Ligand source activities (1 row/activity)





Ligands (move mouse cursor over ligand name to see structure) Receptor Assay information Chemical information
Sel. page Common
name
GPCRdb
ID
#Vendors

Reference
ligand
Fold
selectivity
# Tested
GPCRs
Species

p-value
(-log)
Activity
Type
Activity
Relation
Activity
Value
AssayType

Assay
Description
Source

Mol
weight
Rot
Bonds
H don

H acc

LogP

Smiles

DOI

5572 8709 0 None - 1 Rat 7.6 pA2 = 7.6 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None None
129631922 10553 13 None -34 4 Rat 8.2 pIC50 = 8.2 Functional
NoneNone
Drug Central None None None None None
132274287 10553 13 None -34 4 Rat 8.2 pIC50 = 8.2 Functional
NoneNone
Drug Central None None None None None
132451761 10553 13 None -34 4 Rat 8.2 pIC50 = 8.2 Functional
NoneNone
Drug Central None None None None None
155817470 10553 13 None -34 4 Rat 8.2 pIC50 = 8.2 Functional
NoneNone
Drug Central None None None None None
16132393 10553 13 None -34 4 Rat 8.2 pIC50 = 8.2 Functional
NoneNone
Drug Central None None None None None
16133850 10553 13 None -34 4 Rat 8.2 pIC50 = 8.2 Functional
NoneNone
Drug Central None None None None None
4448 10553 13 None -34 4 Rat 8.2 pIC50 = 8.2 Functional
NoneNone
Drug Central None None None None None
4514 10553 13 None -34 4 Rat 8.2 pIC50 = 8.2 Functional
NoneNone
Drug Central None None None None None
91933454 10553 13 None -34 4 Rat 8.2 pIC50 = 8.2 Functional
NoneNone
Drug Central None None None None None
CHEMBL525610 10553 13 None -34 4 Rat 8.2 pIC50 = 8.2 Functional
NoneNone
Drug Central None None None None None
DB06285 10553 13 None -34 4 Rat 8.2 pIC50 = 8.2 Functional
NoneNone
Drug Central None None None None None
129631922 10553 13 None -7 4 Human 8.1 pIC50 = 8.1 Functional
NoneNone
Drug Central None None None None None
132274287 10553 13 None -7 4 Human 8.1 pIC50 = 8.1 Functional
NoneNone
Drug Central None None None None None
132451761 10553 13 None -7 4 Human 8.1 pIC50 = 8.1 Functional
NoneNone
Drug Central None None None None None
155817470 10553 13 None -7 4 Human 8.1 pIC50 = 8.1 Functional
NoneNone
Drug Central None None None None None
16132393 10553 13 None -7 4 Human 8.1 pIC50 = 8.1 Functional
NoneNone
Drug Central None None None None None
16133850 10553 13 None -7 4 Human 8.1 pIC50 = 8.1 Functional
NoneNone
Drug Central None None None None None
4448 10553 13 None -7 4 Human 8.1 pIC50 = 8.1 Functional
NoneNone
Drug Central None None None None None
4514 10553 13 None -7 4 Human 8.1 pIC50 = 8.1 Functional
NoneNone
Drug Central None None None None None
91933454 10553 13 None -7 4 Human 8.1 pIC50 = 8.1 Functional
NoneNone
Drug Central None None None None None
CHEMBL525610 10553 13 None -7 4 Human 8.1 pIC50 = 8.1 Functional
NoneNone
Drug Central None None None None None
DB06285 10553 13 None -7 4 Human 8.1 pIC50 = 8.1 Functional
NoneNone
Drug Central None None None None None
155817427 10006 0 None -158 3 Rat 5.5 pIC50 = 5.5 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
1788 10006 0 None -158 3 Rat 5.5 pIC50 = 5.5 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
129316189 10003 0 None -35 3 Rat 6.8 pIC50 = 6.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
155817471 10003 0 None -35 3 Rat 6.8 pIC50 = 6.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
16201228 10003 0 None -35 3 Rat 6.8 pIC50 = 6.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
4449 10003 0 None -35 3 Rat 6.8 pIC50 = 6.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
1824 8784 0 None - 1 Human 7.0 pIC50 = 7 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 10537121
155817427 10006 0 None -1 3 Human 7.5 pIC50 = 7.5 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
155817427 10006 0 None -1 3 Human 7.5 pIC50 = 7.5 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 8702701
1788 10006 0 None -1 3 Human 7.5 pIC50 = 7.5 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
1788 10006 0 None -1 3 Human 7.5 pIC50 = 7.5 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 8702701
129631922 10553 13 None -7 4 Human 7.8 pIC50 = 7.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
129631922 10553 13 None -7 4 Human 7.8 pIC50 = 7.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 8702701
132274287 10553 13 None -7 4 Human 7.8 pIC50 = 7.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
132274287 10553 13 None -7 4 Human 7.8 pIC50 = 7.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 8702701
132451761 10553 13 None -7 4 Human 7.8 pIC50 = 7.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
132451761 10553 13 None -7 4 Human 7.8 pIC50 = 7.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 8702701
155817470 10553 13 None -7 4 Human 7.8 pIC50 = 7.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
155817470 10553 13 None -7 4 Human 7.8 pIC50 = 7.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 8702701
16132393 10553 13 None -7 4 Human 7.8 pIC50 = 7.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
16132393 10553 13 None -7 4 Human 7.8 pIC50 = 7.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 8702701
16133850 10553 13 None -7 4 Human 7.8 pIC50 = 7.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
16133850 10553 13 None -7 4 Human 7.8 pIC50 = 7.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 8702701
4448 10553 13 None -7 4 Human 7.8 pIC50 = 7.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
4448 10553 13 None -7 4 Human 7.8 pIC50 = 7.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 8702701
4514 10553 13 None -7 4 Human 7.8 pIC50 = 7.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
4514 10553 13 None -7 4 Human 7.8 pIC50 = 7.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 8702701
91933454 10553 13 None -7 4 Human 7.8 pIC50 = 7.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
91933454 10553 13 None -7 4 Human 7.8 pIC50 = 7.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 8702701
CHEMBL525610 10553 13 None -7 4 Human 7.8 pIC50 = 7.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
CHEMBL525610 10553 13 None -7 4 Human 7.8 pIC50 = 7.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 8702701
DB06285 10553 13 None -7 4 Human 7.8 pIC50 = 7.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
DB06285 10553 13 None -7 4 Human 7.8 pIC50 = 7.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 8702701
3624 10597 0 None -5 2 Rat 8.1 pIC50 = 8.1 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
1815 10598 0 None 25 3 Human 8.4 pIC50 = 8.4 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 10854439
1815 10598 0 None 25 3 Human 8.4 pIC50 = 8.4 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
3624 10597 0 None 5 2 Human 8.8 pIC50 = 8.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
155817432 10007 0 None -446 3 Rat 5.3 pIC50 None 5.3 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
16144017 10007 0 None -446 3 Rat 5.3 pIC50 None 5.3 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
1822 10007 0 None -446 3 Rat 5.3 pIC50 None 5.3 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
155817428 10008 0 None -6 2 Human 5.7 pIC50 None 5.7 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 8702701
1790 10008 0 None -6 2 Human 5.7 pIC50 None 5.7 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 8702701
155817432 10007 0 None -70 3 Human 6.1 pIC50 None 6.1 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
16144017 10007 0 None -70 3 Human 6.1 pIC50 None 6.1 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
1822 10007 0 None -70 3 Human 6.1 pIC50 None 6.1 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
155817433 10600 0 None -125 3 Rat 6.1 pIC50 None 6.1 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
16134968 10600 0 None -125 3 Rat 6.1 pIC50 None 6.1 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
1827 10600 0 None -125 3 Rat 6.1 pIC50 None 6.1 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
1825 8777 0 None - 1 Human 6.2 pIC50 None 6.2 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
1820 8279 0 None -10 2 Rat 6.3 pIC50 None 6.3 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
1807 9878 0 None -5 2 Human 6.3 pIC50 None 6.3 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 8702701
129631922 10553 13 None -34 4 Rat 6.3 pIC50 None 6.3 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
132274287 10553 13 None -34 4 Rat 6.3 pIC50 None 6.3 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
132451761 10553 13 None -34 4 Rat 6.3 pIC50 None 6.3 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
155817470 10553 13 None -34 4 Rat 6.3 pIC50 None 6.3 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
16132393 10553 13 None -34 4 Rat 6.3 pIC50 None 6.3 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
16133850 10553 13 None -34 4 Rat 6.3 pIC50 None 6.3 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
4448 10553 13 None -34 4 Rat 6.3 pIC50 None 6.3 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
4514 10553 13 None -34 4 Rat 6.3 pIC50 None 6.3 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
91933454 10553 13 None -34 4 Rat 6.3 pIC50 None 6.3 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
CHEMBL525610 10553 13 None -34 4 Rat 6.3 pIC50 None 6.3 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
DB06285 10553 13 None -34 4 Rat 6.3 pIC50 None 6.3 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
155817434 10601 0 None -50 2 Rat 6.5 pIC50 None 6.5 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
1828 10601 0 None -50 2 Rat 6.5 pIC50 None 6.5 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
1794 8711 0 None 19 3 Human 6.6 pIC50 None 6.6 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 8702701
155817429 10009 0 None -3 2 Human 6.7 pIC50 None 6.7 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11046116
1814 10009 0 None -3 2 Human 6.7 pIC50 None 6.7 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11046116
1801 8782 0 None -3 2 Human 6.8 pIC50 None 6.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 10537121
1819 8280 0 None -3 2 Human 6.9 pIC50 None 6.9 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11046116
1821 8783 0 None -1 2 Human 7.0 pIC50 None 7 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 10537121
1815 10598 0 None -25 3 Rat 7.0 pIC50 None 7 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
155817433 10600 0 None -12 3 Human 7.1 pIC50 None 7.1 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11046116
155817433 10600 0 None -12 3 Human 7.1 pIC50 None 7.1 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
16134968 10600 0 None -12 3 Human 7.1 pIC50 None 7.1 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11046116
16134968 10600 0 None -12 3 Human 7.1 pIC50 None 7.1 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
1827 10600 0 None -12 3 Human 7.1 pIC50 None 7.1 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11046116
1827 10600 0 None -12 3 Human 7.1 pIC50 None 7.1 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
1800 8781 0 None -3 2 Human 7.2 pIC50 None 7.2 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 10537121
1820 8279 0 None 10 2 Human 7.3 pIC50 None 7.3 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
1799 8780 0 None -1 2 Human 7.3 pIC50 None 7.3 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 10537121
1808 10644 0 None 2 2 Human 7.4 pIC50 None 7.4 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 9360953
1809 10643 0 None 1 2 Human 7.5 pIC50 None 7.5 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 8702701
1798 8779 0 None -1 2 Human 7.6 pIC50 None 7.6 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 10537121
1798 8779 0 None -1 2 Human 7.6 pIC50 None 7.6 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 8702701
1797 8785 0 None 1 2 Human 7.7 pIC50 None 7.7 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 9360953
155817434 10601 0 None 50 2 Human 8.2 pIC50 None 8.2 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
1828 10601 0 None 50 2 Human 8.2 pIC50 None 8.2 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
129316189 10003 0 None 15 3 Human 8.4 pIC50 None 8.4 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 10537121
129316189 10003 0 None 15 3 Human 8.4 pIC50 None 8.4 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 10854439
129316189 10003 0 None 15 3 Human 8.4 pIC50 None 8.4 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
155817471 10003 0 None 15 3 Human 8.4 pIC50 None 8.4 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 10537121
155817471 10003 0 None 15 3 Human 8.4 pIC50 None 8.4 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 10854439
155817471 10003 0 None 15 3 Human 8.4 pIC50 None 8.4 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
16201228 10003 0 None 15 3 Human 8.4 pIC50 None 8.4 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 10537121
16201228 10003 0 None 15 3 Human 8.4 pIC50 None 8.4 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 10854439
16201228 10003 0 None 15 3 Human 8.4 pIC50 None 8.4 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
4449 10003 0 None 15 3 Human 8.4 pIC50 None 8.4 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 10537121
4449 10003 0 None 15 3 Human 8.4 pIC50 None 8.4 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 10854439
4449 10003 0 None 15 3 Human 8.4 pIC50 None 8.4 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681




Ligands (move mouse cursor over ligand name to see structure) Receptor Assay information Chemical information
Sel. page Similar-
ity
Common
name
GPCRdb
ID
#Vendors

Reference
ligand
Fold
selectivity
# Tested
GPCRs
Species

p-value
(-log)
Activity
Type
Activity
Relation
Activity
Value
Assay
Type
Assay
Description
Source

Mol
weight
Rot
Bonds
H don

H acc

LogP

Smiles

DOI