894X(97)00421-6
CHEMBL1190394 19880 0 None - 1 Rat 8.6 pEC50 = 8.6 Functional
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 519 10 3 4 4.1 CC(C)(N)C(=O)N[C@H](CCCc1ccccc1)C(=O)N1CCC2(CC1)CC(CCC(=O)O)c1ccccc12 10.1016/S0960-894X(97)00421-6
CHEMBL540800 19880 0 None - 1 Rat 8.6 pEC50 = 8.6 Functional
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 519 10 3 4 4.1 CC(C)(N)C(=O)N[C@H](CCCc1ccccc1)C(=O)N1CCC2(CC1)CC(CCC(=O)O)c1ccccc12 10.1016/S0960-894X(97)00421-6
44314888 20456 0 None - 1 Rat 8.6 pEC50 = 8.6 Functional
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 491 8 3 4 3.4 CC(C)(N)C(=O)N[C@H](CCCc1ccccc1)C(=O)N1CCC2(CC1)C[C@@H](C(=O)O)c1ccccc12 10.1016/S0960-894X(97)00421-6
CHEMBL1194776 20456 0 None - 1 Rat 8.6 pEC50 = 8.6 Functional
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 491 8 3 4 3.4 CC(C)(N)C(=O)N[C@H](CCCc1ccccc1)C(=O)N1CCC2(CC1)C[C@@H](C(=O)O)c1ccccc12 10.1016/S0960-894X(97)00421-6
CHEMBL553290 20456 0 None - 1 Rat 8.6 pEC50 = 8.6 Functional
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 491 8 3 4 3.4 CC(C)(N)C(=O)N[C@H](CCCc1ccccc1)C(=O)N1CCC2(CC1)C[C@@H](C(=O)O)c1ccccc12 10.1016/S0960-894X(97)00421-6
44314948 20235 0 None - 1 Rat 8.5 pEC50 = 8.5 Functional
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 521 9 2 6 3.0 CCOC(=O)[C@H]1CC2(CCN(C(=O)[C@@H](COCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21 10.1016/S0960-894X(97)00421-6
CHEMBL1193173 20235 0 None - 1 Rat 8.5 pEC50 = 8.5 Functional
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 521 9 2 6 3.0 CCOC(=O)[C@H]1CC2(CCN(C(=O)[C@@H](COCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21 10.1016/S0960-894X(97)00421-6
CHEMBL544536 20235 0 None - 1 Rat 8.5 pEC50 = 8.5 Functional
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 521 9 2 6 3.0 CCOC(=O)[C@H]1CC2(CCN(C(=O)[C@@H](COCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21 10.1016/S0960-894X(97)00421-6
44314963 20566 0 None - 1 Rat 7.6 pEC50 = 7.6 Functional
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 544 8 3 5 3.9 CCOC(=O)C[C@H]1CC2(CCN(C(=O)[C@@H](Cc3c[nH]c4ccccc34)NC(=O)C(C)(C)N)CC2)c2ccccc21 10.1016/S0960-894X(97)00421-6
CHEMBL1195548 20566 0 None - 1 Rat 7.6 pEC50 = 7.6 Functional
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 544 8 3 5 3.9 CCOC(=O)C[C@H]1CC2(CCN(C(=O)[C@@H](Cc3c[nH]c4ccccc34)NC(=O)C(C)(C)N)CC2)c2ccccc21 10.1016/S0960-894X(97)00421-6
CHEMBL554852 20566 0 None - 1 Rat 7.6 pEC50 = 7.6 Functional
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 544 8 3 5 3.9 CCOC(=O)C[C@H]1CC2(CCN(C(=O)[C@@H](Cc3c[nH]c4ccccc34)NC(=O)C(C)(C)N)CC2)c2ccccc21 10.1016/S0960-894X(97)00421-6
9872740 33238 37 None - 1 Rat 8.5 pEC50 = 8.5 Functional
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 567 10 4 7 3.6 C[C@@H](O)CNC(C)(C)CC(=O)N[C@@H]1CCc2ccccc2N(Cc2ccc(-c3ccccc3-c3nn[nH]n3)cc2)C1=O 10.1016/S0960-894X(97)00421-6
CHEMBL13600 33238 37 None - 1 Rat 8.5 pEC50 = 8.5 Functional
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 567 10 4 7 3.6 C[C@@H](O)CNC(C)(C)CC(=O)N[C@@H]1CCc2ccccc2N(Cc2ccc(-c3ccccc3-c3nn[nH]n3)cc2)C1=O 10.1016/S0960-894X(97)00421-6
44314653 20283 0 None - 1 Rat 8.4 pEC50 = 8.4 Functional
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 493 8 3 5 2.6 CC(C)(N)C(=O)N[C@H](COCc1ccccc1)C(=O)N1CCC2(CC1)C[C@H](C(=O)O)c1ccccc12 10.1016/S0960-894X(97)00421-6
CHEMBL1193574 20283 0 None - 1 Rat 8.4 pEC50 = 8.4 Functional
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 493 8 3 5 2.6 CC(C)(N)C(=O)N[C@H](COCc1ccccc1)C(=O)N1CCC2(CC1)C[C@H](C(=O)O)c1ccccc12 10.1016/S0960-894X(97)00421-6
CHEMBL545003 20283 0 None - 1 Rat 8.4 pEC50 = 8.4 Functional
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 493 8 3 5 2.6 CC(C)(N)C(=O)N[C@H](COCc1ccccc1)C(=O)N1CCC2(CC1)C[C@H](C(=O)O)c1ccccc12 10.1016/S0960-894X(97)00421-6
22867262 20750 0 None - 1 Rat 8.2 pEC50 = 8.2 Functional
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 516 7 4 4 3.5 CC(C)(N)C(=O)N[C@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC2(CC1)C[C@@H](CC(=O)O)c1ccccc12 10.1016/S0960-894X(97)00421-6
CHEMBL1196866 20750 0 None - 1 Rat 8.2 pEC50 = 8.2 Functional
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 516 7 4 4 3.5 CC(C)(N)C(=O)N[C@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC2(CC1)C[C@@H](CC(=O)O)c1ccccc12 10.1016/S0960-894X(97)00421-6
CHEMBL558422 20750 0 None - 1 Rat 8.2 pEC50 = 8.2 Functional
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 516 7 4 4 3.5 CC(C)(N)C(=O)N[C@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC2(CC1)C[C@@H](CC(=O)O)c1ccccc12 10.1016/S0960-894X(97)00421-6
44314767 20472 0 None - 1 Rat 8.2 pEC50 = 8.2 Functional
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 530 7 3 5 3.5 CCOC(=O)[C@H]1CC2(CCN(C(=O)[C@@H](Cc3c[nH]c4ccccc34)NC(=O)C(C)(C)N)CC2)c2ccccc21 10.1016/S0960-894X(97)00421-6
CHEMBL1194891 20472 0 None - 1 Rat 8.2 pEC50 = 8.2 Functional
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 530 7 3 5 3.5 CCOC(=O)[C@H]1CC2(CCN(C(=O)[C@@H](Cc3c[nH]c4ccccc34)NC(=O)C(C)(C)N)CC2)c2ccccc21 10.1016/S0960-894X(97)00421-6
CHEMBL553507 20472 0 None - 1 Rat 8.2 pEC50 = 8.2 Functional
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 530 7 3 5 3.5 CCOC(=O)[C@H]1CC2(CCN(C(=O)[C@@H](Cc3c[nH]c4ccccc34)NC(=O)C(C)(C)N)CC2)c2ccccc21 10.1016/S0960-894X(97)00421-6
44314881 20430 0 None - 1 Rat 8.2 pEC50 = 8.2 Functional
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 521 9 2 6 3.0 CCOC(=O)[C@@H]1CC2(CCN(C(=O)[C@@H](COCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21 10.1016/S0960-894X(97)00421-6
CHEMBL1194592 20430 0 None - 1 Rat 8.2 pEC50 = 8.2 Functional
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 521 9 2 6 3.0 CCOC(=O)[C@@H]1CC2(CCN(C(=O)[C@@H](COCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21 10.1016/S0960-894X(97)00421-6
CHEMBL552911 20430 0 None - 1 Rat 8.2 pEC50 = 8.2 Functional
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 521 9 2 6 3.0 CCOC(=O)[C@@H]1CC2(CCN(C(=O)[C@@H](COCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21 10.1016/S0960-894X(97)00421-6
121879 9015 24 None -1 5 Rat 7.2 pEC50 = 7.2 Functional
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 509 7 3 6 3.6 O=C(CC(N)(C)C)N[C@@H]1CCc2c(N(C1=O)Cc1ccc(cc1)c1ccccc1c1nnn[nH]1)cccc2 10.1016/S0960-894X(97)00421-6
5868 9015 24 None -1 5 Rat 7.2 pEC50 = 7.2 Functional
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 509 7 3 6 3.6 O=C(CC(N)(C)C)N[C@@H]1CCc2c(N(C1=O)Cc1ccc(cc1)c1ccccc1c1nnn[nH]1)cccc2 10.1016/S0960-894X(97)00421-6
CHEMBL308716 9015 24 None -1 5 Rat 7.2 pEC50 = 7.2 Functional
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 509 7 3 6 3.6 O=C(CC(N)(C)C)N[C@@H]1CCc2c(N(C1=O)Cc1ccc(cc1)c1ccccc1c1nnn[nH]1)cccc2 10.1016/S0960-894X(97)00421-6
44314642 20410 0 None - 1 Rat 8.2 pEC50 = 8.2 Functional
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 544 8 3 5 3.9 CCOC(=O)C[C@@H]1CC2(CCN(C(=O)[C@@H](Cc3c[nH]c4ccccc34)NC(=O)C(C)(C)N)CC2)c2ccccc21 10.1016/S0960-894X(97)00421-6
CHEMBL1194442 20410 0 None - 1 Rat 8.2 pEC50 = 8.2 Functional
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 544 8 3 5 3.9 CCOC(=O)C[C@@H]1CC2(CCN(C(=O)[C@@H](Cc3c[nH]c4ccccc34)NC(=O)C(C)(C)N)CC2)c2ccccc21 10.1016/S0960-894X(97)00421-6
CHEMBL552657 20410 0 None - 1 Rat 8.2 pEC50 = 8.2 Functional
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 544 8 3 5 3.9 CCOC(=O)C[C@@H]1CC2(CCN(C(=O)[C@@H](Cc3c[nH]c4ccccc34)NC(=O)C(C)(C)N)CC2)c2ccccc21 10.1016/S0960-894X(97)00421-6
44315063 20645 0 None - 1 Rat 8.1 pEC50 = 8.1 Functional
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 530 7 3 5 3.5 CCOC(=O)[C@@H]1CC2(CCN(C(=O)[C@@H](Cc3c[nH]c4ccccc34)NC(=O)C(C)(C)N)CC2)c2ccccc21 10.1016/S0960-894X(97)00421-6
CHEMBL1196053 20645 0 None - 1 Rat 8.1 pEC50 = 8.1 Functional
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 530 7 3 5 3.5 CCOC(=O)[C@@H]1CC2(CCN(C(=O)[C@@H](Cc3c[nH]c4ccccc34)NC(=O)C(C)(C)N)CC2)c2ccccc21 10.1016/S0960-894X(97)00421-6
CHEMBL555821 20645 0 None - 1 Rat 8.1 pEC50 = 8.1 Functional
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 530 7 3 5 3.5 CCOC(=O)[C@@H]1CC2(CCN(C(=O)[C@@H](Cc3c[nH]c4ccccc34)NC(=O)C(C)(C)N)CC2)c2ccccc21 10.1016/S0960-894X(97)00421-6
1104 8573 0 None - 1 Rat 9.1 pIC50 = 9.1 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 1534126
1122 9478 0 None - 1 Rat 10.2 pIC50 None 10.2 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 9145431
1123 9479 0 None - 1 Rat 10.2 pIC50 None 10.2 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 9145431
1105 8574 0 None - 1 Rat 8.0 pIC50 None 8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 1534126
1103 8572 0 None - 1 Rat 8.2 pIC50 None 8.2 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 1534126
CHEMBL440262 8572 0 None - 1 Rat 8.2 pIC50 None 8.2 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 1534126




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DOI

148124 213878 86 None - 1 Human 9.9 pIC50 = 9.9 Binding
Displacement of [125I]JV1-42 from GHRH receptor expressed in human MX1 cellsDisplacement of [125I]JV1-42 from GHRH receptor expressed in human MX1 cells
ChEMBL 807 8 5 14 3.3 CC(=O)O[C@@]12CO[C@@H]1C[C@H](O)[C@@]1(C)C(=O)[C@H](O)C3=C(C)[C@@H](OC(=O)[C@H](O)[C@@H](NC(=O)OC(C)(C)C)c4ccccc4)C[C@@](O)([C@@H](OC(=O)c4ccccc4)[C@@H]12)C3(C)C 10.1073/pnas.0610860104
CHEMBL3545252 213878 86 None - 1 Human 9.9 pIC50 = 9.9 Binding
Displacement of [125I]JV1-42 from GHRH receptor expressed in human MX1 cellsDisplacement of [125I]JV1-42 from GHRH receptor expressed in human MX1 cells
ChEMBL 807 8 5 14 3.3 CC(=O)O[C@@]12CO[C@@H]1C[C@H](O)[C@@]1(C)C(=O)[C@H](O)C3=C(C)[C@@H](OC(=O)[C@H](O)[C@@H](NC(=O)OC(C)(C)C)c4ccccc4)C[C@@](O)([C@@H](OC(=O)c4ccccc4)[C@@H]12)C3(C)C 10.1073/pnas.0610860104
CHEMBL92 213878 86 None - 1 Human 9.9 pIC50 = 9.9 Binding
Displacement of [125I]JV1-42 from GHRH receptor expressed in human MX1 cellsDisplacement of [125I]JV1-42 from GHRH receptor expressed in human MX1 cells
ChEMBL 807 8 5 14 3.3 CC(=O)O[C@@]12CO[C@@H]1C[C@H](O)[C@@]1(C)C(=O)[C@H](O)C3=C(C)[C@@H](OC(=O)[C@H](O)[C@@H](NC(=O)OC(C)(C)C)c4ccccc4)C[C@@](O)([C@@H](OC(=O)c4ccccc4)[C@@H]12)C3(C)C 10.1073/pnas.0610860104
44387407 148604 0 None - 0 Rat 9.1 pIC50 = 9.1 Binding
Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates
ChEMBL 3354 116 47 46 -12.4 CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)CC(=O)CCc1ccc(O)cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O 10.1021/jm00088a023
91928715 148604 0 None - 0 Rat 9.1 pIC50 = 9.1 Binding
Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates
ChEMBL 3354 116 47 46 -12.4 CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)CC(=O)CCc1ccc(O)cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O 10.1021/jm00088a023
CHEMBL386366 148604 0 None - 0 Rat 9.1 pIC50 = 9.1 Binding
Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates
ChEMBL 3354 116 47 46 -12.4 CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)CC(=O)CCc1ccc(O)cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O 10.1021/jm00088a023
1103 8572 0 None - 0 Rat 9.1 pIC50 = 9.1 Binding
Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates
ChEMBL None None None None 10.1021/jm00088a023
CHEMBL440262 8572 0 None - 0 Rat 9.1 pIC50 = 9.1 Binding
Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates
ChEMBL None None None None 10.1021/jm00088a023
CHEMBL385308 219127 0 None - 0 Rat 8.7 pIC50 = 8.7 Binding
Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates
ChEMBL None None None CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@H](Cc1c[nH]cn1)NC(C)=O)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CO)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1c[nH]cn1)C(=O)N[C@@H](CCC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)[C@@H](C)CC)[C@@H](C)O 10.1021/jm00088a023
CHEMBL412221 219756 0 None - 0 Rat 6.0 pIC50 = 6 Binding
Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates
ChEMBL None None None CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O 10.1021/jm00088a023
CHEMBL269263 217562 0 None - 0 Rat 6.0 pIC50 = 6 Binding
Compound was tested to Inhibit [125I]GRF in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]GRF in rat adenopituitary homogenates
ChEMBL None None None CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O 10.1021/jm00088a023
CHEMBL264522 217403 0 None - 0 Rat 6.9 pIC50 = 6.9 Binding
Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates
ChEMBL None None None CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O 10.1021/jm00088a023
44387431 103296 0 None - 0 Rat 7.9 pIC50 = 7.9 Binding
Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates
ChEMBL 3441 119 50 48 -15.1 CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CCCN)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O 10.1021/jm00088a023
91928702 103296 0 None - 0 Rat 7.9 pIC50 = 7.9 Binding
Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates
ChEMBL 3441 119 50 48 -15.1 CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CCCN)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O 10.1021/jm00088a023
CHEMBL262750 103296 0 None - 0 Rat 7.9 pIC50 = 7.9 Binding
Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates
ChEMBL 3441 119 50 48 -15.1 CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CCCN)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O 10.1021/jm00088a023
44387406 168022 0 None - 0 Rat 6.9 pIC50 = 6.9 Binding
Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates
ChEMBL 3136 108 44 42 -11.2 CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)CC(=O)CCc1ccc(O)cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O 10.1021/jm00088a023
91928713 168022 0 None - 0 Rat 6.9 pIC50 = 6.9 Binding
Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates
ChEMBL 3136 108 44 42 -11.2 CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)CC(=O)CCc1ccc(O)cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O 10.1021/jm00088a023
CHEMBL411913 168022 0 None - 0 Rat 6.9 pIC50 = 6.9 Binding
Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates
ChEMBL 3136 108 44 42 -11.2 CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)CC(=O)CCc1ccc(O)cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O 10.1021/jm00088a023
CHEMBL427794 220163 0 None - 0 Rat 7.8 pIC50 = 7.8 Binding
Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates
ChEMBL None None None CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O 10.1021/jm00088a023
CHEMBL413014 219823 0 None - 0 Rat 7.8 pIC50 = 7.8 Binding
Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates
ChEMBL None None None CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(C)=O)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O 10.1021/jm00088a023
CHEMBL414943 219942 0 None - 0 Rat 7.7 pIC50 = 7.7 Binding
Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates
ChEMBL None None None CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O 10.1021/jm00088a023
CHEMBL437461 220500 0 None - 0 Rat 7.7 pIC50 = 7.7 Binding
Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates
ChEMBL None None None CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)C(C)C)[C@@H](C)O 10.1021/jm00088a023
44387434 175765 0 None - 0 Rat 7.7 pIC50 = 7.7 Binding
Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates
ChEMBL 3497 123 50 48 -13.5 CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CCCCCCCN)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O 10.1021/jm00088a023
91928693 175765 0 None - 0 Rat 7.7 pIC50 = 7.7 Binding
Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates
ChEMBL 3497 123 50 48 -13.5 CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CCCCCCCN)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O 10.1021/jm00088a023
CHEMBL439108 175765 0 None - 0 Rat 7.7 pIC50 = 7.7 Binding
Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates
ChEMBL 3497 123 50 48 -13.5 CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CCCCCCCN)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O 10.1021/jm00088a023
CHEMBL269041 217555 0 None - 0 Rat 6.7 pIC50 = 6.7 Binding
Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates
ChEMBL None None None None 10.1021/jm00088a023
CHEMBL428284 220212 0 None - 0 Rat 6.5 pIC50 = 6.5 Binding
Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates
ChEMBL None None None CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](N)CC(=O)O)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O 10.1021/jm00088a023
CHEMBL439306 220614 0 None - 0 Rat 6.4 pIC50 = 6.4 Binding
Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates
ChEMBL None None None CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O 10.1021/jm00088a023
CHEMBL427665 220142 0 None - 0 Rat 7.4 pIC50 = 7.4 Binding
Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates
ChEMBL None None None CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CO)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1c[nH]cn1)C(=O)N[C@@H](CCC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)[C@@H](C)CC)[C@@H](C)O 10.1021/jm00088a023
CHEMBL262536 217319 0 None - 0 Rat 7.3 pIC50 = 7.3 Binding
Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates
ChEMBL None None None CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O 10.1021/jm00088a023
CHEMBL428135 220197 17 None - 0 Rat 8.3 pIC50 = 8.3 Binding
Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates
ChEMBL None None None CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O 10.1021/jm00088a023
44387430 88670 0 None - 0 Rat 8.2 pIC50 = 8.2 Binding
Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates
ChEMBL 3469 121 50 48 -14.3 CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CCCCCN)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O 10.1021/jm00088a023
91928698 88670 0 None - 0 Rat 8.2 pIC50 = 8.2 Binding
Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates
ChEMBL 3469 121 50 48 -14.3 CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CCCCCN)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O 10.1021/jm00088a023
CHEMBL216479 88670 0 None - 0 Rat 8.2 pIC50 = 8.2 Binding
Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates
ChEMBL 3469 121 50 48 -14.3 CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CCCCCN)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O 10.1021/jm00088a023
CHEMBL438545 220554 0 None - 0 Rat 8.1 pIC50 = 8.1 Binding
Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates
ChEMBL None None None CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O 10.1021/jm00088a023
CHEMBL415373 219965 0 None - 0 Rat 6.1 pIC50 = 6.1 Binding
Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates
ChEMBL None None None CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O 10.1021/jm00088a023
CHEMBL266658 217470 0 None - 0 Rat 8.0 pIC50 = 8.0 Binding
Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates
ChEMBL None None None CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O 10.1021/jm00088a023
CHEMBL265167 217419 13 None - 0 Rat 8.0 pIC50 = 8.0 Binding
Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates
ChEMBL None None None CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@@H](N)Cc1c[nH]cn1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CO)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1c[nH]cn1)C(=O)N[C@@H](CCC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)[C@@H](C)CC)[C@@H](C)O 10.1021/jm00088a023
CHEMBL412558 219782 0 None - 0 Rat 7.0 pIC50 = 7.0 Binding
Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates
ChEMBL None None None CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O 10.1021/jm00088a023
148124 213878 86 None - 1 Human 8.0 pIC50 = 8.0 Binding
Displacement of [125I]JV1-42 from GHRH receptor expressed in human MX1 cellsDisplacement of [125I]JV1-42 from GHRH receptor expressed in human MX1 cells
Drug Central 807 8 5 14 3.3 CC(=O)O[C@@]12CO[C@@H]1C[C@H](O)[C@@]1(C)C(=O)[C@H](O)C3=C(C)[C@@H](OC(=O)[C@H](O)[C@@H](NC(=O)OC(C)(C)C)c4ccccc4)C[C@@](O)([C@@H](OC(=O)c4ccccc4)[C@@H]12)C3(C)C None
CHEMBL3545252 213878 86 None - 1 Human 8.0 pIC50 = 8.0 Binding
Displacement of [125I]JV1-42 from GHRH receptor expressed in human MX1 cellsDisplacement of [125I]JV1-42 from GHRH receptor expressed in human MX1 cells
Drug Central 807 8 5 14 3.3 CC(=O)O[C@@]12CO[C@@H]1C[C@H](O)[C@@]1(C)C(=O)[C@H](O)C3=C(C)[C@@H](OC(=O)[C@H](O)[C@@H](NC(=O)OC(C)(C)C)c4ccccc4)C[C@@](O)([C@@H](OC(=O)c4ccccc4)[C@@H]12)C3(C)C None
CHEMBL92 213878 86 None - 1 Human 8.0 pIC50 = 8.0 Binding
Displacement of [125I]JV1-42 from GHRH receptor expressed in human MX1 cellsDisplacement of [125I]JV1-42 from GHRH receptor expressed in human MX1 cells
Drug Central 807 8 5 14 3.3 CC(=O)O[C@@]12CO[C@@H]1C[C@H](O)[C@@]1(C)C(=O)[C@H](O)C3=C(C)[C@@H](OC(=O)[C@H](O)[C@@H](NC(=O)OC(C)(C)C)c4ccccc4)C[C@@](O)([C@@H](OC(=O)c4ccccc4)[C@@H]12)C3(C)C None
9114 8899 0 None - 0 Human 9.9 pIC50 = 9.9 Binding
Measuring displacement of [<sup>12</sup>5I]JV-1-42 in a radioligand binding assay.Measuring displacement of [<sup>12</sup>5I]JV-1-42 in a radioligand binding assay.
Guide to Pharmacology None None None None 17261802
1109 8940 0 None - 1 Rat 10.1 pKi = 10.1 Binding
UnclassifiedUnclassified
Guide to Pharmacology None None None None 10542394
1109 8940 0 None - 1 Rat 10.1 pKi = 10.1 Binding
UnclassifiedUnclassified
Guide to Pharmacology None None None None 14755056
1109 8940 0 None - 1 Rat 10.1 pKi = 10.1 Binding
UnclassifiedUnclassified
Guide to Pharmacology None None None None 9892695
1107 8938 0 None - 1 Rat 10.3 pKi = 10.3 Binding
UnclassifiedUnclassified
Guide to Pharmacology None None None None 10542394
1107 8938 0 None - 1 Rat 10.3 pKi = 10.3 Binding
UnclassifiedUnclassified
Guide to Pharmacology None None None None 14755056
1107 8938 0 None - 1 Rat 10.3 pKi = 10.3 Binding
UnclassifiedUnclassified
Guide to Pharmacology None None None None 9892695
1110 8941 0 None - 1 Rat 10.1 pKi None 10.1 Binding
UnclassifiedUnclassified
Guide to Pharmacology None None None None 9892695
1115 8946 0 None - 1 Rat 10.2 pKi None 10.2 Binding
UnclassifiedUnclassified
Guide to Pharmacology None None None None 14755056
1116 8947 0 None - 1 Rat 10.2 pKi None 10.2 Binding
UnclassifiedUnclassified
Guide to Pharmacology None None None None 14755056
1121 9477 0 None - 1 Rat 10.2 pKi None 10.2 Binding
UnclassifiedUnclassified
Guide to Pharmacology None None None None 9145431
1124 9480 0 None - 1 Rat 10.2 pKi None 10.2 Binding
UnclassifiedUnclassified
Guide to Pharmacology None None None None 9892695
1106 8937 0 None - 1 Rat 10.3 pKi None 10.3 Binding
UnclassifiedUnclassified
Guide to Pharmacology None None None None 9892695
1118 9473 0 None - 1 Rat 10.3 pKi None 10.3 Binding
UnclassifiedUnclassified
Guide to Pharmacology None None None None 7991622
1108 8939 0 None - 1 Rat 10.4 pKi None 10.4 Binding
UnclassifiedUnclassified
Guide to Pharmacology None None None None 9892695
1111 8942 0 None - 1 Rat 10.4 pKi None 10.4 Binding
UnclassifiedUnclassified
Guide to Pharmacology None None None None 9892695
1112 8943 0 None - 1 Rat 10.4 pKi None 10.4 Binding
UnclassifiedUnclassified
Guide to Pharmacology None None None None 9892695
1113 8944 0 None - 1 Rat 10.4 pKi None 10.4 Binding
UnclassifiedUnclassified
Guide to Pharmacology None None None None 9892695
1114 8945 0 None - 1 Rat 10.4 pKi None 10.4 Binding
UnclassifiedUnclassified
Guide to Pharmacology None None None None 9892695
1117 9472 0 None - 1 Rat 10.4 pKi None 10.4 Binding
UnclassifiedUnclassified
Guide to Pharmacology None None None None 7991622
1119 9474 0 None - 1 Rat 10.4 pKi None 10.4 Binding
UnclassifiedUnclassified
Guide to Pharmacology None None None None 7991622
1125 7069 0 None - 1 Rat 8.4 pKi None 8.4 Binding
UnclassifiedUnclassified
Guide to Pharmacology None None None None 14755056
1125 7069 0 None - 1 Rat 8.4 pKi None 8.4 Binding
UnclassifiedUnclassified
Guide to Pharmacology None None None None 7991622
1125 7069 0 None - 1 Rat 8.4 pKi None 8.4 Binding
UnclassifiedUnclassified
Guide to Pharmacology None None None None 9145431
1125 7069 0 None - 1 Rat 8.4 pKi None 8.4 Binding
UnclassifiedUnclassified
Guide to Pharmacology None None None None 9892695
1120 9476 0 None - 1 Rat 9.9 pKi None 9.9 Binding
UnclassifiedUnclassified
Guide to Pharmacology None None None None 7991622
1120 9476 0 None - 1 Rat 9.9 pKi None 9.9 Binding
UnclassifiedUnclassified
Guide to Pharmacology None None None None 9145431