GPCR CLASS (FAMILY)
Class A (Rhodopsin)
PDB CODE
SPECIES
Homo sapiens
RESOLUTION
3.3 Å
PREFERRED CHAIN
A
REFERENCE
PUBLICATION DATE
April 12, 2023
LIGAND INTERACTIONS
LIGANDS
nalfurafine - Agonist pubchem gtoplig chembl_ligand drug_central drugbank
PHYSIOLOGICAL LIGANDS
[Met]enkephalin (Human), β-neoendorphin (Human), dynorphin A (Human), dynorphin A-(1-8) (Human), dynorphin A-(1-13) (Human), big dynorphin (Human), β-endorphin (Mouse), β-endorphin (Rat), dynorphin B (Human), β-endorphin (Human), α-neoendorphin (Human), [Leu]enkephalin (Human)