Mutant Browser

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Protein name Generic number Position Segment Mutation FoldChange or Qual Exp Type Ligand Reference Review
oprx_human 6.52x52 280 TM6 Q => H N/A N/A Mollereau C et al (1996)
oprx_human 2.66x66 113 TM2 L => M N/A N/A Bes B et al (2003)
oprx_human 3.32x32 130 TM3 D => A N/A N/A Mouledous L et al (2000)
oprx_human 3.32x32 130 TM3 D => E N/A N/A Mouledous L et al (2000)
oprx_human 3.32x32 130 TM3 D => N N/A N/A Mouledous L et al (2000)
oprx_human 3.33x33 131 TM3 Y => A N/A N/A Mouledous L et al (2000)
oprx_human 3.33x33 131 TM3 Y => F N/A N/A Mouledous L et al (2000)
oprx_human 3.35x35 133 TM3 N => W N/A N/A Kam KW et al (2002)
oprx_human 5.43x44 220 TM5 F => A N/A N/A Mouledous L et al (2000)
oprx_human 5.47x47 224 TM5 F => A N/A N/A Mouledous L et al (2000)
oprx_human 6.48x48 276 TM6 W => A N/A N/A Mouledous L et al (2000)
oprx_human 6.52x52 280 TM6 Q => H N/A N/A Mollereau C et al (1996)
oprx_human 6.58x58 286 TM6 Q => A N/A N/A Mouledous L et al (2000)
oprx_human 6.58x58 286 TM6 Q => E N/A N/A Mouledous L et al (2000)
oprx_human 7.29x28 295 TM7 E => D N/A N/A Mouledous L et al (2000)
Protein name Generic number Segment Position Mutation FoldChange or Qual Exp Type Ligand Reference Review


Residue

Diagrams

ICL1 T K M K ICL1ECL1 F W P F ECL1ICL2 P I R A L D V R ICL2ECL2 S A Q V E D E E I E C L V E I P T ECL2ICL3 R L L S G ICL3ECL3 V Q P S ECL3N-term M E P L F P A P F W E V I Y G S H L Q G N L S L L S P N H S L L P P H L L L N A S H G A F L P N-termC-term A S A L R R D V Q V S D R V R S I A K D V A L A C K T S E T V P R P A C-term L G L K V T I V G L Y L A V C V G G L L G N C L V M Y V I L R H T A T N I Y I F N L A L A D T L V L L T L P F Q G T D I L L G G N A L C K T V I A I D Y Y N M F T S T F T L T A M S V D R Y V A I C H T S S K A Q A V N V A I W A L A S V V G V P V A I M G P Q D Y W G P V F A I C I F L F S F I V P V L V I S V C Y S L M I R R L R G V S R E K D R N L R R I T R L V L V V V A V F V G C W T P V Q V F V L A Q G L G S E T A V A I L R F C T A L G Y V N S C L N P I L Y A F L D E N F R K F K A C F C C
Download: PNG | SVG Increased binding/potency: >5-fold, >10-fold; Reduced binding/potency: >5-fold, >10-fold; No/low effect (<5-fold); and N/A
C N G L L G G V C V A L Y L G V I T V K 1 F N L A L A D T L V L L T L P F Q G T D 2 A T L T F T S T F M N Y Y D I A I V T K 3 A Q A V N V A I W A L A S V V G V P V A 4 Y C V S I V L V P V I F S F L F I C I A F 5 L V V V A V F V G C W T P V Q V F V L A 6 I P N L C S N V Y G L A T C F R L I A 7
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Residue Table


GPCRdb(A)
GPCRdb(A)
NOP receptor
TM2
2x66 2.66x66 L113
TM3
3x32 3.32x32 D130
3x33 3.33x33 Y131
3x35 3.35x35 N133
TM5
5x44 5.43x44 F220
5x47 5.47x47 F224
TM6
6x48 6.48x48 W276
6x52 6.52x52 Q280
6x58 6.58x58 Q286
TM7
7x28 7.29x28 E295