Ligand source activities (1 row/activity)





Ligands (move mouse cursor over ligand name to see structure) Receptor Assay information Chemical information
Sel. page Common
name
GPCRdb
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ligand
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selectivity
# Tested
GPCRs
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p-value
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Activity
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Activity
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Source

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DOI

1079 7688 44 None 63 4 Rat 6.7 pEC50 None 6.7 Functional
UnclassifiedUnclassified
Guide to Pharmacology 292 3 2 2 4.5 OCC(Cc1cc(c(c(c1)C(C)(C)C)O)C(C)(C)C)(C)C 11641424
1079 7688 44 None 63 4 Rat 6.7 pEC50 None 6.7 Functional
UnclassifiedUnclassified
Guide to Pharmacology 292 3 2 2 4.5 OCC(Cc1cc(c(c(c1)C(C)(C)C)O)C(C)(C)C)(C)C 15126507
5024764 7688 44 None 63 4 Rat 6.7 pEC50 None 6.7 Functional
UnclassifiedUnclassified
Guide to Pharmacology 292 3 2 2 4.5 OCC(Cc1cc(c(c(c1)C(C)(C)C)O)C(C)(C)C)(C)C 11641424
5024764 7688 44 None 63 4 Rat 6.7 pEC50 None 6.7 Functional
UnclassifiedUnclassified
Guide to Pharmacology 292 3 2 2 4.5 OCC(Cc1cc(c(c(c1)C(C)(C)C)O)C(C)(C)C)(C)C 15126507
CHEMBL1256697 7688 44 None 63 4 Rat 6.7 pEC50 None 6.7 Functional
UnclassifiedUnclassified
Guide to Pharmacology 292 3 2 2 4.5 OCC(Cc1cc(c(c(c1)C(C)(C)C)O)C(C)(C)C)(C)C 11641424
CHEMBL1256697 7688 44 None 63 4 Rat 6.7 pEC50 None 6.7 Functional
UnclassifiedUnclassified
Guide to Pharmacology 292 3 2 2 4.5 OCC(Cc1cc(c(c(c1)C(C)(C)C)O)C(C)(C)C)(C)C 15126507
2997 199930 35 None -13 4 Human 8.1 pIC50 = 8.1 Functional
NoneNone
Drug Central 270 1 1 2 3.1 O=C1CN=C(c2ccccc2)c2cc(Cl)ccc2N1 None
CHEMBL523 199930 35 None -13 4 Human 8.1 pIC50 = 8.1 Functional
NoneNone
Drug Central 270 1 1 2 3.1 O=C1CN=C(c2ccccc2)c2cc(Cl)ccc2N1 None




Ligands (move mouse cursor over ligand name to see structure) Receptor Assay information Chemical information
Sel. page Similar-
ity
Common
name
GPCRdb
ID
#Vendors

Reference
ligand
Fold
selectivity
# Tested
GPCRs
Species

p-value
(-log)
Activity
Type
Activity
Relation
Activity
Value
Assay
Type
Assay
Description
Source

Mol
weight
Rot
Bonds
H don

H acc

LogP

Smiles

DOI